Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
04/1993
04/07/1993EP0535034A1 Pharmaceutically active benzoquinazoline compounds
04/07/1993CN1070646A Imidazo-fused iso-and heterocycles, process for their preparation, compositions containing them and their use
04/07/1993CN1070641A Herbicidal quinoxalinyloxy ethers
04/06/1993US5200412 Antiinflammatory agents and antiallergens
04/06/1993CA1315790C Method of improving sleep
04/05/1993CA2079735A1 Acylals of imidazole-5-carboxylic acid derivatives, process for their preparation and their use
04/02/1993CA2079281A1 Imidazolyl-propenoic acid derivatives
04/02/1993CA2079268A1 Substituted imidazolyl-propenoic acid derivatives
04/02/1993CA2079266A1 Cyclic-substituted imidazolyl-propenoic acid derivatives
04/01/1993WO1993006092A1 Piperazinyl (sulfonyl)amide derivatives of camphor as oxytocin antagonists
04/01/1993WO1992022583A3 Tri- and tetra-valent monospecific antigen-binding proteins
03/1993
03/31/1993EP0534706A1 Quinazolinones and pyridopyrimidinones useful as angiotensin II antagonists
03/31/1993EP0534443A1 3,6-Disubstituted pyridazine derivatives
03/31/1993EP0534344A1 Substituted 3-amino-2,3,4,5-tetrahydro-1-aryloxy-3-benzazepines, a process for their preparation and their use as modulators of neurotransmitter function
03/31/1993EP0534266A1 Sulfonylaminocarbonyltriazolones with two through oxygen bonded substituents
03/31/1993CN1070399A Substituted amide derivatives of piperizinylcamphorsulfonyl oxytocin antagonists
03/30/1993US5198545 Pharmaceutical epinephrine-pilocarpine compounds and process of preparation thereof
03/30/1993US5198442 (2-imidazolin-2-ylamino) quinoxaline derivatives and methods for using same
03/28/1993CA2079185A1 Dicyclic nitrogens derivatives, preparation process thereof and pharmaceutical compositions containing them
03/27/1993CA2078699A1 3,6-disubstituted pyridazine derivatives
03/26/1993CA2079079A1 Quinazolinones and pyridopyrimidinones
03/24/1993WO1993006079A1 PREPARATION OF SUBSTITUTED ISOSERINE ESTERS USING METAL ALKOXIDES AND β-LACTAMS
03/24/1993EP0533268A1 Benzanilide derivatives as 5-HT1D antagonists
03/24/1993EP0533242A2 Substituted derivatives of piperazinylcamphorsulfonyl oxytocin antagonists
03/24/1993EP0533241A2 Substituted alkyl derivatives of piperazinylcamphorsulfonyl oxytocin antagonists
03/24/1993EP0533240A2 Substituted amine derivatives of piperazinylcamphorsulfonyl oxytocin antagonists
03/24/1993EP0533213A1 Use of azelastin and glycerine ethers for the treatment of psoriasis
03/24/1993EP0533058A1 Imidazo-fused iso- and heterocycles as angiotensin II antagonists
03/24/1993EP0532948A1 Substituted cycloalkenes as herbicides
03/24/1993EP0532918A1 Substituted pyrazolines as pesticides
03/23/1993US5196465 Polymeric thermoplastic materials, comprising 1,2,4-triazolidine-3,5-dione derivatives as stabilizers
03/23/1993US5196444 Angiotensin/II/ antagonists; hypotensive agents
03/23/1993US5196431 2-substituted amino-4, 6-di-tertiary-buthyl-5-hydroxy-1, 3-pyrimidines as antiinflammatory agents
03/23/1993US5196427 Gastrointestinal and central nervous system disorders; hormone inhibitors
03/23/1993CA1314881C Anti-anxiety agents
03/23/1993CA1314879C Anellated indole derivatives
03/19/1993CA2078505A1 Benzanilide derivatives
03/18/1993WO1993005039A1 5-hydroxy-2-pyrimidinylmethylene derivatives useful as antiinflammatory agents
03/18/1993WO1993005036A1 N-substituted carbazole derivative
03/18/1993WO1993005027A1 Triazolylated tertiary amine compound or salt thereof
03/18/1993WO1993005026A1 Peptide isoters containing a heterocycle as h.i.v. inhibitors
03/18/1993WO1993005025A1 C-linked pyrazole derivatives
03/18/1993WO1993005020A1 Indoles as inhibitors of hiv reverse transcriptase
03/18/1993WO1993005014A1 Aromatic sulfonamide derivatives, their use as enzyme inhibitors and pharmaceutical compositions containing them
03/18/1993WO1993004682A1 Novel 4-arylpiperazines and 4-arylpiperidines
03/18/1993DE4130461A1 New 3-amino-5-substd. carboxamide chloro-pyrazine carbamide cpds.
