Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
02/2002
02/26/2002US6350786 Complexes significantly increase the bioavailability of poorly soluble therapeutically active compounds
02/26/2002US6350748 Sulfamoyl compounds and agricultural and horticultural fungicides
02/26/2002US6350747 Protein serine/threonine kinase and protein tyrosine kinase enzyme inhibitors; angiogenesis inhibitors; antitumor and antiproliferative agents
02/26/2002US6350744 Pyrmidine or pyridine derivatives; antiarthritic and antiinflammatory agents; cachexia treatment; interleukin and tumor necrosis factor inhibitors
02/26/2002CA2206776C N-sulfonylindoline derivatives carrying an amide functional group, their preparation and the pharmaceutical compositions in which they are present
02/26/2002CA2178302C Indole, indazole and benzisoxazole derivatives; process for preparing the same and pharmaceutical compositions containing them
02/26/2002CA2081605C Complex salts of hematoporphyrin and of its derivatives, their synthesis and therapeutic agent
02/21/2002WO2002014308A1 Antithrombotic agents
02/21/2002WO2002014307A1 Factor viia inhibitors
02/21/2002WO2002014285A1 Substituted imidazoles as tafia inhibitors
02/21/2002WO2002014274A1 Selective urokinase inhibitors
02/21/2002WO2002014273A1 Indoline derivatives as 5ht2c antagonists
02/21/2002WO2002014271A1 Proline derivatives and use thereof as drugs
02/21/2002WO2002006247A8 Substituted amidoalkyl-uracils as parp inhibitors
02/21/2002WO2001058869B1 Cannabinoid receptor modulators, their processes of preparation, and use of cannabinoid receptor modulators in treating respiratory and non-respiratory diseases
02/21/2002WO2001047510A3 Methods and compositions related to modulators of annexin and cartilage homeostasis
02/21/2002WO2001019791A3 3-vinylpyrrole derivatives, method for the production thereof and their use as medicaments
02/21/2002WO2000054729A8 Heterocyclic aromatic compounds useful as growth hormone secretagogues
02/21/2002US20020022605 Cyclamine sulfonamides as beta-3 adrenergic receptor agonists
02/21/2002DE10039998A1 Neue substituierte Diareno-azepin-Derivate als Integrin Liganden New substituted Diareno-azepine derivatives as integrin ligands
02/20/2002EP1180513A1 Cyclic amide compounds, process for the preparation of the same and uses thereof
02/20/2002EP1180101A1 Compounds having cytokine inhibitory activity
02/20/2002EP0841922B1 1h-4(5)-substituted imidazole derivatives
02/20/2002CN1336930A Bridged heterocyclic derivatives
02/20/2002CN1336925A 4,5,6 and 7-indole and indoline derivatives, their prepn. and use
02/20/2002CN1336924A Amide and urea derivatives as 5-HT reuptake inhibitors and at 5-HT 1B/1D ligands
02/20/2002CN1336919A Phenylphenanthridines with PDE-IV inhibiting activity
02/20/2002CN1336916A Arylpiperazinyl-cyclohexyl indole derivatives for the treatment of depression
02/20/2002CN1336915A Urea of N-heterocyclic carboxylic acid or the isostere of carboxylic acid and aminocarboxylic acid ester
02/20/2002CN1079397C 4-(benzo-1,3-dioxolyl)-pyrrolidine-3-carboxylic acid derivatives as endothelin antagonists
02/20/2002CN1079396C Aromatic amidine derivatives useful as selective thrombin inhibitors
02/19/2002US6348628 Pyridazin-3-one derivatives, their use, and intermediates for their production
02/19/2002US6348627 Aryl and heteroarylcyclopropyl oxime ethers and their use as fungicides
02/19/2002US6348482 Catechols as antimicrobial agents
02/19/2002US6348480 Pharmaceutical compound comprising a pyrazole derivative and methods of using the same for the treatment of calcium release-activated calcium channel associated diseases
02/19/2002US6348461 Central nervous system antagonist with heterocyclic substituents
02/19/2002US6348032 Method of inhibiting neoplastic cells with benzimidazole derivatives
02/19/2002CA2087274C 4-alkylimidazole derivatives
02/14/2002WO2002012442A2 Heterocyclic compounds as ligands of the gabaa receptor
02/14/2002WO2002012228A1 Cinnoline compounds
02/14/2002WO2002012205A1 BENZOTRIAZOLES CONTAINING α-CUMYL GROUPS SUBSTITUTED BY HETEROATOMS AND COMPOSITIONS STABILIZED THEREWITH
02/14/2002WO2002012199A1 Heterocyclic mutilin esters and their use as antibacterials
02/14/2002WO2002012198A2 4-pyrimidinamine derivatives, pharmaceutical compositions and related methods
02/14/2002WO2002012196A2 Lactam compounds and their use as inhibitors of serine proteases and method
02/14/2002WO2001068603A3 Cyclopropyl-fused pyrrolidine-based inhibitors of dipeptidyl iv, processes for their preparation, and their use
02/14/2002WO2001062739A3 Thioimidazolidine derivatives as light stabilizers for polymers
02/14/2002WO2001055119A3 Gonadotropin-releasing hormone receptor antagonists and methods relating thereto
