Patents
Patents for C07D 333 - Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom (32,883)
11/2002
11/21/2002DE10123909A1 Production of ketone compounds useful in pharmacological applications, comprising reacting boronic acid derivatives with carboxylic acid anhydrides in presence of transition metal catalysts, based on palladium, nickel, platinum or copper
11/21/2002CA2447416A1 Substituted benzoylcyclohexenones and their use as herbicidal agents
11/21/2002CA2447314A1 Arginine derivatives
11/21/2002CA2447232A1 Method for producing ketones from carboxylic acid anhydrides
11/21/2002CA2447084A1 Benzamidoacetonitriles and their use as antiparasitics
11/21/2002CA2446797A1 Furan and thiophene derivatives that activate human peroxisome proliferator activated receptors
11/21/2002CA2446593A1 Carboxylic acid derivatives and pharmaceutical compositions comprising the same as an active ingredient
11/21/2002CA2445922A1 Estrogen receptor modulators
11/20/2002EP1258473A1 Benzoic acid derivatives, process for producing the same and drugs containing the same as the active ingredient
11/20/2002EP1257550A1 Platelet adp receptor inhibitors
11/20/2002EP1257264A1 Estrogen receptor modulators
11/20/2002EP1124832B1 Oxime derivatives and the use thereof as latent acids
11/20/2002EP1098645B1 Compositions comprising phenylaminothiophenacetic acid derivatives for the treatment of acute or adult respiratory distress syndrome (ards) and infant respiratory distress syndrome (irds)
11/20/2002EP1077966B1 Biphenyl sulfonyl aryl carboxylic acids useful in the treatment of insulin resistance and hyperglycemia
11/20/2002EP1047688B1 Thiophene nitrone compounds
11/19/2002US6482962 Contacting helminth, nematode, insect or acarid pests or parasites or their food supply, habitat or breeding grounds with a nitroethyl derivative
11/19/2002US6482958 Methods for the preparation of 4-hydroxy benzothiophene
11/19/2002US6482859 Microbicidal N-sulfonylglycin alkynyloxyphenethyl amide derivatives
11/19/2002US6482849 Inhibitors of α4β1 mediated cell adhesion
11/19/2002US6482822 N-(iminomethyl)amines derivatives, their preparation, their use as medicines and compositions containing them
11/14/2002WO2002090348A1 Sulfonamides
11/14/2002WO2002090345A1 3-hydroxymethylbenzo[b]thiophene derivatives and process for their preparation
11/14/2002WO2002090332A2 Novel aeylheteroalkylaminε derivatives
11/14/2002WO2002090330A1 Substituted 2-pyridine-cyclohexane-1,4-diamine derivatives
11/14/2002WO2002090317A1 Substituted cyclohexane-1,4-diamine derivatives
11/14/2002WO2002089801A1 Use of benzothiophenes to treat and prevent prostave cancer
11/14/2002WO2002089792A1 Sulfonamides
11/14/2002WO2002089791A2 Acne treatment with lipooxigenase inhibitors
11/14/2002WO2002089785A1 Sulfonamides
11/14/2002WO2002089783A1 Substituted cyclohexan-1,4-diamine derivatives with constipating and peripheral analgesic properties
11/14/2002WO2002089777A1 Improved transdermal therapeutic system for the treatment of parkinson's disese
11/14/2002WO2002089740A2 Sulfonamides
11/14/2002WO2002072524A3 Method for producing vinyl, aryl and heteroaryl acetic acids and derivatives thereof
11/14/2002WO2002064550A8 Glucocorticoid receptor modulators
11/14/2002WO2001035106A3 Methods for identifying and using amyloid-inhibitory compounds
11/14/2002US20020169203 Modulators of all three classes of calcium channel blocker subtypes (Small, Intermediate and Big conductance K channel (SK, IK and BK)) comprising malonate esters and nitriles; respiratory, brain, cardiovascular, urogenital disorders
11/14/2002US20020169197 Diaryl-enynes
11/14/2002US20020169188 Modulating neurotransmission in the central nervous system
11/14/2002US20020169184 Low molecular weight, non-peptide
11/14/2002US20020169164 Tricyclic sulfonamides and their derivatives as inhibitors of matrix metalloproteinases
11/14/2002CA2446735A1 Substituted cyclohexane-1,4-diamine derivatives with an anti-diarrhoea and peripheral analgesic action
11/14/2002CA2446365A1 Sulfonamides
11/14/2002CA2446120A1 Novel arylheteroalkylamine derivatives
11/14/2002CA2445634A1 Acne treatment comprising lipoxygenase inhibitors
11/14/2002CA2414298A1 3-hydroxymethyl-benzo[b]thiophene derivatives and process for making the same
11/13/2002EP1256576A1 Fused imidazolium derivatives
11/13/2002EP1256342A1 Hypoglycemics comprising organic zinc (ii) complexes
11/13/2002EP1256340A1 Improved transdermal therapeutic system for the treatment of Parkinson's disease
11/13/2002EP1255757A1 Amino acid derivatives and use thereof as nep, ace and ece inhibitors
11/13/2002EP1255553A2 Use of trilostane and its derivatives, optionally in combination with tamoxifen or raloxifene in the treatment of estrogen-dependent cancers e.g. breast, prostate and uterus cancers
11/13/2002EP1255543A2 Use of retinoid-type compounds as antibacterial agents
