Patents
Patents for C07D 409 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms (52,226)
10/2001
10/02/2001US6297259 Substituted N-methyl-N-(4-(piperidin-1-yl)-2-(aryl)butyl) benzamides useful for the treatment of allergic diseases
10/02/2001US6297233 Lactam inhibitors of FXa and method
10/02/2001US6297196 Benzoyl derivatives, process for their preparation and their use as herbicides and plant growth regulators
10/02/2001CA2156908C C9 taxane derivatives and pharmaceutical compositions containing them
10/02/2001CA2037541C Azabicyclo and azacyclo oxime and amine cholinergic agents and methods of treatment
09/2001
09/27/2001WO2001070736A1 N-(heterocyclyl)benzene or pyridine sulphonamides as antithrombotic agents and anticoagulants
09/27/2001WO2001070734A2 Beta-amino acid derivatives as inhibitors of matrix metalloproteases and tnf-alpha
09/27/2001WO2001070729A1 2-amino-3-(alkyl)-pyrimidone derivatives as gsk3.beta. inhibitors
09/27/2001WO2001070727A1 2-(arylalkylamino)pyrimidone derivatives and 2-(heteroarylalkylamino)pyrimidone derivatives
09/27/2001WO2001070700A1 4,5-dihydro-1h-pyrazole derivatives having cb1-antagonistic activity
09/27/2001WO2001070690A1 Heterocyclic side chain containing metalloprotease inhibitors
09/27/2001WO2001070677A1 Sulphonamido-substituted bridged bicycloalkyl derivatives
09/27/2001WO2001070673A2 CYCLIC β-AMINO ACID DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEASES AND TNF-$g(a)
09/27/2001WO2001070269A1 Keratinocyte growth inhibitors and hydroxamic acid derivatives
09/27/2001WO2001070232A1 Protease inhibitors
09/27/2001WO2001070228A1 Antagonists of gonadotropin releasing hormone
09/27/2001WO2001070227A1 Antagonists of gonadotropin releasing hormone
09/27/2001WO2001032654A3 Novel heterocyclic compounds and their use as medicines
09/27/2001WO2001017972A3 Novel herbicides
09/27/2001US20010025105 Anticancer agent; Alzheimer's therapy
09/27/2001US20010025047 Nitrogen containing bicyclic heteroaromatic compound containing sulfonamide and hydroxyamide groups, useful in treatment of arthritis, tumor metastasis, tissue ulceration, abnormal wound healing, bone disease and HIV infections
09/27/2001US20010024749 Surface modified carbonaceous materials
09/27/2001US20010023877 Inverted aerosol dispenser
09/27/2001DE10014006A1 New heterocyclic acylsulfimide derivatives, useful as insecticides, acaricides and nematocides for plant protection or in veterinary medicine
09/27/2001CA2404206A1 Protease inhibitors
09/27/2001CA2404076A1 Heterocyclic side chain containing metalloprotease inhibitors
09/27/2001CA2401870A1 Cyclic .beta.-amino acid derivatives as inhibitors of matrix metalloproteases and tnf-.alpha.
09/27/2001CA2400168A1 Beta-amino acid derivatives as inhibitors of matrix metalloproteases and tnf-alpha
09/26/2001EP1136491A1 2-[(Heteroaryl)alkylamino]pyrimidone derivatives
09/26/2001EP1136482A1 2-Amino-3-(alkyl)-pyrimidone derivatives as GSK3beta inhibitors
09/26/2001EP1136477A1 Benzofuran derivatives, process for the preparation of the same and uses thereof
09/26/2001EP1135386A1 Method for producing pyrazolylbenzoyl derivatives and novel pyrazolylbenzoyl derivatives
09/26/2001EP1135385A1 Thiochromanoylpyrazolone derivatives
09/26/2001EP1135370A2 Carboxylic acids and carboxylic acid isosteres of n-heterocyclic compounds
09/26/2001EP0833825B1 6-carboxamido dihydropyran derivatives
09/26/2001EP0626968B1 Piperidinyl thiacyclic derivatives
09/26/2001CN1314905A Muscarinic antagonists
09/26/2001CN1314883A Amino acid derivatives and drug containing the same as the active ingredient
09/26/2001CN1314346A Process for preparing radio-therapeutic sensitivity intensifier 2-substituted amino-3-cyano-5-nitropyridine
09/26/2001CN1071757C Pyrazol benzoyl derivatives
09/26/2001CN1071756C Pyrazol-4-yl-benzoyl derivatives and their use as herbicides
09/26/2001CN1071755C Heterocyclyycarboxamide derivatives and their use as therapeutic agents
09/26/2001CN1071753C 7-azabicyclo [2,2,1]-heptane and heptene derivatives as cholinergic receptor ligands
09/25/2001US6294677 Thiopyran derivatives
09/25/2001US6294676 As chemical intermediate for preparing herbicides
09/25/2001US6294675 Chemical intermediate
09/25/2001US6294574 Compounds and methods for the treatment of inflammatory and immune disorders
09/25/2001US6294569 Analgesic at central nervous system in the mammalian subject. also, these compounds are inflammatory pain caused, for example by burns (induced by a contact with heat, acid or the other rheumatism or the like, in the said subject.
