Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
06/2009
06/11/2009WO2007109871A3 Acridine derivatives with antitumoral activity
06/11/2009US20090149656 Optical determination of glucose utilizing boronic acid adducts
06/11/2009US20090149652 Affinity for somatostatin receptors; used for the treatment of acromegalia, hypophyseal adenomas or endocrine gastroenteropancreatic tumors including carcinoid syndrome; 4-(urea or thiourea substituted)-1-alkylpiperidines
06/11/2009US20090149651 Processes and intermediates for producing aminobenzimidazole ureas
06/11/2009US20090149528 Cinnamic acid amides
06/11/2009US20090149509 Peptidyl deformylase inhibitors used for inhibiting bacteria or preventing bacterial contamination of a cell culture medium; 2 (S)-hydroxy-3 (R)-[2 (S)-oxazol-2-yl-pyrrolidine-1-carbonyl)-heptanoic acid hydroxamide
06/11/2009US20090149505 Metabotropic Glutamate Receptor-Potentiating Isoindolones
06/11/2009US20090149504 Novel 5-Substituted Indole Derivatives As Dipeptidyl Peptidase IV (DPP-IV) Inhibitors
06/11/2009US20090149500 solid forms of lenalidomide, treating cancer, inflammatory disease, myelodysplastic syndrome, undesired angiogenesis
06/11/2009US20090149499 Polymorphic forms of 3-(4-amino-1-oxo-1,3 dihydro-isoindol-2-yl)-piperidine-2,6-dione)
06/11/2009US20090149493 Inhibitors of the interaction between mdm2 and p53
06/11/2009US20090149476 3-[[6-[4-(1,2,3,4-tetrahydro-1,8-naphthyridin-7-yl)-1-piperidinyl]-2,5-dimethyl-4-pyrimidinyl]amino]-N-[(phenylmethoxy)carbonyl]alanine, used for the treatment of osteoporosis, restenosis, arteriosclerosis, nephropathy or retinopathy
06/11/2009US20090149474 tert-butyl 4-[(4-chlorobenzoyl)amino]-2-(dimethylamino)-1-phenyl-1H-imidazole-5-carboxylate, used for the treatment of gastrointestinal disorders such as gastroesophageal reflux, irritable bowel syndrome, dyspepsia, diarrhea and for the inhibition of transient lower esophageal sphincter relaxations
06/11/2009US20090149472 Salts of substitutted pyrazoline compounds, their preparation and use and medicaments
06/11/2009US20090149469 Phenyl-[4-(3-phenyl-1h-pyrazol-4-yl)-pyrimidin-2-yl]-amine derivatives as igf-ir inhibitors
06/11/2009US20090149468 Substituted heterocyclic compounds and methods of use
06/11/2009US20090149467 Tyrosine Kinase Inhibitors
06/11/2009US20090149463 Therapeutic agents
06/11/2009US20090149460 New Compounds
06/11/2009US20090149459 P38 inhibitors and methods of use thereof
06/11/2009US20090149445 Tricyclic steroid hormone nuclear receptor modulators
06/11/2009US20090149444 Benzylamine analogues
06/11/2009US20090149440 1-(6-Amino-3,5-difluoropyridin-2-yl)-6-fluoro-7-(3-isopropylaminoazetidin-1-yl)-8-methyl-4-oxo-1,4-dihydroquinolin-3-carboxylic acid; antibacterial agent; low toxicity, improved bioavailability, and low binding rate to serum proteins
06/11/2009US20090149439 Pyridylmethysulfone derivative
06/11/2009US20090149415 Compounds for modulating the glycolysis enzyme complex and/or the transaminase complex
06/11/2009US20090148382 Technetium- and rhenium-bis(heteroaryl) complexes, and methods of use thereof
06/11/2009US20090145757 Redox Polymers
06/11/2009US20090144915 incorporation or grafting of hindered 4-aminopiperidines into a polyolefin, a styrene copolymer or an elastomer; stabilizers for protecting against oxidative, thermal, dynamic, light-induced or ozone-induced degradation; storage stability
06/11/2009CA2707989A1 Pyrazole derivatives and use thereof as inhibitors of cyclin dependent kinases
06/11/2009CA2707822A1 New compounds iii
06/11/2009CA2707722A1 Gamma secretase modulators
06/11/2009CA2707671A1 5,6-disubstituted oxindole-derivatives and use thereof for treating vasopressine-dependent diseases
