Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
07/2009
07/22/2009CN101486708A 4-nitro glyoxaline compound, preparation and use thereof
07/22/2009CN101486707A 2-methyl-5-nitro glyoxaline compound, preparation and use thereof
07/22/2009CN101486682A N3 alkylated benzimidazole derivatives as MEK inhibitors
07/22/2009CN101486679A 5HT2c receptor modulators
07/22/2009CN101486678A 5HT2C receptor modulators
07/22/2009CN101486677A 5HT2c receptor modulators
07/22/2009CN101486675A 2- and 2,5-substituted phenylketoenols
07/22/2009CN101485664A 5HT2c receptor modulators
07/21/2009US7563910 Heterocyclic cannabinoid receptor antagonists
07/21/2009US7563908 2-(1H-indolylsulfanyl)-benzyl amine derivatives as SSRI
07/21/2009US7563895 Quinoxaline compounds
07/21/2009US7563894 e.g. [2-(4-Isopropyl-piperazin-1-yl)-benzooxazol-6-yl]-[5-(4-methoxy-phenyl)-pyrimidin-2-yl]-amine; C-kit kinase receptor or stem cell factor inhibitors; anticarcinogenic agents; veterinary medicine
07/21/2009US7563893 3-Phenyl-cinnoline analogue and antitumor agent using the same
07/21/2009US7563784 substituted 1,1,4-1l6-trioxo[1,2]thiazepan-4-ylamide-derived protease inhibitors which inhibit the likes of cathepsin K; treating osteoporosis, osteo- and rheumatoid arthritis and periodontal disease; inhibiting excessive cartilage or matrix degradation
07/21/2009CA2495943C Indoles having anti-diabetic activity
07/16/2009WO2009089042A1 Pyrazole pyrazine amine compounds as kinase inhibitors, compositions thereof and methods of treatment therewith
07/16/2009WO2009088070A1 (heterocyclic methyl)azolylmethylcyclopentanol derivative and intermediate thereof, process for production of the derivative, and agricultural or horticultural preparation and protective agent for industrial material each comprising the derivative
07/16/2009WO2009087649A1 Renin inhibitors
07/16/2009WO2009087127A1 Modulators for amyloid beta
07/16/2009WO2009067686A8 Sunitinib hemi-l-malate, polymorphs and preparation thereof, polymorphs of racemic sunitinib malate, compositins containing sunitinib base and malic acid and preparation thereof
07/16/2009WO2009055335A3 Hcv protease inhibitors
07/16/2009WO2009003999A3 Chemical compounds
07/16/2009WO2008068171A9 Substituted pyrimidines and their use as jnk modulators
07/16/2009US20090182152 Dimer Dianthranilate Bis-[N-Dodecylanilinophenylpyrazolone Carboxamide]Diazo]; for use in hot melt or phase change inks
07/16/2009US20090182151 Method for making amphiphilic dendrimers
07/16/2009US20090182140 Alicyclic Heterocyclic Compound
07/16/2009US20090182114 Tetracarboxylic acid compound, polyimide thereof, and production method thereof
07/16/2009US20090181994 Triazole derivatives as inhibitors of 11-beta-hydroxysteroid dehydrogenase-1
07/16/2009US20090181993 Hiv inhibiting 5-heterocyclyl pyrimidines
07/16/2009US20090181984 Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidinyl derivative and its medical use
07/16/2009US20090181965 Modulators for amyloid beta
07/16/2009US20090181964 Propane-1,3-Dione Derivative or Salt Thereof
07/16/2009US20090181958 Substituted nitrogen-containing heterobicycles, the preparation thereof and their use as pharmaceutical compositions
07/16/2009US20090181953 Compound forms and uses thereof
07/16/2009US20090181952 Compounds useful as alpha7 nicotinic acetylcholine receptor agonists
07/16/2009US20090181949 1h-imidazole derivative having cb1, agonistic, cb1 partial agonistic or cb1 antagnistic activity
