| Patents for C07D 411 - Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms (2,465) |
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| 03/10/2010 | EP2161267A1 A process for stereoselective synthesis of lamivudine |
| 03/09/2010 | US7674823 DNA-PK inhibitors |
| 03/04/2010 | WO2010023676A2 Process for preparing lamivudine polymorph form |
| 02/24/2010 | EP1465631B1 Pyrimidine a2b selective antagonist compounds, their synthesis and use |
| 02/23/2010 | US7667044 treating nervous system diorders such as Alzheimer's disease, Down Syndrome, Parkinson disease and Huntington chorea by administering inhibitors of prolyl endopeptidases |
| 02/16/2010 | US7662811 1,2,3,4-tetrahydropyrazin-2-yl acetamides and methods of use |
| 02/16/2010 | CA2452918C New compounds, which are potent inhibitors of na+/ca2+ exchange mechanism and are useful in the treatment of arrhythmias |
| 02/11/2010 | WO2010016230A1 Sulfoxyimino-substituted benzoyl derivative and herbicide |
| 02/09/2010 | US7659280 2,4-pyrimidinediamine compounds for treating or preventing autoimmune diseases |
| 02/09/2010 | CA2439593C Heterocyclic compounds for aging-related and diabetic vascular complications |
| 02/09/2010 | CA2291065C Raf kinase inhibitors |
| 02/02/2010 | US7655665 Nitromethylene derivatives and their use |
| 01/12/2010 | CA2439831C Polymorphic and other crystalline forms of cis-ftc |
| 01/07/2010 | US20100004263 Mtp inhibiting aryl piperidines or peperazines substituted with5-membered heterocycles |
| 01/06/2010 | CN101619057A N-substituted piperidine derivatives as serotonin receptor agents |
| 01/05/2010 | US7642354 Polycyclic pyrazines as potassium ion channel modulators |
| 12/29/2009 | US7638515 improved selectivity and pharmacokinetic properties; 6-Fluoro-1-[(1 H-indazol-4-yl)amino]-4,4-dimethyl-2-(trifluoromethyl)-1,2,3,4-tetrahydronaphthalene-2,5-diol; cyclization of imines |
| 12/29/2009 | CA2478799C Di-aryl substituted tetrazole modulators of metabotropic glutamate receptor-5 |
| 12/24/2009 | US20090318472 Aminopyrazine derivatives and compositions |
| 12/23/2009 | EP1296972B1 Arylmethylamine derivatives for use as tryptase inhibitors |
| 12/22/2009 | CA2114221C 1, 3-oxathiolane nucleoside analogues |
| 12/15/2009 | CA2481078C Method and compositions for the synthesis of bch-189 and related compounds |
| 12/10/2009 | US20090306114 Polymorphic and Other Crystalline Forms of Cis-FTC |
| 12/09/2009 | EP2130820A1 Antipruritics |
| 12/09/2009 | CN101597281A Preparation method of lamivudine and intermediate thereof |
| 12/08/2009 | US7629343 Carbamic acid compounds comprising a piperazine linkage as HDAC inhibitors |
| 11/19/2009 | US20090286787 Substituted gamma lactams as therapeutic agents |
| 11/18/2009 | EP2018367B1 Novel microbiocides |
| 11/18/2009 | EP0760811B1 Imidazole derivatives as histamine receptor h3 modulators |
| 11/12/2009 | WO2009084033A3 Process for producing 5-fluoro-1-(2r,5s)-[2-(hydroxymethyl)-1,3-oxathiolan-5-yi]cytosine |
| 11/11/2009 | EP1477186B1 Antipruritics |
| 11/05/2009 | WO2009133831A1 Phenylpropionic acid derivative and use thereof |
| 10/29/2009 | US20090270374 Derivatives and analogs of n-ethylquinolones and n-ethylazaquinolones |
| 10/28/2009 | CN101568534A Benzoyl amino heterocyclyl compounds useful in the treatment of a disease mediated through GLK |
| 10/22/2009 | WO2009127996A1 Novel crystalline form of lamivudine |
| 10/14/2009 | EP1658267B1 Inhibitors of cathepsin s |
| 10/14/2009 | CN100548992C Microbiocidal (e.g. fungicidal) 1,2,3-triazole derivatives |
