Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
04/2009
04/23/2009CA2703425A1 Tetrazole derivatives as modulators of metabotropic glutamate receptors (mglurs)
04/23/2009CA2702930A1 Maleate salts of (e)-n-{4-[3-chloro-4-(2-pyridinylmethoxy)anilino]-3-cyano-7-ethoxy-6-quinolinyl}-4-(dimethylamino)-2-butenamide and crystalline forms thereof
04/23/2009CA2702898A1 Inhibitors of c-fms kinase
04/23/2009CA2702837A1 Piperidinyl and piperazinyl modulators of .gamma.-secretase
04/23/2009CA2702834A1 Substituted n-phenyl-pyrrolidinylmethylpyrrolidine amides and therapeutic use thereof
04/23/2009CA2702674A1 Heteroaryl compounds and uses thereof
04/23/2009CA2702563A1 Cgrp antagonists
04/23/2009CA2701792A1 Calcium receptor modulating agents
04/23/2009CA2697974A1 Trisubstituted 1,2,4-triazoles
04/22/2009EP2050745A1 N-pyridylpiperidine compound, method for producing the same, and pest control agent
04/22/2009EP2050744A1 Quinazoline derivatives as angiogenesis inhibitors
04/22/2009EP2050739A1 Quinazoline derivative
04/22/2009EP2050467A1 Therapeutic agent for amyotrophic lateral sclerosis
04/22/2009EP2050450A1 1-Piperidine-2-cyanoimino-1,3-dihydro-2H-benzimidazole derivatives as nociceptin analogs with ORL1 modulating activity for the treatment of pain
04/22/2009EP2049525A1 N-(aminoheteroaryl)-1h-indole-2-carboxamide derivatives, and preparation and therapeutic application thereof
04/22/2009EP2049523A1 Modulators of metabolism and the treatment of disorders related thereto
04/22/2009EP2049522A2 Hepatitis c virus inhibitors
04/22/2009EP2049521A2 Novel pyridazine derivatives
04/22/2009EP2049520A2 Indole compounds
04/22/2009EP2049519A2 Cyclic derivatives as modulators of chemokine receptor activity
04/22/2009EP2049518A2 Indazole and isoindole derivatives as glucokinase activating agents.
04/22/2009EP2049517A1 Amino-piperidine derivatives as cetp inhibitors
04/22/2009EP2049516A2 Pharmaceutical compounds
04/22/2009EP2049515A2 Triazolyl pyridyl benzenesulfonamides as ccr2 or ccr9 modulators for the treatment of atherosclerosis
04/22/2009EP2049514A1 Nitrate esters of piperidines
04/22/2009EP2049513A1 Pieridinyl substituted pyrrolidinones as inhibitors of 11-beta-hydroxysteroid dehydrogenase 1
04/22/2009EP2049502A1 2,4-substituted quinazolines as lipid kinase inhibitors
04/22/2009EP2049501A1 Hydroxylated and methoxylated cyclopenta [d] pyrimidines as akt protein kinase inhibitors
04/22/2009EP2049500A1 Cyclopenta [d] pyrimidines as akt protein kinase inhibitors
04/22/2009EP2049497A2 Pyrimidine derivatives as hsp90 inhibitors
04/22/2009EP2049486A2 Piperidinyl derivatives as modulators of chemokine receptor activity
04/22/2009EP2049484A1 Isoindoline derivatives for the treatment of arrhythmias
04/22/2009EP2049481A2 Novel compounds as antagonists or inverse agonists for opioid receptors
04/22/2009EP2049480A1 2-arylindole derivatives as npges-i inhibitors
04/22/2009EP2049478A1 Substituted n-phenylmethyl -5-oxo-proline-2-amides as p2x7-receptor antagonists and their methods of use
04/22/2009EP2049475A1 Cyclohexyl substituted pyrrolidinones as inhibitors of 11-beta-hydroxysteroid dehydrogenase 1
04/22/2009EP2049473A2 Substituted benzyl amine compounds
