Patents
Patents for C07D 333 - Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom (32,883)
01/2003
01/02/2003EP1109785B1 Indole derivatives and their use in the treatment of malignant and other diseases caused by pathological cell proliferation
01/02/2003EP0891341B1 1,3,4-oxadiazine derivatives and their use as pesticides
01/02/2003EP0804431B9 GLYCOPROTEIN IIb/IIIa ANTAGONISTS
01/02/2003EP0751939B9 Naphthylamides as central nervous system agents
01/02/2003EP0630366B1 Substituted heterocyclic derivatives useful as platelet aggregation inhibitors
01/01/2003CN1388119A Stereoselective preparation for chirality 1-aryl-and 1-heteroaryl-2-substituted-ethyl-2-amine
01/01/2003CN1097588C Dihydrobenzofuran and related compounds used as anti-inflammatory agents
12/2002
12/31/2002US6500865 Sulfonamide derivatives
12/31/2002US6500849 Administering antiinflammatory, antiproliferative, nootropic or antigrowth agents, such as 6-(1-dodecynyl)-2-pyridine-carboxaldehyde and enantiomorphs to mammals; alzheimers disease
12/31/2002US6500832 Administering enzyme inhibitors as viricides for prophylaxis of viral diseases such as aquired immune deficiency syndrome
12/31/2002US6500803 Factor VIIa inhibitors
12/27/2002WO2002102389A1 3, 7 or 3 and 7 thia or oxa prostanoic acid derivatives as agents for lowering intraocular pressure
12/27/2002WO2002082185B1 Perfluoroalkylsulfonic acid compounds for photoresists
12/27/2002WO2001023352A9 Preparation of sulfonyl imine compounds
12/26/2002US20020198383 For use in regioselective and enantioselective alkylations of allylic substrates
12/26/2002US20020198376 As therapeutic agents for autoimmune diseases such as rheumatoid arthritis
12/26/2002US20020198236 Small organic molecule regulators of cell proliferation
12/26/2002US20020198235 Use of benzothiopenes to treat and prevent prostate cancer
12/26/2002US20020198207 Novel Hexanoic acid derivatives
12/26/2002US20020198195 New oxybenzamide derivatives useful for inhibiting factor Xa or VIIa
12/26/2002US20020198184 Matrix metalloproteinase inhibitor is useful as an anticancer agent, angiogenesis inhibitor, a tumor cell infiltration inhibitor or a tumor metastasis inhibitor; inflammatory diseases, osteoarthritis, rheumatoid arthritis
12/26/2002US20020197558 Photoacid generators for use in photoresist compositions
12/25/2002CN1387518A Heterocyclic substd, diphenyl leukotriene antagonists
12/25/2002CN1387507A Diaryl-enynes
12/25/2002CN1097052C Process for production of amidinoindole derivs, and salts thereof
12/25/2002CN1097049C Processes for preparing intermediate product used in method of diastereoselective synthesis of nucleosides
12/24/2002US6498190 Bicyclic amino derivatives and PGD2 antagonist containing the same
12/24/2002US6498187 Fatty acid synthase inhibitors
12/24/2002US6498185 Enzyme factor xa inhibitors
12/24/2002US6498172 Prostaglandin agonists and their use to treat bone disorders
12/24/2002CA2150812C Catechol diethers as selective pde iv inhibitors
12/19/2002WO2002100851A2 Thiophene derivatives as antiviral agents for flavivirus infection
12/19/2002WO2002100849A2 Novel nitriles useful as reversible inhibitors of cysteine proteases
12/19/2002WO2002100846A1 Compounds and methods for the treatment or prevention of flavivirus infections
12/19/2002WO2002100830A1 Pyrrolidine derivatives as factor xa inhibitors
12/19/2002WO2002100825A2 Anthranilic acid amides with a heteroarylsulfonyl side chain, and use thereof as antiarrhythmic active substances
12/19/2002WO2002100822A1 Substituted sulfonamide compounds, process for their use as medicament for the treatment of cns disorders, obesity and type ii diabetes