| 10/14/2009 | CN100548988C Metabolites of ecteinascidin 743 |
| 10/14/2009 | CN100548987C Pesticidal pyridinecarboxamide derivatives |
| 10/06/2009 | US7598397 Sulfonamide peri-substituted bicyclics for occlusive artery disease |
| 10/06/2009 | US7598251 aminopyrazine derivatives; ROCK inhibitors; 3-(1-ethyl-1H-imidazo[4,5-c]pyridin-2-yl)pyrazin-2-amine; antiinflammatory, antidiabetic, antiproliferative agents |
| 10/01/2009 | WO2009118765A2 Novel monoamine re-uptake inhibitor |
| 10/01/2009 | US20090247487 Combination Therapy to Treat Hepatitis B Virus |
| 10/01/2009 | US20090246819 Assay Methods Using Chemiluminescent Detection of Peroxidase |
| 09/30/2009 | CN101544632A Lamivudine diastereoselective synthesis method |
| 09/29/2009 | US7595321 Useful for the prevention and/or treatment of cognitive disorders; 3-Amino-N-(2-cyanoethyl)-6-[4-(pyrrolidin-1-ylsulfonyl)phenyl]pyrazine-2-carboxamide, for example |
| 09/29/2009 | US7595319 Compounds having selective inhibiting effect at GSK3 |
| 09/24/2009 | WO2009116055A1 Lamivudine : zidovudine : water 1 : 1 : 1 cocrystal |
| 09/23/2009 | CN100542535C Preparation method of medicinal composition containing 1,3-oxathin cyclopentane nucleoside analogues |
| 09/22/2009 | CA2209640C Cycloalkano-pyridines |
| 09/16/2009 | CN101531656A Lamivudine crystal form and preparation method thereof |
| 09/11/2009 | WO2009111635A2 Dithiol compounds, derivatives, and uses therefor |
| 09/11/2009 | WO2009111633A2 Mercaptan and seleno-mercaptan compounds and methods of using them |
| 09/11/2009 | WO2009005338A8 Solid forms ult-i, ult-2 and ult-3 of emtricitabine |
| 09/08/2009 | US7585853 Compounds having selective inhibiting effect at GSK3 |
| 09/02/2009 | EP2096110A1 Acridane-9-dithiocarboxylate derivatives for generating chemiluminescence with a peroxidase |
| 09/01/2009 | US7582589 3-carbonylaminothiophenes and their use as fungicides |
| 08/27/2009 | US20090216027 Microbiocidal (e.g. fungicidal) 1,2,3-triazole derivatives |
| 08/27/2009 | US20090216014 Novel compounds and methods of treating cell proliferative diseases, retinopathies and arthritis |
| 08/18/2009 | US7576209 Breast, prostate and ovarian cancer; such as 1-[4-(9-phenyl-3-pyrimidin-2-yl[1,2,4]triazolo[3,4-f]-1,6-naphthyridin-8-yl)phenyl]cyclobutanamine; serine/threonine kinase (Akt) suppression |
| 08/18/2009 | US7576204 (8E,12E,14E)-21-benzoyloxy-3,6-dihydroxy-6,10,12,16,20-pentamethyl-7-((4-methylpiperazin-1-yl)carbonyl)oxy-18,19-epoxytricosa-8,12,14-trien-11-olide; inhibits angiogenesis and inhibits the production of VEGF particularly under hypoxic conditions, which makes it useful as a remedy for solid cancer |
| 08/18/2009 | US7576088 Benzodioxole derivatives |
| 08/18/2009 | US7576086 N1-benzyl-N4-(phenylpropane-2-yl-3-ol)piperazine; triple action on hydroxytryptamine (5-HT), noradrenalin (NA)and dopamine(DA); on brain synapses; cytochrome P-450 monooxygenase enzyme system antagonists; enzyme inhibitors; side effect reduction |
| 08/18/2009 | US7576076 1-Methyl,2,6-dioxo,4-(4-(ethyloxycarbony)piperazin-1-yl-),5-(3-trifluoromethylphenyl)methyl-)-1,2,3,6-tetrahydropyrimidine; antagonist, antagonism; psychoses; antidepressants; schizophrenia; psychological disorders; Alzheimer's disease; neurodegenerative diseases;drug abuse, drug dependence (cocaine) |
| 08/13/2009 | WO2009037538A3 Process for the preparation of lamivudine form i |
| 08/12/2009 | EP2086964A2 Benzoyl amino heterocyclyl compounds useful in the treatment of a disease mediated through glk |
