Patents
Patents for C07D 409 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms (52,226)
08/2006
08/24/2006WO2006088711A1 AZOLYLACYLGUANIDINES AS β-SECRETASE INHIBITORS
08/24/2006WO2006088694A1 SUBSTITUTED THIENYL AND FURYL ACYLGUANIDINES AS β-SECRETASE MODULATORS
08/24/2006WO2006088193A1 Anti-tumor agent
08/24/2006WO2006035067A3 Hiv inhibiting 5-heterocyclyl pyrimidines
08/24/2006WO2004094374A3 Preparation of (s)-clopidogrel and related compounds
08/24/2006US20060189810 Novel sulfonamide inhibitors of aspartyl protease
08/24/2006US20060189805 Characterized by the formation and isolation of intermediate compounds in salified form; by using the intermediate of the present process in the subsequent reductive passage, it is possible to obtain emtricitabine in a purity that allows its direct crystallization; viricides
08/24/2006US20060189681 Inhibitors of hepatitis c virus rna-dependent rna polymerase, and compositions and treatments using the same
08/24/2006US20060189676 Pyrrolcarboxamides and Pyrrolcarbothioamides
08/24/2006US20060189674 Deacetylase inhibitors
08/24/2006US20060189672 2-Heterocyclyl- indole, pyrrolopyridine, pyrrolopyrimidine, or pyrrolopirazine substituted with an N-(amino)sulfonyl(thio)carboxamide: 3-Cyclohexyl-2-furan-3-yl-7-methyl-1H-indole-6-(N-methylsulfonyl)carboxamide; treating a hepatitis virus infection
08/24/2006US20060189629 N-(2-morpholin-4-ylethyl)-1-(4-{[4-(trifluoromethoxy)benzyl]oxy}phenyl)-1H -benzimidazole-5-carboxamide; c-Kit proto-oncogene (stem cell factor receptor) anhibitor; tyrosine kinase inhibitor; antiproliferative, anticarcinogenic agent;
08/24/2006US20060189623 5-Cyano-1H-imidazole-2-carboxylic acid [4-(3,6-dihydro-2H-pyran-4-yl)-2-(4,4-dimethyl-cyclohex-1-enyl)-phenyl]-amide; tyrosine kinase inhibitor; autoimmune diseases, antiinflammatory, anticarcinogenic agent
08/24/2006US20060189622 Pyridazinone and triazinone compounds and use thereof as pharmaceutical preparations
08/24/2006US20060189614 preparing 4-[[4-amino-6-[(2,6-dichlorophenyl)methyl]-1,3,5-triazin-2-yl]amino]benzonitrile by reacting 2,6-dichlorobenzeneethanimidamide with phenyl N'-cyano-N-(4-cyanophenyl)-carbamimidate in a reaction-inert solvent; HIV (Human Immunodeficiency Virus) infection
08/24/2006US20060189613 Sulphonamide Compounds that Modulate Chemokine Receptor Activity (CCR4)
08/24/2006US20060189577 Tyrosine kinase inhibitors
08/24/2006US20060189549 Chalcone derivatives and their use to treat diseases
08/24/2006CA2599046A1 Antitumor agent
08/24/2006CA2598897A1 Fungicidal pyrazine derivatives
08/24/2006CA2598460A1 Amine-linked pyridyl and phenyl substituted piperazine-piperidines with cxcr3 antagonist activity
08/24/2006CA2597594A1 Azolylacylguanidines as beta-secretase inhibitors
08/23/2006EP1693372A1 Novel Sulfamides and their use as endothelin receptor antagonists
08/23/2006EP1693365A1 Inhibitors of dipeptidyl peptidase IV
08/23/2006EP1692124A1 Biaryl sulfonamides as mmp inhibitors
08/23/2006EP1692114A1 Novel benzimidazole and imidazopyridine derivatives and use thereof as a medicament
08/23/2006EP1692113A1 Aryl imidazoles and their use as anti-cancer agents
08/23/2006EP1692111A2 Quinolines useful in treating cardiovascular disease
08/23/2006EP1692085A2 Inhibition of fgfr3 and treatment of multiple myeloma
08/23/2006EP1691810A1 Substituted piperazines
08/23/2006EP1438349B1 Triarylamine containing monomers for optoelectronic devices
08/23/2006EP1345907B1 7-heterocyclyl quinoline and thieno 2,3-b|pyridine derivatives useful as antagonists of gonadotropin releasing hormone
