Patents for C07D 409 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms (52,226) |
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07/24/2008 | CA2675676A1 Nicotinic acetylcholine receptor modulators |
07/24/2008 | CA2674865A1 Indole derivative having i.kappa.b kinase .beta. inhibitory activity |
07/23/2008 | EP1947101A1 Hydrazide compound and thrombopoietin receptor activator |
07/23/2008 | EP1947097A1 BENZOÝb¨THIOPHEN DERIVATIVE AND PROCESS FOR PRODUCTION THEREOF |
07/23/2008 | EP1947096A1 3-HYDROXYMETHYLBENZO[b]THIOPHENE DERIVATIVE AND METHOD FOR PRODUCING SAME |
07/23/2008 | EP1947086A1 Benzene derivative or salt thereof |
07/23/2008 | EP1947085A1 Substituted indole sulfonamide compounds, their preparation and use as medicaments |
07/23/2008 | EP1945617A2 Histone deacetylase inhibitors with aryl-pyrazolyl motifs |
07/23/2008 | EP1945612A2 Heterocyclic compounds as pstat3/il-6 inhibitors |
07/23/2008 | EP1945609A2 Amino acid derivatives as histone deacetylase (hdac) inhibitors |
07/23/2008 | EP1794152B1 Method for manufacturing enantiomeric imidazole compounds |
07/23/2008 | EP1685108B1 1,4-dihydropyridine compounds, pharmaceutical compositions, and methods for the treatment of cardiovascular disease |
07/23/2008 | EP1597247B1 Substituted 3-(benzoylureido)-thiophene derivatives, method for the production and use thereof |
07/23/2008 | EP1567489B1 Pyrrolidin-2-one derivatives as inhibitors of thrombin and factor xa |
07/23/2008 | EP1382603B1 Nitrogenous fused-ring compound having pyrazolyl group as substituent and medicinal composition thereof |
07/23/2008 | EP1071680B1 N,n-disubstituted amides that inhibit the binding of integrins to their receptors |
07/23/2008 | CN101228154A Novel tetracyclic tetrahydrofuran derivatives containing a cyclic amine side chain |
07/23/2008 | CN101228133A Heteroaroyl-substituted serineamides |
07/23/2008 | CN101225084A Dihydropyrimidine compound and use thereof in preparation of medicine treating and preventing virus diseases |
07/23/2008 | CN100404544C 9-ketospinosyn derivatives |
07/23/2008 | CN100404509C Isoquinoline compound, preparation method and application of salt thereof |
07/23/2008 | CN100404508C Tetrahydroquinoline derivatives |
07/22/2008 | US7402696 exert an ACC activity-inhibiting effect that is effective in the treatment of obesity, hyperlipemia, fatty liver, hyperglycemia, impaired glucose tolerance, diabetes, diabetic complications (diabetic peripheral neuropathy, diabetic nephropathy, diabetic retinopathy, and diabetic macroangiopathy, hyperten |
07/22/2008 | US7402683 Cinnamic acid amides |
07/22/2008 | US7402608 Compounds and methods for the treatment or prevention of Flavivirus infections |
07/22/2008 | US7402606 Derivatives of 1-(oxoaminoacetyl) pentylcarbamate as cathepsin K inhibitors for the treatment of bone loss |
07/22/2008 | US7402605 E.g., 17,17-propano-16-hydroxy-5-(4-ethoxycarbonylthiazol-2-yl)-9-oxo-1,2,3,4,20-pentanor-5-thia-8-azaprost-13-ene; EP2 and/or EP4 receptor agonist; immune disease; antiallergens; alopecia; dysmenorrhea; erectile dysfuncction; antiarthritic agents; liver, respiratory, vascular, urogenital disorder |
07/22/2008 | US7402597 e.g. [[7-Allyl-3-[2-[2-(2,4-dichlorophenyl)-5-isopropyl-4-oxazolyl]ethyl]-1,2-benzisoxazol-6-yl]oxy]acetic acid; with vehicles (lactose, D-mannitol, glucose), disintegrators (starch or carboxymethylcellulose calcium ), binders (hydroxypropylcellulose) and lubricants (magnesium stearate or talc) |
07/22/2008 | US7402589 such as 1-(4-Fluorophenyl)-1-{2-[(1S)-2-hydroxy-1,2-dimethyl-propylamino]-pyrimidin-4-yl}-3-o-tolyl-urea; Interleukin-1, Cycloxygenase-2, Tumor Necrosis Factor- alpha antagonist; antiinflammatory agent; rheumatoid arthritis or osteoarthritis |
07/22/2008 | US7402586 3-Benzylsulfonylamino-6-methyl-1-[(3-guanidinooxypropyl)aminocarbonylmethyl]-2-pyridinone trifluoroacetate; anticoagulants either embedded in or physically linked to materials used in the manufacture of devices used in blood collection, blood circulation, and blood storage |
