Patents
Patents for C07D 277 - Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings (33,621)
07/2005
07/28/2005US20050165031 1-(4-(3-(Pyridin-4-yl)propoxy)phenyl)-3-(5-tert-butylisoxazol-3-yl)urea; inhibits protein tyrosine kinases or a specific kinase or kinase class; for for treating and preventing conditions and diseases such as cancer, hematologic malignancies, cardiovascular disease, inflammation or multiple sclerosis
07/28/2005US20050165028 e.g. 4-bromo-N-(2,3-dihydro-1,4-benzodioxin-6-yl)benzamide; analgesics, neuropathic pain, inflammation, arthritis, rheumatic diseases, inflammatory bowel disorders, eye disorders, or bladder disorders, psoriasis, wounds, burns, allergic skin, herpes simplex
07/28/2005US20050165024 Urea derivatives as kinase modulators
07/28/2005CA2551869A1 Alkylamino, arylamino, and sulfonamido cyclopentyl amide modulators of chemokine receptor activity
07/28/2005CA2551415A1 Thiazole derivatives and use thereof
07/28/2005CA2547703A1 Bicyclic pyrazolo-fused compounds as protein kinase modulators
07/27/2005EP1557168A2 Biarylurea Derivatives
07/27/2005EP1556385A1 Heterocyclocarboxamide derivatives
07/27/2005EP1556142A2 Alkyne derivatives as tracers for metabotropic glutamate receptor binding
07/27/2005EP1556059A1 Thrombopoietin mimetics
07/27/2005EP1556040A1 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 and type 2
07/27/2005EP1467980B1 Method for producing halogenated 2-(3-butenylsulfanyl)-1,3-thiazoles
07/27/2005EP1414384A4 Synthesis of epothilones and relates analogs
07/27/2005EP1047418B1 Inhibition of raf kinase using substituted heterocyclic ureas
07/27/2005CN1646518A 3-aminophenol derivatives and dyes that contain these compounds while serving to dye keratin fibers
07/27/2005CN1646507A Aminophenylbenzothiazole compounds
07/27/2005CN1646506A Difluoromethyl thiazolyl carboxanilides
07/27/2005CN1646504A Substituted benzoxazoles and analogues as estrogenic agents
07/27/2005CN1646497A New aryl imidazoles and related compounds as C5a receptor modulators
07/27/2005CN1646123A Therapeutic agent for food competence disorder in stomach
07/27/2005CN1644579A N-alkoxide oxo-2-triazolidone derivative, its preparation and use
07/27/2005CN1212311C Acrylonitrile compounds, process for their prodn, and pesticides containing them
07/27/2005CN1212117C Medicine composition for treating diabetes mellitus
07/26/2005US6921770 Treating 2- phenyliminothiazoline hydrochloride or hydrobromide with a base and extracting with a solvent
07/26/2005US6921760 Psychotherapeutic agents.