11/13/2002EP1187824B1 Novel (2-substituted-5 - 3-thienyl) -benzyl]- 2- ( 2-isopropoxy-5-fluoro] -phenoxy) -ethyl] -amine derivatives, method for the production and use thereof as medicaments
11/13/2002CN1379769A Novel composition and method or stabilizing same
11/13/2002CN1379762A Beta substituted metalloprotease inhibitors
11/13/2002CN1379754A Intermediates for making benzofuran or benzothiophene derivative nitrated in position 5 and uses thereof
11/12/2002US6479554 Immunotherapeutic agents
11/12/2002US6479552 Use of substituted N, N-disubstituted diamino compounds for inhibiting cholesteryl ester transfer protein activity
11/12/2002US6479550 α-sulfenimino acid derivatives
11/12/2002US6479528 Methods for inhibiting or reversing tau filament formation polymerization
11/12/2002US6479524 To prolong the thrombin time
11/12/2002US6479519 Inhibitors of cell adhesion; treatment of asthma or inflammatory bowel disease
11/12/2002US6479517 Treatment of post-menopausal syndrome: osteoporosis, cardiovascular effects such as hyperlipidemia, and estrogen-dependent cancer, particularly breast and uterine cancer
11/12/2002US6479492 Compounds which inhibit leukocyte adhesion mediated by VLA-4
11/12/2002US6479489 Substituted spiroheterocyclic 1H-3-arylpyrrolidine-2,4-dione derivatives, methods of preparing them and their use as pest-control agents
11/12/2002CA2324959C Phthalimido compounds as intermediates for producing substance p receptor antagonists
11/07/2002WO2002088274A1 Double-spiro organic compounds and electroluminescent devices
11/07/2002WO2002056827A3 Substituted felbamate derived compounds
11/07/2002WO2001036365A3 Thyroid receptor antagonists for the treatment of cardiac and metabolic disorders
11/07/2002US20020165398 Amino-thiophene-amido derivatives
11/07/2002US20020165393 Kinetic resolutions of chiral 2- and 3-substituted carboxylic acids
11/07/2002US20020165255 Prostaglandin agonists such as (3-(methanesulfonylamino-methyl)-phenoxy)-acetic acid methyl ester for preventing/ restoring bone mass loss
11/07/2002US20020165236 Such as 3-(3-(4-(4-sulfamoyl-benzylsulfamoyl-phenyl)-ureido)-benzamidine for treatment of malaria
11/07/2002US20020165232 Substituted N, N-disubstituted cycloalkyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
11/07/2002US20020165231 Substituted N-heteroaryl-N-phenyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
11/07/2002US20020165219 Novel heterocycles useful in the treatment of benign prostatic hyperplasia
11/07/2002US20020165218 Mixture of kinase inhibitor and anticancer agents
11/07/2002US20020165215 Organoselenium compounds for cancer chemoprevention
11/07/2002US20020165203 Enzyme inhibitors; antiinflammatory agents; rheumatic diseases; antidiabetic agents
11/07/2002US20020164726 Polyhydroxyalkanoate for use in culturing microorganisms
11/07/2002DE10121252A1 Behandlung der Akne Treatment of acne
11/06/2002EP1254895A1 Nitrogenous cyclic compounds and pharmaceutical compositions containing the same
11/06/2002EP1254136A1 FACTOR Xa INHIBITORS WITH ARYL-AMIDINES AND DERIVATIVES, AND PRODRUGS THEREOF
11/06/2002EP1254135A2 Aminoheterocyclylamides as pesticides and antiparasitic agents
11/06/2002EP1253917A2 Use of substituted 4-amino-1-phenylbutan-2-ol compounds as medicaments
11/06/2002CN1378527A Biaryl ether derivatives useful as monoamine reuptake inhibitors
11/06/2002CN1378450A Novel class of cytodifferentiating agents and histone deactylase inhibitors, and methods of use thereof
11/06/2002CN1377883A Cosmetic preparation containing light stable UV-A light filter agent
11/05/2002US6476264 N-(4-carbamimidoyl-phenyl)-glycine derivatives
11/05/2002US6476075 Use of substituted N, N-bis-benzyl aminoalcohol compounds inhibiting cholesteryl ester transfer protein activity
11/05/2002US6476064 Cyclopentane heptan(ene) acyl sulfonamide, 2-alkyl or 2-arylalkyl, or 2-heteroarylalkenyl derivatives as therapeutic agents
11/05/2002US6476057 Use of substituted N, N-disubstituted cycloalkyl aminoalcohol compounds for inhibiting cholesteryl ester transfer protein activity
11/05/2002US6476026 Compounds and compositions as protease inhibitors
11/05/2002US6476023 Aromatic heterocyclic compounds as anti-inflammatory agents
11/05/2002CA2038379C Trifluoromethyl mercaptan and mercaptoacyl derivatives and method of using same
11/05/2002CA2038029C 1-alkyl-, 1-alkenyl- and 1-alkynylaryl-2-amino-1,3-propanediols and related compounds, a process and intermediates for their preparation and theeir use as medicaments
10/2002
10/31/2002WO2002085838A1 Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds
10/31/2002WO2002085822A1 Compound for organic el element and organic el element
10/31/2002WO2002085301A2 Indole, azaindole and related heterocyclic amidopiperazine derivatives
10/31/2002WO2002069895A3 Heterocyclic analgesic compounds and methods of use thereof
10/31/2002WO2002026720A3 PIPERAZINE BASED INHIBITORS OF FACTOR Xa