08/23/2006EP1337529B1 Heterocyclylalkyl piperidine derivatives, their preparation and compositions containing same
08/23/2006EP1051405B1 Novel dihydroxyhexanoic acid derivatives
08/23/2006EP1027328B1 Substituted anilides
08/23/2006CN1823063A Quinoline derivatives as phosphodiesterase inhibitors
08/23/2006CN1823062A Sulfonyldihydro- benzimidazolone compounds as 5-hydroxytryptamine-6 ligands
08/23/2006CN1823056A Trisubstituted aryl and heteroaryl derivatives as modulatorsof metabolism and the prophylaxis and treatment of disorders related thereto
08/23/2006CN1823046A Phenyl quinolines and their use as estrogenic agents
08/23/2006CN1271069C Diepoxy group containing thioxanthone photoinitiator and preparation method therefor
08/23/2006CN1271066C Aromatic dicarboxylic acid derivatives
08/23/2006CN1271054C Urea compounds having muscarinic receptor antagonist activity
08/23/2006CN1271052C Sulphonamide derivatives, the preparation thereof and the application of same as medicaments
08/22/2006US7094911 Biphenyl and biphenyl-analogous compounds as integrin antagonists
08/22/2006US7094909 Reacting an amide compound containing hydroxy and a carboxyl group and having benzene ring, with a halogenated alkyl aminocarbonyl-pyrrolidine with 2-fluoro groups substituted at the ring carbon, by amindation of amine and carboxyl group
08/22/2006US7094807 Viricides; hepatitis virus
08/22/2006US7094801 Inhibiting the expression of VCAM-1; treating inflammatory disorders including rheumatoid arthritis, atherosclerosis, COPD, asthma, allergic rhinitis and restinosis
08/22/2006US7094788 A tropane ester derivative for treating asthma, chronic obstractive pulmonary disease, vagally induced sinus bradycardia, heart rhythm disorders, spasms in the gastrointestinal or urinary tracts, and menstrual pain
08/22/2006US7094781 Sulfamides and their use as endothelin receptor antagonists
08/22/2006US7094780 3-aminoquinazolin-2,4-dione antibacterial agents
08/22/2006US7094779 2-(3-indolylmethyl)-1-benzoyl-4-oxime-piperazine derivatives, e.g., 1-{(2R)-1-[3,5-bis(trifluoromethyl)benzoyl]-2-(1H-indol-3-ylmethyl)-piperazin-4-yl}-2-propanone O-[2-(dimethylamino)-ethyl]oxime, used for treatment of CNS disorders.
08/22/2006US7094778 Nervous system disorders; muscular disorders; urogenital disorders; gastrointestinal disorders; repiratory system disorders; antiallergens; side effect reduction
08/22/2006US7094777 5-HT2A receptor ligands
08/22/2006CA2242102C Quinazoline derivatives as antitumor agents
08/17/2006WO2006086705A1 Substituted bis aryl and heteroaryl compounds as selective 5ht2a antagonists
08/17/2006WO2006086657A1 Process for preparing 2,3-disubstituted indoles
08/17/2006WO2006085113A2 2-substituted 5-membered heteroaryl carboxylates as hm74a receptor agonists
08/17/2006WO2006085067A1 Atm inhibitors
08/17/2006WO2006076646A3 Heteroaryl substituted quinolin-4-ylamine analogues
08/17/2006WO2006066950A3 Tricyclic aminoalcohols, methods for producing the same and their use as anti-inflammatory agents
08/17/2006WO2006055734A3 3-phenyl-pyrazole derivatives as modulators of the 5-ht2a serotonin receptor useful for the treatment of disorders related thereto
08/17/2006WO2006028977A3 Chiral spiro compounds and their use in asymmetric catalytic reactions
08/17/2006US20060183908 Heterocyclic compounds, methods of making them and their use in therapy
08/17/2006US20060183905 Derivatives of 4-(thio-or selenoxanthene-9-ylidene)-piperidine or acridine and its use as a selective 5-ht2b receptor antagonist
