Patents for C07D 277 - Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings (33,621) |
---|
07/28/2005 | US20050165031 1-(4-(3-(Pyridin-4-yl)propoxy)phenyl)-3-(5-tert-butylisoxazol-3-yl)urea; inhibits protein tyrosine kinases or a specific kinase or kinase class; for for treating and preventing conditions and diseases such as cancer, hematologic malignancies, cardiovascular disease, inflammation or multiple sclerosis |
07/28/2005 | US20050165028 e.g. 4-bromo-N-(2,3-dihydro-1,4-benzodioxin-6-yl)benzamide; analgesics, neuropathic pain, inflammation, arthritis, rheumatic diseases, inflammatory bowel disorders, eye disorders, or bladder disorders, psoriasis, wounds, burns, allergic skin, herpes simplex |
07/28/2005 | US20050165024 Urea derivatives as kinase modulators |
07/28/2005 | CA2551869A1 Alkylamino, arylamino, and sulfonamido cyclopentyl amide modulators of chemokine receptor activity |
07/28/2005 | CA2551415A1 Thiazole derivatives and use thereof |
07/28/2005 | CA2547703A1 Bicyclic pyrazolo-fused compounds as protein kinase modulators |
07/27/2005 | EP1557168A2 Biarylurea Derivatives |
07/27/2005 | EP1556385A1 Heterocyclocarboxamide derivatives |
07/27/2005 | EP1556142A2 Alkyne derivatives as tracers for metabotropic glutamate receptor binding |
07/27/2005 | EP1556059A1 Thrombopoietin mimetics |
07/27/2005 | EP1556040A1 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 and type 2 |
07/27/2005 | EP1467980B1 Method for producing halogenated 2-(3-butenylsulfanyl)-1,3-thiazoles |
07/27/2005 | EP1414384A4 Synthesis of epothilones and relates analogs |
07/27/2005 | EP1047418B1 Inhibition of raf kinase using substituted heterocyclic ureas |
07/27/2005 | CN1646518A 3-aminophenol derivatives and dyes that contain these compounds while serving to dye keratin fibers |
07/27/2005 | CN1646507A Aminophenylbenzothiazole compounds |
07/27/2005 | CN1646506A Difluoromethyl thiazolyl carboxanilides |
07/27/2005 | CN1646504A Substituted benzoxazoles and analogues as estrogenic agents |
07/27/2005 | CN1646497A New aryl imidazoles and related compounds as C5a receptor modulators |
07/27/2005 | CN1646123A Therapeutic agent for food competence disorder in stomach |
07/27/2005 | CN1644579A N-alkoxide oxo-2-triazolidone derivative, its preparation and use |
07/27/2005 | CN1212311C Acrylonitrile compounds, process for their prodn, and pesticides containing them |
07/27/2005 | CN1212117C Medicine composition for treating diabetes mellitus |
07/26/2005 | US6921770 Treating 2- phenyliminothiazoline hydrochloride or hydrobromide with a base and extracting with a solvent |
07/26/2005 | US6921760 Psychotherapeutic agents. |
07/26/2005 | US6921650 Recombinant methods and materials for producing epothilone and epothilone derivatives |
07/26/2005 | CA2193388C Aryl and heteroaryl alkoxynaphthalene derivatives |
07/21/2005 | WO2005066145A1 Heteroaryl-ureas and their use as glucokinase activators |
07/21/2005 | WO2005066114A1 Compounds for diagnosis, treatment and prevention of bone injury and metabolic disorders |
07/21/2005 | WO2005026137A3 Modulators of atp-binding cassette transporters |
07/21/2005 | WO2005013914A3 Heteroarylaminosulfonylphenyl derivatives for use as sodium or calcium channel blockers in the treatment of pain |
07/21/2005 | WO2004050609A8 Substituted ureas and carbamates |
07/21/2005 | US20050159598 Activators of human peroxisome proliferator activated receptors such as {2-[2-fluoro-4-(trifluoromethyl)phenyl]-4-methyl-1,3-thiazol-5-yl}methanol |
