Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
08/2009
08/12/2009EP2086964A2 Benzoyl amino heterocyclyl compounds useful in the treatment of a disease mediated through glk
08/12/2009EP2086960A1 Novel inhibitors of glutaminyl cyclase
08/12/2009EP2086959A1 Substituted 2-imidazoles as modulators of the trace amine associated receptors
08/12/2009EP2086942A2 Novel compounds
08/12/2009EP2086547A2 Solid forms of (3'-chlorobiphenyl-4-yl)(1-(pyrimidin-2-yl)piperidin-4-yl)methanone and methods of their use
08/12/2009EP1910497A4 Compositions and methods for coupling a plurality of compounds to a scaffold
08/12/2009EP1885695B8 Indoline compounds
08/12/2009EP1863871B1 Rubber composition comprising an itaconimido-maleimide
08/12/2009EP1756096B1 Indolyl derivatives as liver-x-receptor modulators
08/12/2009EP1682121B1 Use of crth2 antagonist compounds in therapy
08/12/2009EP1636221B1 3-Heterocyclyl-Azetidine compounds useful as NK1/NK2 receptors antagonists
08/12/2009EP1224170B1 6-position substituted indoline, production and use thereof as a medicament
08/12/2009CN101506202A mGluR5 modulators I
08/12/2009CN101506195A New pyridone derivatives with MCH antagonistic activity and medicaments comprising these compounds
08/12/2009CN101506176A 2-anilino-4-aminoalkyleneaminopyrimidines
08/12/2009CN101506175A 2-anilino-4-(heterocyclic)amino-pyrimidines as inhibitors of protein kinase C-alpha
08/12/2009CN101506162A Substituted isoindoles as bace inhibitors and their use
08/12/2009CN100526308C Arylvinylazacycloalkane compounds and methods of preparation and use thereof
08/12/2009CN100526307C Metalloproteinase inhibitors
08/12/2009CN100526298C Amide derivative and medicine
08/12/2009CN100525763C Mono- and bicyclic azole derivatives that inhibit the interaction of ligands with rage
08/11/2009US7572924 Pyrrole substituted 2-indolinone protein kinase inhibitors
08/11/2009US7572922 Substituted pyrazoles, compositions containing such compounds and methods of use
08/11/2009US7572921 Substituted benzylimidazoles useful for the treatment of inflammatory diseases
08/11/2009US7572914 2-hydroxy-1H-indol derivatives enzyme inhibitors for preventing or treating inflammation, inflammatory bowel disease, psoriasis, dementia related diseases Alzheimer's Disease, Cognitive Impairment, arthritis, neurodegenerative diseases, amyotrophic lateral sclerosis, Down syndrome, Huntington's Disease
08/11/2009US7572913 Inhibitors of Rho kinase; N-Benzyloxycarbonyl-4-[N''-(tert-butyloxycarbonyl)hydrazino]piperidine; 4-{[N''-(tert-butyloxycarbonyl)-N'-(1'-propyl)]hydrazino}piperidine
08/11/2009US7572910 Heteroaromatic substituted sulfonyl or sulfoxide or thio-pyridazinone derivatives, useful for treating diabetic complications and cardiovascular disorders; eg 3-Methoxy-6-(5-chloro-3-methyl-benzofuran-2-sulfenyl)-pyridazine
08/11/2009US7572824 Methods for minimizing thioamide impurities
08/11/2009US7572816 Therapeutic agents for the treatment of cancer, metabolic diseases and skin disorders
08/11/2009US7572812 Treating or preventing pain, UI, an ulcer, IBD, IBS, an addictive disorder, Parkinson's disease, parkinsonism, anxiety, epilepsy, stroke, a seizure, a pruritic condition, psychosis, a cognitive disorder, a memory deficit, restricted brain function, Huntington's chorea, amyotrophic lateral sclerosis
08/11/2009US7572809 (1-Isopropyl-6-methoxy-isoquinolin-3-yl)-(5-methyl-1H-pyrazol-3-yl)-amine; (5-Cyclopropyl-1H-pyrazol-3-yl)-(1-isopropyl-6,7-dimethoxy-isoquinolin-3-yl)-amine; Aurora kinase inhibitors; cancer
