Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
01/2002
01/24/2002US20020010343 Compounds having IgE affecting properties
01/24/2002US20020010204 Use as pesticides.
01/24/2002US20020010203 Methods of modulating c-kit tyrosine protein kinase function with indolinone compounds
01/24/2002US20020010184 Inhibitors of prenyl-protein transferase
01/24/2002US20020010182 Treatment of respiratory diseases such as asthma, bronchitis, rhinitis, cough, expectoration, ophthalmic diseases such as conjunctivitis, dermatitis
01/24/2002US20020010179 Ultraviolet light screening agents; cosmetics
01/24/2002US20020010177 For treating eosinophil-dependent inflammatory diseases, asthma
01/24/2002US20020010174 1,4-diazepine-2-one derivatives as neurokinin antagonist
01/24/2002US20020010120 Composition and method for bleaching a substrate
01/24/2002CA2416667A1 Cyclylamine sulfonamides as beta-3 adrenergic receptor agonists
01/24/2002CA2416245A1 Cyclic amine phenyl beta-3 adrenergic receptor agonists
01/24/2002CA2416036A1 Substituted amidoalkyl-uracils as parp inhibitors
01/24/2002CA2415665A1 Pyrrolidine-2-carboxylic acid hydrazide derivatives for use as metalloprotease inhibitors
01/24/2002CA2415662A1 1-alkyl-3-[1-(substituted phenyl) benzotriazol-6-yl] uracils
01/24/2002CA2415331A1 Beta3 adrenergic agonists
01/23/2002EP1175128A2 Light emitting element and azole compound
01/23/2002EP1173433A1 Cyanopyrroles as progesterone receptor agonists
01/23/2002EP1173424A1 Pyrimidine compounds
01/23/2002EP1173421A2 Indole derivatives as anti-inflammation agents
01/23/2002EP1173414A1 N-protected amines and their use as prodrugs
01/23/2002EP1173169A1 Aryl substituted pyrazoles, imidazoles, oxazoles, thiazoles and pyrroles, and the use thereof
01/23/2002CN1332737A Thrombin inhibitors
01/23/2002CN1332731A Substituted benzimidazoles and their prep. and use
01/23/2002CN1332166A Process for prep. of N-methyl-3-(1-methyl-4-piperidyl)-1H-indole-5-ethyl-sulfonamide
01/23/2002CN1078210C Watersoluble azole antifungals
01/23/2002CN1078208C Pyrrolyl tetrahydrobenzoquinoxaline diones, their preparation and use as glutamate receptor antagonists
01/22/2002US6340758 Conformationally semi-constrained quinoxaline 2,3-diones as neuroprotective agents
01/22/2002US6340700 2-(iminomethyl) amino-phenyl derivatives, preparation, application as medicines and pharmaceutical compositions containing same
01/22/2002US6340685 Antiinflammatory agents
01/22/2002US6340683 Selective NPY (Y5) antagonists (triazines)
01/22/2002US6340678 4,4-difluoro-2,3,4,5-tetrahydro-1H-1-benzoazepine derivatives and drug compositions containing them
01/22/2002CA2043709C Antimigraine alkoxypyrimidine derivatives
01/17/2002WO2002004440A1 Composition and antiviral activity of substituted indoleoxoacetic piperazine derivatives
01/17/2002WO2002004429A1 Pyrimidine derivatives
01/17/2002WO2002004426A1 Squaric acid derivatives containing a bicyclic heteroaromatic ring as integrin antagonists
01/17/2002WO2002004425A2 Viral polymerase inhibitors
01/17/2002WO2002004424A1 Pyrazole derivatives
01/17/2002WO2002003977A2 Combinations of statins, estrogenic agents and optionally estrogens
01/17/2002WO2001062726A3 2-oxo-1-pyrrolidine derivatives, processes for preparing them and their uses
01/17/2002WO2001039759A3 Sulfonic acid or sulfonylamino n-(heteroaralkyl)-azaheterocyclylamide compounds
01/17/2002US20020007075 Neurological disorders including physically damaged nerves and neurodegenerative diseases, and for treating alopecia and promoting hair growth; Alzheimer's, Parkinson's disease; amyotrophic lateral sclerosis
01/17/2002US20020007071 Treating disorders which include neuropeptide Y excess; antagonists, antagonism
01/17/2002US20020006952 Kinase inhibitors; anticancer agents
01/17/2002US20020006948 Central nervous system disorders; antiinflammatory agents
01/17/2002US20020006943 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis
01/17/2002US20020006934 Phenyl-substituted imidazopyridines
01/17/2002US20020006928 Phenyl-substituted indoles and indazoles
01/17/2002CA2415492A1 Pyrazole derivatives
01/17/2002CA2414060A1 Combinations of statins, estrogenic agents and optionally estrogens
01/17/2002CA2413044A1 Composition and antiviral activity of substituted indoleoxoacetic piperazine derivatives
01/16/2002EP1171435A2 Pyrimidine-2-one derivatives as integrin receptor ligands
