Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
01/1993
01/13/1993EP0522887A1 Imidazoles as ACAT- and thromboxane TxA2 inhibitors
01/13/1993EP0522038A1 Substituted pyrimidines, pyrimidinones and pyridopyrimidines
01/13/1993CN1067887A Derivative of 2-aminapyrimidine-4-carboxamide, its preparation and application in therapy
01/13/1993CN1067885A Derivative of 2-aminopyrimidine-4-carboxamide, its preparation and application in therapy
01/13/1993CN1067884A Derives of pyrimidine-4-carboxamide, their preparation and their application in therapeutics
01/12/1993US5179204 N-substituted-4-pyrimidinamines and pyrimidinediamines
01/12/1993US5179112 Heterocyclic amide derivatives and pharmaceutical use
01/12/1993US5179098 Fungicides
01/12/1993US5179096 Therapeutic application of flouroquinolone derivatives
01/07/1993WO1993000341A1 4-(1-h-pyrrol-1-yl)imidazoles with angiotensin ii antagonist activity
01/07/1993WO1993000333A1 Tryptamine analogues, their synthesis and their use as 5-ht1-like or 5-ht2 receptor agonists
01/07/1993WO1993000330A2 Azanorbornane derivatives
01/07/1993WO1993000086A1 Use of tetrahydrocarbazone derivatives as 5ht1 receptor agonists
01/07/1993WO1993000075A1 Methods and compositions for treating emesis, nausea and other disorders using optically pure s(-) ondansetron
01/07/1993WO1992020649A3 Substituted 2-carboxyindoles having pharmaceutical activity
01/07/1993EP0521463A2 Substituted cyclic cycloalkyltriols, process, intermediates for their preparation and their use as antiviral and antiparasitic agents
01/07/1993CA2112488A1 Method and compositions for treating emesis, nausea and other disorders using optically pure s(-) ondansetron
01/07/1993CA2111335A1 Azanorbornane derivatives
01/07/1993CA2110574A1 Tryptamine analogues, their synthesis and their use as 5-ht1-like or 5-ht2 receptor agonists
01/06/1993CN1067654A Processes for diastereoselective synthesis of nucleosides
01/06/1993CN1067651A Pyrimidne or triazine derivative, process for preparing the same and herbicide using the same
01/05/1993US5177223 Indoleacetic acid derivatives, process for their preparation, and medicines containing same as active ingredients
01/05/1993US5177096 Angiotensin II receptor antagonist
01/05/1993US5177095 Hypotensive agents
01/05/1993US5177079 Antiallergen, antiulcer
01/05/1993CA2073111A1 Cycloalkyltriols containing cyclic substituents, processes and intermediate products for their preparation and their use as antiviral and antiparasitic agents
01/05/1993CA2072911A1 Use of benzimidazoline-2-oxo-1-carboxylic acid derivatives
01/05/1993CA1312330C Heterocyclic compounds, a process for their preparation and their use in medicine
12/1992
12/30/1992EP0520883A1 2-Aminopyrimidin-4-carboxamide derivatives, their preparation and their use in therapy
12/30/1992EP0520882A1 2-Aminopyrimidin-4-carboxamide derivatives, their preparation and their application in therapy
12/30/1992EP0520724A1 Angiotensin II antagonists
12/30/1992EP0520423A2 Heterocyclic compounds, their production and use as angiotensin II antagonists
12/30/1992EP0520292A1 Chiral azetidinone derivatives and their use as dopants in liquid crystalline mixtures
12/30/1992EP0519996A1 Imidazoles
12/30/1992CN1067426A 3,4,n-trisubstituted-4,5-dihydro-1h-pyrazole-1-carboxamides and their use as insecticides
12/29/1992US5175293 Pesticides
12/29/1992US5175224 Forming reinforced polyimides
12/29/1992US5175182 Antitumor agent; distamycin A derivatives
12/29/1992US5175180 N-substituted n-(alpha-triazolyl-toluyl)pyrrole compounds and use for treatment of circulatory disorders
12/29/1992US5175176 1-[pyri(mi)dyl-(2)]-hydroxy-pyrazole microbicides
12/29/1992US5175164 Angiotensin ii antagonists incorporating a substituted indole or dihydroindole
12/29/1992US5175163 Tranquilizer, antidepresant, antispasmodic, analgesic and antiinflammatory agent
12/29/1992US5175158 Condensed diazepinones, processes for preparing them and pharmaceutical compositions containing these compounds
12/29/1992US5175157 Cardiovascular disorders
12/29/1992CA1312083C Hydantoin derivatives
12/29/1992CA1312081C Process for the manufacture of substituted pyrrolidinones
12/29/1992CA1312080C Arylpiperazinyl-ethyl(or butyl)-phenyl-heterocyclic compounds
12/29/1992CA1312078C Indolylpropanols, processes for their preparation and their use, and preparations containing the compounds
12/28/1992WO1993000334A1 Indole derivatives, pharmaceutical compositions and methods of treating neurological and psychiatric disorders
