Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
09/2003
09/10/2003EP1341761A1 SUBSTITUTED INDOLES, PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH INDOLES AND THEIR USE AS PPAR-$g(g) BINDING AGENTS
09/10/2003EP1341759A2 3-substituted oxindole beta 3 agonists
09/10/2003EP1341755A1 Carboxylic acid amide derivatives and their use in the treatment of thromboembolic diseases and tumours
09/10/2003EP1341537A2 Pharmaceutically active isoindoline derivatives
09/10/2003EP1159237B1 Method of preparing surface-active alcohols and surface-active alcoholic ethers, products obtained by said method and their use
09/10/2003EP1141153B1 Crosslinking composition for carboxyl-containing polymers in heat-curable systems
09/10/2003EP1137644B1 Benzofuran derivatives, their preparation and use
09/10/2003EP1094813B1 Use of piperine and derivatives thereof for treating skin pigmentation disorders and skin cancer
09/10/2003EP1023063B1 INDENO[1,2-c], NAPHTHO[1,2-c]- AND BENZO[6,7]CYCLOHEPTA[1,2-c]PYRAZOLE DERIVATIVES
09/10/2003EP0983236B1 Process for the preparation of an oxirane, aziridine or cyclopropane
09/10/2003EP0934264B1 Pyrrolidinyl and pyrrolinyl ethylamine compounds as kappa agonists
09/10/2003CN1441800A Beta 3 adrenergic agonists
09/10/2003CN1441794A Lipid-rich plague inhibitors
09/10/2003CN1441791A 四唑衍生物 Tetrazole derivative
09/10/2003CN1441789A Piperazinedione compounds
09/10/2003CN1441788A Novel arylethene-sulfonamides compounds
09/10/2003CN1441787A Modulators of TNF-alpha signaling
09/10/2003CN1441786A Novel diamino pyrazole derivatives and dyes containing said compounds
09/10/2003CN1441785A Tetrahydroixoquinoline analogs useful as growth hormone secretagogues
09/10/2003CN1441783A Medicine comprising dicyanopyridine derivative
09/10/2003CN1441781A Pharmaceutically active piperidine derivatives, in particular as modulators of chemokine receptor activity
09/10/2003CN1441780A Piperidine compounds for use as CCR-3 inhibitors
09/10/2003CN1441775A Hiv整合酶抑制剂 Hiv integrase inhibitors
09/10/2003CN1120838C Dihydrobenzofuran compounds useful as anti-inflammatong agents
09/09/2003US6617451 Amidation of a racemic mixture of a cis-azetidinone having an unsaturated side group with an alkyl phenyl- or phenoxy-acetate in the presence of penicillin G amidase, optionally followed by hydrogenation.
09/09/2003US6617437 Modified oligonucleotide of given formula; useful in diagnostics and therapeutics
09/09/2003US6617347 Selective β3 adrenergic agonists
09/09/2003US6617346 Inhibit the interaction of MDM2 protein with a p53-like peptide and have antiproliferative activity
09/09/2003US6617329 Aminoquinazolines and their use as medicaments
09/09/2003US6617324 Substituted pyrazoles as p38 kinase inhibitors
09/09/2003US6617320 Protease inhibitor; anticoagulants
09/09/2003US6617281 Substituted acylamino phenyl uracils
09/09/2003CA2248953C Novel benzofuranone derivatives and process for producing the same
09/09/2003CA2079413C Pyrimidine nucleoside derivatives having anti-tumor activity, their preparation and use
09/04/2003WO2003072574A1 Piperidine ouracil used as a medicament for treating bacterial infections
09/04/2003WO2003072570A1 Antidiabetic agents
09/04/2003WO2003072569A1 1,4-disubstituted benzofused cycloalkyl urea compounds useful in treating cytokine mediated diseases
09/04/2003WO2003072566A1 Fused tricyclic heterocycles useful for treating hyper-proliferative disorders
09/04/2003WO2003072561A1 Benzofuran and benzothiophene derivatives useful in the treatment of hyper-proliferative disorders
09/04/2003WO2003072552A1 Method for preparing benzisoxazole methane sulfonyl chloride and its amidation to form zonisamide
09/04/2003WO2003072551A1 Uracil-thioether
09/04/2003WO2003072550A1 Novel fused ring indazole compounds
09/04/2003WO2003072541A2 Chemical compounds
09/04/2003WO2003072104A1 Preparation of paroxetine involving novel intermediates
09/04/2003WO2003072103A1 Synthetic derivatives
09/04/2003WO2003062209A3 Substituted quinazolin-4-ylamine analogues as modulators of capsaicin
09/04/2003WO2003047740A3 ENANTIOSELECTIVE TRANSFORMATION OF α,β-UNSATURATED KETONES USING CHIRAL ORGANIC CATALYSTS
09/04/2003WO2003045313A3 2-aminoquinoline compounds
09/04/2003WO2003037891A8 Heteroaryl amines as glycogen synthase kinase 3beta inhibitors (gsk3 inhibitors)
09/04/2003WO2003018002A3 Cyclopropyl and cyclobutyl epothilone analogs
09/04/2003WO2002088106A3 Cysteine protease inhibitors
09/04/2003US20030166938 Preparation of paroxetine involving novel intermediates
09/04/2003US20030166931 Process for synthesis of heteroaryl-substituted urea compounds useful as antiinflammatory agents
