Patents
Patents for C07D 411 - Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms (2,465)
03/2007
03/13/2007CA2351049C Process for recovery of the desired cis-1,3-oxathiolane nucleosides from their undesired trans-isomers
03/08/2007US20070054899 Aromatase inhibitor compounds and uses thereof
03/07/2007CN1923832A Novel pyridazinone compound, preparation method and application thereof
03/01/2007WO2005117882A9 Hydroxamic acid derivatives as metalloprotease inhibitors
02/2007
02/28/2007CN1920050A Method of resolution of 1,3-oxathiolane nucleoside enantiomers
02/27/2007US7183295 Compound for treatment of lipemic agents, antiinflammatory agents and treatment of diabetes
02/20/2007CA2180156C Self-assembled taxo-diperpenoid nanostructures
02/15/2007US20070037977 Substituted-1, 3-oxathiolanes and substituted-1, 3-dioxolanes with antiviral properties
02/15/2007US20070037975 Substituted-1,3-oxathiolanes and substituted-1, 3-dioxolanes with antiviral properties
02/14/2007EP1534391B1 Novel piperazinyl-pyrazinone derivatives for the treatment of 5-ht2a receptor-related disorders
02/13/2007US7176242 N,N′-substituted-1,3-diamino-2-hydroxypropane derivatives
02/06/2007US7173134 retinoid X receptors ("RXRs"); useful for the treatment of diabetes (NIDDIM) and obesity; for example, 3-{4-[(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-2-naphthalenyl)methyl]-2-furyl}-2-propenoic acid
02/06/2007US7173129 Sulfonamide-substituted chalcone derivatives and their use to treat diseases
01/2007
01/31/2007CN1297553C Stereoselective methods for the preparation of nucleosides
01/30/2007CA2297011C Sulfonamide derivatives as therapeutic or prophylactic agent for glomerulopathy
01/18/2007WO2007006739A1 Benzoheterocyclylethylcarboxamide derivatives
01/18/2007WO2007006547A1 Amide derivatives as kinase inhibitors
01/17/2007CN1898210A 2-pyridinylethylcarboxamide derivatives and their use as fungicides
01/17/2007CN1896064A Metabolites of ecteinascidin 743
01/17/2007CN1295228C Nitryl methylene derivatives and uses thereof
01/11/2007US20070010563 Novel methods for the treatment of inflammatory diseases
01/10/2007EP1740544A1 2-pyridinylcycloalkylcarboxamide derivatives useful as fungicides
01/10/2007CN1891221A Combination therapy to treat hepatitis b virus
01/09/2007US7160999 The nucleoside enantiomer (-)-2-hydroxymethyl-5-(5-fluorocytosin-1-yl) -1,3-oxathiolane is an effective antiviral agent against HIV, HBV, and other viruses replicating in a similar manner
01/03/2007EP0958292B1 4-(3-heterocyclyl-1-benzoyl)pyrazoles and their use as herbicides
01/03/2007CN1293058C O-cyclopropyl-carboxanilides and their use as fungicides
12/2006
12/27/2006CN1886403A Use of a compound of formula (i) as an inhibitor of aromatase for therapeutic purposes and compounds of formula (1) thereas
12/26/2006US7153852 Skin disorders; antiinflammatory agents; brain disorders; chronic obstructive pulmonary disease; antiarthritic agents; inflammatory bowel disorders
12/21/2006WO2005092856A8 Tetrahydrocarbazoles and derivatives
12/21/2006US20060287361 Diarylmethylidene piperidine derivatives, preparations thereof and uses thereof as opoid receptors ligands
12/21/2006US20060287293 1-(4-{ethyl-[2-(4-methanesulfonylphenyl)-1-methylethyl]amino}butyl)-4-methanesulfonyl-[1,4]diazepan-2-one; repiratory system disorders: asthma and chronic obstructive pulmonary disease; nervous system, muscular,urogenital, gastrointestinal disorders; antiallergens; side effect reduction
