Patents
Patents for C07D 409 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms (52,226)
09/2006
09/13/2006EP1699780A1 Novel quinoline derivatives
09/13/2006EP1699779A1 1,2,3,4-tetrahydroisoquinoline derivatives, preparations thereof and uses thereof
09/13/2006EP1699778A1 (4-phenylpiperazin-1-yl)acylpiperidine derivatives, preparation thereof and application of same in therapeutics
09/13/2006EP1699762A1 5-amino-4-hydroxy-7-(1h-indolmethyl)-8-methylnonamide derivatives as renin inhibitors for the treatment of hypertension
09/13/2006EP1699761A1 Cb1 modulator compounds
09/13/2006EP1699455A1 Heterocyclic aspartyl protease inhibitors
09/13/2006EP1699454A1 Pyrazole derivatives and use thereof as orexin receptor antagonists
09/13/2006EP1699421A2 Pharmaceutically acceptable salts of quinolinone compounds having improved pharmaceutical properties
09/13/2006EP1442050B1 Linear basic compounds having nk-2 antagonist activity and formulations thereof
09/13/2006EP1412364B1 Platelet adp receptor inhibitors
09/13/2006EP1389206B1 Inhibitors of c-jun n-terminal kinases (jnk) and other protein kinases
09/13/2006EP0917462B1 Cell adhesion inhibitors
09/13/2006CN1832944A Compounds, methods and formulations for the oral delivery of a glucagon like peptide (glp)-1 compound or an melanocortin 4 receptor (mc4) agonist peptide
09/13/2006CN1832939A Triheterocyclic compounds, compositions, and methods for treating cancer or viral diseases
09/13/2006CN1832930A Amide derivative
09/13/2006CN1832927A Novel gamma-secretase inhibitors
09/13/2006CN1832742A Nitrooxy derivatives of losartan, valsatan, candesartan, telmisartan, eprosartan and olmesartan as angiotensin-ii receptor blockers for the treatment of cardiovascular diseases
09/13/2006CN1832740A Indol-5 sulfonamide derivatives, their preparation and their use 5-ht-6 as modulators
09/13/2006CN1832739A Indol-7 sulfonamide derivatives, their preparation and their use 5-ht-6 as modulators
09/13/2006CN1832738A Indol-6 sulfonamide derivatives, their preparation and their use 5-ht-6 as modulators
09/13/2006CN1274676C Quinoline and quinazoline derivatives
09/13/2006CN1274670C Diaminopropionic acid derivatives
09/12/2006US7105708 Method for producing compounds having a CF2O bridge
09/12/2006US7105682 Substituted amine derivatives and methods of use
09/12/2006US7105671 2-Substituted phenyl,3-polar ring,N-heroaromatic propion-amides, e.g., 1-(2-(3,4-Dichlorophenyl)-3-(tetrahydro-furan-2-yl)-propionyl)-3- methylurea; antidiabetic agents; increase the flux of glucose metabolism in beta-cells and hepatocytes
09/12/2006US7105669 Quinazoline derivatives
09/12/2006US7105565 1-methyl-4-trifluoromethyl-1H-pyrrole-3-carboxylic acid [2-(1,3-dimethylbutyl)phenyl]amide; protecting plants against infestation by phytopathogenic microorganisms
09/12/2006US7105564 7-(3-{[5-(Pyrrole-1-sulfonyl)-thiophene-2-carbonyl]-amino}-bicyclo[2.2.1]hept-2-yl)-hept-5-enoic acid; thromboxane A2 receptor and a prostaglandin D2 receptor; for all of eosinophilic infiltration, advance of respiratory anaphylaxis and respiratory contraction
09/12/2006US7105563 5-ureido-3-[(4-(3-methoxyphenyl)pyrrol-2-yl)methylene]indolin-2-one and derivatives; inhibition of phosphoinositide-dependent kinase-1 (PDK-1).
