| Patents for C07D 277 - Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings (33,621) |
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| 10/16/2008 | US20080255123 (2Z)-2-(3-butyl-4,5-dimethyl-1,3-thiazol-2(3H)-ylidene)-1-(5-chloro-2-methoxyphenyl)ethanone; antiinflammatory, analgesic agent; autoimmune diseases; neuroprotectants |
| 10/16/2008 | US20080255108 Novel thiophene sulfoximines, compositions thereof, and methods of treating complement-mediated diseases and conditions |
| 10/16/2008 | US20080255095 Benzylamine analogues |
| 10/16/2008 | US20080255094 Thiazolidine carboxamide derivatives as modulators of the prostaglandin f receptor |
| 10/15/2008 | EP1979335A2 Thiazoles as 11 beta-hsd1 inhibitors |
| 10/15/2008 | EP1979334A1 Novel benzamidine derivatives, process for the preparation thereof and pharmaceutical composition comprising the same |
| 10/15/2008 | EP1979322A1 Cyclohexyl sulfonamide derivatives having h3 receptor activity |
| 10/15/2008 | EP1979320A2 PIPERAZINES AND PIPERIDINES AS mGluR5 POTENTIATORS |
| 10/15/2008 | EP1692124B1 Biaryl sulfonamides as mmp inhibitors |
| 10/15/2008 | EP1567112B1 THIAZOLIDIN-4-ONES FOR INHIBITING hYAK3 PROTEINS |
| 10/15/2008 | EP1476423B1 Arylsulfonamidobenzylic compounds |
| 10/15/2008 | EP1375486B1 Nitrogen-containing heteroaryl compounds having hiv integrase inhibitory activity |
| 10/15/2008 | EP1308436B1 Calcium receptor antagonists |
| 10/15/2008 | EP1142872B1 Aromatic heterocycle compounds having hiv integrase inhibiting activities |
| 10/15/2008 | CN101287718A Substituted heteroaryl- and phenylsulfamoyl compounds |
| 10/15/2008 | CN101284865A New compound and its medicine use |
| 10/15/2008 | CN101284810A Cyano-pyrrolidine and cyano-tetrahydrothiazole derivates |
| 10/15/2008 | CN100425600C Benzothiazole- and benzoxazole-4,7-dione derivatives and their use as CDC25 phosphatase inhibitors |
| 10/15/2008 | CN100425594C PPAR-activating compound and pharmaceutical composition comprising the compound |
| 10/14/2008 | US7435828 immunosuppressive agents; low dosages; 5-[4-(2-hydroxy-ethoxy)-benz[Z]ylidene]-2-([Z]-isopropylimino)-3-o-tolyl-thiazolidin-4-one |
| 10/14/2008 | US7435815 Sulfonylamino-acetic acid derivatives |
| 10/14/2008 | CA2382880C N-cyclopentyl modulators of chemokine receptor activity |
| 10/09/2008 | WO2008121558A1 1, 3-thiazol-2 (3h) -ylidene compounds as cannabinoid receptor ligands |
| 10/09/2008 | WO2008120744A1 Five-membered cyclic amide compound and use thereof |
| 10/09/2008 | WO2008119238A1 Substituted five membered heterocycle compounds, preparation method and medical use thereof |
| 10/09/2008 | WO2008062276A8 Acetylene derivatives as stearoyl coa desaturase inhibitors |
| 10/09/2008 | US20080249130 Oral dosage forms; antiproliferatives, anticholesterol agents; lipid metabolic disorders; myocardial infarction, stroke, restenosis, atherosclerosis |
| 10/09/2008 | US20080249093 immunosuppressive, anti-inflammatory and hemostatic agents to modulate leukocyte trafficking, sequestering lymphocytes in secondary lymphoid tissues, and enhancing vascular integrity; safer and more effective; 3-(4-(5-(3-Cyano-4-isopropyloxyphenyl)-1,2,4-oxadiazol-3-yl)-3-methylphenyl)propanoic acid |
