Patents
Patents for C07D 409 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms (52,226)
06/2008
06/12/2008WO2008070609A1 Thienyl-containing glycopyranosyl derivatives as antidiabetics
06/12/2008WO2008070507A2 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
06/12/2008WO2008070447A2 Anti-viral compounds
06/12/2008WO2008069322A1 Metal coordination compound and light-emitting material using the same
06/12/2008WO2008069313A1 Method for producing pyrrolidine compound
06/12/2008WO2008069242A1 Novel bicyclic heterocyclic compound
06/12/2008WO2008068268A1 Antibacterial quinoline derivatives
06/12/2008WO2008068266A1 Antibacterial quinoline derivatives
06/12/2008WO2008068157A1 2-aminoquinolines as 5-ht(5a) receptor antagonists
06/12/2008WO2008067710A1 Substituted cyclohexane compounds, preparation methods and medicine uses thereof
06/12/2008WO2008067709A1 Substituted cyclobutane compounds, preparation methods and pharmaceutical uses thereof
06/12/2008WO2008067644A1 Inhibitors of hiv replication
06/12/2008US20080139811 Reacting an amino, hydroxy substituted amide with a heterocyclic substituted carboxylic acid to produce (2S,3S,5S)-2-(2,6-Dimethylphenoxyacetyl) amino-3-hydroxy-5-[2S-1-imidazolidin-2-onyl)-3-methyl-butanoyl] amino-1,6-diphenylhexane; inhibitors of HIV infection
06/12/2008US20080139627 Heterocyclic amide and imine derivatives, processes for their preparation, compositions comprising them and their use as pesticides
06/12/2008US20080139561 e.g. 6-(5-Cyclopropyl-1H-pyrazol-3-ylamino)-5-fluoro-2-(1-(4-fluorophenyl)ethylamino) nicotinonitrile; tropomyosin-related kinases (Trk's) inhibitor; anticarcinogenic agent; hormone related cancer, leukemia; antiinflammatory agent; arthritis, restenosis; autoimmune diseases
06/12/2008US20080139536 Benzodiazepines for Treating or Preventing Rsv Infection
06/12/2008CA2671990A1 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
06/12/2008CA2671699A1 Thienyl-containing glycopyranosyl derivatives as antidiabetics
06/12/2008CA2669590A1 2-aminoquinolines as 5-ht(5a) receptor antagonists
06/12/2008CA2668517A1 Antibacterial quinoline derivatives
06/12/2008CA2668515A1 Antibacterial quinoline derivatives
06/11/2008EP1928865A1 Novel high affinity thiophene-based and furan-based kinase ligands
06/11/2008EP1928864A1 Novel cycloalkane carboxamides as factor xa inhibitors
06/11/2008EP1928862A1 2-aminopyrimidine derivatives as modulators of the histamine h4 receptor activity
06/11/2008EP1928859A1 Pyrazole derivates as cannabinoid receptor modulators
06/11/2008EP1928840A1 1h-pyrazole 4-carboxylamides, their preparation and their use as 11beta-hydroxysteroid dehydrogenase
06/11/2008EP1928829A1 Piperidine derivatives as antagonists of the cc chemokine receptor ccr1 and their use as anti-inflammatory agents
06/11/2008EP1928455A1 Anilinopyrazole derivatives useful for the treatment of diabetes
06/11/2008EP1485348B1 Carbonylamino-derivatives as novel inhibitors of histone deacetylase
06/11/2008EP1368032B1 Excitatory amino acid receptor antagonists
06/11/2008EP1313713B1 4-pyrimidinamine derivatives, pharmaceutical compositions and related methods
06/11/2008EP1255739B1 3-aminoquinazolin-2,4-dione antibacterial agents
06/11/2008EP1230235B1 Compounds with antibacterial and antiparasitic properties
06/11/2008CN101198602A Saminopyrimidine derivates with tIE2 inhibiting activity
06/11/2008CN101198594A Process for the production of intermadiates for the preparation of tricyclic benzimidazoles
06/11/2008CN101195604A 4,5-dihydro-1H-pyrazole derivatives having potent CB1-antagonistic activity