12/20/2006EP1732892A1 Tetrahydrocarbazoles and derivatives
12/20/2006EP1732564A1 Biaryl substituted pyrazinones as sodium channel blockers
12/20/2006EP1608644B8 Process and intermediates for preparing emtricitabine
12/20/2006CN1290845C Process for synthesis of nucleoside analogue
12/20/2006CN1290841C Process for the non-enantiomorph selective synthesis of nucleoside analogues
12/14/2006WO2006073589A3 Cycloalkyl keto piperidine tachykinin receptor antagonists
12/07/2006WO2006057977A3 Cycloalkyl piperidine tachykinin receptor antagonists
12/07/2006US20060276492 Treating human immunodeficiency and hepatitis B infections; high activity, low toxicity
12/07/2006US20060276434 3-Carbonylaminothiophenes and their use as fungicides
12/06/2006CN1288157C Dioxadiene pyridine compounds for treating impaired fundic relaxation, method of preparation and use thereof
11/2006
11/30/2006WO2006125972A1 Heteroaryl benzamide derivatives for use as glk activators in the treatment of diabetes
11/30/2006CA2609235A1 Heteroaryl benzamide derivatives for use as glk activators in the treatment of diabetes
11/29/2006EP1725535A2 Hiv integrase inhibitors
11/29/2006CN1871216A Inhibitors of cathepsin s
11/28/2006CA2113603C Tricyclic condensed heterocyclic compounds, their production and use
11/21/2006US7138426 Estrogen receptor modulators
11/16/2006WO2005117882A3 Hydroxamic acid derivatives as metalloprotease inhibitors
11/14/2006US7135495 Indole derivatives
11/14/2006US7135479 Compounds which are both serotonin reuptake inhibitors and antagonists of the 5HT1A receptor
11/09/2006WO2005079802A8 Bipyridyl amides as modulators of metabotropic glutamate receptor-5
11/02/2006US20060247189 Forms of 5-Azacytidine
11/02/2006EP1715867A1 Bipyridyl amides as modulators of metabotropic glutamate receptor-5
11/02/2006EP1608644B1 Process and intermediates for preparing emtricitabine
10/2006
10/26/2006WO2006036941A3 Specific kinase inhibitors
10/26/2006US20060241147 Pyridine derivatives useful for inhibiting sodium/calcium exchange system
10/25/2006CN1281597C New compounds, which are potent inhibitors of Na<+>/Ca<2+> exchange mechanism and are useful in the treatment of arrhythmias
10/24/2006CA2442615C A reduced ignition propensity smoking article
10/24/2006CA2168023C Vasoconstrictive substituted aryloxyalkyl diamines
10/19/2006WO2006109846A1 Triazole derivative and the use thereof
10/19/2006WO2006108791A2 Heterocyclylethylheterocyclylcarboxamide derivatives as fungicides
10/19/2006US20060234987 Neuroprotective benzo 1 3 oxathiol 2 ones
10/17/2006US7122693 Acetaldehyde acetal compounds, their synthesis, and uses thereof
10/11/2006CN1845673A Pyridinylanilides
10/11/2006CN1279034C Dna-pk抑制剂 Dna-pk inhibitors
10/10/2006US7119203 Piperidinyl- and piperazinyl-sulfonylmethyl hydroxamic acids and their use as protease inhibitors
10/10/2006US7119202 Substituted-1,3-oxathiolanes and substituted-1,3-dioxolanes with antiviral properties
10/05/2006WO2006103511A1 Cyclopentapyridine and tetrahydroquinoline derivatives
10/03/2006US7115743 For treatment of leukemia, carcinomas, adenocarcinomas, and melanoma; assaying metabolism via cytochromes
10/03/2006US7115661 Methods and compositions for mitigating pain
09/2006
09/28/2006US20060217379 1,2,3-Trisubstituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto such as diabetes and hyperglycemia
09/27/2006EP1705179A1 N-aroyl cyclic amine derivatives as orexin receptor antagonists