| 10/09/2008 | US20080249071 inhibitory activity against the activation of inflammatory cytokines such as interleukin (IL)-1, IL-6, IL-8 and tumor necrosis factor (TNF- alpha ), NF- kappa K B; inflammatory disorders, autoimmune diseases; side effects reduction; immuno suressants; N-[3,5-bis(trifluoromethyl)phenyl]-2-hydroxybenzamide |
| 10/09/2008 | CA2681586A1 1, 3-thiazol-2 (3h) -ylidene compounds as cannabinoid receptor ligands |
| 10/08/2008 | EP1977749A1 Use of cyclooxygenase-2 inhibitors in the treatment and prevention of neoplasia |
| 10/08/2008 | EP1976839A2 Compounds and methods for modulating protein trafficking |
| 10/08/2008 | EP1976835A2 Histone deacetylase inhibitors |
| 10/08/2008 | EP1697316B1 Novel intermediates for the synthesis of (r)-tamsulosin and of its pharmaceutically acceptable salts and process for their preparation |
| 10/08/2008 | EP1660493B1 Peptidyl heterocyclic ketone derivatives and preparation processes |
| 10/08/2008 | EP1606351A4 Cyanine dye labelling reagents with meso-substitution |
| 10/08/2008 | CN101282957A 新的药物化合物 New pharmaceutical compounds |
| 10/08/2008 | CN101282950A Novel benzothiazolone derivatives |
| 10/08/2008 | CN101282949A Azole and thiazole derivatives and their use |
| 10/08/2008 | CN101282937A Therapeutic agents |
| 10/08/2008 | CN101282920A Fluorination process of anilide derivatives and benzothiazole fluorinate derivatives as in vivo imaging agents |
| 10/07/2008 | US7432392 Ester derivatives and medical use thereof |
| 10/07/2008 | US7432389 Inhibiting beta-secretase enzyme activity and A beta peptide production, to reduce amyloid beta deposits or plaques |
| 10/07/2008 | US7432289 5-Acylamino-1,1′-biphenyl-4-carboxamide derivatives and their use as P38 kinase inhibitors |
| 10/07/2008 | US7432287 e.g. 3-(6-ethanesulfonylpyridin-3-yloxy)-5-(2-hydroxy-1-methyl-ethoxy)-N-(1-methyl-1H-pyrazol-3-yl)benzamide; glucokinase activator; antidiabetic agent; obesity, insulin resistance |
| 10/07/2008 | US7432281 4-(2,2-dichloro)-N-(quinolin-3-yl)benzamide; (1R,2R)2-methyl-N-(quinolin-3-yl)-4-(2-(trifluoromethyl)cyclopropyl)benzamide; inflammation-related conditions in mammals, arthritis, Parkinson's/Alzheimer's diseases, stroke, asthma; acute/chronic or neuropathic pain; VR1 agonist/antagonist |
| 10/07/2008 | US7432254 Method for treating glaucoma IC |
| 10/07/2008 | US7431741 Brightening colorant with indolythiazolium dyes |
| 10/02/2008 | WO2008118122A2 Compounds and amyloid probes thereof for therapeutic and imaging uses |
| 10/02/2008 | WO2008020211A3 Benzimidazole, benzoxazole and benzothiazole derivatives, optical film comprising them and method of production thereof |
| 10/02/2008 | US20080242869 Tri(Cyclo) Substituted Amide Compounds |
| 10/02/2008 | US20080242868 Process for preparing epothilone derivatives by selective catalytic epoxidation |
| 10/02/2008 | US20080242709 2-amido-4-isoxazolyl thiazole compounds exhibiting atp-utilizing enzyme inhibitory activity, and compositions, and uses thereof |
