Patents
Patents for C07D 333 - Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom (32,883)
02/2004
02/24/2004US6696435 For treating atherosclerosis, other coronary artery diseases; 3-((3-(3-trifluoromethoxyphenoxy)phenyl)((3-(1,1,2,2-tetrafluoroethoxy) -phenyl)methyl) amino)-1,1,1-trifluoro-2-propanol for example
02/24/2004US6696216 Thiophene-containing photo acid generators for photolithography
02/24/2004US6696110 Liquid crystalline alkenyl compounds incorporating an heterocyclic five-membered ring
02/24/2004US6695978 Mono-, oligo- and polymers of benzo[b]thiophene and 2,2′-bisbenzo[b]thiophene and their use as charge transport materials
02/24/2004CA2279186C Sulfonyl urea derivatives and their use in the control of interleukin-1 activity
02/19/2004WO2004015024A1 Photochromic and electrochromic compounds and methods of synthesizing and using same
02/19/2004WO2004014867A2 Matrix metalloproteinase inhibitors and methods for identification of lead compounds
02/19/2004WO2004014847A1 Mcp-1 receptor antagonists and method of use thereof
02/19/2004WO2004014844A2 Aryl and heteroaryl compounds and methods to modulate coagulation
02/19/2004WO2004014843A1 Substituted amino compounds and use thereof
02/19/2004WO2004014842A1 Acylated arylcycloalkylamines and their use as pharmaceuticals
02/19/2004WO2004014825A1 Cannabinoid receptor ligands
02/19/2004WO2004014424A1 Releasable polymeric conjugates based on aliphatic biodegradable linkers
02/19/2004WO2004014381A2 Matrix metalloproteinase inhibitors and methods for identification of lead compounds
02/19/2004WO2004014372A1 Acylated, heteroaryl-condensed cycloalkenylamines and their use as pharmaceuticals
02/19/2004WO2003027234A9 Small organic molecule regulators of cell proliferation
02/19/2004US20040034231 Amidinophenyl-4-aminoacetic acid derivative is useful for treating diseases such as thrombosis, apoplexy, cardiac infarction, inflammation and arteriosclerosis, which are associated with coagulation factors xa, IXa and thrombin
02/19/2004US20040034219 Benzothiophene derivative compounds process of preparation and use thereof
02/19/2004US20040034103 Cdc25 photophatase inhibitors
02/19/2004US20040034034 Novel piperazine derivatives
02/19/2004US20040034025 Having a high residual activity, greater activity at lower application rates, curative activity, and a broader spectrum of efficacy; heterocyclic aromatic amides having a hydroxy group adjacent to the amide functionality
02/19/2004US20040033986 Anti tubercular drug: compositions and methods
02/19/2004DE10235206A1 Verfahren zur Herstellung von (S)-3-Methylmino-1-(thien-2-yl)propan-1-ol A process for the preparation of (S) -3-Methylmino-1- (thien-2-yl) propan-1-ol
02/19/2004CA2495067A1 Mcp-1 receptor antagonists and method of use thereof
02/19/2004CA2494920A1 Photochromic and electrochromic compounds and methods of synthesizing and using same
02/19/2004CA2494827A1 Cannabinoid receptor ligands
02/19/2004CA2493008A1 Aryl and heteroaryl compounds and methods to modulate coagulation
02/18/2004EP1389185A2 Aminoalcohol derivatives
02/18/2004EP1389176A1 Method for producing ketones from carboxylic acid anhydrides
02/18/2004EP1244655B1 Antithrombotic agents
02/18/2004EP1233952B1 Pesticidal n-heteroaryl alpha-alkoximino-carboxamides
02/18/2004EP1216238B1 Carboxylic acids and acylsulfonamides, compositions containing such compounds and methods of treatment
02/18/2004EP1178958B1 N-cyanomethyl amides as protease inhibitors
02/18/2004EP1171416B1 3-bicycloaryl-2-aminomethyl bicycloalkanes as serotonine reuptake inhibitors
02/18/2004EP0946166B1 Use of matrix metalloproteinase inhibitors for promoting wound healing
02/18/2004EP0918781B1 Asymmetric synthesis catalyzed by transition metal complexes with cyclic chiral phosphine ligands
02/18/2004CN1138780C Thienopyrimidines
02/18/2004CN1138772C Process for producing benzothiophenecarboxylic acid amide derivatives
02/18/2004CN1138771C 6-hydroxy-3-(4-[2-piperidine-1-group) oxyethyl group] phenoxy)-2-(4-methoxyphenyl) benzo[b] thiophene hydrochloride salt
02/18/2004CN1138770C 6-carbonyl-3-(4-[2-pierid-1-yl)elhoyl]phenoxy)-2-(4-methoxylphenyl) benzo[b] thiophene salt crystal
02/18/2004CN1138760C Preparation and use of ortho-sulfonamido bicyclic heteroaryl hydroxamic acids as matrix metalloproteinase and TACE inhibitors
02/17/2004US6693203 Reacting nopinone enolate with alkyl 7-halo-5-heptynoate, reacting product with hydroxylamine, treating with titanium trichloride and borane reagent, hydrogenating, reacting with 5-hydroxy-4-benzothiophenecarboxylic acid, hydrolyzing
02/17/2004US6693123 (4-(3-pyridylaminomethylene)-2-phenylbenzoyl)-n -methylmethionine, methyl ester for example; restenosis, hyperplasia
02/17/2004US6693117 Compounds with analgesic effect
02/17/2004US6693092 Herbicides; pesticides
02/12/2004WO2004013130A1 Substituted thienyl-hydroxamic acids as histone deacetylase inhibitors
