Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587) |
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08/12/2009 | EP2086964A2 Benzoyl amino heterocyclyl compounds useful in the treatment of a disease mediated through glk |
08/12/2009 | EP2086960A1 Novel inhibitors of glutaminyl cyclase |
08/12/2009 | EP2086959A1 Substituted 2-imidazoles as modulators of the trace amine associated receptors |
08/12/2009 | EP2086942A2 Novel compounds |
08/12/2009 | EP2086547A2 Solid forms of (3'-chlorobiphenyl-4-yl)(1-(pyrimidin-2-yl)piperidin-4-yl)methanone and methods of their use |
08/12/2009 | EP1910497A4 Compositions and methods for coupling a plurality of compounds to a scaffold |
08/12/2009 | EP1885695B8 Indoline compounds |
08/12/2009 | EP1863871B1 Rubber composition comprising an itaconimido-maleimide |
08/12/2009 | EP1756096B1 Indolyl derivatives as liver-x-receptor modulators |
08/12/2009 | EP1682121B1 Use of crth2 antagonist compounds in therapy |
08/12/2009 | EP1636221B1 3-Heterocyclyl-Azetidine compounds useful as NK1/NK2 receptors antagonists |
08/12/2009 | EP1224170B1 6-position substituted indoline, production and use thereof as a medicament |
08/12/2009 | CN101506202A mGluR5 modulators I |
08/12/2009 | CN101506195A New pyridone derivatives with MCH antagonistic activity and medicaments comprising these compounds |
08/12/2009 | CN101506176A 2-anilino-4-aminoalkyleneaminopyrimidines |
08/12/2009 | CN101506175A 2-anilino-4-(heterocyclic)amino-pyrimidines as inhibitors of protein kinase C-alpha |
08/12/2009 | CN101506162A Substituted isoindoles as bace inhibitors and their use |
08/12/2009 | CN100526308C Arylvinylazacycloalkane compounds and methods of preparation and use thereof |
08/12/2009 | CN100526307C Metalloproteinase inhibitors |
08/12/2009 | CN100526298C Amide derivative and medicine |
08/12/2009 | CN100525763C Mono- and bicyclic azole derivatives that inhibit the interaction of ligands with rage |
08/11/2009 | US7572924 Pyrrole substituted 2-indolinone protein kinase inhibitors |
08/11/2009 | US7572922 Substituted pyrazoles, compositions containing such compounds and methods of use |
08/11/2009 | US7572921 Substituted benzylimidazoles useful for the treatment of inflammatory diseases |
08/11/2009 | US7572914 2-hydroxy-1H-indol derivatives enzyme inhibitors for preventing or treating inflammation, inflammatory bowel disease, psoriasis, dementia related diseases Alzheimer's Disease, Cognitive Impairment, arthritis, neurodegenerative diseases, amyotrophic lateral sclerosis, Down syndrome, Huntington's Disease |
08/11/2009 | US7572913 Inhibitors of Rho kinase; N-Benzyloxycarbonyl-4-[N''-(tert-butyloxycarbonyl)hydrazino]piperidine; 4-{[N''-(tert-butyloxycarbonyl)-N'-(1'-propyl)]hydrazino}piperidine |
08/11/2009 | US7572910 Heteroaromatic substituted sulfonyl or sulfoxide or thio-pyridazinone derivatives, useful for treating diabetic complications and cardiovascular disorders; eg 3-Methoxy-6-(5-chloro-3-methyl-benzofuran-2-sulfenyl)-pyridazine |
08/11/2009 | US7572824 Methods for minimizing thioamide impurities |
08/11/2009 | US7572816 Therapeutic agents for the treatment of cancer, metabolic diseases and skin disorders |
08/11/2009 | US7572812 Treating or preventing pain, UI, an ulcer, IBD, IBS, an addictive disorder, Parkinson's disease, parkinsonism, anxiety, epilepsy, stroke, a seizure, a pruritic condition, psychosis, a cognitive disorder, a memory deficit, restricted brain function, Huntington's chorea, amyotrophic lateral sclerosis |
08/11/2009 | US7572809 (1-Isopropyl-6-methoxy-isoquinolin-3-yl)-(5-methyl-1H-pyrazol-3-yl)-amine; (5-Cyclopropyl-1H-pyrazol-3-yl)-(1-isopropyl-6,7-dimethoxy-isoquinolin-3-yl)-amine; Aurora kinase inhibitors; cancer |