07/16/2009US20090181943 Inhibitors of Histone Deacetylase
07/16/2009US20090181939 Azetidinecarboxamide Derivatives And Their Use In The Treatment Of CB1 Receptor Mediated Disorders
07/16/2009US20090181938 Aminopyrimidines useful as kinase inhibitors
07/16/2009CA2703824A1 Modulators for amyloid beta
07/15/2009EP2078011A1 Manufacture of rimcazole
07/15/2009EP2078010A2 Polycyclic heteroaryl substituted triazoles useful as axl inhibitors
07/15/2009EP2078009A1 New fluorene derivatives, compositions containing the same and use thereof as inhibitors of the protein chaperone hsp 90
07/15/2009EP2078000A1 Benzoyl amino heterocyclyl compounds as glucokinase (glk) activators
07/15/2009EP2077998A1 Phthalazine, aza- and diaza-phthalazine compounds and methods of use
07/15/2009EP2077997A1 Pyridazine derivatives
07/15/2009EP2077841A1 Novel substituted pyrimidines as cysteine protease inhibitors
07/15/2009EP2005962A9 Therapeutic agent for inflammatory bowel disease
07/15/2009EP1874304B1 Benzotriazole derivatives as cannabinoid receptor antagonists
07/15/2009EP1426365B1 3-phenoxy-4-pyridazinol derivative and herbicide composition containing the same
07/15/2009EP1379514B1 5-membered heterocycles, preparation and application thereof as medicaments
07/15/2009CN101484444A Novel pyridazine compound and use thereof
07/15/2009CN101484443A Potentiator of radiation therapy
07/15/2009CN101481374A Method for removing trityl group of 1-trityl-5-(1,1'-biphenylyl-2 yl)-1H-tetrazole compound
07/15/2009CN100513398C 2-(2-hydroxybiphenyl-3-yl)-1h-benzoimidazole-5-carboxamidine derivatives as factor VIIA inhibitors
07/14/2009US7560569 (2S,4S)-1-[[(4-carbamoylbicyclo[2.2.2]oct-1-yl)amino]acetyl]-4-fluoropyrrolidine-2-carbonitrile, for treating type II diabetes; increase glucagon-like peptide activity
07/14/2009US7560551 Aurora kinase modulators and method of use
07/14/2009US7560546 Tyrosine kinase inhibitors
07/14/2009US7560483 Synthesizing 1- (acyloxy)-alkyl derivatives from 1-acyl-alkyl derivatives, which typically proceeds stereospecifically, in high yield, does not require the use of activated intermediates and/or toxic compounds and is readily amenable
07/14/2009US7560481 Indoles are cannabinoid receptor ligands
07/14/2009US7560480 Alkyl-containing 5-acylindolinones, the preparation thereof and their use as medicaments
07/14/2009US7560471 5-{4-[1-(2-Ethoxyethyl)-1H-indol-3-yl]piperidin-1-ylmethyl}-2-methoxybenzoic acid; histamine H1 antagonists; bronchial dialtors; asthma; allergic rhinitis; conjunctivitis; dermatitis; urticaria; selective antiallergic effects so less side effect reduction and lower dosage
07/14/2009US7560470 Heterocyclyl-3-sulfonylindazoles as 5-hydroxytryptamine-6 ligands
07/14/2009US7560467 Indazolo-tetrahydropyrimidine-carboxamide derivative kinase inhibitors
07/14/2009US7560466 N4-(2,2-Dimethyl-3-oxo-4H-5-pyrid[1,4]oxazin-6-yl)-N2-(3-chloro-4-methoxyphenyl)-5-fluoro-2,4-pyrimidinediamine; signal transduction cascade inhibitor; Fc receptors for IgE (Fc epsilon RI) and IgG (Fc gamma RI) antagonist; autoimmune diseases, antiinflammatory agent; rheumatoid arthritis
07/14/2009US7560462 Compounds useful for inhibiting CHK1
07/14/2009US7560461 Quinazoline derivatives as kinase inhibitors
07/14/2009US7560460 2-[(4-Chlorophenyl)methyl]-1-(4- {2-[(cyclopropylmethyl)-(methylsulfonyl)amino]phenyl }-piperazinyl) -4-(2-(1,2,3,4-tetrahydroisoquinolyl))butane-1,4-dione; obesity/dietietics; melanocortin receptor angonists; prophylaxis/treatment of diseases involving activation of the melanocortin recepetors (MCR)
