Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397) |
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01/04/2011 | CA2306093C Heteroaryl diazacycloalkanes as cholinergic ligands at nicotinic acetylcholine receptors |
12/30/2010 | US20100331545 Regulator for signaling toll-like receptor, which comprises cathepsin inhibitor as active ingredient |
12/30/2010 | US20100331380 Compounds, Compositions, and Methods for the Treatment of Beta-Amyloid Diseases and Synucleinopathies |
12/30/2010 | US20100331370 Novel isobenzofuran analogs of sclerophytin A |
12/30/2010 | US20100331367 N-aryl-n-piperidin-4-yl-propionamide derivatives and their use as opioid receptor ligands |
12/30/2010 | US20100331346 Beta-amino acid derivatives for treatment of diabetes |
12/30/2010 | US20100331342 Immuno Inhibitory Pyrazolone Compounds |
12/30/2010 | US20100331341 2-carboxamide-7-piperazinyl-benzofuran derivatives 774 |
12/30/2010 | US20100331335 Inhibitors of Jun N-Terminal Kinase |
12/30/2010 | US20100331329 Benzamide derivatives useful as histone deacetylase inhibitors |
12/30/2010 | US20100331317 Benzodiazepine compound and pharmaceutical composition |
12/30/2010 | US20100331315 Rhodanines and related heterocycles as kinase inhibitors |
12/30/2010 | US20100331308 Oxazolidinone derivatives |
12/30/2010 | US20100331307 Therapeutic compounds and compositions |
12/30/2010 | US20100331303 Prolyl hydroxylase inhibitors and methods of use |
12/30/2010 | US20100331298 Carboxamide Compounds and Their Use |
12/30/2010 | US20100330685 Diaminorhodamine derivative |
12/30/2010 | US20100330030 Vasculostatic Agents and Methods of Use Thereof |
12/29/2010 | WO2010150192A1 Heterocyclic sulfonamides, uses and pharmaceutical compositions thereof |
12/29/2010 | WO2010149326A1 Acid-labile trigger units |
12/29/2010 | WO2010129848A3 2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamides |
12/29/2010 | EP2266986A1 Cytotoxins, Prodrugs, Linkers and Stabilizers useful therefor |
12/29/2010 | EP2266983A1 Nitrogenated 5-membered heterocyclic compound |
12/29/2010 | EP2266978A1 Novel physiologically active substances |
12/29/2010 | EP2266977A1 2,4-di[(hetero)arylamino]-pyrimidine derivatives as zap-70 and/or syk inhibitors |
12/29/2010 | EP2266976A1 Fused ring thrombin receptor antagonists |
12/29/2010 | EP2266975A1 1-(2-alkyl-2,3-dihydro-benzofuran-4-yl)-pyrrolidin-3-ylamine acyl compounds |
12/29/2010 | EP2266973A1 Pyrazinylpyrazole |
12/29/2010 | EP2266970A1 Substituted aromatic heterocyclic compounds as fungicides |
12/29/2010 | EP2266965A1 Methods for Isolating Crystalline Form I of 5-Azacytidine |
12/29/2010 | EP2266964A1 Acid-labile trigger units |
12/29/2010 | EP2266958A1 Antiviral agent |
12/29/2010 | EP2265592A1 Substituted pyraz inylmethyl sulfonamides for use as. fungicides |
12/29/2010 | EP2265587A1 Modulators of the histamine h3 receptor useful for the treatment of disorders related thereto |
12/29/2010 | EP2265585A1 Amine and ether compounds which modulate the cb2 receptor |
12/29/2010 | EP2265335A1 Indazole derivatives |
12/29/2010 | EP2265273A1 Hexahydrocyclopentyl[f] indazole sulfonamides and derivatives thereof as selective glucocorticoid receptor modulators |
12/29/2010 | EP2265271A1 Crystalline 2-(4-cyclopropanesulphonyl-phenyl)-n-pyrazin-2-yl-3-(tetrahydropyran-4-yl)-propionamide |
12/29/2010 | EP2265270A1 2-aminopyridine kinase inhibitors |
12/29/2010 | EP2185512B1 Trans-3-aza-bicyclo[3.1.0]hexane derivatives |
12/29/2010 | EP2010514B1 3-(pyridin-2-yl)-[1,2,4]-triazines for use as fungicides |
12/29/2010 | EP1940826B1 Pyrimidinyl amide compounds which inhibit leukocyte adhesion mediated by vla-4 |