09/12/2006US7105546 Useful for treating or preventing neuronal damage associated with neurological diseases
09/12/2006US7105544 N-{3-[1-(3-{[BIS(4-FLUOROPHENYL)ACETYL]AMINO}PROPYL)-4-PIPERIDINYL]PHENYL}-2-METHYLPROPANAMIDE; antagonists for melanin concentrating hormone-1 (MCH1) receptors; treating depression, anxiety, obesity
09/12/2006US7105537 For enhancing bone formation; for therapy of diseases or disorders associated with abnormal bone or mineral homeostasis
09/12/2006US7105536 Compounds
09/12/2006US7105527 such as beta-D-N4-p-bromobenzoyl-2',3'-didehydro-2',3'-dideoxy-5-fluorocytidine; for treating human immunodeficiency virus (HIV) and hepatitis B virus (HBV) infections
09/12/2006US7105519 Inhibitors of macrophage migration inhibitory factor and methods for identifying the same
09/12/2006US7105518 Thiopyrane-4-ones as DNA protein kinase inhibitors
09/12/2006US7105515 Such as N-[3-(2-diethylaminoethyl)-1H-indol-5-yl]-5-chloro-3-methylbenzo[b]thiophene-2-sulphonamide for treating anxiety, depression, cognitive memory disorders and senile dementia, psychosis, infant hyperkinesia (ADHD, attention deficit/hyperactivity disorder)
09/12/2006US7105509 Benzodiazepine derivatives as APP modulators
09/12/2006US7105508 Integrin receptors antagonists
09/12/2006US7105505 Benzimidazole derivatives useful as histamine H3 antagonists
09/12/2006US7105503 Pyrazole compounds
09/12/2006CA2235986C Inhibitors of protein isoprenyl transferases
09/12/2006CA2140929C Hydroxyethylamino sulfonamides useful as retroviral protease inhibitors
09/08/2006WO2006094248A1 Aryl-substituted cyclic sirtuin modulators
09/08/2006WO2006094235A1 Fused heterocyclic compounds and their use as sirtuin modulators
09/08/2006WO2006094034A1 Cinnoline compounds and their use as liver x receptor modilators
09/08/2006WO2006093823A1 2- [ isoquinolin-s - carbonyl ) amino] -propionic acid derivatives as inhibitors of factors xi and ix for the treatment of thrombosis
09/08/2006WO2006093253A1 Novel cyclic compound having quinolylalkylthio group
09/08/2006WO2006093247A1 NOVEL AMINOPYRIDINE COMPOUND WITH Syk INHIBITORY ACTIVITY
09/08/2006WO2006092059A1 Design and synthesis of novel antimicrobials
09/08/2006WO2006080043A3 Organic compounds useful for the treatment of alzheimer's disease, their use and method of preparation
09/08/2006WO2006067414A3 Glycine transport inhibitors
09/08/2006WO2005086700A3 Hiv integrase inhibitors
09/08/2006CA2603534A1 Design and synthesis of novel antimicrobials
09/08/2006CA2599992A1 Acridine and quinoline dervatives as sirtuin modulators
09/08/2006CA2599987A1 Fused heterocyclic compounds and their use as sirtuin modulators
09/08/2006CA2599808A1 2- [ isoquinolin-s - carbonyl ) amino] -propionic acid derivatives as inhibitors of factors xi and ix for the treatment of thrombosis
09/08/2006CA2599688A1 Cinnoline compounds and their use as liver x receptor modulators
09/08/2006CA2599544A1 Novel aminopyridine compound with syk inhibitory activity
09/07/2006US20060199964 preparation of 6-haloalkyl-3-nicotinic acid esters and also to novel enamine intermediates
09/07/2006US20060199960 e.g. 6-Methyl-3-(pyridin-3-ylamino)-pyridine-2-carboxylic acid (4-methyl-thiazol-2-yl)-amide; metabotropic glutamate receptor antagonists (mGluR); central nervous system disorders, antidepressant, anxiolytc agent; psychosis, epilepsy, schizophrenia, Alzheimer's disease, cognitive disorders
09/07/2006US20060199957 Novel bicyclic and tricyclic cannabinoids
09/07/2006US20060199847 Stable ammonium salts of alpha-liponic acid, the production thereof and the use of the same
09/07/2006US20060199845 Thiophene compounds for inflammation and immune-related uses