07/26/2005US6921650 Recombinant methods and materials for producing epothilone and epothilone derivatives
07/26/2005CA2193388C Aryl and heteroaryl alkoxynaphthalene derivatives
07/21/2005WO2005066145A1 Heteroaryl-ureas and their use as glucokinase activators
07/21/2005WO2005066114A1 Compounds for diagnosis, treatment and prevention of bone injury and metabolic disorders
07/21/2005WO2005026137A3 Modulators of atp-binding cassette transporters
07/21/2005WO2005013914A3 Heteroarylaminosulfonylphenyl derivatives for use as sodium or calcium channel blockers in the treatment of pain
07/21/2005WO2004050609A8 Substituted ureas and carbamates
07/21/2005US20050159598 Activators of human peroxisome proliferator activated receptors such as {2-[2-fluoro-4-(trifluoromethyl)phenyl]-4-methyl-1,3-thiazol-5-yl}methanol
07/21/2005US20050159460 2-[(1R,3S,4S)-1-benzyl-4-t-butoxycarbonylamino-3-hydroxy-5-phenylpentyl]-5-butyl-thiazole; for inhibiting beta-secretase-mediated cleavage of amyloid precursor protein, particularly to inhibit production of A beta peptide; treatment of diseases associated with a pathological form of A beta peptide
07/21/2005US20050159459 inhibitors of the beta-secretase enzyme that are useful in the treatment of Alzheimer's disease and other diseases characterized by deposition of A beta peptide in a mammal. The compounds of the invention are useful to reduce forming beta peptides
07/21/2005US20050159427 N-acylsulfonamide apoptosis promoters
07/21/2005US20050159423 Antibacterial compounds
07/21/2005US20050159405 Substituted 10-aryl-11h-benzo[b]fluourenes and 7-aryl-5, 6-dihydro-benzo[a]anthracenes for selective effects on estrogen receptors
07/21/2005US20050156336 Process for exchanging functional groups by halogen-metal exchange reaction
07/20/2005EP1555257A1 Process for producing aromatic nitrile compound
07/20/2005EP1554260A1 Aryloxyalkylamine derivatives as h3 receptor ligands
07/20/2005EP1554239A2 Sulfonylamino-acetic acid derivatives and their use as orexin receptor antagonists
07/20/2005EP1286673B8 Ligands of integrin receptors
07/20/2005EP0784430B1 Method for reducing unwanted cellular adhesions
07/20/2005CN1642929A Kappa-opioid receptor agonist comprising 2-phenylbenzothiazoline derivative
07/20/2005CN1642918A Novel hererocyclic compound and preparation thereof and medicine composition containing same and use thereof in medicine
07/20/2005CN1642915A Benzamide derivatives useful as histone deacetylase inhibitors
07/20/2005CN1642879A Process for producing biaryl compound
07/20/2005CN1211375C Thiazole-derivatives
07/20/2005CN1211374C Heterocyclic derivative, its preparation method and medicine compositioncontaining them
07/20/2005CN1211367C Prostaglandin agonists and their use to treat bone disorders
07/19/2005US6919482 A 1,4-bis(N-(2-(4-hydroxy-3-hydroxymethylphenyl) -2-hydroxyethyl)amino)-cyclohexane or alkyl-cyclohexane or -pyrazine derivatives; treating respiratory diseases disorders, asthma, bronchitis, nervous system injury
07/19/2005US6919470 Aryl and heteroaryl sulfonates
07/19/2005US6919379 Compounds useful in reflux disease
07/19/2005US6919375 Sulfonated amino acid derivatives and metalloproteinase inhibitors containing the same
07/19/2005US6919367 Substituted thioacetamides
07/19/2005US6919362 For use as hypoglycaemic and hypolipidaemic agents
07/19/2005US6919361 Five-membered-ring compound
07/19/2005US6919358 Substituted acid derivatives useful as antidiabetic and antiobesity agents and method
07/14/2005WO2005064006A1 OPTICALLY ACTIVE, HETEROAROMATIC β-HYDROXY ESTERS, PROCESSES FOR THEIR PREPARATION FROM β-KETO ESTERS AND PROCESSES FOR THE PREPARATION OF THESE β-KETO ESTERS
07/14/2005WO2005063729A1 3-(4-benzyloxyphenyl)propanoic acid derivatives
07/14/2005WO2005063725A1 Phenylpropanoic acid derivatives
07/14/2005WO2005063724A1 1-(azolin-2-yl) amino-1,2-diphenylethane compounds for combatting insects, arachnids and nematodes