07/22/2008 | US7402583 Substituted quinolines as antitumor agents |
07/22/2008 | US7402581 3,5-Dibromo-N-[(2S)-2-(4-fluorophenyl)-4-(3-morpholin-4-ylazetidin-1-yl)butyl]-N-methylbenzamide; neurokinin 1 and 2 (NK1,2) receptors, antagonist; improved pharmacokinetics: not inhibit liver enzyme cytochrome P450, prevent drug-drug interactions, oral bioavailability, antiinflammatory and analgesic |
07/22/2008 | US7402580 Polymerase inhibitors; antiischemic agents; brain disorders; cardiovascular disorders; antiinflammatory agents; antiarthritic agents; neurodegenerative agents; Alzheimer's disease; muscular disorders; antidiabetic agents; kidney disorders; viricides; anticancer agents; immunosuppressants |
07/22/2008 | CA2474511C Benzofuran and benzothiophene derivatives useful in the treatment of hyper-proliferative disorders |
07/22/2008 | CA2388076C Novel substituted succinic acid metallo-beta-lactamase inhibitors and their use in treating bacterial infections |
07/22/2008 | CA2372840C Substituted bicyclic compounds |
07/22/2008 | CA2278223C 1,4-dihydropyridin derivatives and their use in therapy |
07/22/2008 | CA2238171C Quinoline derivatives as nk3 antagonists |
07/17/2008 | WO2008086226A2 Factor xa inhibitors |
07/17/2008 | WO2008086188A2 Thiophene carboxamides as factor xa inhibitors |
07/17/2008 | WO2008084671A1 Process for producing 1-substituted-2-pyridone-3-carboxylic acid derivative |
07/17/2008 | WO2008084073A1 Heteroaryl-substituted serine amides |
07/17/2008 | WO2008084004A1 Sulfonamide derivatives as chymase inhibitors |
07/17/2008 | WO2008067219A3 Quinazolinone modulators of tgr5 |
07/17/2008 | WO2008056257A3 Novel triazinedione derivatives as gaba-b receptor modulators |
07/17/2008 | WO2008045564A8 Carboxamide compounds and their use as antagonists of the chemokine ccr2 receptor |
07/17/2008 | US20080171882 [(4S)-4-Methyl-2,5-dioxoimidazolidin-4-yl]methanesulfonyl chloride and [(4R)-4-methyl-2,5-dioxoimidazolidin-4-yl]methanesulfonyl chloride; chemical intermediates for enzyme inhibitors |
07/17/2008 | US20080171767 N-substituted-2-alkylthio-2-(substituted aryloxy and heteroaryloxy)alkylamides and their sulphinyl and sulphonyl derivatives such as 2-(3,5-dichlorophenoxy)-2-methylthio-N-2-methylprop-2-yl acetamide; fungal infections of plants |
07/17/2008 | US20080171733 Antiinflammatory agents, antidepressants, analgesics, purinergic receptor antagonists; neurodegenerative diseases, spinal cord injuries; 1-(2,3-dichlorophenyl)-N-[(2-methylphenyl)methyl]-1H-tetraazol-5-amine |
07/17/2008 | US20080171692 Substituted amides |
07/17/2008 | US20080171050 Treatment of hyperproliferative diseases with epidermal growth factor receptor antagonists |
07/17/2008 | DE4345588B4 Selbstlade-Granatwerfer Self-loading grenade launcher |
07/17/2008 | CA2674924A1 Factor xa inhibitors |
07/17/2008 | CA2674843A1 Factor xa inhibitors |
07/17/2008 | CA2674644A1 Sulfonamide derivatives as chymase inhibitors |
07/17/2008 | CA2673377A1 Heteroaryl-substituted serineamides |
07/16/2008 | EP1944308A1 Process for production of ortho-metallized 1:3 complex of iridium with homoligand |
07/16/2008 | EP1944305A1 Quinoline derivatives as phosphodiesterase inhibitors |
07/16/2008 | EP1943245A2 1,3-disubstituted indole derivatives for use as ppar modulators |
07/16/2008 | EP1943242A1 Piperidin-4-yl-pyridazin-3-ylamine derivatives as fast dissociating dopamine 2 receptor antagonists |
07/16/2008 | EP1943222A1 Antibacterial active 5-chinolin derivative |
07/16/2008 | EP1943221A1 Piperazine amidines as antiviral agents |
07/16/2008 | EP1556376B1 Large conductance calcium-activated k channel opener |
07/16/2008 | EP1527049B1 Fused heterocyclic compounds as peptidase inhibitors |
07/16/2008 | EP1476151B1 1-arylsulfonyl-3-substitued indole and indoline derivates useful in the treatment of central nervous system disorders |