04/22/2009EP2049472A2 Cyclopropyl amine derivatives as histamin h3 receptor modulators
04/22/2009EP2049120A1 Urotensin ii receptor antagonists
04/22/2009EP2049116A2 Hepatitis c virus inhibitors
04/22/2009EP2049115A2 Alkyne-substituted pyridone compounds and methods of use
04/22/2009EP1934199B1 Indane derivatives as mch receptor antagonists
04/22/2009EP1931654B1 Modulators of metabolism and the treatment of disorders related thereto
04/22/2009EP1802572B1 Indol derivatives as inhibitors of soluble adenylyl cyclase
04/22/2009EP1718632B1 Pyrimidine derivatives as orexin receptor antagonists
04/22/2009EP1673354B1 Arylindenopyridines and arylindenopyrimidines and their use as adenosine a2a receptor antagonists
04/22/2009EP1628972B1 INDAZOLE-DERIVATIVES AS FACTOR Xa INHIBITORS
04/22/2009EP1592389B1 Piperazine-2-carboxamide derivatives
04/22/2009EP1587805B1 Pharmaceutical process and compounds prepared thereby
04/22/2009EP1507529B1 Combination comprising valsartan, amlodipine and hydrochlorothiazide
04/22/2009CN101415700A Active ingredient combinations with insecticidal properties
04/22/2009CN101415698A Fungicide n-cyclopropyl-sulfonylamide derivatives
04/22/2009CN101415687A Binding inhibitor of sphingosine-1-phosphate
04/22/2009CN101415683A New compounds
04/22/2009CN101415681A Pyridine and pyrimidine derivatives as mGluR2 antagonists
04/22/2009CN101415675A Inhibitors of the 11-beta-hydroxysteroid dehydrogenase type 1 enzyme
04/22/2009CN101415674A Pyrrolidine derivatives as ERK inhibitors
04/22/2009CN101412710A Omeprazole sodium compound and preparation thereof
04/22/2009CN101412709A Morpholinyl containing benzimidazoles as inhibitors of respiratory syncytial virus replication
04/22/2009CN101412692A 1-(3-amino propyl) piperidine-4-aminoamide compounds, and pharmaceutical composition, preparation and use thereof
04/22/2009CN100480248C Malonamide derivatives as gamma-secretase inhibitors
04/22/2009CN100480242C CDK-inhibitory pyrimidines, and production and use thereof as pharmaceutical agents
04/21/2009US7521562 Filters for electronic display devices
04/21/2009US7521561 Biphenyl-2-ylcarbamic acid 1-[2-(2-chloro-4-{[(R)-2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroquinolin-5-yl)ethylamino]methyl}-5-methoxyphenyl-carbamoyl)ethyl]piperidin-4-yl ester; beta 2 adrenergic receptor agonist and muscarinic receptor antagonist; bronchodilator agent; pulmonary disorders, asthma
04/21/2009US7521471 CB1cannabinoid receptor antagonists; e.g. 5-(4-chlorophenyl)-4-cyano-1-(2,4-dichlorophenyl)-N-piperidin-1-yl-1H-pyrazole-3-carboxamide; various psychological, neurodegenerative, pain and cardiovascular disorders
04/21/2009US7521464 drugs have beta-amyloid peptide production inhibitory activity, such as 2-(2-benzo[b]thiophen-4-yl-acetylamino)-N-(5-phenyl-2H-pyrazol-3-yl)-propionamide, useful for treatment of Alzheimer's disease and Down's Syndrome
04/21/2009US7521462 4-Amino-piperidine derivatives as monoamine uptake inhibitors
04/21/2009US7521455 Histamine H3 receptor antagonist or inverse agonist activity; metabolic diseases, circulatory diseases, or nervous system diseases; e.g. 3-(4-((1-cyclobutyl-4-piperidinyl)oxy)phenyl)-2-ethylpyrido(2,3-d)pyrimidin-4(3H)-one
