Patents
Patents for C07D 277 - Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings (33,621)
02/2005
02/16/2005EP1506180A1 Thiazolidine-4-one derivative, method for preparing the same, and pharmaceutical composition containing the same
02/16/2005EP1506162A2 Synthesis of benzonitriles and benzimidates
02/16/2005EP1505968A1 Multicyclic compounds for use as melanin concentrating hormone antagonists in the treatment of obesity and diabetes
02/16/2005EP1425258A4 Hydroxyeicosenoic acid analogs
02/16/2005EP1395553B1 Pyrrolidine derivatives as factor xa inhibitors
02/16/2005EP1215203B1 Hydroxamic acid derivatives, process for the production thereof and drugs containing the same as the active ingredient
02/16/2005CN1582269A Hydroxyeicosenoic acid analogs
02/16/2005CN1582149A Dipeptidyl peptidase IV inhibitors and their uses for lowering blood pressure levels
02/16/2005CN1580056A Heterocyclic derivatives their preparing methods and uses
02/15/2005US6855843 Antihistamines; rheumatic diseases; antidiabetic agents; inflammatory bowel disorders
02/15/2005US6855832 O- or S-substituted tetrahydronaphthalene derivatives having retinoid and/or retinoid antagonist-like biological activity
02/15/2005US6855715 Drugs such as 1-(3-Amino-4-chlorobenzoyl-D-phenylglycinyl)-4-(4-fluoro-2 -methylsulphonylphenyl)piperazine, used as anticoagulants
02/10/2005WO2005012297A1 Benzimidazole, benzthiazole and benzoxazole derivatives and their use as lta4h modulators
02/10/2005WO2005012296A1 Benzimidazole, benzthiazole and benzoxazole derivatives and their use as lta4h modulators
02/10/2005WO2005012273A2 Process for the preparation of substituted thiazoles
02/10/2005WO2005012249A2 Adamantyglycine- based inhibitors of dipeptidyl peptidase iv for the treatment of diabetes
02/10/2005WO2005012231A1 Aminocarbonyl naphthol derivative, cyanonaphthol derivative, and method for producing them
02/10/2005WO2005012228A1 O-coordinated metal chelates and their use in optical recording media having high storage capacity
02/10/2005WO2005011812A1 Cyanoamide compounds useful as malonyl-coa decarboxylase inhibithors
02/10/2005WO2005011685A1 Aryl dicarboxamides
02/10/2005WO2004112701A3 Cyclohexylglycine derivatives as dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes
02/10/2005WO2004110983A3 New benzamides as pparϒ modulators
02/10/2005WO2004103976A3 Method for synthesising heterocyclic compounds from thiourea derivatives
02/10/2005US20050033059 Synthesis of epothilones, intermediates thereto, analogues and uses thereof
02/10/2005US20050033057 Thiazoline acid derivatives
02/10/2005US20050033005 Sulfonamide anions as catalysts for NCO oligomerization
02/10/2005US20050032865 Cyanomethyl substituted thiazoliums and imidazoliums and treatments of disorders associated with protein aging
02/10/2005US20050032864 Azolidinedione derivatives such as 5-[4-[[3-methyl-4-oxo-3,4-dihydro-2-quinazolinyl]methoxy]phenylmethyl]thiazolidine-2,4-dione potassium salt; dyslipidaemia; eating, cardiovascular and kidney disorders; atherosclerosis, obesity, psoriasis, polycystic ovarian syndrome; hypotensive agents
02/10/2005US20050032858 Novel heterocyclic compound and anti-inflamatory agent
02/10/2005US20050032856 Use of pramipexole to treat amyotrophic lateral sclerosis
02/10/2005US20050032824 E. g., 1-Cyano-3-(2-mercaptobenzothiazol-6-yl)-2-phenylisourea; metabolic diseases; management of the glucose/fatty acid pathway; antilipemic agents; cardiovascular diseases; antidiabetic agents; anticarcinogenic agents; obesity; more profound effects in metabolism shift than ranolazine or trimetazidine
