Patents
Patents for C07D 409 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms (52,226)
01/2005
01/20/2005US20050014802 Prevent reproduction of virus; antitumor agents
01/20/2005US20050014796 Mediators of hedgehog signaling pathways, compositions and uses related thereto
01/20/2005US20050014788 Piperidine derivatives and their use as modulators of chemokine receptor activity (especially ccr5)
01/20/2005US20050014786 Tetrahydroquinoline derivatives as cannabinoid receptor modulators
01/20/2005US20050014757 Serotonin receptor antagonist; psychological disorders; side effect reduction
01/20/2005US20050014750 Isochroman compounds for treatment of cns disorders
01/20/2005US20050014749 Piperazine derivatives and methods of use
01/20/2005US20050014705 E.g., dimethylcarbamic acid, 2-oxo-3-benzyl-4-methyl-2H-1-benzopyran; affects both the Tumor Necrosis Factor alpha level and transcription activity of NuclearFactor kappa Beta; antiimmunoinflammatory agents and autoimmune properties; antiarthritis agents; rheummatic diseases; osteoporosis; leukemia
01/20/2005US20050014700 Cbi analogues of cc-1065 and the duocarmycins
01/20/2005US20050014650 Delta 1-pyrrolines used as pesticides
01/20/2005DE102004014061A1 Amid-substituierte 1,2,4-Triazin-5(2H)-one Amide substituted 1,2,4-triazine-5 (2H) -ones
01/20/2005CA2530737A1 Cck-1 receptor modulators
01/20/2005CA2529739A1 Aspartyl protease inhibitors
01/20/2005CA2528626A1 Indoles useful in the treatment of inflammation
01/20/2005CA2526725A1 Mch antagonists for the treatment of obesity
01/19/2005EP1498419A1 Process for preparing alkali metal salts of hydrophobic sulfonamides
01/19/2005EP1498418A1 Sulfonamides for treatment of endothelin-mediated disorders
01/19/2005EP1498411A1 Diketohydrazine derivative compounds and drugs containing the compounds as the active ingredient
01/19/2005EP1497287A1 Quinolinone derivatives
01/19/2005EP1497284A2 Pyrrolidinium derivatives as antagonists of m3 muscarinic receptors
01/19/2005EP1497283A1 Maleic acid salt of(2s)-n-(5(amino(imino)methyl)-2-thienyl)methyl-1-(2r)-2-((2r)-2-((carboxymethyl)amino)3,3-diphenylpropanoyl)-2-pyrrolidine carboxamide and a process for
01/19/2005EP1497278A1 Heterocyclic amide derivatives as cytokine inhibitors
01/19/2005EP1497240A1 Non-heating clay composites for building materials
01/19/2005EP1496906A1 Inhibitors of akt activity
01/19/2005EP1496896A1 Inhibitors of akt activity
01/19/2005EP1496892A2 1h-benzo(f)indazol-5-yl derivatives as selective glucocorticoid receptor modulators
01/19/2005EP1496838A2 Substituted amides
01/19/2005EP1395574B1 4-(phenyl-piperidin-4-ylidene-methyl)-benzamide derivatives and their use for the treatment of pain, anxiety or gastrointestinal disorders
01/19/2005CN1568323A Activator for peroxisome proliferator-activated receptor delta
01/19/2005CN1568322A Pharmaceutically active sulfonamide derivatives bearing both lipophilic and ionisable moieties as inhibitors of protein junkinases
01/19/2005CN1568185A Compounds effecting glucokinase
01/19/2005CN1566098A Isoquinoline compound, preparation method and application of salt thereof
01/19/2005CN1566096A Prostaglandin agonists and their use to treat bonedisorders
01/19/2005CN1566091A Molindone derivatives and use for preparing antineoplastic medicine thereof
01/19/2005CN1185228C Hydroxyphenyl-piperidin-4-ylidene-methyl-benzamide derivatives for treatment of pain
01/19/2005CN1185227C Novel compounds