04/21/2009US7521453 e.g. 5-Bromo-2-(3-methylisoxazol-5-ylmethylamino)-4-(5-cyclopropyl- 1H-pyrazol-3-ylamino)pyrimidine; anticarcinogenic, antitumor agents; breast, prostate, colon cancer
04/21/2009US7521451 e.g. 5,6-dimethyl-3a,4,7,7a-tetrahydro-2-benzofuran-1,3-dione;intravenous, water-soluble compounds useful for manufacturing an anasthetic, sedative agents; side effect reduction
04/21/2009US7521448 N-substituted benzimidazolyl c-Kit inhibitors
04/21/2009US7521447 2-aza-[4.3.0]bicyclic heteroaromatic rings; useful for the treatment of inflammation, osteoarthritis, rheumatoid arthritis, psoriasis, Crohn's disease, inflammatory bowel disease, cancer, autoimmune diseases, and for the treatment of other cytokine-mediated diseases
04/21/2009US7521445 Heterocyclic substituted carbonyl derivatives and their use as dopamine D3 receptor ligands
04/21/2009US7521396 processes for their preparation, and to their use as herbicides.
04/21/2009US7521062 Thiosemicarbazones as anti-virals and immunopotentiators
04/21/2009CA2499329C Indole-3-carboxamides as glucokinase (gk) activators
04/21/2009CA2362003C Heterocyclic urea and related compounds useful as anti-inflammatory agents
04/21/2009CA2356263C Aminopyrazole derivatives
04/21/2009CA2228038C 2(1h)-quinolone derivatives, their preparation and their use in therapy
04/21/2009CA2157855C Benzoylguanidines substituted by heterocyclic n-oxide, process for their preparation, their use as a medicament or diagnostic agent, medicament containing them and intermediate products for their preparation
04/16/2009WO2009049305A2 5- (2-hydroxyphenyl) tetrazoles as hsp90 inhibitors against cancer
04/16/2009WO2009049132A1 Quinoline derivatives for modulating dna methylation
04/16/2009WO2009048765A1 5-ht7 receptor antagonists
04/16/2009WO2009048752A2 Insecticidal substituted azinyl derivatives
04/16/2009WO2009048751A1 Insecticidal pyrimidinyl aryl hydrazones
04/16/2009WO2009048101A1 Amide compound
04/16/2009WO2009047775A2 Polymorphs of esomeprazole salts
04/16/2009WO2009047514A1 [1,2,4]triazolo[1,5-a]pyridine and [1,2,4]triazolo[1,5-c]pyrimidine compounds and their use
04/16/2009WO2009047359A1 Inhibitors of protein kinases
04/16/2009WO2009047264A1 Spiropyrrolidines and their use against hcv and hiv infection
04/16/2009WO2009047240A1 Indole derivatives useful as ppar activators
04/16/2009WO2009047161A1 Chiral cis-imidazolines
04/16/2009WO2009046804A1 Imidazole derivatives
04/16/2009WO2009046802A1 N- ( pyrazole- 3 -yl) -benzamide derivatives as glucokinase activators
04/16/2009WO2009046784A1 Pyridine derivatives useful as glucokinase activators
04/16/2009WO2009021965A3 Substituted quinoline derivatives as h1 receptor antagonists
04/16/2009WO2009010660A3 Substituted indazoles, the preparation thereof, and use of same in therapeutics
04/16/2009WO2008108380A3 Pyrrole compounds
04/16/2009WO2008103277A3 Nitrogen-containing heterocyclyl ketones and their use as c-met inhibitors
04/16/2009WO2008032072A8 2-benzimidaz0lyl-6-m0rph0lin0-4-piperidin-4-ylpyrimidine derivatives as pi3k and mtor inhibitors for the treatment of proliferative disorders