| 10/02/2008 | US20080242708 Fungicides/bactericides for plant protection; exhibit a strong fortifying effect in plants; for controlling cereal diseases against Puccinia species, and diseases in viticulture and fruit and vegetable production against Botrytis, Venturia or Alternaria species; low toxicity; tolrerance |
| 10/02/2008 | US20080242671 Selective in presence of at least one other cathepsin isozyme; such as N-{-2-[2-(4-methoxy-phenylamino)-ethylcarbamoyl]-cyclohexyl}-3-methyl-benzamide |
| 10/02/2008 | US20080242656 N-Substituted-N-Sulfonylaminocyclopropane Compounds and Pharmaceutical Use Thereof |
| 10/02/2008 | US20080242654 Novel compounds as cannabinoid receptor ligands |
| 10/02/2008 | CA2677991A1 Thiazolidine derivatives |
| 10/01/2008 | EP1973890A2 Indane modulators of glucocorticoid receptor, ap-1, and/or nf-kb activity and use thereof |
| 10/01/2008 | EP1973875A1 Compounds and methods for inhibiting the interaction of bcl proteins with binding partners |
| 10/01/2008 | EP1973404A1 Malononitrile compounds |
| 10/01/2008 | EP1496877B1 Method and composition for treatment of diabetes, hypertension, chronic heart failure and fluid retentive states |
| 10/01/2008 | CN101277933A Substituted propylamine derivatives and methods of their use |
| 10/01/2008 | CN101274920A Bis(2-benzothiazolydiazoamino)-biphenyl, preparation and application thereof |
| 10/01/2008 | CN101274919A 1,8-bis(2-benzothiazolydiazoamino)- naphthaline, preparation and application thereof |
| 10/01/2008 | CN101274918A Substitutive five membered heterocyclic compound, preparation and medical use thereof |
| 10/01/2008 | CN100422185C Novel derivatives of cycloalcanodiones, method for the production thereof and their pharmacological applications |
| 10/01/2008 | CN100422179C 2-amino-5-benzoylthiazole npy antagonists |
| 10/01/2008 | CN100422163C Compound for preparing fluorescein and its preparation method |
| 09/30/2008 | US7429659 Isopropyl-piperazin-1-yl)-(5-piperidin-1-ylmethyl-furan-2-yl)-methanone; 5-(4-Fluoro-piperidin-1-ylmethyl)-furan-2-yl]-(4-isopropyl-piperazin-1-yl)-methanone, fumarate salt; insomnia, attention deficit hyperactivity disorders, learning disorders, cognitive dysfunction, eating disorders, obesity |
| 09/30/2008 | US7429618 substituted triarylmethane compounds for immunosuppressive treatment of autoimmune disorders or inflammatory diseases; [Tris-(4-fluoro-phenyl)-methyl]-phosphonic acid dimethyl ester; Gardos channel antagonists |
| 09/30/2008 | US7429587 e.g. 2-(4-Chlorophenyl)-N-{(3S)-1-[(1S)-1-methyl-2-morpholin-4-yl-2-oxoethyl]-2-oxopyrrolidin-3-yl}ethenesulfonamide; blood coagulation factor and trypsin-like serine protease inhibitor; anticoagulant, antiinflammatory agent; atherosclerotic plaque, myocardial infarction and unstable angina |
| 09/30/2008 | US7429586 Non-imidazole aryloxyalkylamines |
| 09/30/2008 | US7429278 N-(2-Thiophen-2-ylethyl)benzene-1,4-diamine; hair dye; very strong and sparingly selective coloration of keratin fibers, light fast, avoiding the degradation of the fibers |
| 09/30/2008 | US7429274 Agent and method for the oxidative coloring of keratin fibers |
| 09/30/2008 | CA2381001C Carbamate derivative and agricultural/horticultural fungicide |
| 09/30/2008 | CA2355470C Benzoheterocycles and their use as mek inhibitors |
| 09/25/2008 | WO2008115433A1 Desferrithiocin polyether analogues |