08/11/2009 | US7572796 excitatory amino acid antagonists for treating neurodegenerative diseases as cerebrovascular diseases, epilepsy, schizophrenia, Alzheimer's disease, Parkinson's disease, Huntington's disease, cerebral ischaemia, infarction, psychoses; 6-{3-[4-(4-fluorobenzyl)-1-piperidyl]propyl}-1H-indole-3-carbonitrile |
08/11/2009 | US7572793 Tau protein kinase 1 inhibitors; treatment for neurodegenerative disorders; Alzheimer's Disease, Parkinson's disease, Pick's Disease, vision defects; antiischemic, antidiabetic, anticarcinogenic, antitumor agents, antidepressants |
08/11/2009 | US7572788 Compositions and methods relating to novel compounds and targets thereof |
08/11/2009 | CA2527933C Substituted 3-alkyl and 3-alkenyl azetidine derivatives |
08/11/2009 | CA2395846C Diazepan derivatives or salts thereof |
08/11/2009 | CA2219359C Hydantoin derivatives as intermediates for pharmaceutical active compounds |
08/06/2009 | WO2009097306A1 Substituted pyridazine derivatives which have histamine h3 antagonist activity |
08/06/2009 | WO2009096526A1 Carboxylic acid compound or salt thereof |
08/06/2009 | WO2009095933A2 Improved and novel process for the preparation of bosentan |
08/06/2009 | WO2009095773A2 Novel heterocycles |
08/06/2009 | WO2009095399A2 Pyrazine derivatives and their use as protein kinase inhbitors |
08/06/2009 | WO2009095394A1 Diazepanes as histamine h3 receptor antagonists |
08/06/2009 | WO2009095163A2 Cyclic indole-3-carboxamides, their preparation and their use as pharmaceuticals |
08/06/2009 | WO2009094866A1 Dicycloazaalkane derivates, preparation processes and medical uses thereof |
08/06/2009 | WO2009094845A1 5-(3-heteroaromatic ring substituted phenyl) tetrazole compounds and their uses for anti-hiv/aids |
08/06/2009 | WO2009054952A3 Small molecule inhibitors of parp activity |
08/06/2009 | US20090198060 Nitrogen-containing heterocyclic compound and thrombopoietin receptor activator |
08/06/2009 | US20090198056 such as N-[(1S,2R)-1-Benzyl-2-hydroxy-3-(1H-imidazol-2-ylamino)-3-oxopropyl]-5-[methyl(methylsulfonyl)amino]-N'-[(1R)-1-phenylethyl]isophthalamide, used for the for treatment of Alzheimer's disease |
08/06/2009 | US20090198052 Method for preparing optically active piperidine compounds |
08/06/2009 | US20090198049 Methods and intermediates for the synthesis of porphyrins |
08/06/2009 | US20090197899 3-(Dihydro-1H-pyrazolo[4,3-d]pyrimidin-5-yl)-4-propoxybenzenesulfonamide Derivatives and Methods of Use |
08/06/2009 | US20090197886 Hexahydro-cycloheptapyrazole cannabinoid modulators |
08/06/2009 | US20090197885 Compositions and treatments using pyridazine compounds and cholinesterase inhibitors |
08/06/2009 | US20090197883 Diphenyl Substituted Cycloalkanes, Compositions Containing Such Compounds and Methods Of Use |
08/06/2009 | US20090197882 Indazole derivatives for the treatment of hsp90-induced diseases |
08/06/2009 | US20090197879 Vanilloid receptor ligands and their use in treatments |
08/06/2009 | US20090197860 Biaryl substituted diazabicycloalkane derivatives |
08/06/2009 | CA2715069A1 Novel heterocycles |
08/06/2009 | CA2713553A1 Pyrazine derivatives and their use as protein kinase inhibitors |
08/06/2009 | CA2712885A1 Substituted pyridazine derivatives which have histamine h3 antagonist activity |
08/06/2009 | CA2712854A1 Cyclic indole-3-carboxamides, their preparation and their use as pharmaceuticals |
08/06/2009 | CA2712352A1 Dicycloazaalkane derivates, preparation processes and medical uses thereof |
08/05/2009 | EP2085395A1 Arylvinylazacycloalkane compounds and methods of preparation and use thereof |