07/16/2008 | EP1392655B1 Potassium channel openers |
07/16/2008 | EP1386913B1 Pyrrole derivative |
07/16/2008 | EP1286966B1 4-aminopiperidine derivatives and their use as medicine |
07/16/2008 | EP1165551B1 C10 carbamoyloxy substituted taxanes as antitumor agents |
07/16/2008 | EP1054004B1 Novel pyrimidine-5-carboxamide derivatives |
07/16/2008 | CN101223164A Substituted piperidines as renin inhibitors |
07/16/2008 | CN101223155A Benzoheterocyclylethylcarboxamide derivatives |
07/16/2008 | CN101223154A 噻吩化合物和血小板生成素受体激活剂 Thiophene compounds and thrombopoietin receptor activators |
07/16/2008 | CN101223147A Pyrimidindione derivatives as prokineticin 2 receptor antagonists |
07/16/2008 | CN101223146A Modulators of ATP-binding cassette transporters |
07/16/2008 | CN101223144A Pyrazole-4- carboxamide derivatives as microbiocides |
07/16/2008 | CN101223140A Piperidine derivatives useful in the diagnostic and therapeutic treatment of diseases depending on renin activity |
07/16/2008 | CN101222924A Substituted piperidine derivatives as somatostatin sst1 receptor antagonists |
07/16/2008 | CN100402526C Lysotropic-photodiscolour diaryl ethylene and preparation and application thereof |
07/16/2008 | CN100402525C Pyridine derivatives as fungicidal compounds |
07/16/2008 | CN100402521C 4-imidazolin-2-one compounds |
07/16/2008 | CN100402501C Aminoquinoline derivatives and their use as adenosine A3 ligands |
07/16/2008 | CN100402499C 2-iminopyrrolidine derivatives |
07/15/2008 | US7399865 such as (E)-N-{4-[4-(benzyloxy)-3-chloroanilino]-3-cyano-7-ethoxy-6-quinolinyl}-4-(dimethylamino)-2-butenamide used as antineoplastic agents, or inhibitors of the HER-2 gene or proteins and epidermal growth factor receptor enzymes |
07/15/2008 | US7399781 N-substituted benzothiophenesulfonamide derivatives |
07/15/2008 | US7399780 pyridin-2-yl-1H-indole or pyrimidin-4-yl-1H-indole derivatives; enzyme inhibitor of glycogen synthase kinase-3; treating dementia, Alzheimer's Disease, Parkinson's Disease, amyotrophic lateral sclerosis, corticobasal degeneration, Down syndrome, Huntington's Disease |
07/15/2008 | US7399778 by targeting beta and gamma secretase enzyme decreases production of amyloid precursor protein; 5-Chloro-N-{2-ethyl-1-[1-(4-methoxybenzyl)-1H-pyrazol-5-yl]butyl}thiophene-2-sulfonamide; Alzheimer's Disease, Down's Syndrome, cognitive decline |
07/15/2008 | US7399776 Antiinflamamtory agents; immunology disorders; autoimmune diseases; antiallergens; aids viricides; antiarthritic agents; muscular disorders; Parkinson's disease; Alzheimer's disease; kidney damage |
07/15/2008 | US7399774 6-substituted nicotinamide derivatives as opioid receptor antagonists |
07/15/2008 | US7399771 Piperidine derivatives as CCR5 inhibitors |
07/15/2008 | US7399770 N-(hydroxy)-2-(4'-chlorobiphenyl-4-sulfonyl)-4-hydroxy-1,2,3,4-tetrahydrobenzo[4,5]thieno[3,2-c]pyridine-1-carboxamide; collagenase inhibitor; antiinflammatory, angiogenesis agent, wound healing agent; arthritis, multiple sclerosis, osteoarthrosis, atherosclerosis, restenosis, myocardial infarction |
07/15/2008 | US7399767 Heterocyclic benzo[c]chromene derivatives useful as modulators of the estrogen receptors |
07/15/2008 | US7399765 Substituted diazabicycloalkane derivatives |
07/15/2008 | US7399761 Phthalazine derivatives with angiogenesis inhibiting activity |
07/15/2008 | US7399749 For therapy and prophylaxis of disorders associated with the HCV protease |
07/15/2008 | US7399432 Charge transport compositions and electronic devices made with such compositions |
07/15/2008 | CA2421120C Quinolinone derivatives as tyrosine kinase inhibitors |
07/10/2008 | WO2008083124A1 N-substituted-heterocycloalkyloxybenzamide compounds and methods of use |
07/10/2008 | WO2008082487A2 Novel jnk inhibitors |
07/10/2008 | WO2008081476A2 Process for preparing duloxetine hydrochloride |