09/27/2006EP1383757B1 Antagonists of mcp-1 function and methods of use thereof
09/21/2006WO2006096954A1 Process and methods for the preparation of optically active cis-2-hydroxymethyl-4-(cytosin-1´-yl)-1,3-oxathiolane or pharmaceutically acceptable salts thereof
09/20/2006EP0889889B1 Piperazine and piperidine compounds
09/19/2006US7109334 Predominantly cis nucleosides or nucleoside analogues and derivatives from 2-oxymethyl- thiolane-S-oxide, oxathiolane-S-oxide or dithiolane-S-oxide and a pyridine, pyrimidine or triazine base
09/19/2006US7109234 Benzoxathiepine derivatives and their use as medicines
09/14/2006US20060205722 Such as N-{1-[2-(1,3-dioxan-2-yl)ethyl]piperidin-4-yl}-N-(4-fluorobenzyl)-2-[4-(2-hydroxy-2-methylpropoxy)phenyl]acetamide; selective inverse agonists of 5-HT2A receptor with minimal monamine receptors subtype activity; antipsychotics with reduced side effects
09/13/2006CN1274687C Suitqable to industrialized method for preparing emtricitabine
09/13/2006CN1274686C Suitable industrialized method of preparing Lamivudine
09/08/2006WO2005086700A3 Hiv integrase inhibitors
09/07/2006US20060199818 Inhibiting the activity of a 5-hydroxytryptamine 2A by administering a N-heterocyclyl (preferably 1,3-dioxan-5-yl)-4-[(N-substituted)(hetero)arylamino]piperidine in which the N-substituant is arylalkanoyl, arylthioalkanoyl, arylalkylaminocarbonyl or arylalkylaminothiocarbonyl group
09/05/2006US7101867 Benzofuran derivatives, their production and use
08/2006
08/31/2006WO2006062984A3 Inhibitors of protein kinases
08/30/2006EP1694649A1 2-pyridinylethylcarboxamide derivatives and their use as fungicides
08/30/2006EP1412343B1 Compounds, which are potent inhibitors of na+/ca2+ exchange mechanism and are useful in the treatment of arrhythmias
08/29/2006US7098234 Indole derivatives, process for preparation of the same and use thereof
08/24/2006WO2006088711A1 AZOLYLACYLGUANIDINES AS β-SECRETASE INHIBITORS
08/24/2006US20060189805 Characterized by the formation and isolation of intermediate compounds in salified form; by using the intermediate of the present process in the subsequent reductive passage, it is possible to obtain emtricitabine in a purity that allows its direct crystallization; viricides
08/24/2006CA2597594A1 Azolylacylguanidines as beta-secretase inhibitors
08/23/2006EP1693373A1 Enantiomerically pure beta-D-(-)-dioxolane-nucleosides
08/22/2006US7094778 Nervous system disorders; muscular disorders; urogenital disorders; gastrointestinal disorders; repiratory system disorders; antiallergens; side effect reduction
08/17/2006US20060183899 Having a predominantly cis configuration by coupling an S-oxide of a 2-oxymethyl- thiolane, dithiolane or oxathiolane with a nucleoside base in the presence of a tertiary amine, a Lewis acid of a Group 1B or 2B metal catalyst and deprotecting the intermediate formed
08/17/2006US20060183749 Novel compounds and methods of treating cell proliferative diseases, retinopathies and arthritis
08/10/2006WO2006062982A3 Urea inhibitors of map kinases
08/10/2006US20060178513 Pyridinylanilides
08/09/2006EP1687301A1 Thiaepothilone for treating cancerous diseases
08/09/2006EP1597253B1 Compounds and methods of treating cell proliferative diseases, retinopathies and arthritis
08/03/2006WO2006051477A3 Fused tricyclic compounds as inhibitors of tumor necrosis factor-alpha
08/03/2006CA2595855A1 Pyrazine compounds for inflammation and immune-related uses
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