Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
09/2010
09/30/2010WO2010111460A1 Inhibitors of nf-kb
09/30/2010WO2010110409A1 Process for producing pyrone and pyridone derivatives
09/30/2010WO2010110353A1 Novel amide derivative and skin whitening agent
09/30/2010WO2010110231A1 Substituted 3-hydroxy-4-pyridone derivative
09/30/2010WO2010108608A1 Substituted piperidines as par-1 antagonists
09/30/2010WO2010108584A1 Synthesis of n-substituted furan-2(5h)-ones
09/30/2010US20100249205 Metabolites of Wortmannin Analogs and Methods of Using Same
09/30/2010US20100249181 HIV Protease Inhibiting Compounds
09/30/2010US20100249176 Heterocycle amide t-type calcium channel antagonists
09/30/2010US20100249175 Dicationic compounds which selectively recognize G-quadruplex DNA
09/30/2010US20100249161 2- ( 2 -hydroxyphenyl) -quinazolin-4-ones useful for treating obesity and diabetes
09/30/2010US20100249159 Rho-kinase inhibitors
09/30/2010US20100249129 Compounds as cannabinoid receptor ligands
09/30/2010US20100249113 Modulators of atp binding cassette transporters
09/30/2010US20100249097 Novel substituted tetrahydronaphthalenes, process for the preparation thereof and the use thereof as medicaments
09/30/2010US20100249094 Compounds for the Treatment of Hepatitis C
09/30/2010US20100249092 Heteroaryl compounds and uses thereof
09/30/2010US20100249049 Arylalkylamine compound and process for preparing the same
09/30/2010US20100248264 Capture compounds, collections thereof and methods for analyzing the proteome and complex compositions
09/30/2010DE102009014484A1 Substituierte Piperidine Substituted piperidines
09/30/2010CA2756376A1 Process for the preparation of doxazosin and salts thereof
09/30/2010CA2756255A1 Substituted bicyclic hcv inhibitors
09/30/2010CA2756178A1 Compounds as cannabinoid receptor ligands
09/30/2010CA2756172A1 Inhibitors of hepatitis c virus replication
09/30/2010CA2756005A1 Substituted piperidines as par-1 antagonists
09/30/2010CA2755910A1 Inhibitors of nf-kb
09/30/2010CA2755348A1 Antiviral compounds and uses thereof
09/29/2010EP2233472A1 Heterocyclic compounds and uses thereof in the treatment of sexual disorders
09/29/2010EP2233470A1 Histamine H3 receptor antagonists
09/29/2010EP2231679A1 Synthesis of biguanidines and triazines, and biguanidino-aluminium complexes as intermediates
09/29/2010EP2231646A1 Bis-pyridylpyridones as melanin-concentrating hormone receptor 1 antagonists
09/29/2010EP2231640A1 Beta-amino acid derivatives for treatment of diabetes
09/29/2010EP2231638A1 Phthalazinone derivatives
09/29/2010EP2231620A1 Diaminopyridines for the treatment of diseases which are characterised by excessive or anomal cell proliferation
09/29/2010EP2231611A1 Novel 2-pyrrolidinyl-3-amido-6-amino-pyridine derivatives useful as potassium channel activators
09/29/2010EP2231606A2 Processes for producing cycloalkylcarboxiamido-pyridine benzoic acids
09/29/2010EP2231602A1 Gamma secretase modulators
09/29/2010EP2231600A1 Carboxamide, sulfonamide and amine compounds for metabolic disorders
09/29/2010EP2231558A1 3,4-substituted pyrrolidine beta-secretase inhibitors for the treatment of alzheimer's disease
09/29/2010EP1638957B1 N-heterocyclyl phenyl-substituted cyclic ketoenols
09/29/2010EP1628957B1 Sulfopyrroles
09/29/2010EP1615889B1 Biphenyl derivatives having beta2 adrenergic receptor agonist and muscarinic receptor antagonist activity
09/29/2010EP1534695B1 Tyrosine kinase inhibitors