07/21/2005 | US20050159460 2-[(1R,3S,4S)-1-benzyl-4-t-butoxycarbonylamino-3-hydroxy-5-phenylpentyl]-5-butyl-thiazole; for inhibiting beta-secretase-mediated cleavage of amyloid precursor protein, particularly to inhibit production of A beta peptide; treatment of diseases associated with a pathological form of A beta peptide |
07/21/2005 | US20050159459 inhibitors of the beta-secretase enzyme that are useful in the treatment of Alzheimer's disease and other diseases characterized by deposition of A beta peptide in a mammal. The compounds of the invention are useful to reduce forming beta peptides |
07/21/2005 | US20050159427 N-acylsulfonamide apoptosis promoters |
07/21/2005 | US20050159423 Antibacterial compounds |
07/21/2005 | US20050159405 Substituted 10-aryl-11h-benzo[b]fluourenes and 7-aryl-5, 6-dihydro-benzo[a]anthracenes for selective effects on estrogen receptors |
07/21/2005 | US20050156336 Process for exchanging functional groups by halogen-metal exchange reaction |
07/20/2005 | EP1555257A1 Process for producing aromatic nitrile compound |
07/20/2005 | EP1554260A1 Aryloxyalkylamine derivatives as h3 receptor ligands |
07/20/2005 | EP1554239A2 Sulfonylamino-acetic acid derivatives and their use as orexin receptor antagonists |
07/20/2005 | EP1286673B8 Ligands of integrin receptors |
07/20/2005 | EP0784430B1 Method for reducing unwanted cellular adhesions |
07/20/2005 | CN1642929A Kappa-opioid receptor agonist comprising 2-phenylbenzothiazoline derivative |
07/20/2005 | CN1642918A Novel hererocyclic compound and preparation thereof and medicine composition containing same and use thereof in medicine |
07/20/2005 | CN1642915A Benzamide derivatives useful as histone deacetylase inhibitors |
07/20/2005 | CN1642879A Process for producing biaryl compound |
07/20/2005 | CN1211375C Thiazole-derivatives |
07/20/2005 | CN1211374C Heterocyclic derivative, its preparation method and medicine compositioncontaining them |
07/20/2005 | CN1211367C Prostaglandin agonists and their use to treat bone disorders |
07/19/2005 | US6919482 A 1,4-bis(N-(2-(4-hydroxy-3-hydroxymethylphenyl) -2-hydroxyethyl)amino)-cyclohexane or alkyl-cyclohexane or -pyrazine derivatives; treating respiratory diseases disorders, asthma, bronchitis, nervous system injury |
07/19/2005 | US6919470 Aryl and heteroaryl sulfonates |
07/19/2005 | US6919379 Compounds useful in reflux disease |
07/19/2005 | US6919375 Sulfonated amino acid derivatives and metalloproteinase inhibitors containing the same |
07/19/2005 | US6919367 Substituted thioacetamides |
07/19/2005 | US6919362 For use as hypoglycaemic and hypolipidaemic agents |
07/19/2005 | US6919361 Five-membered-ring compound |
07/19/2005 | US6919358 Substituted acid derivatives useful as antidiabetic and antiobesity agents and method |
07/14/2005 | WO2005064006A1 OPTICALLY ACTIVE, HETEROAROMATIC β-HYDROXY ESTERS, PROCESSES FOR THEIR PREPARATION FROM β-KETO ESTERS AND PROCESSES FOR THE PREPARATION OF THESE β-KETO ESTERS |
07/14/2005 | WO2005063729A1 3-(4-benzyloxyphenyl)propanoic acid derivatives |
07/14/2005 | WO2005063725A1 Phenylpropanoic acid derivatives |
07/14/2005 | WO2005063724A1 1-(azolin-2-yl) amino-1,2-diphenylethane compounds for combatting insects, arachnids and nematodes |
07/14/2005 | WO2005063705A1 Benzene compounds disubstituted with cyclic groups at the 1- and 2-positions |
07/14/2005 | WO2005063692A1 (hetero)cyclyl carboxanilides for controlling harmful fungi |
07/14/2005 | WO2005063689A1 Benzamide derivative |
07/14/2005 | WO2005063222A1 Hsp90 FAMILY PROTEIN INHIBITOR |
07/14/2005 | WO2005051946A3 Compounds having beta2 adrenergic receptor agonist and muscarinic receptor antagonist activity |