09/04/2003US20030166930 Process for synthesis of heteroaryl-substituted urea compounds useful as antiinflammatory agents
09/04/2003US20030166697 Divalent aromatic heterocyclic compounds useful in prevention or treatment of hyperlipidemia, arteriosclerosis, diabetes mellitus, hypertension, obesity, and the like
09/04/2003US20030166690 Use of compounds for decreasing activity of hormone-sensitive
09/04/2003US20030166685 Acid derivatives of benzene useful as anticoagulants in treating and preventing cardiovascular diseases, as anti-inflammatory agents, and as metastasis inhibitors in treating cancer
09/04/2003US20030166684 3-phenyl-furan-(5H)-2-one and dihydrofuran-2-one derivatives as antibacterial agents
09/04/2003US20030166680 For treating serine protease or dual-serine protease mediated disorders
09/04/2003US20030166665 4-,5-,6-And 7-indole derivatives useful for the treatment of CNS disorders
09/04/2003US20030166664 E.g. 3-(1-(2-(5-(acetylamino)-2-methylphenyl)ethyl)piperidin--4-yl)-6-chloro-1H -indole; potent dopamine D4 ligands, dopamine antagonists; antiseratonin agents; psychoses; anxiolytic agents; antidepressants; side effects reduction
09/04/2003US20030166649 E.g., 4-(2-(1-Benzhydryl-2-(2-((benzylsulfonyl)amino)ethyl)-5-chloro-1H-indol-3 -yl)ethoxy)benzoic acid; inhibitors of phospholipase enzymes, esp. phospholipase A2; antiarthritic and -inflammatory agents; analgesics; rheumatoid diseases
09/04/2003US20030166645 Novel nitrofuran-containing heterocyclic compounds and uses thereof
09/04/2003US20030166644 Compounds and uses thereof for decreasing activity of hormone-sensitive lipase
09/04/2003US20030166638 Technical field
09/04/2003US20030166633 Pyridinylimidazoles
09/04/2003US20030166619 N2O2- functionality is bound direct to a carbon atom; treating biological disorders hypertension, restenosis, impotency, genetic disorders or infections
09/04/2003US20030166590 Microsomal triglyceride transfer protein
09/04/2003US20030165432 Versatile hydrophilic dyes
09/04/2003CA2477287A1 Uracil-thioether
09/04/2003CA2477224A1 Piperidine ouracil used as a medicament for treating bacterial infections
09/04/2003CA2476723A1 Preparation of paroxetine involving novel intermediates
09/04/2003CA2475598A1 Method for preparing benzisoxazole methane sulfonyl chloride and its amidation to form zonisamide
09/03/2003EP1341403A1 Luminescent element material and luminescent element comprising the same
09/03/2003EP1340981A2 Antibodies for detecting amphetamine derivatives
09/03/2003EP1340754A1 Substituted heterocyclic compounds, process for their preparation and pharmaceutical compositions containing them
09/03/2003EP1340753A1 Carbamate derivatives, process for producing the same and use thereof
09/03/2003EP1340500A1 Antidiabetic agents
09/03/2003EP1339723A1 Process and ester derivatives useful for preparation of cephalosporins
09/03/2003EP1339699A1 Substituted amidoalkyl uracils and the use thereof
09/03/2003EP1339695A1 Farnesyltransferase inhibitors
09/03/2003EP1339694A1 Substituted 2-phenylaminoimidazoline phenyl ketone derivatives as ip antagonists
09/03/2003EP1339693A1 Diaminopyrazole derivatives and their use for oxidation dyeing of keratinous fibres
09/03/2003EP1339692A1 Novel compounds for use as hiv protease inhibitors
09/03/2003EP1339690A1 N-type calcium channel antagonists for the treatment of pain
09/03/2003EP1339688A1 N-type calcium channel antagonists for the treatment of pain
09/03/2003EP1339687A1 4-6-diphenyl pyridine derivatives as antiinflammatory agents
09/03/2003EP1339684A1 Mch antagonists and their use in the treatment of obesity
09/03/2003EP1339683A2 Estrogen receptor modulators
09/03/2003EP1339681A1 Synthesis of fused pyrrolecarboxamides
09/03/2003EP1339678A2 Ep4 receptor selective agonists in the treatment of osteoporosis
09/03/2003EP1339677A1 Aminoalkylpyrrolidine serotonin receptor ligands and compositions, their pharmaceutical uses, and methods for their synthesis
09/03/2003EP1339406A2 Piperazine derivatives, their preparation and their use for treating central nervous system (cns) disorders
09/03/2003EP1214300B1 Rate-controlled particles
09/03/2003EP1077947B1 Novel 1,5 and 3-o-substituted 1h-indazoles with anti-asthmatic, anti-allergic, anti-inflammatory, immuno-modulating and neuro-protective effect, method for the production and use thereof as medicaments
09/03/2003EP1060178B1 Heterocyclic compounds as inhibitors of rotamase enzymes
09/03/2003EP0993454B1 Benzo(5,6)cyclohepta(1,2b)pyridine derivatives useful for inhibition of farnesyl protein transferase
09/03/2003EP0984936B1 Cyanoguanidines as cell proliferation inhibitors
09/03/2003EP0977741B1 Substituted phenyl derivatives, their preparation and use
09/03/2003EP0945445B1 1,5-benzodiazepine derivatives