02/10/2005US20050032790 For example, 1-(2-Amino-4-chlorobenzoyl-D-phenylglycinyl)-4,4'-bispiperidine; for treatment of thrombosis, emphysema, cirrhosis; antiarthritic agents, anticancer agents, antihistamines
02/10/2005US20050032788 treating fibrotic lung diseases and fibrotic hypertrophy or fibrosis of prostate, liver, the pleura, pancreas or bowel wall with saturated and unsaturated azoles and salts, e.g., 3-[2-phenyl-2-oxoethyl]-4,5-dimethyl-thiazolium salt
02/10/2005US20050032787 Pheny (alkyl)carboxylic acid derivatives and dionic phenylalkylheterocyclic derivatives and their use as medicines with serum glucose and/or serum lipid lowering activity
02/10/2005US20050029705 Extrusion die
02/10/2005CA2534212A1 Benzimidazole, benzthiazole and benzoxazole derivatives and their use as lta4h modulators
02/10/2005CA2533658A1 Process for the preparation of substituted thiazoles
02/10/2005CA2529662A1 Aryl dicarboxamides
02/09/2005EP1504759A1 Oral therapeutic or preventive drugs for pollakiuria and urinary incontinence or oral sleep inducers, containing tropolone derivatives
02/09/2005EP1503761A1 Substituted piperazines as melanocortin receptor ligands
02/09/2005EP1503756A1 Epothilone derivative for the treatment of hepatoma and other cancer diseases
02/09/2005EP1436252A4 Hydroxyfattysulfonic acid analogs
02/09/2005EP1087951B1 Carbon substituted aminothiazole inhibitors of cyclin dependent kinases
02/09/2005EP0900210B1 Antivirally active heterocyclic azahexane derivatives
02/09/2005CN1578910A Neurofibrillary labels
02/09/2005CN1578663A Inhibitors of histone deacetylase
02/09/2005CN1578659A Modulators of peroxisome proliferator activated receptors (ppar)
02/09/2005CN1188403C Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
02/08/2005US6852856 Dissolving a 4-(4,6-dialkyl-aryloxy-s-triazin-2-yl)-), 4-methylmorpholinium halide in water and freezing; or, decreasing the content of a 4,6-dialkyl-s-triazine impurity; condensation agents for amidation and esterification reactions
02/08/2005US6852751 Difluorobutyric acid metalloprotease inhibitors
02/08/2005US6852731 3-Substituted-7-oxo-4,7-dihydro-thieno(3,2-b)pyridine-6-carboxylic acid benzylamide derivatives; for herpes viruses
02/08/2005US6852720 Thiazol-2-yl-imine compounds as PDE-7 inhibitors
02/08/2005US6852711 HIV protease inhibitors
02/08/2005US6852548 Produce light energy when decomposed; stable at room temperature
02/03/2005WO2005010028A1 Alpha-amino acid benzothiazolylthio ester as intermediates for manufacture of ace inhibitors and process for preparation thereof
02/03/2005WO2005009941A1 Indane derivates as muscarinic receptor agonists
02/03/2005WO2005009940A1 Novel aminobenzophenone compounds
02/03/2005WO2005009437A1 Design and synthesis of optimized ligands for ppar
02/03/2005WO2004100881A3 Preparation and use of aryl alkyl acid derivatives for the treatment of obesity
02/03/2005US20050027128 Substituted thiazoles
02/03/2005US20050027125 Intensifiers of adenosine receptors for cardiac arrhythmia
02/03/2005US20050026974 Immunogenic conjugates of nitroaromatic compounds and proteins; monoclonal antibodies specific for nitroaromatic compounds , their protein conjugates
02/03/2005US20050026973 New heterocyclic oxime compounds
02/03/2005US20050026966 Coupling a benzylcarbamate compound containing carboxylic group with an amine to form amide, deprotecting the amide to form free amine, reducing free amine, forming an amine salt with toulene sulfonic acid, coupling bis-toulenesulfonic acid salt with a thiazole derivative to form the end product
02/03/2005US20050026945 Cyanoamide compounds useful as malonyl-CoA decarboxylase inhibitors
02/03/2005US20050026943 Oxazolo, thiazolo and selenazolo [4,5-c]-quinolin-4-amines and analogs thereof