07/14/2005 | US20050154202 Substituted aryl amides |
07/14/2005 | US20050154056 Inhibitors of HCV NS5B polymerase |
07/14/2005 | US20050154031 which are selective against serotonin 5-HT2A and 5-HT2C receptors; 2-amino-5-methyl-4-(naphth-1-yl)thiazole; irritable bowel syndrome, dyspepsia, gastroesophageal reflux, tachygastria; migraine, neurogenic pain, anxiety, depression, sleep disorder, asthma, incontinence, endometriosis, and fibrosis |
07/14/2005 | US20050153995 Nonnucleoside inhibitors of reverse transcriptase, composite binding pocket and methods for use thereof |
07/14/2005 | US20050153977 N-[4-(4-chlorothiophen-2-yl)-5-(4-cyclohexylpiperazin-1-yl)thiazol-2-yl]-3-fluoro-4-hydroxybenzamide; nonpeptide c-mpl ligand; low immunogenicity; proliferate human c-mpl-Ba/F3 cells; increase platelets by promoting the formation of megakaryocytic colonies; orally |
07/14/2005 | US20050153973 (4R)-3-(2-{[8-(2-Pyrimidinyl)-8-azabicyclo[3.2.1]oct-3-yl]exo-amino}acetyl)thiazolidine-4-carbonitrile; enzyme inhibitors; diabetes |
07/14/2005 | US20050153962 2,4-dichloro-N-(4-chloro-3-methoxy-phenyl)-N-[4-(pyrrolidine-1-carbonyl)thiazole-2-yl]-benzamide; cannabionic receptor (CB1) antagonist and inverse agonists; side effects reduction; amidation of aminothiazol derivatives with acid chloride and coupling by dehydroxylation with alcohol or amine derivatives |
07/14/2005 | US20050153958 Substituted aryl ketones |
07/14/2005 | US20050153950 Broad -spectrum cephem compounds |
07/14/2005 | US20050153366 Protein-protein interaction antagonist screening libraries based upon 1,4-disubstituted naphthalenes and related scaffolds |
07/14/2005 | CA2551610A1 3-(4-benzyloxyphenyl)propanoic acid derivatives |
07/14/2005 | CA2546981A1 Optically active, heteroaromatic .beta.-hydroxy esters, processes for their preparation from .beta.-keto esters and processes for the preparation of these .beta.-keto esters |
07/13/2005 | EP1553091A1 Heteroaromatic pentacyclic compound and medicinal use thereof |
07/13/2005 | EP1551816A1 Thiazolyl biphenyl amides |
07/13/2005 | EP1551815A1 Thiazole compounds for the treatment of neurodegenerative disorders |
07/13/2005 | EP1551799A1 Cyclohexyl sulphones as gamma-secretase inhibitors |
07/13/2005 | EP1551798A1 Novel sulphones for inhibition of gamma secretase |
07/13/2005 | EP1551797A1 Cyclohexyl sulphone derivatives as gamma-secretase inhibitors |
07/13/2005 | EP1551795A1 Inhibitors of histone deacetylase |
07/13/2005 | EP1178969B1 Gastrin and cholecystokinin receptor ligands |
07/13/2005 | EP1161415B1 N-cyanomethylamides as protease inhibitors |
07/13/2005 | EP1144364B1 Multicyclic compounds which inhibit leukocyte adhesion mediated by vla-4 |
07/13/2005 | CN1639158A Thiazole derivatives as NPY receptor antagonists |
07/13/2005 | CN1639157A 2-acylaminothiazole derivative or salt thereof |
07/13/2005 | CN1639139A 5-phenylthiazole derivatives and use as PI3 kinase inhibitors |
07/13/2005 | CN1639138A Biphenylmethyl-thiazolidinediones and analogues and their use as PPAR-gamma activators |
07/13/2005 | CN1639128A O-cyclopropyl-carboxanilides and their use as fungicides |
07/13/2005 | CN1639119A Substituted 2-amino-cycloalkanecarboxamides and their use as cysteine protease inhibitors |
07/13/2005 | CN1639096A Process for producing trans-4-amino-1-cyclohexanecarboxylic acid derivative |
07/13/2005 | CN1638768A Thiazole and oxazole derivatives that modulate PPAR activity |
07/13/2005 | CN1638757A 组织蛋白酶半胱氨酸蛋白酶抑制剂 Cathepsin cystatin |
07/13/2005 | CN1637018A Novel effectors of dipeptidyl peptidase IV |