01/16/2002EP1171428A1 Fab i inhibitors
01/16/2002EP1171424A1 Cyclo-alkyl substituted benzimidazoles and their use as parp inhibitors
01/16/2002EP1171122A1 Pyrrolidine modulators of chemokine receptor activity
01/16/2002EP0880517B1 Quinazoline compounds
01/16/2002EP0766678B1 Optical brightening agents
01/16/2002EP0638075B1 Thiazole or imidazole derivatives as maillard reaction inhibitors
01/16/2002CN1331693A 1,2-annelated quinoline derivatives
01/16/2002CN1331691A Piperidines as CCR5 modulators
01/16/2002CN1331689A 4-and 5-alkynyloxindoles and 4-and 5-alkenyloxindoles
01/16/2002CN1331682A Substituted 2-phenylbenzimidazoles, prodn. thereof and their use
01/16/2002CN1331679A 3-azabicyclo [3.1.0] hexane derivatives as opiate receptors ligands
01/16/2002CN1331677A Pyrrolidine derivatives-CCR-3 receptor antagonists
01/16/2002CN1331591A Piperidines as CCR5 modulators
01/15/2002US6339101 Administering n-linked sulfonamide of an n-heterocyclic carboxylic acid derivative for therapy of nerve-related vision disorder, improving vision, therapy memory impairment or enhancing memory performance in an animal
01/15/2002US6339099 Guanidine mimics as factor Xa inhibitors
01/15/2002CA2028302C Benzimidazole derivatives, their production and use
01/10/2002WO2002002554A1 Sulfonyl-pyrrolidine derivatives useful for the treatment of neurological disorders
01/10/2002WO2002002551A1 4-heteroaryl-3-heteroarylidenyl-2-indolinones and their use as protein kinase inhibitors
01/10/2002WO2002002539A1 Aryl phenylheterocyclyl sulfide derivatives and their use as cell adhesion-inhibiting anti-inflammatory and immune-suppressive agents
01/10/2002WO2002002533A1 Propane-1,3-dione derivatives
01/10/2002WO2002002531A1 Nonpeptide substituted spirobenzoazepines as vasopressin antagonists
01/10/2002WO2002002523A1 Process for preparing distamycin derivatives
01/10/2002WO2002002488A2 Methods and compounds for modulating nuclear receptor coactivator binding
01/10/2002WO2001056993A3 Pyrazole compositions useful as inhibitors of erk
01/10/2002US20020004600 Process for the preparation of substituted pyrimidines
01/10/2002US20020004503 Viricides
01/10/2002US20020004501 Therapy for muscular disorders, urogenital disorders, gastrointestinal disorders, respiratory system disorders
01/10/2002US20020004494 Muscular disorders, gastrointestinal disorders, respiratory system disorders
01/10/2002US20020004032 Macrocyclic chelants for metallopharmaceuticals
01/10/2002CA2415103A1 Methods and compounds for modulating nuclear receptor coactivator binding
01/10/2002CA2414468A1 4-heteroaryl-3-heteroarylidenyl-2-indolinones and their use as protein kinase inhibitors
01/10/2002CA2414461A1 Aryl phenylheterocyclyl sulfide derivatives and their use as cell adhesion-inhibiting anti-inflammatory and immune-suppressive agents
01/10/2002CA2413243A1 Sulfonyl-pyrrolidine derivatives useful for the treatment of neurological disorders
01/09/2002EP1170290A2 Compounds having ultra-violet absorption properties
01/09/2002EP1170289A2 Retroviral protease inhibiting compounds
01/09/2002EP1169320A1 Farnesyl transferase inhibitors having a pyrrole structure and process for preparation thereof
01/09/2002EP0996617B1 2,4-Dithi(oxo)-pyridin-5-yl compounds bearing a tricyclic substituent useful as P2 purinoceptor antagonists
01/09/2002EP0918768B1 Aromatic amidine derivatives useful as selective thrombin inhibitors
01/09/2002EP0607439B1 Nitrogenous heterocyclic compound
01/09/2002CN1330654A 4,5-pyrrolo-oxindoles
01/09/2002CN1330648A 4-aryloxindoles as inhibitor of JNK protein kinases
01/09/2002CN1330647A 4-alkenyl (and alkynyl) oxindoles as inhibitors of cell cycle protein dependent kinases, in particular CDK2
01/09/2002CN1330634A Carboxylic acids and carboxylic acid isosteres of N-heterocyclic compounds
01/09/2002CN1077572C 取代的吡咯 Substituted pyrrole
01/09/2002CN1077571C Substituted bisindolylmaleimides for inhibition of cell proliferation
01/08/2002US6337344 Anticoagulants and enzyme inhibitors for cardiovascular disorders
01/08/2002US6337342 Bis-aryl or heteroaryl indoles
01/08/2002US6337340 Carboxylic acids and isosteres of heterocyclic ring compounds having multiple heteroatoms for vision and memory disorders
01/08/2002US6337335 Enzyme inhibitors for autoimmune diseases, transplant rejection, grant versus host disease, hyperproliferative disorders and diseases in which cells receive pro-inflammatory signals.