06/11/2009CA2707669A1 5-halogen-substituted oxindole derivatives and use thereof for treating vasopressine-dependent diseases
06/11/2009CA2707667A1 Amidomethyl-substituted oxindole derivatives and the use thereof for the treatment of vasopressin-dependent illnesses
06/11/2009CA2707653A1 Diaminopyridines for the treatment of diseases which are characterised by excessive or anomal cell proliferation
06/11/2009CA2707651A1 1,2-disubstituted-4-benzylamino-pyrrolidine derivatives as cetp inhibitors useful for the treatment of diseases such as hyperli pidemia or arteriosclerosis
06/11/2009CA2707565A1 Renin inhibitors
06/11/2009CA2706420A1 Compounds for therapy and diagnosis
06/11/2009CA2705489A1 Pyridylmethyl-sulfonamide compounds
06/10/2009EP2067776A1 Piperidine compounds and pharmaceutical compositions containing them
06/10/2009EP2066659A1 Substituted sulfonamide derivatives
06/10/2009EP2066658A1 Pyridine- and quinoline-pyrimidine-derivatives
06/10/2009EP2066657A1 Substituted oxindole derivatives and their use as vasopressin and/or oxytocin receptor ligands
06/10/2009EP2066656A2 5-substituted quinazolinone derivatives as antitumor agents
06/10/2009EP2066655A2 Pyridinyl-pyrimidine derivatives useful as potassium channel modulating agents
06/10/2009EP2066654A1 N-(1-hetarylpiperidin-4-yl)(het)arylamides as ep2 receptor modulators
06/10/2009EP2066653A1 6-1h-imidazo-quinazoline and quinolines derivatives, new potent analgesics and anti-inflammatory agents
06/10/2009EP2066645A2 2 amino-pyrimidine derivatives as h4 receptor antagonists, processes for preparing them and their use in pharmaceutical compositions
06/10/2009EP2066637A1 Novel substituted bipyridine derivatives and their use as adenosine receptor ligands
06/10/2009EP2066636A1 5-phenyl-nicotinamide derivatives
06/10/2009EP2066630A1 Piperidine derivatives
06/10/2009EP2066318A2 Oxindole derivatives as anticancer agents
06/10/2009EP1805142A4 Novel pyridine compounds, process for their preparation and compositions containing them
06/10/2009EP1414797B9 Hepatitis c virus polymerase inhibitors with a heterobicylic structure
06/10/2009EP0976737B1 Pyrazole derivatives, process for preparing the same, intermediates, and pest control agent containing the same as active ingredient
06/10/2009EP0854870B1 Substituted imidazoles having anti-cancer and cytokine inhibitory activity
06/10/2009CN101454311A Salt of phenoxypyridine derivative or crystal thereof and process for producing the same
06/10/2009CN101454310A Inhibitors of 11-beta-hydroxysteroid dehydrogenase 1
06/10/2009CN101454309A Synthesis and uses of pyroglutamic acid derivatives
06/10/2009CN101454308A Process for preparing heterocyclic derivatives
06/10/2009CN101450939A Novel benzimidazoles compounds
06/10/2009CN101450938A 7-(4-oximido-3-amido-3-alkyl-1-piperidine)quinoline carboxylic acid derivates and preparation method thereof
06/10/2009CN101450934A Sulfonyl-derivatives as novel inhibitors of histone deacetylase
06/10/2009CN100497334C Indole derivatives useful as histamine h3 antagonists
06/10/2009CN100497333C Dihydrobenzodiazepin-2-one derivatives for the treatment of neurological disorders
06/10/2009CN100497332C Compound for preparing nifeviroc and its preparing process
06/10/2009CN100497331C 7-(4-oxime-3-amino-1-piperidine) quinoline carboxylic acid derivative and method for making same
06/10/2009CN100497314C Substituted 4-phenyltetrahydroisoquinolinium, process for their preparation, their use as a medicament, and medicament containing them
06/10/2009CN100497302C Diarylurea derivatives and their use as chloride channel blockers