02/03/2005US20050026929 2-Phenyl-4-(piperidin-1-ylcarbonyl)-oxazole derivatives; capsase activators; cancer, autoimmune diseases, rheumatoid arthritis, inflammatory bowel disease, or psoriasis
02/03/2005US20050026907 For treating disease, such as cancer, neurological disorders, including polyglutamine-repeat disorders, anemias, thalassemias, inflammatory conditions, autoimmune diseases and cardiovascular conditions
02/03/2005US20050026906 Such as N-4-methoxy-7-morpholin-4-yl-benzothiazol-2-yl)-2-methyl-isonicotinamide; for control or prevention of illnesses based on the modulation of the adenosine system, such as Alzheimer's disease, Parkinson's disease, neuroprotection, schizophrenia, anxiety, pain
02/03/2005US20050026875 Treating bacterial, viral, or fungal infections, cancer, a lung injury, an eye disorder, neurological disorder or stroke
02/03/2005US20050026785 Novel phenyl-propargylether derivatives
02/03/2005DE10330358A1 New arylalkanol derivatives used for treating e.g. respiratory diseases, joint diseases, vascular inflammations, skin disorders, kidney and liver diseases and neurological diseases
02/03/2005CA2533417A1 Design and synthesis of optimized ligands for ppar
02/03/2005CA2530302A1 Novel aminobenzophenone compounds
02/03/2005CA2529036A1 Indane derivates as muscarinic receptor agonists
02/02/2005EP1502590A1 Heterocyclic oxime derivatives, process for their preparation and use thereof in the treatment of type II diabetes
02/02/2005EP1502576A2 Composition containing a 2-thioacetamide and use thereof for stimulating growth or preventing fall out of keratin fibres
02/02/2005EP1501815A1 Substituted phenylacetamides and their use as glucokinase activators
02/02/2005EP1501812A1 Pna monomer and precursor
02/02/2005EP1501811A1 Process for preparing thiazole derivative and the intermediate compounds for preparing the same
02/02/2005EP1501800A1 Bombesin antagonists
02/02/2005EP1501794A1 Thiazolidinones and the use thereof as polo-like kinase inhibitors
02/02/2005EP1501509A2 Aryl-link-aryl substituted thiazolidine-dione and oxazolidine-dione as sodium channel blockers
02/02/2005EP1501508A1 Inhibitors of histone deacetylase
02/02/2005EP1181283B1 Diaminothiazoles and their use for inhibiting protein kinases
02/02/2005CN1575287A Alpha-form or beta-form crystal of acetanilide derivative
02/02/2005CN1575286A Thiophene-amd thiazolesulfonamides as antineoplastic agents
02/02/2005CN1575283A Piperazine derivatives with CCRI receptor antagonist activity
02/02/2005CN1575280A Urea and thiourea derivatives as non-nucleoside reverse transcriptase inhibitors
02/02/2005CN1575279A Substituted thioacetamides
02/02/2005CN1575275A Novel alpha-oxygenated or alpha-thiolated carboxylic acid penethylamide derivatives
02/02/2005CN1575273A 3, 4-di-substituted cyclobutene-1, 2-diones as CXC-chemokine receptor antagonists
02/02/2005CN1575171A Novel anti-diabetic agents
02/01/2005US6849742 Binaphthol derivative and process for producing the same
02/01/2005US6849741 Method for preparing compounds derived from thiazolidinedione, oxazolidinedione or hydantoin
02/01/2005US6849651 Synthesis of epothilones, intermediates thereto, analogues and uses thereof
02/01/2005US6849632 Heteroaryl alkyl piperazine derivatives
02/01/2005US6849097 I.e., N-(thiophen-2 or-3-ylmethyl)-, N-(furan-3-ylmethyl)-, N-(1H-imidazol-2-ylmethyl)- and N-(pyrrol-2-ylmethyl)-p-phenylenediamines; developers for hair dyes
01/2005
01/27/2005WO2005007798A2 Hydroxypropyl methacrylamide polymers and copolymers comprising reactive thiazoline-2-thione
01/27/2005WO2005007616A1 Diphenylamino ketone derivatives as mek inhibitors