08/05/2009 | EP2085394A2 Metronidazole derivatives as antiparasitic agents |
08/05/2009 | EP2085391A2 Inhibitors of factor XA and other serine proteases involved in the coagulation cascade |
08/05/2009 | EP2084152A2 Substituted 4-imidazoles |
08/05/2009 | EP2084151A1 Substituted dihydropyrazolones for treating cardiovascular and haematological diseases |
08/05/2009 | EP2084148A1 Fungicide n-cycloalkyl-carboxamide, thiocarboxamide and n-substituted-carboximidamide derivatives |
08/05/2009 | EP2084131A1 Indole and benzofuran 2-carboxamide derivatives |
08/05/2009 | EP2083818A2 Melatonin derivatives and their use as antioxidants |
08/05/2009 | EP1924560B1 6-substituted- 2,3,4,5-tetrahydro-1h-benzo[d]azepines as 5-ht2c receptor agonists |
08/05/2009 | EP1877398B1 Quinazoline derivatives as egf and/or erbb2 tyrosine kinase inhibitors |
08/05/2009 | EP1781606B1 Azetidine derivatives as ccr-3 receptor antagonists |
08/05/2009 | EP1699454B1 Pyrazole derivatives and use thereof as orexin receptor antagonists |
08/05/2009 | EP1631292B1 4-anilino-quinazoline derivatives as antiproliferative agents |
08/05/2009 | EP1531822B1 1-aryl-4-substituted piperazine derivatives for use as ccr1 antagonists for the treatment of inflammation and immune disorders |
08/05/2009 | EP1501797B1 3-(substituted amino)-1h-indole-2-carboxylic acid ester and 3-(substituted amino)-benzo[b]thiophene-2-carboxylic acid ester derivatives as interleukin-4 gene expression inhibitors |
08/05/2009 | EP1491534B1 Novel hairpin polyamide |
08/05/2009 | EP1465880B1 5-sulphanyl-4h-1,2,4-triazole derivatives and their use to treat disorders associated with somatostatine |
08/05/2009 | EP1445253B1 4,4-difluoro-1, 2, 3, 4-tetrahydro-5h-1-benzazepine derivatives or salts thereof |
08/05/2009 | EP1399116B1 Use of dicationic compounds for dyeing human keratinous fibres and compositions containing same |
08/05/2009 | EP1357111B1 2-pyridone derivatives having affinity for cannabinoid type 2 receptor |
08/05/2009 | EP1296974B1 2-cyanopyrrolidine derivatives and their use as medicaments |
08/05/2009 | CN101501023A Phenyl substituted heteroaryl-derivatives and use thereof as anti-tumor agents |
08/05/2009 | CN101501021A Muscarinic receptor agonists that are effective in the treatment of pain, alzheimer's disease and schizophrenia |
08/05/2009 | CN101501008A Arylpiperazine derivatives and uses thereof |
08/05/2009 | CN101501006A Pyridinone and pyridazinone derivatives as inhibitors of poly(ADP-ribose)polymerase (PARP) |
08/05/2009 | CN101500995A 1-oxo-isoindoline compounds for the treatment of spinal muscular atrophy and other uses |
08/05/2009 | CN101500994A 1,3-disubstituted 4-methyl-1h-pyrrole-2-carboxamides and their use for the manufacture of medicaments |
08/05/2009 | CN101497607A Process for synthesizing sunitinib |
08/05/2009 | CN100522960C Thioamide derivatives as progesterone receptor modulators |
08/05/2009 | CN100522947C CCK-1 receptor modulators |
08/05/2009 | CN100522161C (Indol-3-yl)-heterocycle derivatives as agonists of the cannabinoid CB1 receptor |
08/04/2009 | US7569724 Antiproliferative agnets; anticancer agents; skin disorders |
08/04/2009 | US7569700 Substituted, bicyclic 8-pyrrolidinobenzimidazoles, methods for their production and their use as medicaments |
08/04/2009 | US7569689 Modulators of the glucocorticoid receptor, AP-1, and/or NF-κB activity and use thereof |
08/04/2009 | US7569688 Propane-1, 3-dione derivative |
08/04/2009 | US7569678 Protease inhibitor conjugates and antibodies useful in immunoassay |
08/04/2009 | US7569592 Heteroaryl substituted pyrazole modulators of metabotropic glutamate receptor-5 |