Patents
Patents for C07D 409 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms (52,226)
01/2002
01/02/2002EP1165513A1 Indolinone compounds as kinase inhibitors
01/02/2002EP1165510A1 1-arenesulfonyl-2-aryl-pyrrolidine and piperidine derivatives for the treatment of cns disorders
01/02/2002EP1165197A1 Crystallization process for producing fine crystal products
01/02/2002EP1165068A1 C10 heterosubstituted acetate taxanes as antitumor agents
01/02/2002EP0912553B1 BENZO[g]QUINOLINE DERIVATIVES
01/02/2002EP0835256B1 Microbicidal benzotriazoles
01/02/2002EP0764157B1 Benzopyrans and their use as therapeutic agents
01/02/2002EP0731091B1 2-oxoindoline derivatives as cholecystokinin receptor antagonists
01/02/2002CN1329609A Tetrahydrobenza epine derivatives useful as modulators of dopamine D3 receptors (antipsychotic agents)
01/02/2002CN1329607A Substituted benzopyran analogs for treatment of inflammation
01/02/2002CN1329597A Pyridinium derivatives for treatment of diabetic and aging-related vascular complications
01/02/2002CN1077106C 吡唑衍生物 Pyrazole derivative
01/01/2002US6335460 Treating retroviral infections, including human immunodeficiency virus, and aids
01/01/2002US6335452 1-substituted 2,5-dithienyl pyrrole derivatives and film-forming materials
01/01/2002US6335445 Derivatives of 2-(iminomethyl)amino-phenyl, their preparation, their use as medicaments and the pharmaceutical compositions containing them
01/01/2002US6335362 Antitumor and anticarcinogenic agents for leukemia
01/01/2002US6335357 1-aryl-3-cyano-5-(het)arylalkylaminopyrazole derivatives; insecticides for agriculture and horticulture
01/01/2002US6335334 Hypertensive agents, anticoagulants; cardiovascular and sexual disorders, angina pectoris, and atherosclerosis
01/01/2002US6335329 Carboxylic acid substituted heterocycles, derivatives thereof and methods of use
01/01/2002US6335327 1-benzazepine derivatives; agonists or antagonists of vasopressin and/or oxytocin
01/01/2002CA2056799C 1,4-dihydropyridine derivatives and methods of producing the same
01/01/2002CA2029105C Halogenated sulphonylaminocarbonyltriazolinones
12/2001
12/27/2001WO2001098310A1 Novel chromophores for polymeric thin films and optical waveguides and devices comprising the same
12/27/2001WO2001098291A2 1,3-bis-(substituted-phenyl)-2-propen-1-ones and their use to treat vcam-1 mediated disorders
12/27/2001WO2001098290A2 Thiophene derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
12/27/2001WO2001098289A1 Novel non-psychotropic cannabinoids
12/27/2001WO2001098286A1 Nitrosated and nitrosylated taxanes, compositions and methods of use
12/27/2001WO2001098272A1 Novel compounds
12/27/2001WO2001032646A3 Sulfonamide derivatives
12/27/2001WO2000064864A9 N-protected amines and their use as prodrugs
12/27/2001US20010056184 Pipecolinic acid derivatives, method of manufacturing the same and therapeutic agents containing these compounds
12/27/2001US20010056107 Cyano and carboxy derivatives of substituted styrenes are inhibitors of tumor necrosis factor alpha , nuclear factor kappa B, and phosphodiesterase and can be used to treat cachexia, endotoxic shock, inflammatory conditions etc.
12/27/2001US20010056105 Useful as cosmetic for hair and body hygiene, and for treatment of dermatological complaints, with an inflammatory and/or immunoallergic component of rheumatic or respiratory type, cardivascular and opthalmogical disorders
12/27/2001US20010056100 Carboxylic acid or tetrazole derivatives containing carbamate groups are useful for treating the conditions associated with the urinary tract, pain, inflammation, respiratory states, edema formation of hypotensive vascular diseases
12/27/2001US20010056096 Administering to a patient suffering from hypercholesterolemia, hyperlipedimea and other metabolic disorders an effective amount of hydrozone, oxime or imine derivatives
12/27/2001CA2414085A1 Thiophene derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
12/27/2001CA2413878A1 1,3-bis-(substituted-phenyl)-2-propen-1-ones and their use to treat vcam-1 mediated disorders
12/27/2001CA2411963A1 Novel chromophores for polymeric thin films and optical waveguides and devices comprising the same
12/27/2001CA2411585A1 Novel non-psychotropic cannabinoids
12/27/2001CA2411255A1 Novel compounds
12/27/2001CA2410632A1 Nitrosated and nitrosylated taxanes, compositions and methods of use
12/26/2001CN1328552A Pyrimidone derivatives
12/26/2001CN1328549A Substituted benzo [de] isoquinoline-1,3-diones
12/26/2001CN1328546A Pyrrolidines as inhibitors of neuraminidases
12/26/2001CN1328455A Use of N-substituted azabicycloalkane derivatives for treating diseases of central nervous system