01/19/2005CN1185223C Novel Compounds and methods for synthesis and therapy
01/19/2005CN1185217C Propanolamine derivatives, processes for their preparation, pharmaceuticals comprising these compounds, and their use
01/19/2005CN1185216C Fungicides
01/19/2005CN1185213C Azetidine derivatives, preparation and pharmaceutical compositions thereof
01/18/2005US6844446 Catalysts containing per-ortho aryl substituted aryl or heteroaryl substituted nitrogen donors
01/18/2005US6844367 Benzamides and related inhibitors of factor Xa
01/18/2005US6844357 Anticarcinogenic agents
01/18/2005US6844347 Substituted 4-amino-2aryl-pyrimidines, their production and use and pharmaceutical preparations containing same
01/18/2005US6844344 Depression, anxiety; tobacco or nicotine withdrawal; such as 1-(benzofuran-4-yl)oxy-3-(4-(6-methoxybenzo(b)thiophen-2-yl)piperidinyl)-2 -propanol oxalate
01/18/2005US6844335 2-amino-3-(alkyl)-pyrimidone derivatives as GSK3.β.inhibitors
01/18/2005CA2158458C Taxanes prepared by beta-lactams and ammonium alkoxides
01/13/2005WO2005003131A1 Tricyclic delta opioid modulators
01/13/2005WO2005003118A1 Amide-substituted 1,2,4-triazin-5(2h)-ones for the treatment of chronically inflammatory diseases
01/13/2005WO2005003115A1 Thiophene amino acid derivatives, process for preparing them and pharmaceutical compositions containing them
01/13/2005WO2005003114A1 5-fluoro-thiopen-compounds,the process for their preparation,the pharmaceutical compositions containing them and their use as metallopotenases inhibitors
01/13/2005WO2005003103A2 2, 4, 6-tri-substituted 6-membered heterocycles and their use in the treatment of neurodegenerative diseases
01/13/2005WO2005003102A1 Methods of preparation of dehydro-diketopiperazines in liquid phase or of solid supported phase
01/13/2005WO2005003101A2 Pyrazine and pyridine derivatives as rho kinase inhibitors
01/13/2005WO2005003099A2 Pyrimidines useful as modulators of voltage-gated ion channels
01/13/2005WO2005003097A1 Cis-2,4,5-triaryl-imidazolines
01/13/2005WO2005003089A2 7-ethynyl-2,4,9-trithiaadamantane and related methods
01/13/2005WO2005002552A2 Benzimidazole derivatives and their use as protein kinases inhibitors
01/13/2005WO2005002514A2 Compounds having inhibitibe activity of phosphatidylinositol 3-kinase and methods of use thereof
01/13/2005WO2004106329A3 Novel antiinfective compounds and their pharmaceutical compositions
01/13/2005WO2004099192A3 Heterocycle substituted carboxylic acids as inhibitors of protein tyrosine phosphatase-1b
01/13/2005WO2004082623A3 Substituted piperidine compounds
01/13/2005WO2004064764A3 Substituted alkyl amido piperidines
01/13/2005WO2004050035A3 Benzimidazoles and analogs thereof as antivirals
01/13/2005US20050009894 Benzimidazole derivatives and their use as KDR kinase protein inhibitors
01/13/2005US20050009876 Indazole compounds, compositions thereof and methods of treatment therewith
01/13/2005US20050009870 3-(amino)sulfonylamino-substituted, e.g., N-(1,6-Dibenzyl-2-oxo-1,2,3,4-tetrahydroquinolin-3-yl)-benzenesulfonamide and N-(1-Benzyl-2-oxo-6-(thiophen-3-yl)-1,2,3,4-tetrahydroquinolin-3-yl)benzenesulfonamide; eating, metabolic, obesity, cognitive, neurological, pain, inflammatory and psychiatric disorders
01/13/2005US20050009864 Substituted 4-phenyltetrahydroisoquinolinium, process for their preparation, their use as a medicament, and medicament containing them
