Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
03/2003
03/06/2003WO2003018021A1 2,4-disubstituted pyrimidinyl derivatives for use as anticancer agents
03/06/2003WO2003018017A1 3-substituted 6,7-dihydroxytetrahydroisoquinoline derivatives for use as antibacterial agents
03/06/2003WO2003018008A1 Apo ai expression accelerating agent
03/06/2003WO2003018002A2 Cyclopropyl and cyclobutyl epothilone analogs
03/06/2003WO2003018000A1 Novel ascorbic acid compounds, methods of synthesis and application
03/06/2003WO2002102382A9 A PROCESS FOR PREPARING PAROXETINE HCl WHICH LIMITS FORMATION OF PINK COLORED COMPOUNDS
03/06/2003WO2002100844A3 Hiv protease inhibitors, compositions containing the same, their pharmaceutical uses and materials for their synthesis
03/06/2003WO2002072570A3 Non-imidazole compounds as histamine h3 antagonists
03/06/2003WO2002066443A3 2-thioxo-1,2,3,4-tetrahydropyrimidine derivatives
03/06/2003WO2002057224A3 Synthesis and antimicrobial activityof novel dicationic 'reversed amidines'
03/06/2003US20030045717 Suitable as fluorescent dyes (fluorophores) for used in optical determination and demonstration methods in medicine, pharmacology and biological and environmental sciences; photostability, storage stability
03/06/2003US20030045711 Epothilone derivatives and methods for making and using the same
03/06/2003US20030045705 Backbone modified oligonucleotide analogues
03/06/2003US20030045560 6-(Aryl-amido or aryl-amidomethyl)-naphthalen-2-yloxy-acidic derivatives as inhibitors of plasminogen activator inhibitor type-1 (PAI-1)
03/06/2003US20030045552 Isoindole-imide compounds, compositions, and uses thereof
03/06/2003US20030045551 Pseudopolymorph of ( - ) -cis -2-(2 -chlorophenyl) -5, 7-dihydroxy-8 [4R- ( 3S-hydroxy -1-methyl)piperidinyl ] -4H -1 -benzopyran-4-one
03/06/2003US20030045528 Antibacterial and antiprotozoal agents
03/06/2003US20030045525 Particularly in the treatment of benign prostatic hyperplasia.
03/06/2003US20030045519 Treating allergy, allergy-induced airway responses, and congestion (e.g., nasal congestion)
03/06/2003US20030045516 Chemokine receptor antagonists and methods of use therefor
03/06/2003US20030045479 Novel N-formyl hydroxylamine compounds, compositions and methods of use
03/06/2003US20030045444 High thermal stability, are used as stabilizers for organic polymers to counter damage thereto caused by light, oxygen and heat, as light stabilizers for textile fiber materials and as sunscreens for the human skin.
03/06/2003US20030044399 Method of treatment
03/06/2003CA2458477A1 3-substituted 6,7-dihydroxytetrahydroisoquinoline derivatives for use as antibacterial agents
03/06/2003CA2458344A1 Ascorbic acid derivatives, methods of synthesis and pharmaceutical use thereof
03/06/2003CA2457838A1 2,4-disubstituted pyrimidinyl derivatives for use as anticancer agents
03/06/2003CA2456280A1 Cyclopropyl and cyclobutyl epothilone analogs
03/06/2003CA2455842A1 Process for the preparation of indole derivatives
03/06/2003CA2455311A1 Rapamycin dialdehydes
03/06/2003CA2455308A1 Rapamycin 29-enols
03/05/2003WO2002020507A1 Chromanone derivatives
03/05/2003EP1288214A1 Paroxetine methanesulfonate
03/05/2003EP1288202A1 N-acyltetrahydroisoquinoline derivatives
03/05/2003EP1287011A1 Hygromycin a derivatives for the treatment of bacterial and protozoal infections
03/05/2003EP1286986A1 Quinolinyl-piperidin-4-ylidene-methyl-benzamide derivatives for the treatment of pain
03/05/2003EP1286985A1 Substituted pyridine herbicides
03/05/2003EP1286967A1 Cyclohexane derivatives and their use as therapeutic agents
03/05/2003EP1286966A1 4-aminopiperidine derivatives and their use as medicine
03/05/2003EP1286965A1 Piperidine compounds and process for providing such
03/05/2003EP1286955A1 Aryl and heteroarylcyclopropyl oxime ethers and their use as fungicides
03/05/2003EP1286949A2 Process for the preparation of aniline compounds
03/05/2003EP1202984B1 diphenyl-piperidine derivate
03/05/2003EP1194427B1 Thiophene-ethyl thiourea compounds and use in the treatment of hiv
03/05/2003EP1119560B1 Naphthopyrans annelated in c5-c6, their preparation and compositions and (co) polymer matrices containing them
03/05/2003EP1021411B1 Benzamide derivatives as thrombin inhibitors
03/05/2003EP0966447B1 Small molecules useful in the treatment of inflammatory disease
03/05/2003EP0945438B1 Pyrazole derivatives
03/05/2003EP0942901B1 Cyclic imines as pesticides
03/05/2003EP0896577B1 Taxane derivatives having a Pyridyl substituted C13 side chain and their use as anti-tumor agents