06/11/2008CN100393715C Imidazole deriviatives and their use as peripherally-selective inhibitors of dopamine-beta-hydroxylase
06/10/2008US7385067 Process for the preparation of compounds having a CF2O bridge
06/10/2008US7385063 Method for preparing imidazole derivatives
06/10/2008US7385059 3,4-disubstituted 1H-pyrazole compounds and their use as cyclin dependent kinase and glycogen synthase kinase-3 modulators
06/10/2008US7384962 Heterocyclic compounds useful for the treatment of inflammatory and allergic disorders: process for their preparation and pharmaceutical compositions containing them
06/10/2008US7384957 3,4-dihydro-1H-isoquinolin-2-yl-derivatives
06/10/2008US7384947 Treating cancer with anticarcinogenic agents 3-Amino-9-chloro-5,6,7,8-tetrahydro-naphtho[2,3-b]furan-2-yl))-(2-methyl-pyridin-3-yl)-methanone; antiproliferative agents
06/10/2008US7384944 Organ grafting; antiarthritic agents; inflammatory bowel disease
06/10/2008CA2129046C Opioid diarylmethylpiperazines and piperidines
06/05/2008WO2008067219A2 Quinazolinone modulators of tgr5
06/05/2008WO2008065754A1 Substituted carbinol compound
06/05/2008WO2008043791A3 Thiophene derivatives for treating hepatitis c
06/05/2008WO2008043788A3 Novel compounds
06/05/2008WO2008024765B1 Therapeutic substituted thiazolidinones, oxazolidinones, and related compounds
06/05/2008US20080132562 Tetronic and tetramic acids
06/05/2008US20080132558 1-arylpyrazoles and their use as pesticide
06/05/2008US20080132557 Heterocyclic Carboxamides with Microbiocidal Activity
06/05/2008US20080132550 4,5-diphenyl-2-amino-4,5-dihydro-imidazole derivatives; antiinflammatory agent, neurodegenerative diseases; inflammatory bowel disease, rheumatoid arthritis and diseases associated with central nervous system, such as Alzheimer's disease
06/05/2008US20080132540 Such as trans-N-(1-Acetyl-2,3-dihydro-1H-indol-6-yl)-N-(1-benzyl-piperidin-4-yl)-3-phenyl-acrylamide; for treating/preventing anxiolytic disorders/depression, injured mammalian nerve tissue, conditions, neurological disorders, bone loss, substance related disorders, and obesity; neuropeptide y (NPY Y2)
06/05/2008US20080132521 Isoquinolinone Derivatives and Their Use As Therapeutic Agents
06/05/2008US20080132503 Inhibitors of Histone Deacetylase
06/05/2008US20080132496 Anticoagulants; factor Xa inhibitors; compounds are N-(benzimidazolyl, imidazo(4,5-b)pyridyl- or indolyl)-substituted benzamides
06/05/2008US20080132481 Use of 3-substituted amino-2-carboxy-substituted indoles or benzo(b)thiophenes or esters thereof that modulate T helper (Th) cells; treating allergy, asthma, rhinitis, dermatitis, B-cell lymphomas, tumors and diseases associated with bacterial, rhinovirus or respiratory syncytial virus (RSV) infections
06/05/2008US20080132459 Inhibitors of Histone Deacetylase
06/05/2008DE19946341B4 Verfahren zur Herstellung substituierter Phenylsulfonylharnstoffe aus Sulfohalogeniden A process for the preparation of substituted phenylsulfonylureas of Sulfohalogeniden
06/05/2008DE102006056526A1 Verfahren zur stereoselektiven Synthese von chiralen Epoxiden durch ADH-Reduktion von alpha-Abgangsgruppen-substituierten Ketonen und Cyclisierung Method for the stereoselective synthesis of chiral epoxides by ADH reduction of alpha-leaving group-substituted ketones and cyclization
06/04/2008EP1927594A1 1,2,3-Trisubstituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto such as diabetes and hyperglycemia
06/04/2008EP1927589A1 Quinoline derivatives
06/04/2008EP1926826A2 Class iia histone deacetylase (hdac) substrate
06/04/2008EP1926724A1 Analogs of dehydrophenylahistins and their therapeutic use