08/17/2006US20060183899 Having a predominantly cis configuration by coupling an S-oxide of a 2-oxymethyl- thiolane, dithiolane or oxathiolane with a nucleoside base in the presence of a tertiary amine, a Lewis acid of a Group 1B or 2B metal catalyst and deprotecting the intermediate formed
08/17/2006US20060183791 Substituted p-diaminobenzene derivatives
08/17/2006US20060183785 For the treatment of pain; epilepsy, manic depression, bipolar disorder, depression, anxiety and diabetic neuropathy; 5-Methyl-1-[2'-(trifluoromethoxy)-1,1'-biphenyl-3-yl]-1H-pyrazole-3-carboxamide
08/17/2006US20060183784 Human growth hormone antagonists
08/17/2006US20060183762 3-aminoquinazolin-2,4-dione antibacterial agents
08/17/2006US20060183752 Process for preparing 2, 3-disubstituted indoles
08/17/2006US20060183741 Treatment of associated conditions and disorders such as gastrointestinal reflux disorders, eating disorders leading to obesity and irritable bowel syndrome
08/17/2006US20060183736 Selective estrogen receptor modulators containing a phenylsulfonyl group
08/17/2006US20060183732 Novel lactams and uses thereof
08/17/2006CA2598429A1 Substituted bis aryl and heteroaryl compounds as selective 5ht2a antagonists
08/17/2006CA2597680A1 Process for preparing 2,3-disubstituted indoles
08/16/2006EP1691586A1 Charge-transporting organic material containing compound having 1,4-dithiin ring
08/16/2006EP1690854A1 Heterocyclic urea and related compounds useful as anti-inflammatory agents
08/16/2006EP1689744A1 Antiresorptive mutual salt of raloxifene and bisphosphonic acid
08/16/2006EP1689743A2 Piperidinyl-and piperazinyl-sulfonylmethyl hydroxamic acids and their use as protease inhibitors
08/16/2006EP1689729A1 Tetronic and tetramic acids as inhibitors of beta-secrease
08/16/2006EP1689722A2 4-aminopyrimidine derivatives for treatment of hyperproliferative disorders
08/16/2006EP1689720A1 Pyrazolyl derivatives in the form of drugs for treating acute or chronic neuronal regressions
08/16/2006EP1689712A1 4-phenylpiperidine derivatives as renin inhibitors
08/16/2006EP1689710A1 Indole derivatives for use as chemical uncoupler
08/16/2006EP1689403A2 Heteroaryl-hydrazone compounds
08/16/2006EP1689394A1 Amino substituted pyridinyl methanone compounds useful in treating kinase disorders
08/16/2006EP1487437B1 Use of selective ep4 receptor agonists for the treatment of diseases
08/16/2006EP1432702B1 Nitrogen-containing heterocyclic compounds and their use as raf inhibitors
08/16/2006EP1368320B1 Substituted 2-oxy-3,5-dicyano-4-aryl-6-aminopyridines and use thereof
08/16/2006EP1337247B1 Use of Gaboxadol for the treatment of premenstrual disorder, postnatal depression or postmenopausal related dysphoric disorder
08/16/2006EP1261603B1 Flavone derivatives, preparation method and use as medicines
08/16/2006CN1820005A Photochromic diarylethene-containing coordination compounds and the production thereof
08/16/2006CN1269804C Metalloproteinase inhibitors
08/16/2006CN1269801C Amino acid derivatives and drug containing the same as the active ingredient
08/15/2006US7091353 Isoindole-imide compounds, compositions, and uses thereof
08/15/2006US7091343 Compositions useful as inhibitors of protein kinases
08/15/2006US7091247 urotensin antagonists; vasoactive agents
08/15/2006US7091238 substiuted with 3,4-methylenedioxybenzene; treating congestive heart failure and muscle fatigue; nontoxic
08/15/2006US7091237 Furan and thiophene derivatives that activate human peroxisome proliferator activated receptors
08/15/2006US7091234 Thio-oxindole derivatives