08/11/2009US7572796 excitatory amino acid antagonists for treating neurodegenerative diseases as cerebrovascular diseases, epilepsy, schizophrenia, Alzheimer's disease, Parkinson's disease, Huntington's disease, cerebral ischaemia, infarction, psychoses; 6-{3-[4-(4-fluorobenzyl)-1-piperidyl]propyl}-1H-indole-3-carbonitrile
08/11/2009US7572793 Tau protein kinase 1 inhibitors; treatment for neurodegenerative disorders; Alzheimer's Disease, Parkinson's disease, Pick's Disease, vision defects; antiischemic, antidiabetic, anticarcinogenic, antitumor agents, antidepressants
08/11/2009US7572788 Compositions and methods relating to novel compounds and targets thereof
08/11/2009CA2527933C Substituted 3-alkyl and 3-alkenyl azetidine derivatives
08/11/2009CA2395846C Diazepan derivatives or salts thereof
08/11/2009CA2219359C Hydantoin derivatives as intermediates for pharmaceutical active compounds
08/06/2009WO2009097306A1 Substituted pyridazine derivatives which have histamine h3 antagonist activity
08/06/2009WO2009096526A1 Carboxylic acid compound or salt thereof
08/06/2009WO2009095933A2 Improved and novel process for the preparation of bosentan
08/06/2009WO2009095773A2 Novel heterocycles
08/06/2009WO2009095399A2 Pyrazine derivatives and their use as protein kinase inhbitors
08/06/2009WO2009095394A1 Diazepanes as histamine h3 receptor antagonists
08/06/2009WO2009095163A2 Cyclic indole-3-carboxamides, their preparation and their use as pharmaceuticals
08/06/2009WO2009094866A1 Dicycloazaalkane derivates, preparation processes and medical uses thereof
08/06/2009WO2009094845A1 5-(3-heteroaromatic ring substituted phenyl) tetrazole compounds and their uses for anti-hiv/aids
08/06/2009WO2009054952A3 Small molecule inhibitors of parp activity
08/06/2009US20090198060 Nitrogen-containing heterocyclic compound and thrombopoietin receptor activator
08/06/2009US20090198056 such as N-[(1S,2R)-1-Benzyl-2-hydroxy-3-(1H-imidazol-2-ylamino)-3-oxopropyl]-5-[methyl(methylsulfonyl)amino]-N'-[(1R)-1-phenylethyl]isophthalamide, used for the for treatment of Alzheimer's disease
08/06/2009US20090198052 Method for preparing optically active piperidine compounds
08/06/2009US20090198049 Methods and intermediates for the synthesis of porphyrins
08/06/2009US20090197899 3-(Dihydro-1H-pyrazolo[4,3-d]pyrimidin-5-yl)-4-propoxybenzenesulfonamide Derivatives and Methods of Use
08/06/2009US20090197886 Hexahydro-cycloheptapyrazole cannabinoid modulators
08/06/2009US20090197885 Compositions and treatments using pyridazine compounds and cholinesterase inhibitors
08/06/2009US20090197883 Diphenyl Substituted Cycloalkanes, Compositions Containing Such Compounds and Methods Of Use
08/06/2009US20090197882 Indazole derivatives for the treatment of hsp90-induced diseases
08/06/2009US20090197879 Vanilloid receptor ligands and their use in treatments
08/06/2009US20090197860 Biaryl substituted diazabicycloalkane derivatives
08/06/2009CA2715069A1 Novel heterocycles
08/06/2009CA2713553A1 Pyrazine derivatives and their use as protein kinase inhibitors
08/06/2009CA2712885A1 Substituted pyridazine derivatives which have histamine h3 antagonist activity
08/06/2009CA2712854A1 Cyclic indole-3-carboxamides, their preparation and their use as pharmaceuticals
08/06/2009CA2712352A1 Dicycloazaalkane derivates, preparation processes and medical uses thereof
08/05/2009EP2085395A1 Arylvinylazacycloalkane compounds and methods of preparation and use thereof