03/18/1993CA2095847A1 Novel 4-arylpiperazines and 4-arylpiperidines
03/17/1993EP0532410A1 N-substituted heterocyclic derivatives as angiotensin II inhibitors
03/17/1993EP0532097A1 Piperazinyl(sulfon)amide derivatives of camphor as oxytocin antagonists
03/17/1993EP0532054A1 Process for preparing alpha,alpha-disubstituted aromatics and heteroaromatics as cognition enhancers
03/17/1993EP0531883A1 Condensed 5-membered ring heterocycles, process for their preparation and medicaments containing them
03/17/1993EP0531382A1 N-substituted-1,2,4-triazolone compounds for treatment of cardiovascular disorders
03/17/1993CN1069974A Triazolyl-substituted tertiary amino compounds and their salts
03/17/1993CN1069971A Novel sulfonamide fibrinogen receptor antagonists
03/17/1993CN1069882A Compounds and methods for inhibition of HIV and related viruses
03/17/1993CN1020101C Process for preparation of tricycle kentones
03/17/1993CA2078264A1 Substituted derivatives of piperizinylcamphorsulfonyl oxytocin antagonists
03/17/1993CA2078263A1 Substituted alkyl derivatives of piperizinylcamphorsulfonyl oxytocin antagonists
03/17/1993CA2078025A1 Substituted amine derivatives of piperizinylcamphorsulfonyl oxytocin antagonists
03/16/1993US5194622 Chemical condensation of an aldehyde of an azole and a phosphonium derivative
03/16/1993US5194605 Cyclic renin inhibitors containing 2-substituted (3S,4S)-4-amino-5-cyclohexyl-3-hydroxy pentanoic acid, 2-substituted (3S,4S)-5-cyclohexyl-3,4-di-hydroxy pentanoic acid or 2-substituted (4S,5S)-5-amino-6-cyclohexyl-4-hydroxyhexanoic acid or its analogs
03/16/1993US5194436 For trating psychosis
03/16/1993US5194369 Silver halide color photographic material
03/16/1993CA1314551C Poly-4-aminopyrrole-2-carboxamido derivatives and their use as site specific alkylating agents
03/15/1993CA2078058A1 Imidazo-fused iso- and heterocycles, process for their preparation, compositions containing them and their use
03/14/1993CA2077922A1 Substituted amide derivatives of piperizinylcamphorsulfonyl oxytocin antagonists
03/12/1993WO1993004684A1 Novel 4-arylpiperazines and 4-arylpiperidines
03/12/1993CA2095826A1 4-arylpiperazines and 4-arylpiperidines
03/11/1993CA2077967A1 N-substituted heterocyclic derivatives, their preparation and the pharmaceutical compositions in which they are present
03/10/1993EP0530907A1 Indoles as inhibitors of HIV reverse transcriptase
03/10/1993EP0530616A1 Pyrazolylsulfonylguanidino pyrimidines as herbicides
03/10/1993EP0530264A1 Arthropodicidal tetrahydropyridazines.
03/10/1993CN1069730A 2-Piperazinone compounds their production and use
03/10/1993CN1069729A Dihydropyridazinones, pyridazinones and related compounds as fungicides
03/10/1993CN1069726A Medicaments
03/10/1993CA2077620A1 Substituted cycloalkenes
03/09/1993US5192795 Cognition activators
03/09/1993US5192773 Immunosuppressive compounds
03/09/1993US5192647 Forming latent images
03/07/1993CA2077577A1 Condensed 5-membered heterocyclic compounds, processes for preparing them and pharmaceutical preparations containing these compounds
03/07/1993CA2077283A1 Inhibitors of hiv reverse transcriptase
03/04/1993WO1993004065A1 NEW 3-(SUBSTITUTED TETRAZOLYL)-4-OXO-4H-PYRIDO-[1,2-a]PYRIMIDINES, SALTS THEREOF, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESS FOR PREPARING SAME
03/04/1993WO1993004059A1 4-acylaminoimidazole derivative
03/04/1993WO1993004052A1 Amide tetrazole acat inhibitors
03/04/1993WO1993004048A1 New pyrazine derivatives, their preparation and their use
03/04/1993WO1993004046A1 Angiotensin ii receptor blocking imidazolinone derivatives
03/04/1993WO1993004045A1 Angiotensin ii receptor blocking imidazolinone derivatives
03/04/1993WO1993004041A1 Synthetic heteroaryl polyamines as excitatory amino acid neurotransmitter antagonists
03/04/1993WO1993000330A3 Azanorbornane derivatives
03/04/1993WO1992018089A3 Use of steroidal and non-steroidal amines to sensitize multidrug-resistant cells
03/04/1993CA2115990A1 Angiotensin ii receptor blocking imidazolinone derivatives
03/04/1993CA2115989A1 Angiotensin ii receptor blocking imidazolinone derivatives
03/04/1993CA2115755A1 New pyrazine derivatives, their preparation and their use
03/04/1993CA2114935A1 Synthetic heteroaryl polyamines as excitatory amino acid neurotransmitter antagonists
03/04/1993CA2114145A1 New 3-/substituted tetrazolyl/-4-oxo-4h-pyrido-/1,2-a/- pyrimidines, salts thereof, pharmaceutical compositions containing them and process for preparing same
03/03/1993EP0530149A1 Parasiticide
03/03/1993EP0529858A1 2-Piperazinone compounds, their production and use
03/03/1993EP0529451A1 Substituted pyrazolines as pesticides
03/03/1993EP0529292A2 Substituted aralkylsulfonyl-aminoguanidinoazines as herbizides
03/03/1993EP0529253A1 Phenylalkylderivatives, compounds containing them and process for their fabrication