01/13/2005US20050009860 Tricyclic delta-opioid modulators
01/13/2005US20050009853 Pyrimidine derivatives for the treatment of abnormal cell growth
01/13/2005US20050009844 Inhibitors of p38
01/13/2005US20050009840 2-amino- pyridines and pyrazines additionally substituted witn one or more carbocyclic or heterocyclic groups, e.g., 4-[6-amino-5-(2,6-dichloro-benzyloxy)-pyridin-3-yl]-phenol, for treating many kinds of cancer
01/13/2005US20050009839 Novel azoles having an insecticidal action
01/13/2005US20050009838 Piperidinyl-and piperazinyl-sulfonylmethyl hydroxamic acids and their use as protease inhibitors
01/13/2005US20050009829 1-Substituted 2-carboxamide derivatives of fused ring imidazoles, e.g., -[5-(5-Chloro-thiophen-2-yl)-isoxazol-3-ylmethyl]-1H-benzoimidazole-2-carboxylic acid (1-isopropyl-piperidin-4-yl)-amide
01/13/2005US20050009820 Thiochromenones used to combat painful conditions and neurodegenerative diseases
01/13/2005US20050009819 1-Aryl-or 1-alkylsulfonylbenzazole derivatives as 5-hydroxytryptamine-6 ligands
01/13/2005US20050009817 Substituted heteroaryls
01/13/2005US20050009812 Remedies for stress diseases comprising mitochondrial benzodiazepine receptor antagonists
01/13/2005US20050009804 N-heterocyclyl- or cycloalkyl-N-(2-carboxy-5-aryl-3-thiophenyl)cycloalkanecarboxamides, e.g., 5-(3-fluorophenyl)-3-[isopropyl-(4-methylcyclohexanecarbonyl)amino]-thiophene-2-carboxylic acid; especially for prevention and treatment of HVC
01/13/2005US20050009755 (74)(3S)-3-amino-1-(1-benzyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-4-yl)-5-methyl-2-heptanone for example; cysteine protease inhibitors; treating bone resorption diseases such as osteoporosis
01/13/2005US20050006246 Nitrogen atom transfer
01/13/2005DE10328479A1 6-Arylamino-5-cyano-4-pyrimidinone 6-arylamino-5-cyano-4-pyrimidinones
01/13/2005DE10328400A1 One-pot synthesis of carbocyclic or heterocyclic compounds, especially pyrimidine useful as components of natural products or drugs, from acid halide, alkyne and active hydrogen compound
01/13/2005CA2531327A1 Compounds and therapeutical use thereof
01/13/2005CA2531061A1 Pyrimidines useful as modulators of voltage-gated ion channels
01/13/2005CA2531050A1 Pharmaceutical compounds
01/13/2005CA2530816A1 Amide-substituted 1,2,4-triazin-5(2h)-ones for the treatment of chronic inflammatory diseases
01/13/2005CA2530389A1 Pyrazine and pyridine derivatives as rho kinase inhibitors
01/13/2005CA2528119A1 Cis-2,4,5-triaryl-imidazolines
01/12/2005EP1495017A2 Novel heteroaryl alkylamide derivatives useful as bradykinin receptor modulators
01/12/2005EP1495004A2 Benzenesulfonamide derivatives and their use as dopamine d3 and d2 receptor ligands
01/12/2005EP1495003A1 Fredericamycin derivatives
01/12/2005EP1495002A1 Benzamide derivatives useful as histone deacetylase inhibitors
01/12/2005EP1495001A1 Antibacterial agents
01/12/2005EP1494672A1 Aminocarbonyl substituted pyridines, pyridazines, pyrimidines, pyrazines and triazines having antiangiogenic activity
01/12/2005EP1494671A1 1-(4-piperidinyl)benzimidazolones as histamine h3 antagonists
01/12/2005EP1494668A2 Use of benzimidazole analogs in the treatment of cell proliferation
01/12/2005EP1494663A1 Derivatives of 1-(oxoaminoacetyl) pentylcarbamate as cathepsin k inhibitors for the treatment of bone loss
01/12/2005EP1171423B1 Carbamic acid derivatives and their use as metabotropic glutamate receptor ligands