08/05/2009EP2085394A2 Metronidazole derivatives as antiparasitic agents
08/05/2009EP2085391A2 Inhibitors of factor XA and other serine proteases involved in the coagulation cascade
08/05/2009EP2084152A2 Substituted 4-imidazoles
08/05/2009EP2084151A1 Substituted dihydropyrazolones for treating cardiovascular and haematological diseases
08/05/2009EP2084148A1 Fungicide n-cycloalkyl-carboxamide, thiocarboxamide and n-substituted-carboximidamide derivatives
08/05/2009EP2084131A1 Indole and benzofuran 2-carboxamide derivatives
08/05/2009EP2083818A2 Melatonin derivatives and their use as antioxidants
08/05/2009EP1924560B1 6-substituted- 2,3,4,5-tetrahydro-1h-benzo[d]azepines as 5-ht2c receptor agonists
08/05/2009EP1877398B1 Quinazoline derivatives as egf and/or erbb2 tyrosine kinase inhibitors
08/05/2009EP1781606B1 Azetidine derivatives as ccr-3 receptor antagonists
08/05/2009EP1699454B1 Pyrazole derivatives and use thereof as orexin receptor antagonists
08/05/2009EP1631292B1 4-anilino-quinazoline derivatives as antiproliferative agents
08/05/2009EP1531822B1 1-aryl-4-substituted piperazine derivatives for use as ccr1 antagonists for the treatment of inflammation and immune disorders
08/05/2009EP1501797B1 3-(substituted amino)-1h-indole-2-carboxylic acid ester and 3-(substituted amino)-benzo[b]thiophene-2-carboxylic acid ester derivatives as interleukin-4 gene expression inhibitors
08/05/2009EP1491534B1 Novel hairpin polyamide
08/05/2009EP1465880B1 5-sulphanyl-4h-1,2,4-triazole derivatives and their use to treat disorders associated with somatostatine
08/05/2009EP1445253B1 4,4-difluoro-1, 2, 3, 4-tetrahydro-5h-1-benzazepine derivatives or salts thereof
08/05/2009EP1399116B1 Use of dicationic compounds for dyeing human keratinous fibres and compositions containing same
08/05/2009EP1357111B1 2-pyridone derivatives having affinity for cannabinoid type 2 receptor
08/05/2009EP1296974B1 2-cyanopyrrolidine derivatives and their use as medicaments
08/05/2009CN101501023A Phenyl substituted heteroaryl-derivatives and use thereof as anti-tumor agents
08/05/2009CN101501021A Muscarinic receptor agonists that are effective in the treatment of pain, alzheimer's disease and schizophrenia
08/05/2009CN101501008A Arylpiperazine derivatives and uses thereof
08/05/2009CN101501006A Pyridinone and pyridazinone derivatives as inhibitors of poly(ADP-ribose)polymerase (PARP)
08/05/2009CN101500995A 1-oxo-isoindoline compounds for the treatment of spinal muscular atrophy and other uses
08/05/2009CN101500994A 1,3-disubstituted 4-methyl-1h-pyrrole-2-carboxamides and their use for the manufacture of medicaments
08/05/2009CN101497607A Process for synthesizing sunitinib
08/05/2009CN100522960C Thioamide derivatives as progesterone receptor modulators
08/05/2009CN100522947C CCK-1 receptor modulators
08/05/2009CN100522161C (Indol-3-yl)-heterocycle derivatives as agonists of the cannabinoid CB1 receptor
08/04/2009US7569724 Antiproliferative agnets; anticancer agents; skin disorders
08/04/2009US7569700 Substituted, bicyclic 8-pyrrolidinobenzimidazoles, methods for their production and their use as medicaments
08/04/2009US7569689 Modulators of the glucocorticoid receptor, AP-1, and/or NF-κB activity and use thereof
08/04/2009US7569688 Propane-1, 3-dione derivative
08/04/2009US7569678 Protease inhibitor conjugates and antibodies useful in immunoassay
08/04/2009US7569592 Heteroaryl substituted pyrazole modulators of metabotropic glutamate receptor-5