12/29/2010 | EP1861377B1 Benzimidazolone derivatives as cb2 receptor ligands |
12/29/2010 | EP1791830B1 Diaminotriazole compounds useful as protein kinase inhibitors |
12/29/2010 | EP1001946B1 QUINOXALINE COMPOUNDS WHICH INHIBIT PLATELET-DERIVED GROWTH FACTOR AND/OR p56lck TYROSINE KINASES |
12/29/2010 | CN1926132B Pyrazole compounds useful as protein kinase inhibitors |
12/29/2010 | CN1922139B Bicyclic amide derivatives |
12/29/2010 | CN101928284A Nitrogen-containing heterocyclic derivatives and drugs containing the same as the active ingredient |
12/29/2010 | CN101928282A Preparing method of pyridine compound |
12/29/2010 | CN101928281A Bicyclo-substituted pyrazolone azo derivative, preparation method thereof and application thereof in medicaments |
12/29/2010 | CN101928280A Pepperphentonamine derivative containing naphthalene rings |
12/29/2010 | CN101928279A 3-amino-2-pyrones cyclooxygenase inhibitors as well as preparation method and application thereof |
12/29/2010 | CN101928274A Peperphentonamine derivative |
12/29/2010 | CN101928244A Structural analogue and derivative of isochromanone-4 compound with cardiovascular activity, preparation method and application thereof |
12/29/2010 | CN101928243A Acenaphtho heterocyclic compounds, and cyclodextrin inclusion compounds or conjugates thereof and application thereof in preparing Bcl-2 family protein inhibitors |
12/29/2010 | CN101445504B Dioxane-2-alkyl carbamates derivatives |
12/29/2010 | CN101391994B Synthetic method of itraconazole key intermediate triazole compounds |
12/29/2010 | CN101200465B Decahydronaphthalene compounds and medical uses thereof |
12/29/2010 | CN101142193B Propane-1,3-dion derivative or salt thereof |
12/29/2010 | CA2766320A1 Acid-labile trigger units |
12/29/2010 | CA2766104A1 Heterocyclic sulfonamides, uses and pharmaceutical compositions thereof |
12/28/2010 | USRE42015 N4-acylcytosine-1,3-dioxolane nucleosides for treatment of viral infections |
12/28/2010 | US7858794 such as 5-Chloro-thiophene-2-carboxylic acid (1-acetyl-7-dimethylamino-4-methyl-4-phenyl-1,2,3,4-tetrahydro-quinolin-6-yl)-amide, having follicle stimulating hormone modulatory activity, used to regulate fertility as contraceptives and for treatment of breast cancer, prostate cancer and endometriosis |
12/28/2010 | US7858792 Biphenyl-2-ylcarbamic Acid 1-(2-{5-[2-(4-Hydroxyphenyl)ethylamino]pentylcarbamoyl}ethyl)piperidin-4-yl Ester, used for the treatment of respiratory system disorders such as chronic obstructive pulmonary disease and asthma |
12/28/2010 | US7858789 Affinity for somatostatin receptors; used for the treatment of acromegalia, hypophyseal adenomas or endocrine gastroenteropancreatic tumors including carcinoid syndrome; 4-(urea or thiourea substituted)-1-alkylpiperidines |
12/28/2010 | US7858781 inflammatory conditions, allergies, autoimmune diseases, chronic pain, graft rejection, cancers which involve leukocyte filtration, stenosis or restenosis, atherosclerosis, rheumatoid arthritis, osteoarthritis; e.g. 4-Isobutoxy-1H-indole-2-carboxylic acid [4-(2-azepan-1-yl-ethyl)-phenyl]-amide |
12/28/2010 | US7858776 (2,3-cis)-3-amino-2-phenyl-2,3-dihydro-1,5-benzoxazepin-4(5H)-one; for treatment of neurological disorders related to amyloid beta protein production such as Alzheimer's disease; inhibit gamma secretase and thereby inhibit the production of amyloid beta protein |
12/28/2010 | US7858657 treating lung cancer with PI-3 kinase inhibitor acetic acid 4-diallylaminomethylene-6-hydroxy-1- alpha -methoxymeth-yl-10 beta ,13 beta -dimethyl-3,7,17-trioxo-1,3,4,7,10,11 beta ,12,13,14 alpha ,15,16,17-dodecahydro-2-oxa-cyclopenta [ alpha ]phenanthren-11-yl ester |