09/07/2006US20060199844 Inhibitors of raf-kinase; Hyperproliferative disorders
09/07/2006US20060199840 Chemical derivatives and their application as antitelomerase agent
09/07/2006US20060199828 Pyrazine-2-carboxyamide derivatives
09/07/2006US20060199827 Inhibitors of macrophage migration inhibitory factor and methods for identifying the same
09/07/2006US20060199826 Cyclopropane compounds and pharmaceutical use thereof
09/07/2006US20060199825 4-Aminating a 4-chloro-2-hydroxy-3-nitrodihydroquinoline with a N-(hetero)cyclylpiperazine, and alkylating the remaining amine group in the quinoline ring to produce a 4-(4-(hetero)cyclylpiperazinyl)-3-nitro-1-alkyldihydroquinolinone
09/07/2006US20060199786 Process and methods for the preparation of optically active cis-2-hydroxymethyl-4- (cytosin-1'-yl) -1,3-oxathiolane or pharmaceutically acceptable salts thereof
09/07/2006DE102005009440A1 Thienopyridinderivate Thienopyridine derivatives
09/07/2006DE102005008649A1 Neue substituierte Pyrrolidinone, deren Herstellung und deren Verwendung als Arzneimittel New substituted pyrrolidinones, their preparation and their use as medicaments
09/06/2006EP1698627A1 Pyrazole compounds useful as protein kinase inhibitors
09/06/2006EP1698375A1 Azetidine ring compounds and drugs comprising the same
09/06/2006EP1698335A1 Preventive and/or therapeutic agent for disease in which mitochondrial benzodiazepine receptor participates
09/06/2006EP1697351A1 2,6-bisheteroaryl-4-aminopyrimidines as adenosine receptor antagonists
09/06/2006EP1697348A1 Hiv protease inhibiting compounds
09/06/2006EP1697329A1 Optically active carboxamides and use thereof to combat undesirable microorganisms
09/06/2006EP1697312A2 Hydroxamic acid esters and pharmaceutical use thereof
09/06/2006EP1697307A1 Opioid receptor antagonists
09/06/2006EP1697292A1 Method for the production of tetrahydrogeranylacetone
09/06/2006EP1696915A1 Benzenesulfonylamino-pyridin-2-yl derivatives and related compounds as inhibitors of 11-beta-hydroxysteroid dehydrogenase type 1 (11-beta-hsd-1) for the treatment of diabetes and obesity
09/06/2006EP1401441A4 Allosteric adenosine receptor modulators
09/06/2006EP1223933B1 5-membered heterocycle derivatives and use thereof as monoaminoxidase inhibitors
09/06/2006CN1829939A Second order nonlinear optical chromophores, polymers containing same, and electro-optic devices therefrom
09/06/2006CN1829712A Nicotinamide derivatives useful as PDE4 inhibitors
09/06/2006CN1829711A Novel heterocyclic compounds useful for the treatment of inflammatory and allergic disorders: process for their preparation and pharmaceutical compositions containing them
09/06/2006CN1829709A Bicyclic imidazol derivatives against flaviviridae
09/06/2006CN1829701A Piperazine derivatives and their use as therapeutic agents
09/06/2006CN1829698A Pyridazine derivatives and their use as therapeutic agents
09/06/2006CN1829695A Aminoquinoline derivatives and their use as adenosine A3 ligands
09/06/2006CN1829508A Indol-4 sulfonamide derivatives, their preparation and their use 5-ht-6 as modulators
09/06/2006CN1829507A 酪氨酸激酶抑制剂 Tyrosine kinase inhibitor
09/06/2006CN1827616A Synthesis and uses of indole analogs of 1-benzyl-3-(5'-hydroxymethy 1-2' -furyl) indazole
09/06/2006CN1827603A Novel pyrazole analogs acting on cannabinoid receptors
09/06/2006CN1273450C 1-aryl-or 1-alkylsulfonylbenzazole derivatives as 5-hydroxytryptamine-6ligands
09/06/2006CN1273444C Dipeptide nitriles
09/06/2006CN1273128C Substituted N-[(aminoiminomethyl or aminomethyl) phenyl] propyl amides
09/05/2006USRE39265 Heteroarylpiperidines, and their use as antipsychotics and analgetics