12/19/2002WO2002100819A1 N-arylphenylacetamide derivatives and medicinal compositions containing the same
12/19/2002WO2002100813A2 Modulators of peroxisome proliferator activated receptors
12/19/2002WO2002100802A2 Fluorous triphase and other multiphase systems
12/19/2002WO2002100403A1 Modulators of peroxisome proliferator activated receptors (ppar)
12/19/2002WO2002100388A2 Cyclopentane heptan (ene) acyl sulfonamide, 2-alkyl or 2-arylalkyl, or 2-heteroarylalkenyl derivatives as therapeutic agents for the treatment of ocular hypertension
12/19/2002WO2002100344A2 Amino acid conjugates providing for sustained systemic concentrations of gaba analogues
12/19/2002WO2002100341A2 Compounds for the treatment of metabolic disorders
12/19/2002US20020193614 Treatment of cardiovascular disorders
12/19/2002US20020193596 Inhibitors of protein isoprenyl transferases
12/19/2002US20020193578 Compounds having activity as inhibitors of cytochrome P450RAI
12/19/2002US20020193383 1-(N-phenylalkylaminoalkyl)piperazine derivatives substituted at position 2 of the phenyl ring
12/19/2002US20020189033 Substituted 2-aminoalkyl-1,4diaminobenzene compounds and oxidation dye precursor compositions containing same
12/19/2002DE10128331A1 New 2-(heteroarylsulfonyl-amino)-benzamide derivatives, which are potassium ion channel blocking antiarrhythmic agents, useful for e.g. treating atrial fibrillation or flutter
12/19/2002CA2450220A1 Cyclopentane heptan (ene) acyl sulfonamide, 2-alkyl or 2-arylalkyl, or 2-heteroarylalkenyl derivatives as therapeutic agents for the treatment of ocular hypertension
12/19/2002CA2449629A1 Pyrrolidine derivatives as factor xa inhibitors
12/19/2002CA2449256A1 Modulators of peroxisome proliferator activated receptors
12/19/2002CA2448764A1 N-arylphenylacetamide derivatives and pharmaceutical compositions containing the same
12/19/2002CA2448552A1 Modulators of peroxisome proliferator activated receptors (ppar)
12/19/2002CA2445653A1 Substituted sulfonamide compounds, process for their use as medicament for the treatment of cns disorders, obesity and type ii diabetes
12/18/2002EP1266898A1 Processes for the production of thienopyrimidine derivatives
12/18/2002EP1265891A2 Novel lipoic acid heterocyclic or benzene derivatives, preparation and use thereof as medicines
12/18/2002EP1265865A2 Difluorobutyric acid derivatives and their use as metalloprotease inhibitors
12/18/2002EP1265857A1 Sulfonamide derivatives
12/18/2002EP1265855A1 Novel cd23 inhibitors
12/18/2002EP0934300B1 The preparation and use of ortho-sulfonamido heteroaryl hydroxamic acids as matrix metalloproteinase and tace inhibitors
12/18/2002CN1386124A Method of preparing a polymer, method of preparing a compound, compounds, polymers, and method for manufacturing and electronic device
12/18/2002CN1096446C N-(ortho-substd-benzyloxy)imine derivs, and their use as fungicides, acaricides or insecticides
12/17/2002US6495702 Process for preparing 5-hydroxybenzo [b] thiophene-3-carboxylic acid derivatives
12/17/2002US6495699 Antiarthritic agents; osteoporosis
12/17/2002US6495691 Their pharmaceutically acceptable salts, wherein the meaning of x is hydrogen, carboxyl, alkoxycarbonyl, aryloxycarbonyl, nitrile, or carbamoyl of the formula ticlopidine, is an antithrombotic drug with platelet aggregation inhibiting
12/17/2002US6495683 Herpes virus
12/17/2002US6495607 Benzocycloheptenes, process for their production, pharmaceutical preparations that contain the latter as well as their use for the production of pharmaceutical agents
12/17/2002US6495557 Condensed thienopyrimidines with phosphodiesterase-v inhibiting action
12/17/2002US6495554 Phosphodiesterase v inhibitors, treating cardiovascular disorders, and therapy of erectile dysfunction.
12/17/2002US6495552 Treatment or prevention of the diseases and conditions which respond to treatment by retinoids and or which in healthy mammals, including humans, are controlled by natural retinoic acid.
12/17/2002CA2064783C Cytoprotective fatty moiety compounds
12/12/2002WO2002098901A2 Peptide deformylase inhibitors
12/12/2002WO2002098870A1 Substituted oxime derivatives and the use thereof as latent acids
12/12/2002WO2002098851A1 Derivatives 0f n,s-substitutions n'-1 [(hetero)aryl] alkyl-n'-[hetero) aryl] methyl isothioureas, method for producing salts and bases thereof, physiologically active n,s-substitutions n'-1 [(hetero)aryl] alkyl-n'-[hetero) aryl] methyl isothioureas, a pharmaceutical composition and curing method
12/12/2002WO2002098850A2 Chemical compounds and pharmaceutical compositions as cathepsin s inhibitors
12/12/2002WO2002098849A2 Hydroxy alkyl amine derivatives as beta-secretase inhibitors and their use for the treatment of alzheimer’s disease and similar diseases
12/12/2002WO2002098848A1 Benzoylsulfonamides and sulfonylbenzamidines for use as antitumour agents
12/12/2002WO2002098840A1 Carboxylic acid derivative and medicine comprising salt or ester of the same
12/12/2002WO2002098420A1 4-substituted-1-(arylmethylidene)thiosemicarbazide, 4-substituted-1-(arylcarbonyl)thiosemicarbazide and analogs as activators of caspases and inducers of apoptosis and the use thereof
12/12/2002WO2002057252A3 Heterocyclic sulfonamide inhibitors of beta amyloid production
12/12/2002US20020188139 P-thienylbenzylamides as agonists of angiotensin-(1-7) receptors, and methods of their preparartion and use
12/12/2002US20020188136 Pesticides and herbicides
12/12/2002US20020188120 Such as 4-(4-methyoxy-benzenesulfonyl)-1-(3-phenyl-propyl)-piperidine-4-carboxylic acid hydroxyamide for treatment of arthritis, tumor metastasis, tissue ulceration, abnormal wound healing, periodontal disease, bone diseases, diabetes, and HIV
12/12/2002US20020188043 Photochromic diarylethene substituted with isoxazole group
12/12/2002US20020188017 Thienylazolylalkoxyethanamines, their preparation and their application as medicaments
12/12/2002US20020187982 Glucagon antagonists/inverse agonists
12/12/2002US20020187961 Omega-cycloalkyl 17-heteroaryl prostaglandin E2 analogs as EP2-receptor agonists
12/12/2002DE10205367A1 Verbindung mit Phenylacetylenstruktur, Flüssigkristallzusammensetzung, Polymer, optisch anisotropes Produkt, optisches oder Flüssigkristall-Element, Dibenzothiophenverbindung, Zwischenprodukt und Verfahren zum Herstellen derselben Compound with Phenylacetylenstruktur, liquid crystal composition, Polymer, optically anisotropic product, or the liquid crystal optical element, Dibenzothiophenverbindung, intermediate and process for producing same
12/12/2002CA2448834A1 Hydroxy alkyl amine derivatives as beta-secretase inhibitors and their use for the treatment of alzheimer's disease and similar diseases
12/12/2002CA2448418A1 Chemical compounds and pharmaceutical compositions as cathepsin s inhibitors
12/12/2002CA2446719A1 Benzoylsulfonamides and sulfonylbenzamidines for use as antitumour agents
12/11/2002EP1264820A1 Novel amide compounds
12/11/2002EP1263763A2 Tubulin binding ligands and corresponding prodrug constructs
12/11/2002EP1263743A1 Heterocycle substituted diphenyl leukotriene antagonists
12/11/2002EP1263714A1 Novel phenylheteroalkylamine derivatives
12/11/2002EP1263711A1 Novel use of phenylheteroalkylamine derivatives
12/11/2002EP0937064B1 Substituted oximes derivatives useful as neurokinin antagonists
12/11/2002EP0863891B1 (methylsulfonyl)phenyl-2-(5h)-furanones as cox-2 inhibitors