03/05/2003EP0832069B1 BIPHENYL-2-CARBOXYLIC ACID-TETRAHYDRO-ISOQUINOLIN-6-YL AMIDE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS INHIBITORS OF MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN AND/OR APOLIPOPROTEIN B (Apo B) SECRETION
03/05/2003EP0831830B1 Imidazole compounds
03/05/2003CN1400970A Substituted arylpyrazines
03/05/2003CN1400969A Fused imidazolium derivatives
03/05/2003CN1400968A Method for preparing alpha sulfonyl hydroxamic acid derivatives
03/05/2003CN1102592C 2R, 4S, S,S-and 2S, 4R, S,S-hydroxyitraconazole
03/05/2003CN1102580C Arylethenesulfonamide derivatives and drug composition containing the same
03/05/2003CN1102376C Improved anti dandruff shampoo
03/05/2003CA2421287A1 Chromanone derivatives
03/04/2003US6528661 Providing atorvastatin ester derivative; converting the atorvastatin ester derivative to atorvastatin hemi-calcium with calcium hydroxide
03/04/2003US6528538 Cyclic compounds useful in the treatment of dyslipidaemia, atherosclerosis and diabetes, pharamaceutical compositions and preparation process
03/04/2003US6528535 Bicyclic inhibitors of protein farnesyl transferase
03/04/2003US6528532 Benzenesulfonamide group
03/04/2003US6528531 Aliphatic hydroxy substituted piperidyl diaryl pyrrole derivatives as antiprotozoal agents
03/04/2003US6528526 Inhibition of cell proliferation and/or cell matrix production and/or cell movement (chemotaxis) and/or T cell activation and proliferation
03/04/2003US6528510 HIV protease inhibitors
03/04/2003US6528509 Pyrazole compositions useful as inhibitors of ERK
03/04/2003CA2218913C Substituted oximes, hydrazones and olefins as neurokinin antagonists
03/04/2003CA1341424C Diketohexanoic acids and 2- and 3-diloweralkyl derivatives thereof
02/2003
02/27/2003WO2003016306A1 Hiv inhibiting pyrimidines derivatives
02/27/2003WO2003016292A1 Ultraviolet light absorbers
02/27/2003WO2003016289A1 Triazine derivatives and their use as sunscreens
02/27/2003WO2003016286A1 3-phenoxy-4-pyridazinol derivative and herbicide composition containing the same
02/27/2003WO2003016276A2 3-substituted oxindole beta-3 agonists
02/27/2003WO2003016275A1 Antiviral agent
02/27/2003WO2003016265A1 Cyclic compound and ppar agonist
02/27/2003WO2003015785A1 2h-phthalazin-1-ones and methods for use thereof
02/27/2003WO2003015774A1 Compounds effecting glucokinase
02/27/2003WO2003015769A1 Aminoalkyl-substituted aromatic bicyclic compounds, method for the production thereof and their use as medicaments
02/27/2003WO2003015517A1 Agonists and antagonists of 5h3-like receptors of invertebrate s as pesticides
02/27/2003WO2002098865A3 Cyclic nucleotide phosphodiesterase inhibitors, preparation and uses thereof
02/27/2003WO2002094180A3 Pharmaceutically active isoindoline derivatives
02/27/2003WO2002092588A3 Aromatic sulfone hydroxamates and their use as protease inhibitors
02/27/2003WO2002089782A3 Dioxanes and uses thereof
02/27/2003WO2002089749A3 Arylsulfonamide ethers, and methods of use thereof
02/27/2003WO2002085301A3 Indole, azaindole and related heterocyclic amidopiperazine derivatives
02/27/2003WO2002079149A3 Novel cyano-substituted dihydropyrimidine compounds and their use to treat diseases
02/27/2003WO2002067675A3 Substituted 4,5-dihydro-1,2,4-triazin-6-ones, 1,2,4-triazin-6-ones, and their use as fungicides and insecticides
02/27/2003US20030040639 Reacting polymer bound chemical intermediate compound with complex to produce complex compound; reacting with nucleophile(s); benzene derivative is decomplexed, optionally derivatised, cleaved from the support
02/27/2003US20030040631 As chemical intermediates used for the preparation of S-alpha-ethyl-2-oxo-1-pyrrolidine acetamide
02/27/2003US20030040536 For therapy of disease states in mammals that are alleviated by a protein kinase inhibitor, particularly diseases such as cancer, inflammatory disorders, restenosis, and cardiovascular disease
02/27/2003US20030040532 Methods for treating dementia due to HIV disease
02/27/2003US20030040437 Substituted pyridine herbicides
02/27/2003CA2457037A1 Aminoalkyl-substituted aromatic bicyclic compounds, method for the production thereof and their use as medicaments
02/27/2003CA2456985A1 2h-phthalazin-1-ones and methods for use thereof
02/27/2003CA2456290A1 Agonists and antagonists of 5h3-like receptors of invertebrate s as pesticides
02/27/2003CA2454080A1 Ultraviolet light absorbers
02/26/2003EP1285920A1 C10 Ester sustituted taxanes as antitumor agents
02/26/2003EP1285918A1 C7 Ester substituted taxanes as antitumor agents
02/26/2003EP1284966A2 Process for the synthesis of amine ethers from secondary amino oxides
02/26/2003EP1284741A2 3'-or 2'-hydroxymethyl substituted nucleoside derivatives for treatment of hepatitis virus infections