07/14/2005WO2005063705A1 Benzene compounds disubstituted with cyclic groups at the 1- and 2-positions
07/14/2005WO2005063692A1 (hetero)cyclyl carboxanilides for controlling harmful fungi
07/14/2005WO2005063689A1 Benzamide derivative
07/14/2005WO2005063222A1 Hsp90 FAMILY PROTEIN INHIBITOR
07/14/2005WO2005051946A3 Compounds having beta2 adrenergic receptor agonist and muscarinic receptor antagonist activity
07/14/2005US20050154202 Substituted aryl amides
07/14/2005US20050154056 Inhibitors of HCV NS5B polymerase
07/14/2005US20050154031 which are selective against serotonin 5-HT2A and 5-HT2C receptors; 2-amino-5-methyl-4-(naphth-1-yl)thiazole; irritable bowel syndrome, dyspepsia, gastroesophageal reflux, tachygastria; migraine, neurogenic pain, anxiety, depression, sleep disorder, asthma, incontinence, endometriosis, and fibrosis
07/14/2005US20050153995 Nonnucleoside inhibitors of reverse transcriptase, composite binding pocket and methods for use thereof
07/14/2005US20050153977 N-[4-(4-chlorothiophen-2-yl)-5-(4-cyclohexylpiperazin-1-yl)thiazol-2-yl]-3-fluoro-4-hydroxybenzamide; nonpeptide c-mpl ligand; low immunogenicity; proliferate human c-mpl-Ba/F3 cells; increase platelets by promoting the formation of megakaryocytic colonies; orally
07/14/2005US20050153973 (4R)-3-(2-{[8-(2-Pyrimidinyl)-8-azabicyclo[3.2.1]oct-3-yl]exo-amino}acetyl)thiazolidine-4-carbonitrile; enzyme inhibitors; diabetes
07/14/2005US20050153962 2,4-dichloro-N-(4-chloro-3-methoxy-phenyl)-N-[4-(pyrrolidine-1-carbonyl)thiazole-2-yl]-benzamide; cannabionic receptor (CB1) antagonist and inverse agonists; side effects reduction; amidation of aminothiazol derivatives with acid chloride and coupling by dehydroxylation with alcohol or amine derivatives
07/14/2005US20050153958 Substituted aryl ketones
07/14/2005US20050153950 Broad -spectrum cephem compounds
07/14/2005US20050153366 Protein-protein interaction antagonist screening libraries based upon 1,4-disubstituted naphthalenes and related scaffolds
07/14/2005CA2551610A1 3-(4-benzyloxyphenyl)propanoic acid derivatives
07/14/2005CA2546981A1 Optically active, heteroaromatic .beta.-hydroxy esters, processes for their preparation from .beta.-keto esters and processes for the preparation of these .beta.-keto esters
07/13/2005EP1553091A1 Heteroaromatic pentacyclic compound and medicinal use thereof
07/13/2005EP1551816A1 Thiazolyl biphenyl amides
07/13/2005EP1551815A1 Thiazole compounds for the treatment of neurodegenerative disorders
07/13/2005EP1551799A1 Cyclohexyl sulphones as gamma-secretase inhibitors
07/13/2005EP1551798A1 Novel sulphones for inhibition of gamma secretase
07/13/2005EP1551797A1 Cyclohexyl sulphone derivatives as gamma-secretase inhibitors
07/13/2005EP1551795A1 Inhibitors of histone deacetylase
07/13/2005EP1178969B1 Gastrin and cholecystokinin receptor ligands
07/13/2005EP1161415B1 N-cyanomethylamides as protease inhibitors
07/13/2005EP1144364B1 Multicyclic compounds which inhibit leukocyte adhesion mediated by vla-4
07/13/2005CN1639158A Thiazole derivatives as NPY receptor antagonists
07/13/2005CN1639157A 2-acylaminothiazole derivative or salt thereof
07/13/2005CN1639139A 5-phenylthiazole derivatives and use as PI3 kinase inhibitors
07/13/2005CN1639138A Biphenylmethyl-thiazolidinediones and analogues and their use as PPAR-gamma activators
07/13/2005CN1639128A O-cyclopropyl-carboxanilides and their use as fungicides
07/13/2005CN1639119A Substituted 2-amino-cycloalkanecarboxamides and their use as cysteine protease inhibitors
07/13/2005CN1639096A Process for producing trans-4-amino-1-cyclohexanecarboxylic acid derivative
07/13/2005CN1638768A Thiazole and oxazole derivatives that modulate PPAR activity
07/13/2005CN1638757A 组织蛋白酶半胱氨酸蛋白酶抑制剂 Cathepsin cystatin
07/13/2005CN1637018A Novel effectors of dipeptidyl peptidase IV