Patents
Patents for C07D 409 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms (52,226)
02/2005
02/02/2005CN1187349C 3-(4, 5-dihydroisoxazole-5-yl)-benzoylpyrazole
02/02/2005CN1187342C Substituted 1-aminoalkyl-lactams compound and their use as muscarinic receptor antagonists
02/02/2005CN1187336C New imidazole derivatives
02/02/2005CN1187333C Certain substituted caprolactams, pharmaceutical compositions containing them and their use in treating tumors
02/02/2005CN1187325C Pharmaceutical compositions containing 3-amino-azetidine derivatives, novel derivatives and preparation thereof
02/01/2005US6849744 3-(substituted phenyl),4-substituted-5H-1,2-oxathiole 2-oxide or 2,2-dioxide compounds useful as agricultural fungicides, insecticides, herbicides
02/01/2005US6849739 N-heterocyclic derivatives as NOS inhibitors
02/01/2005US6849733 Compounds containing amidated guanidine derivative type functional group of structure N-C(=N)-N-CO-N-C=N or N-C(=N)-N-CO-N
02/01/2005US6849713 Topisomerase inhibitor
02/01/2005US6849660 Antimicrobial biaryl compounds
02/01/2005US6849658 Biaromatic compounds and pharmaceutical and cosmetic compositions comprising them
02/01/2005US6849643 Indazolyl-substituted pyrroline compounds as kinase inhibitors
02/01/2005US6849639 Anticancer agents, antiinflamatory agents, osteoporosis, atherosclerosis
02/01/2005US6849636 Useful for treatment of noninsulin-dependent diabetes, hyperglycemia, obesity, insulin resistance, dyslipidemia, hyperlipidemia, hypertension, Metabolic Syndrome
02/01/2005US6849635 Sulfonamides
02/01/2005US6849634 Potassium channel inhibitors
02/01/2005US6849629 Heteroaromatic substituted sulfonyl or sulfoxide or thio-pyridazinone derivatives, useful for treating diabetic complications and cardiovascular disorders
02/01/2005US6849622 May be useful for the prophylaxis and treatment of diabetes, particularly type 2 diabetes, and for prophylaxis and treatment of other diseases induced or exacerbated by impaired glucose tolerance
02/01/2005US6849621 Treating: allergy, allergy-induced airway responses, congestion, hypotension, cardiovascular disease, hypotension, diseases of the GI tract, hyper and hypo motility and acidic secretion of the gastrointestinal tract, obesity, sleep
01/2005
01/27/2005WO2005007647A1 Trisubstituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto
01/27/2005WO2005007635A2 Combretastatin derivatives with cytotoxic action
01/27/2005WO2005007628A1 Tetrahydroquinoline derivatives as cannabinoid receptor modulators
01/27/2005WO2005007157A1 Pyrazolines as par-1 antagonists for treatment of cardiovascular diseases
01/27/2005WO2005007111A2 Tetrahydroquinoline derivatives as cannabinoid receptor modulators
01/27/2005WO2004087647A3 4-substituted quinolein derivatives with antimicrobial activity
01/27/2005US20050020659 Substituted pyrazole derivatives and related compounds as bradykinin B1 receptor antagonists
01/27/2005US20050020639 Novel compounds
01/27/2005US20050020635 C7 carbamoyloxy substituted taxane compositions
01/27/2005US20050020630 Antiinflammatory agents; cardiovascular disorders; anticancer agents; antiarthritic agents; skin disorders; autoimmune disease; cardiovascular disorders
01/27/2005US20050020629 Pain management
01/27/2005US20050020624 Dihydroindole and tetrahydroquinoline derivatives
01/27/2005US20050020618 Antidiabetic agents; obesity
01/27/2005US20050020611 Phosphodiesterase inhibitor; antihistamines; antiallergens
01/27/2005US20050020605 Quinolyl amide derivatives as CCR-5 antagonists
01/27/2005US20050020604 5-HT receptor ligands and uses thereof
01/27/2005US20050020597 Attention deficit disorders; hyperactivity; post-trauma stress disorders; anxiolytic agents; obsessive compulsive disorders; analgesics; Parkinson's disease
01/27/2005US20050020588 Cysteine protease inhibitors
01/27/2005US20050020583 Amino-phthalazinone derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions containing them
01/27/2005US20050020578 Oxidoreductase enzyme inhibitors such as (R)-1-[4-(2-methyl-4-phenyl-5,8-dihydro-6H-pyrido[3,4-d]pyrimidin-7-yl)-pyrimidin-2-yl-ethanol, used as antidiabetic agents
01/27/2005US20050020575 Sulfonyldihydrobenzimidazolone compounds as 5-hydroxytryptamine-6 ligands
01/27/2005US20050020573 5HT2c receptor modulators
01/27/2005US20050020540 Biphenylcarboxylic amide derivatives as p38-kinase inhibitors
01/27/2005CA2532316A1 Pyrazolines as par-1 antagonists for treatment of cardiovascular diseases
01/27/2005CA2532152A1 Trisubstituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto
01/27/2005CA2531389A1 Combretastatin derivatives with cytotoxic action
01/27/2005CA2529790A1 Heteroaryloxy nitrogenous saturated heterocyclic derivative
01/26/2005EP1500657A1 Substituted pyrazoles as P38 kinase inhibitors