06/04/2008EP1926721A2 Thiophene and thiazole substituted trifluoroethanone derivatives as histone deacetylase (hdac) inhibitors
06/04/2008EP1926712A1 6-substituted 2,3,4,5-tetrahydro-1h-benzo[d]azepines as 5-ht2c receptor agonists
06/04/2008EP1926708A1 Biaryl substituted heterocycle inhibitors of lta4h for treating inflammation
06/04/2008EP1532134B1 Novel thiophene acyl hydrazino derivatives, method for preparing same, use thereof as medicines, pharmaceutical compositions and novel use
06/04/2008EP1487817B1 Piperidine derivatives useful as modulators of chemokine receptor activity
06/04/2008EP1343775B1 Piperazine derivatives
06/04/2008EP1237887B1 9-(piperazinylalkyl)carbazoles as bax-modulators
06/04/2008EP1204643B1 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
06/04/2008CN101193887A 新颖的三环血管紧张素Ⅱ激动剂 Novel tricyclic angiotensin Ⅱ agonists
06/04/2008CN101193886A New tricyclic angiotensin II agonists
06/04/2008CN101193881A New bicyclic angiotensin II agonists
06/04/2008CN101193874A 6-oxazol-4-ylmethoxy-alkoxymethyl substituted benzoic acid derivatives forming PPAR ligands, methods for production and the use thereof in the form of drugs
06/04/2008CN101193869A Glucocortioid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
06/04/2008CN101193867A N-substituted benzimidazolyl c-Kit inhibitors and combinatorial benzimidazole library
06/04/2008CN101193631A Inhibitors of soluble adenylate cyclase
06/04/2008CN100391954C Enantiomers of thiophene hydroxamic acid derivatives and their use as hdac inhibitors
06/04/2008CN100391944C Indoles useful in the treatment of androgen-receptor related diseases
06/04/2008CN100391942C Pure enantiomer basic aryl-cycloalkyl-hydroxycarboxylic acid esters, process for preparing same and their use in medicaments
06/03/2008US7381824 Quinoline derivatives
06/03/2008US7381741 In which the amino is substituted by arylmethyl- or heteroarylmethyl- group, e.g., 2-Methoxybenzyl)-(2-phenylpyrrolidin-3-yl)-amine and 5-{[2-(3-Chloro-phenyl)-pyrrolidin-3-ylamino]-methyl}-6-methoxy-3-methyl-1,1a,3,7b-tetrahydro-3-aza-cyclopropa[a]naphalen-2-one; neurokinin 1 (Substance P) inhititors
06/03/2008US7381739 Antiserotonine agents; central nervous system disorders; Alzheimer's disease; Parkinson's disease; Huntington's disease; sleep disorders
06/03/2008US7381725 Pyridazine derivatives as ligands for GABA receptors
06/03/2008US7381721 Substituted piperidine compounds
06/03/2008US7381719 To treat obesity and Related Diseases; oral bioavailablility, oral administration; inhibition of orexigenic effects; side effects reduction; weight loss while maintaining or minimizing the loss of lean muscle mass; 6-[4-(2-Benzylamino-ethyl)-phenoxy]-nicotinamide
06/03/2008US7381537 Use of inhibitors of glutaminyl cyclases for treatment and prevention of disease
06/03/2008CA2401711C Cyclic amide derivatives
06/03/2008CA2389360C Urea derivatives as anti-inflammatory agents
05/2008
05/29/2008WO2008062878A1 Novel pyrazole derivative, harmful organism control agent, and use of the control agent
05/29/2008WO2008062770A1 Quinolone derivative or pharmaceutically acceptable salt thereof
05/29/2008WO2008062739A1 Pyrazoles and use thereof as drugs
05/29/2008WO2008062424A2 Substituted 4,5-dihydro-1h-pyrazole derivatives as cannabinoid modulators
05/29/2008WO2008062012A1 Pyridazin-4-ylmethyl-sulfonamides used as fungicides and against arthropods
05/29/2008WO2008062011A1 Pyrimidylmethyl-sulfonamide compounds useful as fungicides and against arthropods
05/29/2008WO2008061740A1 Pyrimidines and their use as cxcr2 receptor antagonists