12/28/1992CA2090240A1 Indole derivatives, pharmaceutical compositions and methods of treating neurological and psychiatric disorders
12/28/1992CA2072528A1 4-pyrimidinecarboxamide derivatives, their preparation and their application in therapy
12/28/1992CA2072433A1 2-aminopyrimidine-4-carboxamide derivatives, their preparation and their use in therapeutics
12/26/1992CA2071086A1 Heterocyclic compounds
12/25/1992CA2072282A1 Polyfluoroalkylthiopoly(ethylimidazolium) compounds, process for their preparation, and their use as biocides
12/23/1992WO1992022583A2 Tri- and tetra-valent monospecific antigen-binding proteins
12/23/1992WO1992022294A1 Immunomodulatory azaspiranes
12/23/1992EP0519831A1 N-Substituted heterocyclic derivatives, their preparation, and pharmaceutical compositions containing them
12/23/1992EP0519464A1 Nucleoside derivatives and production thereof
12/23/1992EP0519211A1 Substituted 4-aminopyrimidine, process for their preparation and their use as parasiticide
12/23/1992CN1067245A Processes for diastereoselective synthesis of nucleosides
12/23/1992CN1067244A Pyrrolidones
12/23/1992CN1019574B Process for preparing pyrimidine derivatives with insect-and mite-killing activity
12/23/1992CA2110577A1 Immunomodulatory azaspiranes
12/22/1992US5173512 An aqueous oil-in-water emulsion of perfluoro-N-cyclohexylmorpholine or a mixture with perfluoro-N-hexylmorpholine; synthetic blood
12/22/1992US5173503 Derivatives of N,N-dimethyl-4-phenylalkylenesulfonyl-imidazole -1-sulphonamides; phytopathogenic fungi
12/22/1992US5173496 Antiinflammatory agents
12/22/1992US5173489 α,α-disubstituted aromatics and heteroaromatics as cognition enhancers
12/22/1992CA1311760C Pyrazoline derivatives and agents for treating cerebrovascular diseases containing the same as active ingredient
12/22/1992CA1311755C 4-(aroylamino)piperidinebutanamide derivatives
12/17/1992DE4117121A1 New 1-(1,4-bi:phenyl-methyl) benzimidazole(s) as angiotensin II antagonists
12/16/1992EP0518676A2 Cyclic renin inhibitors
12/16/1992EP0518672A2 Cyclic renin inhibitors
12/16/1992EP0518033A1 Fused heterocyclic compounds, their production and use
12/16/1992EP0517812A1 Angiotensin ii antagonists incorporating a substituted benzyl element
12/16/1992CN1067053A Pyrazine derivatives and process for preparing same
12/16/1992CN1067052A Substituted diaminophthalimides and analogues
12/15/1992US5171748 For hypertension, cardiovascular disorders
12/15/1992US5171746 Thiazole and imidazole derivatives and antiulcer composition containing same
12/15/1992US5171744 3-Quinuclidinyl propanoates
12/15/1992CA2071181A1 Benzodiazepine analogs
12/12/1992CA2070983A1 Cyclic renin inhibitors
12/12/1992CA2070972A1 Cyclic renin inhibitors
12/10/1992WO1992021339A1 Isoxazole and isothiazole compounds that enhance cognitive function
12/09/1992EP0517658A1 Stabilisation of polymeric organic materials by using synergistic mixtures comprising sterically hindered cyclic amines and derivatives of 3-pyrazolidinone or 1,2,4-triazolidine-3,5-dione
12/09/1992EP0517357A1 Angiotensin II antagonists incorporating a substituted indole or dihydroindole
12/09/1992EP0517325A2 Drug hapten analogues for immunoassays
12/09/1992EP0517052A1 Substituted imidazolinyl-pyrimidines
12/09/1992CN1066847A Angiotensin ii receptor blocking 2,3,6 substituted quinazolinones
12/09/1992CN1066844A Azole derivate, manufacturing method and application thereof
12/08/1992US5169945 Reacting imide with secondary amine to form amide which protects amine during nucleophilic reactions
12/08/1992CA2070717A1 Substituted imidazolinylpyrimidines
12/08/1992CA2062239A1 Hydantoin derivatives for competitive enzyme immunoassays
12/08/1992CA2062101A1 Hydantoin derivatives for competitive enzyme immunoassays
12/08/1992CA1311242C Pesticidal method using n-phenylpyrazoles
12/06/1992CA2065078A1 Angiotensin ii antagonists incorporating a substituted indole or dihydroindole
12/05/1992CA2070193A1 Stabilisation of polymeric organic materials by using synergistic mixutres comprising sterically hindered cyclic amines and derivatives of 3-pyrazolidinone or 1,2,4-triazolidine-3,5-dione
12/02/1992EP0516588A1 Substituted diaminophtalimides and analogues
12/02/1992EP0516486A2 Azetidinone derivatives useful in the preparation of carbapenem antibiotics
12/02/1992EP0515893A1 Substituted 4-heteroarylpyrazolines
12/02/1992EP0515548A1 Imidazole angiotensin ii antagonists incorporating a substituted benzyl element