09/25/2001US6294558 Antiinflammatory agents and prostaglantins
09/25/2001US6294557 Analgesic at central nervous system in the mammalian subject. also, these compounds are inflammatory pain caused, for example by burns (induced by a contact with heat, acid or the other rheumatism or the like, in the said subject.
09/25/2001US6294551 N-linked sulfonamides of heterocyclic thioesters
09/25/2001US6294536 Triazine derivatives, their production and use
09/25/2001CA2029132C Sulphonylaminocarbonyltriazolinones having substituents which are bonded via sulphur
09/20/2001WO2001068652A1 Condensed imidazoles as histamine h3 receptor ligands
09/20/2001WO2001068647A1 Medicaments against viral diseases
09/20/2001WO2001068643A2 Novel lipoic acid heterocyclic or benzene derivatives, preparation and use thereof as medicines
09/20/2001WO2001068637A2 Method for the preparation of tetrahydrobenzothiepines
09/20/2001WO2001068616A1 Substituted 1-aryl-cyclopropylmethylamino-1,3,5-triazines
09/20/2001WO2001068607A1 Amide compounds and use thereof
09/20/2001WO2001068591A1 Carboxylic acid derivatives as ip antagonists
09/20/2001WO2001068585A1 Novel amide compounds
09/20/2001WO2001068140A2 Opioid formulations
09/20/2001WO2001068096A2 Combination therapy for the prophylaxis and treatment of hyperlipidemic conditions and disorders
09/20/2001WO2001034591A3 Substituted 4h-chromene and analogs as activators of caspases and inducers of apoptosis and the use thereof
09/20/2001WO2001019819A3 Carboxylic acids and acylsulfonamides, compositions containing such compounds and methods of treatment
09/20/2001US20010023295 By reacting a 3-((alkyl, alkoxy, phenyl or heteroaryl)carbonylamino)thiophene with a ketone in the presence of an acid and reducing the reaction mixture; agricultural fungicides
09/20/2001US20010023255 Phosphonooxymethyl ethers of taxane derivatives
09/20/2001US20010023248 Antiinflammatory agents, central nervous system disorders
09/20/2001DE10012820A1 New N2-(cyclopropyl-aryl-methyl)-1,3,5-triazine-2,4-diamine derivatives useful as pre- or post-emergence, total or selective herbicides or as pesticides, e.g. insecticides
09/20/2001DE10012549A1 New heterocyclic-substituted dihydropyrimidine derivatives useful for treatment of viral infections, especially hepatitis B infections
09/20/2001CA2402898A1 Novel lipoic acid heterocyclic or benzene derivatives, preparation and use thereof as medicines
09/20/2001CA2402865A1 Opioid formulations
09/19/2001EP1134213A2 Process for the preparation of substituted N-(indole-2-carbonyl)- glycinamides
09/19/2001EP1133489A1 Isonipecotamides for the treatment of integrin-mediated disorders
09/19/2001EP1133475A1 Substituted benzo de]isoquinoline-1,3-diones
09/19/2001EP1133293A1 Use of n-substituted azabicycloalkane derivatives for treating diseases of the central nervous system
09/19/2001EP0869954B1 Heterocyclic compounds for use in the treatment of neurogenic inflammation
09/19/2001EP0839144B1 Piperazine derivatives as therapeutic agents
09/19/2001CN1313856A Thiazoline acid derivatives
09/19/2001CN1313853A Oxindole derivatives as growth hormone releasers
09/19/2001CN1313280A Benzheterocyclic derivatives
09/19/2001CN1071331C Anti-helicobacter acyl derivatives of azolones
09/18/2001US6291682 Pyrazol-4-ylbenzoyl derivatives and their use as herbicides
09/18/2001US6291679 Process for preparing benzoperhydroisoindole compounds
09/18/2001US6291672 Human NK3 receptor-selective antagonist compounds, method for obtaining them and pharmaceutical compositions containing them
09/18/2001US6291514 Heteroaryl amidines, methylamidines and guanidines, preparation thereof, and use thereof as protease inhibitors
09/18/2001US6291510 Small molecule inhibitors of rotamase enzyme activity
09/18/2001US6291505 Pyrazole estrogen receptor agonist and antagonist
09/18/2001US6291504 Potent inhibitors of the class of enzymes known as cyclin dependent kinases
09/18/2001US6291486 Polycyclic Dihydrothiazoles, their preparation and use as pharmaceuticals
09/18/2001US6291484 Treatment of the various medical conditions associated with postmenopausal syndrome
09/18/2001US6291480 Diaryl piperidyl pyrrole derivatives as antiprotozoal agents
09/18/2001US6291450 Carboxylic acid substituted heterocycles, derivatives thereof and methods of use
09/18/2001US6291400 Herbicidal compounds
09/18/2001US6289745 High temperature insertion type flow element and mounting extension
09/13/2001WO2001066525A1 New ccr5 modulators: benzimidazoles or benzotriazoles
09/13/2001WO2001066521A1 Azacyclic compounds for use in the treatment of serotonin related diseases
09/13/2001WO2001066520A1 Indole derivatives, process for preparation of the same and use thereof
09/13/2001WO2001009138A3 Chemokine receptor antagonists and methods of use therefor
09/13/2001US20010021780 Anticonvulsants, psychological disorders