07/14/2009US7560458 Triazolopyrimidine derivatives as glycogen synthase kinase 3 inhibitors
07/14/2009US7560456 Pesticidal pyridinecarboxamide derivatives
07/14/2009US7560454 1-(4-(10,11-dihydro-5H-pyrrolo[2,1-c](1,4)benzodiazepine-10-ylcarbonyl)-2-methyl-benzylcarbamoyl)-4methoxy-L-proline-N,N-dimethylamide; vasopressin agonists particularly useful in the treatment of urogenital disorders central diabetes insipidus, nocturnal enuresis and nocturia; blood disorders
07/10/2009WO2008083367A2 Polycyclic heteroaryl substituted triazoles useful as axl inhibitors
07/10/2009WO2008083357A1 Bridged bicyclic aryl and bridged bicyclic heteroaryl substituted triazoles useful as axl inhibitors
07/10/2009CA2710234A1 Polycyclic heteroaryl substituted triazoles useful as axl inhibitors
07/10/2009CA2710230A1 Bridged bicyclic aryl and bridged bicyclic heteroaryl substituted triazoles useful as axl inhibitors
07/09/2009WO2009086041A1 Herbicidal pyridazinone derivatives
07/09/2009WO2009084695A1 2-aminoquinazoline derivative
07/09/2009WO2009084614A1 Imidazole carbonyl compound
07/09/2009WO2009084029A2 Improved process for the preparation of (2r,3s)-2-(2,4- difluqrophenyl)-3-(5-fluoropyrimidin-4-yl)-1-(1h-1,2,4-triazol-1-yl) butan-2-ol
07/09/2009WO2009084028A2 Improved process for manufacturing anhydrous (e)-3-[2-butyl-1- {(4-carboxyphenyl) methyl}-1h-imidazole-5-yl]-(thiophen-2- ylmethyl)prop-2-enoic acid methane sulfonate
07/09/2009WO2009083553A1 Azine compounds as glucokinase activators
07/09/2009WO2009083076A1 2-benzylpyridazinone derivatives as met kinase inhibitors
07/09/2009WO2009082845A1 N-{1-[3-(2-ethoxy-5-(4-ethylpiperazinyl)benzenesulfonyl)-4,5-dihydro-5-oxo-1,2,4-triazin-6-yl]ethyl}butyramide, the preparation method and use thereof
07/09/2009WO2009057811A3 Heterocyclic compound and pharmaceutical composition thereof
07/09/2009WO2008130368A3 Transcription factor modulating compounds and methods of use thereof
07/09/2009WO2008039087A8 Indoline derivatives and uses thereof
07/09/2009US20090176988 Preparation and Use of Magnesium Amides
07/09/2009US20090176984 Isotopically Enriched N-Substituted Piperazine Acetic Acids And Methods For The Preparation Thereof
07/09/2009US20090176981 Stereoisomerically Enriched 3-Aminocarbonyl Bicycloheptene Pyrimidinediamine Compounds And Their Uses
07/09/2009US20090176973 Thrombopoietin mimetics
07/09/2009US20090176859 Cathepsin cysteine protease inhibitors
07/09/2009US20090176858 Hcv protease inhibitors and uses thereof
07/09/2009US20090176849 Process for the preparation of 2-alkyl-1-((2'-substituted-biphenyl-4-yl) Methyl)-imidazole, dihydroimidazole or benzimidazloe derivatives
07/09/2009US20090176840 Use of galr3 receptor antagonists for the treatment of depression and/or anxiety and compounds useful in such methods
07/09/2009US20090176806 protein kinase C or glycogen synthase kinase-3-beta inhibitors such as 3-(2-chlorophenyl)-4-[1-(3-hydroxypropyl)-1H-pyrrolo[2,3-b]pyridin-3-yl]-1H-pyrrole-2,5-dione, used for treating cardiovascular, skin, nervous system disorders and immunological disorders, diabetes, inflammatory diseases and cancer
07/09/2009US20090176799 Phosphodiesterase 4 inhibitors
07/09/2009US20090176798 New compounds III
07/09/2009US20090176794 1h-indol-1-yl-urea compounds
07/09/2009US20090176782 Inhibitors of tace
07/09/2009US20090176781 Acetylenic Heteroaryl Compounds