Patents
Patents for C07D 333 - Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom (32,883)
04/2004
04/28/2004EP1412335A2 ENANTIOSELECTIVE TRANSFORMATION OF $g(a), $g(b)-UNSATURATED ALDEHYDES USING CHIRAL ORGANIC CATALYSTS
04/28/2004EP1412327A2 Inhibitors of protein kinase for the treatment of disease
04/28/2004EP1412325A1 Substituted sulfonamide compounds, process for their use as medicament for the treatment of cns disorders, obesity and type ii diabetes
04/28/2004EP1412324A2 Amino acid conjugates providing for sustained systemic concentrations of gaba analogues
04/28/2004EP1313724B1 N-heteroarylmethyl-p-phenylendiamine derivatives and compounds containing oxidation colouring agents
04/28/2004EP1263714B1 Novel phenylheteroalkylamine derivatives
04/28/2004EP1051394B1 Potassium channel inhibitors
04/28/2004EP1042313B1 Benzopyran and benzothiopyran derivatives having retinoid antagonist like activity
04/28/2004EP0403618B2 Methyl esters of aldimino- or ketimino-oxy-ortho-tolylacrylic acid, manufacturing process and fungicides containing them
04/28/2004CN1491937A 农药 Pesticide
04/28/2004CN1147461C 3-amino-3-aryl-1-alcohol derivatives and preparation and use thereof
04/28/2004CN1147459C Galcium receptor-active compound
04/27/2004US6727258 Allosteric adenosine receptor modulators
04/27/2004US6727255 Brain, nervous system and psychological disorders
04/27/2004US6727250 Administering compounds such as trans-3-(naphth-2-yl)-but-2-enoic acid-n-(2-carboxy-phenyl)-amide or like for therapy of conditions associated with increased telomerase activity, e.g. tumour diseases
04/27/2004US6727238 Sulfonylbenzene compounds as anti-inflammatory/analgesic agents
04/27/2004CA2136745C Heterocyclically disubstituted sulphonylamino(thio)carbonyl compounds
04/22/2004WO2004033419A1 Sulfonamides having antiangiogenic and anticancer activity
04/22/2004WO2004032871A2 Piperazine and piperazinone inhibitors of factor xa
04/22/2004WO2004026806A3 Diastereoselective method of preparing olefins by means of the horner-wadsworth-emmons reaction, comprising the addition of a tris-(polyoxaalkyl)-amine sequestering agent
04/22/2004WO2003082263A8 Sulfamic acids as inhibitors of human cytoplasmic protein tyrosine phosphatases
04/22/2004WO2003041728A9 Novel phenyl-propargylether derivatives
04/22/2004WO2002094794A8 4 (phenyl-piperazinyl-methyl) benzamide derivatives and their use for the treatment of pain anxiety or gastrointestinal disorders
04/22/2004US20040077905 Catalyst containing a Group VIII metal encapsulated in a polymer that has side chains containing an aromatic substituent; stable even in air, easy to recover, and reusable
04/22/2004US20040077896 Compounds for the treatment of metabolic disorders
04/22/2004US20040077867 Amine compounds, their production and use
04/22/2004US20040077864 A ketoxime of given formula, palladium as a reduction and racemization catalyst, lipase as a stereoselective acylation catalyst, an acyl donor, and a tertiary amine react in an organic solvent to provide a chiral amide which is hydrolyzed
04/22/2004US20040077854 4-chloro-N-((5-((4-(hexylamino)piperidin-1-yl)sulfonyl)thien-2 -yl)methyl)benzamide for example; JUN kinase inhibitors to treat nervous system disorders, cancer, cardiovascular and autoimmune disorders
04/22/2004US20040077630 Allosteric adenosine receptor modulators
04/22/2004US20040077502 Stable ethylene inhibiting compounds and methods for their preparation
04/22/2004DE10247226A1 New heteroaryl-substituted carboxylic acid amide derivatives, useful as factor Xa and factor VIIa inhibitors for e.g. treating thrombosis, myocardial infarction, arteriosclerosis, inflammation or tumors
04/22/2004CA2501520A1 Sulfonamides having antiangiogenic and anticancer activity
04/21/2004EP1409483A1 Arylsulfonamide derivatives as c-jun-n-terminal kinases (jnk's) inhibitors
04/21/2004EP1409476A1 Pharmaceutical compounds with serotonin receptor activity
04/21/2004EP1409468A2 Guanidinobenzamides as mc4-r agonists
04/21/2004EP1409450A1 N-(3-amino-2-hydroxy-propyl) substituted alkylamide compounds
04/21/2004EP1409440A1 A method to inhibit ethylene responses in plants
04/21/2004EP0904262B1 Conformationally restricted aromatic inhibitors of microsomal triglyceride transfer protein and method
04/21/2004CN1491221A Thiophene substituted amine derivatives as GLYT-1 inhibitors
04/21/2004CN1491207A Acylated indanyl amines and their use as pharmaceuticals
04/21/2004CN1491197A Tropolone derivative
04/21/2004CN1146542C Benzamide derivatives and their use as cytokine inhibitors
04/21/2004CN1146540C Novel compound with analgesic effect and use thereof
04/20/2004US6723857 Processes for the preparation of bicyclic aminoalcohols
04/20/2004US6723848 Method for producing benzo annelated heterocycles
04/20/2004US6723753 Substituted n-benzyl-n-phenyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
04/20/2004US6723752 (R)-chiral halogenated substituted n-benzyl-n-phenyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
04/20/2004US6723745 Prevention or treatment of autoimmune disease in warm blooded animal
04/20/2004US6723743 Treating patient suffering from rheumatoid arthritis, psoriasis, bronchial asthma, alzheimer's disease, myocardial infarction or atherosclerosis