| 08/12/2009 | CN101506206A Inhibitors of Akt activity |
| 08/12/2009 | CN100526310C Cyclopropyl-thienyl-carboxamide as fungicides |
| 08/11/2009 | US7572800 Administering anti-hepatitis B virus agents in combination or alternation such asbeta-2-hydroxymethyl-5-(5-fluorocytosin-1-yl-1,3-oxathiolane or a salt and one another antihepatitis B agent |
| 08/06/2009 | US20090197925 O-cyclopropyl-carboxanilides and their use |
| 07/30/2009 | US20090192310 Process and Intermediates for Preparing Emtricitabine |
| 07/23/2009 | WO2009005338A3 Solid forms ult-i, ult-2 and ult-3 of emtricitabine |
| 07/23/2009 | US20090186932 Pesticidal N-Phenylpyrazole Derivatives |
| 07/22/2009 | CN100516066C Compounds for treating impaired fundic relaxation |
| 07/16/2009 | WO2009058800A3 Synthesis of nucleosides |
| 07/14/2009 | US7560556 Assay methods using chemiluminescent detection of peroxidase |
| 07/14/2009 | US7560466 N4-(2,2-Dimethyl-3-oxo-4H-5-pyrid[1,4]oxazin-6-yl)-N2-(3-chloro-4-methoxyphenyl)-5-fluoro-2,4-pyrimidinediamine; signal transduction cascade inhibitor; Fc receptors for IgE (Fc epsilon RI) and IgG (Fc gamma RI) antagonist; autoimmune diseases, antiinflammatory agent; rheumatoid arthritis |
| 07/14/2009 | US7560462 Compounds useful for inhibiting CHK1 |
| 07/14/2009 | US7560460 2-[(4-Chlorophenyl)methyl]-1-(4- {2-[(cyclopropylmethyl)-(methylsulfonyl)amino]phenyl }-piperazinyl) -4-(2-(1,2,3,4-tetrahydroisoquinolyl))butane-1,4-dione; obesity/dietietics; melanocortin receptor angonists; prophylaxis/treatment of diseases involving activation of the melanocortin recepetors (MCR) |
| 07/14/2009 | US7560456 Pesticidal pyridinecarboxamide derivatives |
| 07/14/2009 | US7560451 Aspartyl protease inhibitors |
| 07/09/2009 | WO2009084033A2 Process for producing 5-fluoro-1-(2r,5s)-[2-(hydroxymethyl)-1,3-oxathiolan-5-yi]cytosine |
| 07/09/2009 | US20090176801 Novel lapachone compounds and methods of use thereof |
| 07/08/2009 | CN100509804C N-substituted piperidine derivatives as serotonin receptor agents |
| 07/02/2009 | US20090171086 2,4-pyrimidinediamine compounds and their uses |
| 06/25/2009 | WO2009077954A1 Aminopyrazole derivatives |
| 06/25/2009 | CA2706836A1 Aminopyrazole derivatives |
| 06/18/2009 | WO2009074019A1 Proteinase inhibitors useful for treating cancer |
| 06/18/2009 | US20090156628 Aminothiazoles and their Uses |
| 06/18/2009 | US20090156574 N-(4-(5-Butyl-2-methoxyphenyl)-1,3-thiazol-2-yl)-4-((4-oxopiperidin-1-yl)carbonyl)benzamide; antiinflammatory, anticarcinogenic, antidiabetic, analgesic agents |
| 06/16/2009 | US7547782 Met kinase inhibitors |
| 06/09/2009 | US7544692 Dissolved in water; recrystallized, dehydrated; lymphadenopathy associated virus, human T-cell leukemia/lymphoma virus, hepatitis virus |
| 06/04/2009 | WO2009069014A1 Amorphous lamivudine and its preparation |
| 06/04/2009 | WO2009069013A1 Crystalline form i of lamivudine and its preparation |
| 06/04/2009 | WO2009069012A1 Process and intermediates for the preparation of substituted 1, 3-oxathiolanes, especially lamivudine |
| 06/04/2009 | WO2009069011A1 Process for the preparation of substituted 1,3-oxathiolanes |
| 06/02/2009 | US7541472 3-Aryl-3-hydroxy-2-methylenepropionic acid esters as fungicides |
| 06/02/2009 | US7541368 Pyrazoles as inhibitors of tumor necrosis factor |
| 05/28/2009 | US20090137570 Inhibitors of cathepsin s |
| 05/22/2009 | WO2009010260A3 Condensed anthranilamide insecticides |