12/28/2010 | US7858644 administering prostaglandin receptor antagonists such as N-[4-(4'-Methoxy-biphenyl-4-yloxymethyl)-5-methyl-furan-2-carbonyl]-benzenesulfonamide, used analgesics, neuroprtectants and diuretics, or for the treament of diabetes, tinitus, cancer, bone, blood, sleep, cardiovascular and sexual disorders |
12/28/2010 | US7858642 Substituted hydroxyethylamine aspartyl protease inhibitors |
12/28/2010 | US7858633 Cycloalkyl substituted pyrimidinediamine compounds and their uses |
12/28/2010 | US7858632 Purinergic receptor antagonists; genitourinary and pain-related diseases; for example, 5-(2-isopropyl-4,5-dimethoxybenzyl)-pyrimidine-2,4-diamine |
12/28/2010 | US7858629 3-{(3S)-4-{[1-(3-ethoxyphenyl)-2-(4-methylphenyl)-1H-imidazol-4-yl]carbonyl}-3 -[(isopropylamino)carbonyl]-1-piperazinyl}-1-naphthoic acid, useful for the treatment, control, or prevention of obesity and diabetes |
12/28/2010 | US7858624 such as methyl 2-((R)-((R)-1-((2S,3S)-5-(butylamino)-1-cyclohexyl-3-hydroxy-5-oxopentan-2-ylcarbamoyl)piperidin-3-yl)(3-chlorophenyl)methoxy)ethylcarbamate, used as hypotensive agents or for the treatment of cardiovascular disorders, vision defects, aldosteronism and obesity |
12/23/2010 | WO2010148209A2 Preparation of montelukast |
12/23/2010 | WO2010147922A1 Deuterated i soindoline- i, 3-dione derivatives as pde4 and tnf-alpha inhibitors |
12/23/2010 | WO2010147898A2 Small molecule inhibitors of spleen tyrosine kinase (syk) |
12/23/2010 | WO2010147791A1 Azetidine 2 -carboxamide derivatives which modulate the cb2 receptor |
12/23/2010 | WO2010147430A2 Novel c-aryl glucoside sglt2 inhibitors and pharmaceutical composition comprising same |
12/23/2010 | WO2010147375A2 Method for screening for substance which inhibits interaction between beta amyloid peptide and vegf and inhibitor searched by same |
12/23/2010 | WO2010146488A1 Bicyclic and tricyclic compounds as kat ii inhibitors |
12/23/2010 | WO2010146299A1 Azetidine-derived esters, preparation thereof, and therapeutic use thereof as cannabinoid receptor modulators |
12/23/2010 | WO2010146173A1 Quinazoline derivatives as histamine h4-recept0r inhibitors for use in the treatment of inflammatory disorders |
12/23/2010 | WO2010146116A1 Triazole compounds carrying a sulfur substituent |
12/23/2010 | WO2010146115A1 Triazole compounds carrying a sulfur substituent |
12/23/2010 | WO2010146114A1 Triazole compounds carrying a sulfur substituent |
12/23/2010 | WO2010145989A1 1-(2-alkyl-2,3-dihydro-benzofuran-4-yl)-pyrrolidin-3-ylamine acyl compounds |
12/23/2010 | WO2010145764A1 Substituted enamino carbonyl compounds |
12/23/2010 | WO2010144959A1 Analogues of anti-fibrotic agents |
12/23/2010 | WO2010128528A3 Piperidine derivatives useful for treatment of diebetes |
12/23/2010 | WO2010072770A3 Griseofulvin analogues for the treatment of cancer by inhibition of centrosomal clustering |
12/23/2010 | WO2009146555A8 Hiv integrase inhibitors from pyridoxine |
12/23/2010 | US20100324296 Dichroic-photochromic compounds and devices |
12/23/2010 | US20100324266 Photocleavable Protecting Groups |
12/23/2010 | US20100324128 9, 10-Alpha, Alpha-OH-Taxane Analogs and Methods for Production Thereof |
12/23/2010 | US20100324094 Conformationally Restrained Epothilone Analogues as Anti-Leukemic Agents |
12/23/2010 | US20100324093 Ccr9 inhibitors and methods of use thereof |
12/23/2010 | US20100324053 Trisubstituted 1,2,4 triazoles |
12/23/2010 | US20100324043 Bicyclic And Tricyclic Compounds As KAT II Inhibitors |
12/23/2010 | US20100324030 5-Quinoline derivatives having an anti-bacterial activity |