09/29/2010EP1086950B1 Heterocyclic indole derivatives and mono- or diazaindole derivatives
09/29/2010CN101848898A Phthalazinone derivatives as inhibitors of PARP-1
09/29/2010CN101848897A Gamma secretase modulators
09/29/2010CN101845016A Method for synthesizing derivatives of chiral tetrahydroquinoline by catalyzing asymmetric hydrosilylation with iridium
09/29/2010CN101061110B Heterlcyclic diamide insecticides
09/29/2010CN101006082B Histamine H3 receptor agents, preparation and therapeutic uses
09/29/2010CN101006076B Modulators of ATP-binding cassette transporters
09/28/2010US7803944 Viral polymerase inhibitors
09/28/2010US7803939 N2,N4-bis(4-ethoxyphenyl)-5-fluoro-2,4-pyrimidinediamine; inhibit the IgE and/or IgG receptor signaling cascades that lead to the release of chemical mediators; Syk kinase inhibitors
09/28/2010US7803841 EP2 receptor agonists
09/28/2010US7803836 (3-{[4-amino-3-(1-cyclopentyl-pyrrolidin-3-ylamino)-benzenesulfonyl]-isobutyl-amino}-1-benzyl-2-hydroxy-propyl)-carbamic acid hexahydro-furo[2,3-b]furan-3-yl ester; active against wild-type HIV and show broad-spectrum activity against mutant HIV exhibiting resistances against known protease inhibitors
09/28/2010US7803831 3-(2-hydroxy-phenyl)-1H-pyrazole-4-carboxylic acid amide derivatives as HSP90 inhibitors for the treatment of cancer
09/28/2010US7803814 Tricyclic steroid hormone nuclear receptor modulators
09/28/2010US7803813 selective serotonin receptor agonists, such as 2-chloro-4-fluoro-N-(3-(1-methylpiperidin-4-ylamino)phenyl)benzamide fumarate, used fot the treatment or prevention of neuronal protein extravasation and/or headaches
09/28/2010US7803807 such as trans-2-[3'-oxospiro [cyclohexane- 1,1'(3'H)-isobenzofuran]-4yl]-5-(2-pyridyl) imidazo[4,5-b]pyridine, exhibiting neuropeptide Y antagonistic effects, used for the treatment of cardiovascular, nervous system, metabolic, gastrointestinal, sexual and respiratory system disorders; pharmacokinetics
09/28/2010US7803795 and nitric oxide synthase inhibitor; e.g. 1-(phenylmethyl)-4-piperidyl-6-phthalazine-3one; antiinflammatory agent; preserve the cellular energy level: survival of ischaemic tissues after insult; neurodegenerative diseases: stroke, Alzheimer's and Parkinson's diseases, atherosclerosis, osteoarthritis
09/28/2010CA2527587C Heteroaryl-substituted imidazole derivatives as glutamate receptor antagonists
09/28/2010CA2527129C Benzopyran derivatives substituted with a benzimidazole derivative, pharmaceutically acceptable salts thereof, their preparations and pharmaceutical compositions containing them
09/28/2010CA2481707C Benzopyran derivatives substituted with secondary amines having tetrazole, method for the preparation thereof and pharmaceutical compositions containing them
09/28/2010CA2395772C Sulfonamide-containing heterocyclic compounds
09/28/2010CA2387016C Acrylamide derivatives as fab i inhibitors
09/28/2010CA2383524C Thiazolyl alkynyl compounds and methods of use thereof
09/28/2010CA2383257C Substituted (aminoiminomethyl or aminomethyl) dihydrobenzofurans and benozopyrans
09/28/2010CA2308201C Use of anti-fungal agents for the treatment of fungus-induced mucositis
09/23/2010WO2010107115A1 Glycine transporter inhibitor
09/23/2010WO2010106097A1 Substituted pyrimidines for the treatment of cancer
09/23/2010WO2010105779A1 Novel method for producing enaminocarbonyl compounds
09/23/2010WO2010105772A1 Novel method for producing enaminocarbonyl compounds