12/25/2001US6333425 Ionic compounds derived from malononitrile in which anionic charge is delocalized; excellent properties of solubility and dissociation
12/25/2001US6333346 Aminofuranoneureas or thioureas 4-amino-2(5h)-thiophenones as antitumor agents
12/25/2001US6333344 Prolines as antimicrobial agents
12/25/2001US6333341 Tumor necrosis factor, antiinflammatory agents and analgesics
12/25/2001US6333338 Anticoagulants, cardiovascular disorders
12/25/2001US6333324 For therapy and prophylaxis of matrix metalloproteinases (mmp) or tumor necrosis factor .alpha. (tnf.alpha.), mediated diseases
12/25/2001CA2052424C 2-(4-piperidinyl)-1h-pyrido¬4,3-b|indol-1-ones and related compounds, intermediates and a process for their preparation
12/20/2001WO2001096331A1 Lactam inhibitors of factor xa and method
12/20/2001WO2001096330A2 Thrombin receptor antagonists
12/20/2001WO2001096323A1 Serine protease inhibitors
12/20/2001WO2001096314A1 Fungicidal 5-phenyl substituted 2-(cyanoamino) pyrimidines
12/20/2001WO2001096313A1 Distamycin a analogs
12/20/2001WO2001096308A1 1,2-dihydropyridine compounds, process for preparation of the same and use thereof
12/20/2001WO2001096303A1 Serine protease inhibitors
12/20/2001WO2001096302A1 Piperidines for use as orexin receptor antagonists
12/20/2001WO2001096299A2 Indole derivatives and their use as 15-lipoxygenase inhibitors
12/20/2001WO2001096295A2 2-cyanopyrrolidine derivatives and their use as medicaments
12/20/2001WO2001095911A1 Protease inhibitors
12/20/2001WO2001095858A2 Piperazinedione compounds
12/20/2001WO2001040223A3 Aminoheterocyclylamides as pesticides and antiparasitic agents
12/20/2001WO2001016108A3 Bicyclic androgen and progesterone receptor modulator compounds and methods
12/20/2001WO1999019304A3 Alpha-alkylthio substituted pyrimidine ethers and thioethers as viral reverse transcriptase inhibitors
12/20/2001US20010053788 4,5-dihydro-1H-pyrazole derivatives having CB1-antagonistic activity
12/20/2001CA2719176A1 2-cyanopyrrolidine derivatives and their use as medicaments
12/20/2001CA2412353A1 Protease inhibitors
12/20/2001CA2412216A1 Lactam inhibitors of factor xa and method
12/20/2001CA2412010A1 Fungicidal 5-phenyl substituted 2-(cyanoamino) pyrimidines
12/20/2001CA2411805A1 Serine protease inhibitors
12/20/2001CA2411116A1 Indole derivatives and their use as 15-lipoxygenase inhibitors
12/19/2001EP1164134A1 Benzimidazole compounds and their use as modulators of the GABA A receptor complex
12/19/2001EP1163238A1 Chemokine recpetor binding heterocyclic compounds
12/19/2001EP1163237A1 Amide derivatives
12/19/2001EP1163236A1 Aromatic heterocyclic compounds as anti-inflammatory agents
12/19/2001EP1163229A1 2,4-diamino-1,3,5-triazines, method for producing them and their use as herbicides and plant growth regulators
12/19/2001EP1163221A1 Sulfonamide derivatives as 5ht7 receptor antagonists
12/19/2001EP0785794B1 Enteric coated compositions of 1,5-benzodiazepine derivatives having cck antagonistic or agonistic activity
12/19/2001EP0639080B1 Non-azo naphthalimide dyes and use as alkylating agents
12/19/2001CN1327443A Substituted anilides
12/18/2001US6331640 Diaminopropionic acid derivatives
12/18/2001US6331639 By reacting a 3-((alkyl, alkoxy, phenyl or heteroaryl)carbonylamino)thiophene with a ketone in the presence of an acid and reducing the reaction mixture; agricultural fungicides
12/18/2001US6331637 N-Alkyl, N-Alkenyl, N-Alkynyl, N-Aryl and N-fused bicyclo or tricyclo thienyl-, furyl-,and Pyrrolyl-sulfonamides and derivatives thereof that modulate the activity of endothelin
12/18/2001US6331634 Process for preparing 2-alkyl-3-aminothiophene derivative and 3-aminothiophene derivative
12/18/2001US6331563 N-Hydroxy-2-(Alkyl, Aryl, or Heteroaryl, Sulfanyl, Sulfinyl or Sulfonyl)-3-Substituted Alkyl, Aryl or Heteroarylamides as Matrix Metalloproteinase inhibitors
12/18/2001US6331554 Antipicornaviral compounds, compositions containing them, and methods for their use
12/18/2001US6331545 Heterocycyclic piperidines as modulators of chemokine receptor activity
12/18/2001US6331544 Treating positive and negative symptoms of schizophrenia and other psychoses
12/18/2001US6331537 Treating neurological disorders in animals
12/18/2001US6331507 Substituted aromatic thiocarboxylic acid amides and their use as herbicides
12/18/2001CA2213815C Pyrrolidinyl hydroxamic acid compounds and their production process
12/13/2001WO2001094339A1 Substituted pyridine herbicides
12/13/2001WO2001094317A2 Method for synthesis of substituted azole libraries
12/13/2001WO2001093841A2 Barbituric acid analogs as therapeutic agents
12/13/2001WO2001093682A1 N-phenyl-4-(4-pyridyl)-2-pyrimidineamine derivatives
12/13/2001WO2001068140A3 Opioid formulations
12/13/2001WO2001049275A3 Methods and compositions for mitigating pain using nitrate esters