01/26/2005EP1500653A1 Substituted arylpyrazines
01/26/2005EP1500652A1 Quinazoline derivative and medicine
01/26/2005EP1499898A2 Regulation of tnf-alpha
01/26/2005EP1499612A1 Piperidine ouracil used as a medicament for treating bacterial infections
01/26/2005EP1499609A2 Pesticidal heterocycles
01/26/2005EP1499598A1 Chemical compounds with dual activity, processes for their preparation and pharmaceutical compositions
01/26/2005EP1499597A2 Compounds and methods for inducing apoptosis in proliferating cells
01/26/2005EP1499594A1 Process for the preparation of 7-substituted-3-quinoline and 3-quinol-4-one carbonitriles
01/26/2005EP1499593A1 Quinoline derivatives as caspase-3 inhibitor, preparation for producing the same and pharmaceutical composition comprising the same
01/26/2005EP1499591A1 Carboxylic acid amides
01/26/2005EP1499577A1 2-(2,6-dichlorophenyl)-diarylimidazoles
01/26/2005EP1499316A1 (1-4-piperidinyl)benzimidazole derivatives useful as histamine h3 antagonists
01/26/2005EP1499314A1 N-acyl piperidine derivatives for use as melanocortin receptor ligands in the treatment of feeding disorders
01/26/2005EP1499311A1 Substituted benzazoles and use thereof as raf kinase inhibitors
01/26/2005EP1499308A2 Tri-substituted heteroaryls and methods of making and using the same
01/26/2005EP1243579B1 Process for the production of pyridine derivatives
01/26/2005EP0983267B1 Amidoaromatic ring sulfonamide hydroxamic acid compounds
01/26/2005EP0844877B1 Use of oxido-squalene cyclase inhibitors to lower blood cholesterol
01/26/2005CN1571786A Alkyl ether derivatives or salts thereof
01/26/2005CN1571781A 4-imidazolin-2-one compounds
01/26/2005CN1571667A Inhibitors of dipeptidyl peptidase ó¶
01/26/2005CN1186341C Diaryl perfluoro cyclopentene photochromic compounds and its preparing method and use
01/26/2005CN1186340C C10 carbonate substituted taxanes as antitumor agents
01/26/2005CN1186328C Substd. 5-benzyl-2, 4-diaminopyrimidines
01/25/2005US6846954 α- and β-amino acid hydroxyethylamino sulfonamides useful as retroviral protease inhibitors
01/25/2005US6846919 Non-endogenous, constitutively activated human serotonin receptors and small molecule modulators thereof
01/25/2005US6846839 Identifying indolinone compounds that inhibit growth factor stimulated cell proliferation by contacting cells with compounds and with selected growth factors and monitoring inhibitory effect
01/25/2005US6846829 N-heterocyclic derivatives as NOS inhibitors
01/25/2005US6846828 Aminopyrimidine and aminopyridine anti-inflammation agents
01/25/2005US6846821 Tetrahydrothiopy ranphthalazinone derivatives as PDE4 inhibitors
01/25/2005US6846819 Bactericides compound containing acrylamide group
01/25/2005US6846817 Nicotine receptor ligands
01/25/2005CA2309352C Heterocyclic-substituted tricyclics as thrombin receptor antagonists
01/25/2005CA2103383C Quinazoline derivatives
01/20/2005WO2005005419A1 Mch antagonists for the treatment of obesity
01/20/2005WO2005005415A1 Indoles useful in the treatment of inflammation
01/20/2005WO2005005411A1 Substituted indole ligands for the orl-1 receptor
01/20/2005WO2005005393A2 Cck-1 receptor modulators
01/20/2005WO2005005392A1 Azacyclic compounds as inhibitors of sensory neurone specific channels
01/20/2005WO2005005374A1 Aspartyl protease inhibitors
01/20/2005WO2005004606A2 Pyridinylanilides
01/20/2005WO2004096129A3 Inhibitors of akt activity
01/20/2005WO2004074218A3 Inhibitors of macrophage migration inhibitory factor and methods for identifying the same
01/20/2005WO2004069793A3 Novel 2-substituted cyclic amines as calcium sensing receptor modulators
01/20/2005WO2004069792A3 Quinoline-derived amide modulators of vanilloid vr1 receptor
01/20/2005US20050014942 Transforming growth factor inhibitor; controllign cell differentiation, cell proliferation
01/20/2005US20050014939 E.g., N-[4-(2-Pyrrolidinylethoxy)phenyl]-4-oxo-4,5,6,7-tetrahydro-1H-indole-3-carboxamide; treating diseases associated with pathogenic agonism, inverse agonism or antagonism of the GABAA receptor such as anxiety, depression, a sleep disorder, or cognitive impairment
01/20/2005US20050014840 Thiol sulfonamide metalloprotease inhibitors
01/20/2005US20050014817 Fluorothiophene derivatives, process for preparing them and pharmaceutical compositions containing them
01/20/2005US20050014816 Thiophene amino acid derivatives, process for preparing them and pharmaceutical compositions containing them
01/20/2005US20050014815 Substituted 2-pyrrolidine-2-yl-1H-indole compounds
01/20/2005US20050014811 Such as 4-cyclopentylamino-benzenesulfonic acid 2-(3,4-dimethoxy-phenylamino)-1H-benzoimidazol-5-yl ester; cyclin-dependent kinase inhibitors that are aimed to be more active than flavopiridol
01/20/2005US20050014809 Substituted thien-3-yl-sulphonylamino(thio)carbonyl-triazolin(thi)ones