09/23/2010WO2009065897A3 Inhibitors of malt1 proteolytic activity and uses thereof
09/23/2010US20100240725 Novel 1,3-dihydro-5-isobenzofurancarbonitrile derivatives and pharmaceutical composition thereof for the treatment of premature ejaculation
09/23/2010US20100240707 1,3,5-trisubstituted triazole derivative
09/23/2010US20100240706 1,3-disubstituted-4-phenyl-1h-pyridin-2-ones
09/23/2010US20100240705 Substituted enaminocarbonyl compounds used as insecticides
09/23/2010US20100240679 4-Phenylpiperidine Derivatives as Renin Inhibitors
09/23/2010US20100240670 4-[(arylmethyl)aminomethyl]piperidine derivatives, their preparation and their therapeutic application
09/23/2010US20100240653 Biphenyl sulfonyl and phenyl-heteroaryl sulfonyl modulators of the histamine h3-receptor useful for the treatment of disorders related thereto
09/23/2010US20100240650 Substituted pyrrolines as kinase inhibitors
09/23/2010US20100240639 Sulfonyl-Derivatives as Novel or Histone Deacetylase
09/23/2010US20100239496 Imaging agents for detecting neurological disorders
09/23/2010CA2755759A1 Substituted pyrimidines for the treatment of cancer
09/22/2010EP2230237A1 New method for producing enaminocarbonyl compounds
09/22/2010EP2230236A1 New method for producing enaminocarbonyl compounds
09/22/2010EP2229376A1 Indole-substituted 3-cyanopyridines as kinase inhibitors
09/22/2010EP2229356A1 1,2-disubstituted-4-benzylamino-pyrrolidine derivatives as cetp inhibitors useful for the treatment of diseases such as hyperli pidemia or arteriosclerosis
09/22/2010EP1836163B1 Pyrrolidine derivatives for the treatment of a disease depending on the activity of renin
09/22/2010EP1692114B1 Novel benzimidazole and imidazopyridine derivatives and use thereof as a medicament
09/22/2010EP1618092B1 Aryl-substituted pyrazole-amide compounds useful as kinase inhibitors
09/22/2010EP1599464B1 Novel cyclic urea derivatives, preparation method thereof and pharmaceutical use of same as kinase inhibitors
09/22/2010CN1976705B 1,1,1- trifluoro-4-phenyl-4-methyl-2-(1H-pyrrolo not 2,3-C|pyridin-2-ylmethyl)pentan-2-ol derivatives and related compounds as glucocorticoid ligands for the treatment of inflammatory diseases and dia
09/22/2010CN1788001B 2, 4- di (phenylamino) pyrimidines useful in the treatment of neoplastic diseases, inflammatory and immune system disorders
09/22/2010CN101842369A 2,3-dihydrobenzo(1,4) dioxin-2-ylmethyl derivatives as alpha2C antagonists for use in the treatment of peripheric and central nervous system diseases
09/22/2010CN101842360A Anti-infective pyrimidines and uses thereof
09/22/2010CN101838271A Bicyclic [3.1.0] derivatives as glycine transporter inhibitors
09/22/2010CN101838239A Pyrazole compound as well as composition and application thereof
09/22/2010CN101837127A Medical use of inhibitors of glutaminyl and glutamate cyclases
09/21/2010US7799922 adenosine A3 receptor antagonists; improved bioavailability; treatment of diseases such as asthma, COPD and ARDS, glaucoma, tumor, allergic and inflammatory diseases, ischemia, hypoxia, arrythmia and renal diseases; e.g. 4-Methoxy-N-[6-(morpholin-4-yl)-4-benzylamino-3-cyanoquinolin-2-yl]-benzamide
09/21/2010US7799916 reacting 5-bromobenzofuran-2-carboxamide with 3-(4-piperazin-1-ylbutyl)indole-5-carbonitrile by transition-metal-catalysed coupling by means of a Pd complex (tris(dibenzylideneacetone)-dipalladium to form 5-(4-[4-(5-cyano-3-indolyl)butyl]-1-piperazinyl)benzofuran-2-carboxamide; reductive amination