02/14/2002US20020019531 Indoles
02/14/2002US20020019527 Antitumor, antcarcinogenic agents
02/14/2002US20020019525 Pyrido [2,3-b] indolizine derivatives and aza analogues thereof; CRF1 specific ligands
02/14/2002US20020019434 Indole derivatives having an antiviral activity
02/14/2002US20020019424 1-sulfonyl pyrrolidine derivatives
02/14/2002US20020019411 Cyclopropyl-fused pyrrolidine-based inhibitors of dipeptidyl peptidase IV and method
02/14/2002US20020019408 New isoxazole-sulfonamide endothelin antagonists
02/14/2002US20020019405 Nitrosated and nitrosylated phosphodiesterase inhibitors, compositions and methods of use
02/14/2002US20020019402 Integrin inhibitors and their methods of use
02/14/2002US20020019401 Psychological disorders; adjustment of dopamine concentration
02/14/2002US20020019390 Imidazole and imidazoline derivatives and uses thereof
02/14/2002US20020019389 3-(N-(5,6-dimethyl-2-methoxypyridin-3-yl)aminocarbonyl)-7,8-dimethoxy-1-phenyl-2,3,4,5-tetrahydro-3H-benzazepine, for example
02/14/2002US20020019383 3-amido or 3-sulfonylamino azetidine compounds and their preparation; high affinity for cannabinoid receptor CB1 type, useful in treating central nervous system, immune, gastrointestinal or cardiovascular disorders, drug abuse
02/14/2002CA2420967A1 Heterocyclic compounds as ligands of the gabaa receptor
02/14/2002CA2419030A1 4-pyrimidinamine derivatives, pharmaceutical compositions and related methods
02/14/2002CA2418995A1 Lactam compounds and their use as inhibitors of serine proteases and method
02/14/2002CA2415022A1 Cinnoline compounds
02/13/2002EP1178983A1 Indole-type derivatives as inhibitors of p38 kinase
02/13/2002EP1178981A1 Substituted 3-pyridyl-4-arylpyrroles, and related therapeutic and prophylactic methods
02/13/2002EP1178973A2 Novel compounds, their use and preparation
02/13/2002EP1178969A1 Gastrin and cholecystokinin receptor ligands
02/13/2002EP1042320B1 New compounds which are p2-purinoceptor 7-transmembrane (tm) g-protein coupled receptor antagonists
02/13/2002EP0869942B1 4-((heterocycloalkyl or heteroaromatic)-substituted phenyl]-2-azetidinones useful as hypolipidemic agents
02/13/2002EP0711768B1 Benzimidazole derivative
02/13/2002CN1335839A Bis-sulfonamides
02/13/2002CN1335838A Pyrimidine compounds
02/13/2002CN1335836A Tricyclic pyrazole derivatives
02/13/2002CN1335834A Aromatic heterocycle compounds having HIV integrase inhibiting activities
02/13/2002CN1335773A Method of using (2-imidazolin-2-ylamino) quinoxalines in treating neural injury
02/13/2002CN1335316A New N-triazolyl methyl piperazine derivate using as neurokinin receptor antagonistic agent
02/13/2002CN1079097C Bicyclic heterocyclic sulfonamide and sulfonic ester derivatives
02/13/2002CN1079096C Arylsulfonylimidazolone derivatives as antitumor agent
02/12/2002US6346625 Protein kinase inhibitors
02/12/2002US6346621 Indole or quinoline compounds substituted with amino compounds on nitrogen
02/12/2002US6346620 Methods for preparation of 2-(4-(4-(4,5-dichloro-2-methylimidazol-1-yl)butyl)-1-piperazinyl)-5-fluoropyrimidine and salts thereof
02/12/2002US6346522 1-arylpyrazoles; systemic pesticides, insecticides, larvicides, miticides, antiprotozoa, and anthelmintic agents; agriculture, horticulture, animal husbandry, public health and veterinary medicine
02/12/2002US6346503 Substituted 2-amino-4-alkylamino-1,3,5-triazines as herbicides
02/12/2002CA2088742C Benzimidazole and imidazopyridine derivatives and their application
02/12/2002CA2067877C Polycyclic amine compounds and their enantiomers, their method of preparation and pharmaceutical compositions in which they are present
02/07/2002WO2002010158A2 3-indolyl-4-phenyl-1h-pyrrole-2,5-dione derivatives as inhibitors of glycogen synthase kinase-3beta
02/07/2002WO2002010154A2 Substituted heterocyclic amides
02/07/2002WO2002010141A1 Imidazole derivatives
02/07/2002WO2002010140A2 Imidazolyl derivatives
02/07/2002WO2002010137A2 Indazole derivatives as jnk inhibitors
02/07/2002WO2002009648A2 Antimicrobial biaryl compounds
02/07/2002WO2001085700A3 Hiv replication inhibiting pyrimidines and triazines
02/07/2002WO2001062744A3 Substituted piperazine compounds
02/07/2002WO2001060806A3 Substituted arylpyrazines
02/07/2002WO2001030333A3 Tissue factor antagonists and methods of use thereof
02/07/2002US20020016498 Jet streams of solvent impinge creating high turbulence at point of impact on chemical intermediates; eliminates need for high intensity milling
02/07/2002US20020016459 Substituted 2-amino-4-alkylamino-1,3,5-triazines as herbicides
02/07/2002US20020016333 Pyrazoles and pyrazolopyrimidines having crf antagonistic activity
02/07/2002US20020016327 Compounds and methods of use for treatment of neurogenic inflammation