| 09/25/2008 | WO2008115141A1 4, 5-dihydro-1,3-thiazol-2-amine derivatives and their use in the treatment of respiratory, cardiovascular, neurological or gastrointestinal disorders |
| 09/25/2008 | WO2008113760A2 Arylsulphonyglycine derivatives as suppressors of the interaction of glycogen phosphorylase a with the gl subunit of glycogen-associated protein phosphatase 1 (ppl) for the treatment of metabolic disorders, particulary diabetes |
| 09/25/2008 | WO2008113255A1 Benzamide derivatives with anti-proliferative activity, pharmaceutical preparations thereof |
| 09/25/2008 | WO2007146349A3 Cgrp receptor antagonists |
| 09/25/2008 | US20080234344 Amino Acid and Peptide Conjugates of Arylalkylic Acids for Cosmetic Use |
| 09/25/2008 | US20080234292 Such as S)-(1-(1-Aminobicyclo[2.2.2]oct-4-yl)aminoacetyl)-2-cyanopyrrolidine; inhibitors of the enzyme dipeptidyl peptidase; antidiabetic agents |
| 09/25/2008 | US20080234273 Such as 3-{[4-(azetidin-1-ylcarbonyl)-2-chlorophenyl]oxy}-5-({(1S)-2-[(difluoromethyl)oxy]-1-methylethyl}oxy)-N-(1-methyl-1H-pyrazol-3-yl)benzamide; glucokinases (Glk) |
| 09/25/2008 | US20080233163 4-[4-Methyl-5-(2-nitrooxy-ethyl)-thiazol-2-yl]-phenylamine; N-{4-[4-Methyl-5-(2-nitrooxy-ethyl)-thiazol-2-yl]-phenyl}-acetamide; or4-Methyl-5-(2-nitrooxy-ethyl)-2-(4-nitro-phenyl)-thiazole; cardiovascular, gastrointestinal, inflammatory, respiratory disease |
| 09/25/2008 | CA2681124A1 New substituted arylsulphonylglycines, the preparation thereof and the use thereof as pharmaceutical compositions |
| 09/25/2008 | CA2680592A1 Desferrithiocin polyether analogues and uses thereof in treating pathological conditions |
| 09/24/2008 | EP1972621A1 Method for producing thiazole compound |
| 09/24/2008 | EP1971602A2 Niacin receptor agonists, compositions containing such compounds and methods of treatment |
| 09/24/2008 | EP1971584A2 Isotopically-labeled benzothiazole compounds as imaging agents for amyloidogenic proteins |
| 09/24/2008 | CN101273048A Sulfonamide derivatives as glycokinase activators useful in the treatment of type 2 diabetes |
| 09/24/2008 | CN101273023A 5-substituted thiazol-2-yl amino compounds and compositions as protein kinase inhibitors |
| 09/24/2008 | CN101273022A Thiazoles derivatives as AMPK activator |
| 09/24/2008 | CN101273019A Novel benzimidazole and benzothiazole derivatives, method for preparing same, use thereof as drugs, pharmaceutical compositions and novel use especially as C-Met inhibitors |
| 09/24/2008 | CN101273015A 3-cyclyl-2- (4-sulfamo yl-phenyl) -N-cyclyl-propionamide derivatives useful in the treatment of impaired glucose tolerance and diabetes |
| 09/24/2008 | CN101270099A Method for preparing N-[2-(1-ethoxycarbonyl-3-phenylpropylamino)-tauryl]-thiazolidinecarboxylic acid and its derivant |
| 09/24/2008 | CN100420678C Cyclization process for substituted benzothiazole derivatives |
| 09/24/2008 | CN100420677C Substituted aryl methylene sulfonylated aza cyclo-pentanone compounds, its medicine compositions and its preparing process and use |
| 09/24/2008 | CN100420672C Selective COX-2 inhibitory novel esters from indolealkanols and novel amides from indolealkylamines |