06/09/2009US7544812 For example, 2-(4-{2-[1-(4-tert-Butyl-benzyl)-3-methyl-2-oxo-imidazolidin-4-yl]-ethoxy}-2-methyl-phenoxy)-2-methyl-propionic acid, 2-(4-{3-[1-(4-tert-Butyl-benzyl)-3-methyl-2-oxo-imidazolidin-4-yl]-propyl}-2-methyl-phenoky)-2-methyl-propionic acid; for treating diabetes mellitus
06/09/2009US7544807 Ionic liquids
06/09/2009US7544806 Piperidine-substituted indoles-or heteroderivatives thereof
06/09/2009US7544803 2-(2,2,2-Trifluoro-ethyl)-1,2,3,4-tetrahydro-isoquinoline-6-carboxylic acid quinolin-7-ylamides; treatment of acute, inflammatory and neuropathic pain, dental pain, general headache, migraine, cluster headache, mixed-vascular and non-vascular syndromes, arthritis, gastrointestinal disorders
06/09/2009US7544799 Crystal modification of a N-phenyl-2-pyrimidineamine derivative, processes for its manufacture and its use
06/09/2009US7544709 Derivatives of andrimide and moiramide B having antibacterial properties
06/09/2009US7544708 To treat diseases of respiratory, urinary and gastrointestinal systems; highly selective; significant potency; (2R,2S)(1 alpha ,5 alpha ,6 alpha )-N-{-[4-(1,3-dioxo-1,3-dihydro-isoindol-2-yl)-butyl]-3-azabicyclo[3.1.0]hex-6-yl-methyl}-2-hydroxy-2-cyclopentyl-2-phenylacetamide
06/09/2009US7544703 N-(3,5-Dimethylphenyl)-2-[2-(4-methylpiperazin-1-yl)pyridin-4-ylmethylthio]pyridine-3-carboxamide; 2-(2-Cyclopropylaminopyridin-4-ylmethylthio)-N-(3,5-dimethylphenyl)pyridine-3-carboxamide; cancer, rheumatoid arthritis, age-related macular degeneration, diabetic retinopathy, retinopathy of prematurity
06/09/2009US7544690 MCH receptor antagonists
06/09/2009US7544688 Hetereoaryl nitrile derivatives
06/09/2009US7544687 (2S)-3-{4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-ethoxy]-phenyl}-2-(4-m-tolyl-piperazin-1-yl)-propionic acid; hyperglycemia, dyslipidemia, type II diabetes mellitus; (2S)-2-[4-(4-nitro-benzenesulfonyl)-piperazin-1-yl]-3-{4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-ethoxy]-phenyl}-propionic acid;
06/09/2009US7544686 Piperazinylalkylpyrazole derivatives useful as selective T-type calcium channel blockers and preparation method thereof
06/09/2009US7544675 Chemical compounds with dual activity, processes for their preparation and pharmaceutical compositions
06/09/2009US7544312 Charge transport compositions and electronic devices made with such compositions
06/09/2009US7544215 Neutral and cationic naphthalene and colorants for keratin fibers containing these compounds
06/09/2009CA2583764C Thrombopoietin activity modulating compounds and methods
06/09/2009CA2424470C Treatment of gastrointestinal stromal tumors
06/09/2009CA2401812C Use of pdgf receptor tyrosine kinase inhibitors for the treatment of diabetic nephropathy
06/09/2009CA2162900C New peptide derivatives
06/04/2009WO2009070693A2 Modulators of ocular oxidative stress
06/04/2009WO2009070645A1 Indoles, derivatives, and analogs thereof and uses thereof
06/04/2009WO2009070116A1 A quinoline derivative acting as a p2x7-receptor antagonist
06/04/2009WO2009069736A1 Nitrogenated compound
06/04/2009WO2009069680A1 Medicinal composition for treating gastrointestinal stromal tumor (gist) and kit and method for estimating the prognosis of patient suffering from gastrointestinal stromal tumor
06/04/2009WO2009068652A1 2, 6-disubstituted pyridines and 2, 4-disubstituted pyrimidines as soluble guanylate cyclase activators
06/04/2009WO2009068552A1 Piperazinyl-sulfonamide derivatives useful in the treatment of gpr38 receptor mediated diseases
06/04/2009WO2009068512A1 2 -amino-pyrimidine derivatives as histamine h4 antagonists
06/04/2009WO2009068468A2 Pyridine compounds
06/04/2009WO2009068194A2 Halogen-substituted δ1 pyrrolines
06/04/2009WO2009045992A3 C-met protein kinase inhibitors
06/04/2009WO2009004427A3 Benzimidazole derivatives