04/15/2004WO2004031405A1 Substrates for o6-alkylguanine-dna alkyltransferase
04/15/2004WO2004031194A1 Process and intermediates for the preparation of the thienopyrrole derivatives
04/15/2004WO2004031193A1 Process and intermediates for the preparation of thienopyrrole derivatives
04/15/2004WO2004031169A1 Antibacterial agent having thiophene skeleton
04/15/2004WO2004031168A2 Processes and intermediates for the preparation of optically active 3-amino-1-(2-thienyl)-1-propanol derivatives
04/15/2004WO2004031139A1 Cyclohexyl sulphones as gamma-secretase inhibitors
04/15/2004WO2004031138A1 Novel sulphones for inhibition of gamma secretase
04/15/2004WO2004031137A1 Cyclohexyl sulphone derivatives as gamma-secretase inhibitors
04/15/2004WO2004031128A1 Improved method for the production of n-substituted amides from nitriles
04/15/2004WO2004031109A2 Chiral diols, their manufacture and ligands and catalysts derived therefrom
04/15/2004WO2004020445A3 4-(3,3-dihalo-allyloxy) phenol derivatives having pesticidal properties
04/15/2004WO2004018436A3 Compounds derived from aryl carbamates, preparation thereof and uses of same
04/15/2004WO2004010987A3 Use of s1p receptor agonists in heart diseases
04/15/2004WO2004005220A3 Method for asymmetric resolution of a racemic using diprogulic acid and use of said acid as asymmetric resolution agent
04/15/2004WO2003053359A3 1,3-bis-(substituted-phenyl)-2-propyn-1-ones and their use to treat disorders
04/15/2004WO2002083111A3 Imidazole, thiazole and oxazole derivatives and their use for the manufacture of a medicament for the treatment and/or prevention of pollakiuria or urinary incontinence
04/15/2004US20040072880 Cycloalkyl inhibitors of potassium channel function
04/15/2004US20040072878 2,3-Diphenylpropionic acid derivatives or their salts, medicines or cell adhesion inhibitors containing the same, and their usage
04/15/2004US20040072871 Novel thiophene derivatives, their process of preparation and the pharmaceutical compositions which comprise them
04/15/2004US20040072868 Liver disorders; anticholesterol agents; cardiovascular disorders
04/15/2004US20040072097 Photosensitive composition and acid generator
04/15/2004CA2501063A1 Substrates for o6-alkylguanine-dna alkyltransferase
04/15/2004CA2500969A1 Cyclohexyl sulphones as gamma-secretase inhibitors
04/15/2004CA2500966A1 Novel sulphones for inhibition of gamma secretase
04/15/2004CA2500145A1 Process and intermediates for the preparation of the thienopyrrole derivatives
04/15/2004CA2498843A1 Process and intermediates for the preparation of thienopyrrole derivatives
04/14/2004EP1408027A1 DIAMINE DERIVATIVE,PROCESS FOR PRODUCING THE SAME, AND BACTERICIDE CONTAINING THE SAME AS ACTIVE INGREDIENT
04/14/2004EP1406900A1 Novel compounds, their preparation and use
04/14/2004EP1406889A2 Interaction inhibitors of tcf-4 with beta-catenin
04/14/2004EP1406870A1 Taxol enhancer compounds
04/14/2004EP1406869A1 Taxol enhancer compounds
04/14/2004EP1406868A1 Synthesis of taxol enhancers
04/14/2004EP1406859A1 Substituted 4-aminocyclohexanol derivatives
04/14/2004EP1406858A1 Substituted 4-aminocyclohexanols
04/14/2004EP1406622A2 Dipeptidyl peptidase inhibitors for the treatment of diabetes
04/14/2004EP1406605A1 Carbamates of 2-heterocyclic-1,2-ethanediols
04/14/2004EP1305270B1 Kinetic resolutions of chiral 2- and 3-substituted carboxylic acids
04/14/2004CN1489576A Cannabinod receptor ligands
04/14/2004CN1489458A Inhibitors against the production and releaseof inflammator cytokines
04/13/2004US6720425 Alkyl or aryl substituted dihydronaphthalene derivatives having retinoid and/or retinoid antagonist-like biological activity
04/13/2004US6720338 Bcl-x1 inhibiting compositions and methods of promoting apoptosis in a mammal
04/13/2004US6720317 Inhibitors of factor Xa
04/08/2004WO2004029060A1 Novel herbicides, usage thereof, novel thienopyrimidine derivatives, intermediates of the same, and process for production thereof
04/08/2004WO2004029047A1 Derivative of dihydro-dibenzo (a) anthracenes and their use as selective estrogen receptor modulators
04/08/2004WO2004029046A2 Novel raloxifene acid addition salts and/or solvates thereof, improved method for purification of said raloxifene acid addition salts and/or solvates thereof and pharmaceutical compositions comprising these
04/08/2004WO2004029037A1 Novel aromatic sulfonium salt compound, photo-acid generator comprising the same and photopolymerizable composition containing the same, resin composition for optical three-dimensional shaping, and method of optically forming three-dimensional shape
04/08/2004WO2004029036A1 Novel method for the industrial synthesis of strontium ranelate and the hydrates thereof
04/08/2004WO2004029035A1 Novel method for the industrial synthesis of the methyl diester of 5-amino-3-carboxymethyl-4-cyano-2-thiophenecarboxylic acid and application of divalent salts of ranelic acid and the hydrates thereof in said synthesis
04/08/2004WO2004029034A1 Synthesis of thiophenecarboxylic acid esters for the production of ranelic acid salts
04/08/2004WO2003057225A3 Phosphate transport inhibitors
04/08/2004WO2003051276B1 Therapeutic heterocycles