02/12/2004WO2004013123A1 Method for the production of (s)-3-methylamino-1-(thien-2-yl)propan-1-ol
02/12/2004WO2004013122A2 Octupolar molecules used as organic semi-conductors
02/12/2004WO2004013094A2 Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds
02/12/2004WO2004013087A1 Anthranyl derivatives having an anticholecystokinin activity (anti-cck-1), a process for their preparation, and pharmaceutical use thereof
02/12/2004WO2004013080A1 Spirobifluorene derivatives, their preparation and uses thereof
02/12/2004WO2004012730A1 Improved transdermal delivery system for the administration of rotigotine
02/12/2004WO2003101381A3 1,2 diamido cycloalkyl sodium channel blockers
02/12/2004WO2003037916A3 Linear basic compounds having nk-2 antagonist activity and formulations thereof
02/12/2004WO2002100344A3 Amino acid conjugates providing for sustained systemic concentrations of gaba analogues
02/12/2004WO2002042289A8 Process for preparing 3-aryl-benzo[b]thiophenes
02/12/2004US20040030189 Compounds having fungicidal activity and processes to make and use same
02/12/2004US20040030181 Process for stereoselectively reducing 4-aryl-4-oxobutanoic acid derivatives
02/12/2004US20040030156 Substituted amino-furan-2-yl-acetic acid and amino-thien-2-yl-acetic acid derivatives and their use in the treatment of migraine and pain
02/12/2004US20040030141 Biphenyl derivatives substituted with an aromatic or heteroaromatic radical, and pharmaceutical and cosmetic compositions containing them
02/12/2004US20040030137 Novel heterocyclic amide derivatives and their use as dopamine D3 receptor ligands
02/12/2004US20040030132 Anticancer agents; arterosclerosis; bone disorders; antiarthritic agents; vision defects
02/12/2004US20040030131 Central nervous system disorders
02/12/2004US20040030054 Quaternary ammonium, phosphonium compound
02/12/2004US20040029945 Method of inhibiting matrix metalloproteinases
02/12/2004US20040029932 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
02/12/2004US20040029876 Acylamino cyclopropane derivatives
02/12/2004US20040029862 Alzheimer's disease
02/12/2004US20040029814 Cathepins inhibitor; antiinflammatory agents; antiarthritic agents
02/12/2004US20040029771 Methods for treating diseases related to intraocular pressure
02/12/2004DE10234188A1 Oktupolare Moleküle als organische Halbleiter Octupolar molecules as organic semiconductors
02/12/2004CA2494404A1 Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds
02/12/2004CA2494114A1 Substituted thienyl-hydroxamic acids as histone deacetylase inhibitors
02/12/2004CA2491366A1 Improved transdermal delivery system for the administration of rotigotine
02/11/2004EP1388537A1 Arginine derivatives
02/11/2004EP1388535A1 Acylated arylcycloalkylamines and their use as pharmaceuticals
02/11/2004EP1388529A2 Stable ethylene inhibiting compounds and methods for their preparation
02/11/2004EP1388342A1 Acylated, heteroaryl-condensed cycloalkenylamines and their use as pharmaceuticals
02/11/2004EP1387827A2 Synthesis of cyclopentadiene derivatives
02/11/2004EP1387821A2 Estrogen receptor modulators
02/11/2004EP0797567B1 Novel amino acid derivatives with improved multi-drug resistance activity
02/11/2004CN1474803A Novel amide derivatives and medicinal use thereof
02/11/2004CN1474689A CDC25 phosphatase inhibitors
02/11/2004CN1473814A Intemediate for preparing alkyl-dihalogeno phenyl substituted keto-enol
02/10/2004US6689801 Certain heteroaryl substituted thiol inhibitors of endothelin-converting enzyme
02/10/2004US6689786 Sulfonylurea, sulfonylthiourea, sulfonylguanidine, sulfonylcyanoguanidine and acylsulfonamide derivatives; antithrombotics
02/05/2004WO2004011452A1 Process for the preparation of 3-hydroxy-(2-thienyl)propanamines
02/05/2004WO2004011418A1 3,4-di-substituted cyclobutene-1, 2-diones as cxc-chemokine receptor ligands
02/05/2004WO2004011417A1 N-bisaryl- and n-aryl-cycloalkylidenyl-alpha-hydroxy-and alpha-alkoxy acid amides
02/05/2004WO2004011410A1 Chemical compounds
02/05/2004WO2004010987A2 Use of s1p receptor agonists in heart diseases
02/05/2004WO2003076388A3 Bis-aniline derivatives useful as potassium channels modulators
02/05/2004WO2003074475A3 Substituted aryl ketones
02/05/2004US20040024229 Production method for biarylalanine
02/05/2004US20040024190 Viral polymerase inhibitors
02/05/2004US20040024066 E.g., N-(2-(Benzo(b)thiophen-5-ylmethanesulfonyl)-1-(3,4-dichloro- phenyl)- ethyl)-N-hydroxyformamide; gene expression inhibitors of s-CD23; autoimmune disease; antiallergens; matrix metalloprotease enzyme inhibitors
02/05/2004US20040024059 Novel pleuromutilin derivatives
02/05/2004US20040024045 Glucagon antagonists/inverse agonists
02/05/2004US20040024019 Drug composition antagonistic to both pgd2/txa2 receptors
02/05/2004US20040023999 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof