Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005) |
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07/01/2010 | CA2740928A1 New retinoid derivatives endowed with cytotoxic and/or antiangiogenic properties |
06/30/2010 | EP2202222A2 Indene derivatives, their preparation and use as medicaments |
06/30/2010 | EP2201946A1 Pai-1 production inhibitor |
06/30/2010 | EP2200970A1 Aldehydes containing hydroxyl groups |
06/30/2010 | EP1735270B1 Diamino alcohols and their use as renin inhibitors |
06/30/2010 | CN101765585A antibacterial agents |
06/30/2010 | CN101759668A Cinnamamide derivative and application as cerebral nerve protective agent |
06/30/2010 | CN101759667A Preparation method of novel antidepressant moclobemide |
06/30/2010 | CN101759666A Preparation method of pinaverium bromide |
06/30/2010 | CN101759665A Substituent phenylpiperazine aryl alkanol derivant and application thereof in preparing analgesics |
06/30/2010 | CN101759633A Reagents for analyzing N-linked sugar chain |
06/30/2010 | CN101759604A Guanidyl substitutional tetracycline derivative |
06/30/2010 | CN101759599A Tetracycline compound with amino isonitroso |
06/30/2010 | CN101759598A Tetracycline compound with amino acid amidine |
06/29/2010 | US7745626 Stereoselective alkylation of chiral 2-methyl-4-protected piperazines |
06/29/2010 | US7745465 Antiischemic agents; antiinflammatory agents; antiallergens; autoimmune disease |
06/29/2010 | US7745464 heterocyclic compounds that bind to disease-related proteins, used for treating and modulating disorders associated with hyperproliferation, such as cancer |
06/29/2010 | US7745463 useful for the treatment of human immunodeficiency virus (HIV) and acquired immunodeficiency syndrome (AIDS) |
06/29/2010 | US7745456 2,5-bis{[alkyl(or aryl)imino]aminophenyl}furans and thiophenes; "reversed" amidines; DNA-binding affinities; microbiocide; mycobacterial, fungal, protozoal infection; Mycobacterium tuberculosis, Trypanosoma spp., Candida albicans, Aspergillus spp., Cryptosporidium parvum, Giardia lamblia, Plasmodium spp. |
06/29/2010 | US7745451 2,3-Difluoro-benzyl)-[6-(5-methyl-pyridin-2-yl)-5,6,7,8-tetrahydro-pyrido[4,3-d]pyrimidin-4-yl]-amine, useful for the prevention and treatment of pain, inflammation, cognitive disorders, anxiety and depression in humans |
06/29/2010 | US7745441 Urokinase inhibitors |
06/29/2010 | US7745439 Indene derivatives and process for the preparation thereof |
06/29/2010 | US7745436 Disalt inhibitors of IL-12 production |
06/29/2010 | US7745413 Collection of traceable compounds and uses thereof |
06/29/2010 | CA2442885C Sulphones which modulate the action of gamma secretase |
06/29/2010 | CA2442881C New process for the industrial synthesis of the tetraesters of 5-[bis(carboxymethyl)amino]-3-carboxymethyl-4-cyano-2-thiophenecarboxylic acid, and application to the synthesis ofbivalent salts of ranelic acid and their hydrates |
06/24/2010 | WO2010071567A1 (4-tert-butylpiperazin-2-yl)(piperazin-1-yl)methanone-n-carboxamide derivatives |
06/24/2010 | WO2010070615A1 Cysteine protease inhibitors |
06/24/2010 | WO2010070371A1 Process for the preparation of piperazine derivatives |
06/24/2010 | WO2010070370A1 Process for the preparation of piperazine compounds and hydrochloride salts thereof |
06/24/2010 | WO2010070369A1 Piperazine salt and a process for the preparation thereof |
06/24/2010 | WO2010069758A1 Polymerizable photoinitiators and radiation curable compositions |
06/24/2010 | US20100160343 Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by vla-4 |
06/24/2010 | US20100160341 Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by vla-4 |
06/24/2010 | US20100160331 Novel carbamoyloxy arylalkan arylpiperazine compound, pharmaceutical compositions comprising the compound and method for treating pain, anxiety and depression by administering the compound |
06/24/2010 | US20100160289 Sulfonamides as trpm8 modulators |
06/24/2010 | US20100158996 Ester compound and medical use thereof |
06/24/2010 | US20100158818 Antimicrobial n-chlorinated compositions |
06/24/2010 | CA2746990A1 (4-tert-butylpiperazin-2-yl)(piperazin-1-yl)methanone-n-carboxamide derivatives |
06/24/2010 | CA2744888A1 Cysteine protease inhibitors |
06/24/2010 | CA2744073A1 Process for the preparation of piperazine compounds and hydrochloride salts thereof |
06/24/2010 | CA2743924A1 Piperazine salt and a process for the preparation thereof |
06/23/2010 | EP2199282A1 Amide compound |
06/23/2010 | EP2199273A1 Polymerizable photoinitiators and radiation curable compositions |
06/23/2010 | EP2197830A2 Method for producing amines from sugar alcohols |
06/23/2010 | CN1906155B Novel hydroxamic acid ester derivant and pharmaceutical use thereof |
06/23/2010 | CN101754958A Method for the production of highly pure 2,4'-dimethyl-3-piperidino-propiophenone (tolperisone), pharmaceutical compositions containing the same, and agent formulations containing tolperisone |
06/23/2010 | CN101747295A Methanesulfonic acid cinepazide crystal form and preparation method |
06/23/2010 | CN101747294A Method for purifying N-(2,6-xylyl)-2-(1-piperazinyl)acetamide |
06/23/2010 | CN101747293A Naftopidil preparing method |
06/23/2010 | CN101747292A Benzoylguanidine-trimetazidine conjugate, as well as preparation method and medical application thereof |
06/23/2010 | CN101747243A Ionic liquid prepared through diimine (vikane) and (perfluoroalkglsulfonyl fluorosulfonyl group) imine alkali salt |
06/23/2010 | CN101161645B Urea derivatives as well as preparation method and uses thereof |
06/22/2010 | US7741480 Process for the preparation of linezolid and related compounds |
06/22/2010 | US7741328 Treating inflammatory diseases such as rheumatoid arthritis, multiple sclerosis or Crohn's disease; Very Late Antigen-4 (VLA-4), also called alpha 4 beta 1 integrin; N-(sulfonamido-substituted pyrimidyl, pyridyl or pyrazyl)-L-4-(N,N-dimethylcarbamyloxy)phenylalanine compounds |
06/22/2010 | US7741323 6-methoxy-1-(trans-methylimino-N-oxy)-3-phenyl-1H-indene-2-carboxylate ethyl ester, used for selectively modulating the activities of peroxisome proliferator activated receptors; excellent effect in lowering both blood glucose and insulin levels; side effect reduction |
06/22/2010 | US7741318 used for treating central nervous system diseases such as depression, cognitive diseases and neurodegenerative diseases such as Parkinson's disease, alzheimer's disease or psychoses, and stroke |
06/22/2010 | US7741316 Pharmacological uses of azetidine derivatives |
06/22/2010 | CA2541131C Derivatives of piperazine, process for their preparation and pharmaceutical compositions containing them |
06/22/2010 | CA2441398C Lipid lowering biphenylcarboxamides |
06/22/2010 | CA2420996C Substituted heterocyclic compounds for treating multidrug resistance |
06/22/2010 | CA2315715C Inhibition of p38 kinase using symmetrical and unsymmetrical diphenyl ureas |
06/17/2010 | WO2010066010A1 Process for the preparation of asymmetrical bis(thiosemicarbazones) |
06/17/2010 | US20100152220 Indene derivatives as pharmaceutical agents |
06/17/2010 | US20100150836 Radiolabelled benzamide analogues, their synthesis and use in diagnostic imaging |
06/17/2010 | CA2746070A1 Process for the preparation of asymmetrical bis(thiosemicarbazones) |
06/16/2010 | EP2195293A2 Cycloptopyl amide derivatives |
06/16/2010 | CN1993337B Method for improving a piperazine colour stability |
06/16/2010 | CN1839124B Succinate and malonate salt of trans-4-(1R,3S)-6-chloro-3-phenylindan-1-yl)-1,2,2-trimethylpiperazine and the use as a medicament |
06/16/2010 | CN101735173A Heavy metal chelating agent and preparation method thereof |
06/16/2010 | CN101735172A Cinepazide monohydrate, crystal forms and preparation method thereof |
06/16/2010 | CN101735113A Urea derivatives, preparation method and use thereof |
06/16/2010 | CN101735102A Method for synthesizing 2,2-disubstituted acetaldehyde hydrazone at room temperature under low pressure by taking acetylene as raw material |
06/16/2010 | CN101735090A Process for preparing secondary amides by carbonylation of a corresponding tertiary amine |
06/16/2010 | CN101735079A Derivative of beta-amine methyl cyclopentanol and cyclopentyl ester, preparation method and application thereof |
06/16/2010 | CN101177420B Method for intermittent azeotropic rectifying separating N-ethylpiperazine-ethanolamine |
06/15/2010 | US7737286 α-Hydroxy-benzeneacetic acid derivatives, and compounds having two 5-membered latone rings fused to central cyclohexa-1,4-diene nucleus based upon the same, and uses of the compounds |
06/15/2010 | US7737283 Urea substituted with a 5 member nitrogen-containing ring; biological conjugated drug used to modulate of the activation state of p38 kinase protein; antiinflammatory agents; rheumatoid arthritis, asthma, sepsis, toxic shock syndrome, adult respiratory distress syndrome, stroke, reperfusion injury |
06/15/2010 | US7737143 such as 6-(1H-Benzimidazol-1-yl)-N-benzylpyrazin-2-amine, used as antidiabetic, anticarcinogenic and antiarthritic agents or for treating autoimmune diseases |
06/15/2010 | US7737142 (Thio) carbamoyl-cyclohexane derivatives as D3/D2 receptor antagonists |
06/15/2010 | CA2441309C Biguanide derivatives |
06/15/2010 | CA2328440C Heterocyclically substituted amides used as calpain inhibitors |
06/10/2010 | WO2010065801A1 Amine substituted piperazine melanocortin receptor-specific compounds |
06/10/2010 | WO2010065512A2 Compounds for treating proliferative disorders |
06/10/2010 | WO2010064631A1 Photobase generator |
06/10/2010 | WO2010063774A1 Novel 4-(azacycloalkyl)benzene-1,3-diol compounds as tyrosinase inhibitors, process for the preparation thereof and use thereof in human medicine and in cosmetics |
06/10/2010 | WO2010063403A2 Radioisotope-labeled lysine and ornithine derivatives, their use and processes for their preparation |
06/10/2010 | WO2010044940A3 2,5-linked polyfluorenes for optoelectronic devices |
06/10/2010 | WO2010043976A3 Highly pure ranolazine or a pharmaceutically acceptable salt thereof |
06/10/2010 | WO2009147170A3 Drug combinations comprising a dgat inhibitor and a ppar-agonist |
06/10/2010 | US20100145048 Compounds for the treatment of inflammatory disorders |
06/10/2010 | US20100144720 Inhibitors of human tumor-expressed ccxckr2 |
06/10/2010 | US20100144588 Proton acceptor iminium/carbocation-type coupling agents |
06/10/2010 | US20100143455 Triazole antifungal agents |
06/10/2010 | CA2745364A1 Radioisotope-labeled lysine and ornithine derivatives, their use and processes for their preparation |
06/10/2010 | CA2745065A1 Compounds for treating proliferative disorders |
06/10/2010 | CA2744711A1 Bcl-2-selective apoptosis-inducing agents for the treatment of cancer and immune diseases |
06/10/2010 | CA2744708A1 Apoptosis-inducing agents for the treatment of cancer and immune and autoimmune diseases |
06/10/2010 | CA2742709A1 Novel 4- (azacycloalkyl) benzene-1,3-diol compounds as tyrosinase inhibitors, process for the preparation thereof and use thereof in human medicine and in cosmetics |
06/09/2010 | EP2049508B1 N-hydroxy-3-(4-{3-phenyl-3-oxo-propenyl}-phenyl)-acrylamide derivatives and related compounds as histone deacetylase inhibitors for the treatment of cancer |