Patents for C07D 271 - Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms (7,144) |
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06/10/2008 | US7384963 2′-Methyl-5-(1,3,4-oxadiazol-2-yl)1, 1′-biphenyl-4-carboxaide derivatives and their use as p38 kinase |
06/10/2008 | US7384929 N-aryl azaspiroalkene and azaspiroalkane compounds and methods of preparation and use thereof |
06/04/2008 | CN101190917A 3,4-dihydro-3-methyl-4-oxomidazo[5,1-d]-1,2,3,5-tetrazine-8-formic acid benzenesulfonyl furoxan esters compound, preparation method and use thereof |
06/03/2008 | US7381821 Reacting 4-(alpha-(p-chlorophenyl)benzyl)-1-leaving group-alkylpiperazine with protected 1-hydroxy-1-(4-(p-hydroxyphenyl)-3-butynyl)urea to form 1-(4-(p-(4-(alpha-(p-chlorophenyl)benzyl)-1-piperazin-1-ylalkyl)phenyl)-3-butynyl)-1-hydroxyurea; preparation of intermediates |
05/29/2008 | WO2008064320A2 Hydrindane analogs having sphingosine 1-phosphate receptor agonist activity |
05/29/2008 | WO2008064315A1 Tetralin analogs having sphingosine 1-phosphate agonist activity |
05/29/2008 | US20080125433 Method of treating hair loss using thyromimetic compounds |
05/29/2008 | CA2669104A1 Hydrindane analogs having sphingosine 1-phosphate receptor agonist activity |
05/29/2008 | CA2669102A1 Tetralin analogs having sphingosine 1-phosphate agonist activity |
05/28/2008 | CN100390135C Novel derivatives of dicarboxylic acid having pharmaceutical properties |
05/27/2008 | US7378529 Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4 |
05/27/2008 | US7378409 Substituted cycloalkylamine derivatives as modulators of chemokine receptor activity |
05/22/2008 | WO2008059128A1 Phenylic derivatives and use thereof as drugs |
05/22/2008 | US20080119486 Benzoyl-piperazine derivatives |
05/21/2008 | EP1482924B1 Cathepsin cysteine protease inhibitors |
05/21/2008 | CN101184739A Polycyclic oxadiazoles or isoxazoles and their use as S1P receptor ligands |
05/20/2008 | US7375134 N1-(1-cyanocyclopropyl)-4-fluoro-N2-{(1S)-2,2,2-trifluoro-1-[4'-(methylsulfonyl)-1,1'-biphenyl-4-yl]ethyl}-L-leucinamide; osteoporosis and other bone loss disorders |
05/15/2008 | WO2008058178A1 N-hydroxyamidinoheterocycles as modulators of indoleamine 2,3-dioxygenase |
05/15/2008 | WO2008057775A2 Heterocyclic amide compounds useful as kinase inhibitors |
05/15/2008 | US20080114002 3-[2-(3-Cyanophenoxy)-4-(trifluoromethyl)phenyl]propanoic acid;prostaglandin D2 inhibitor, orphan receptor CRTH2 antagonist; antiinflammatory, analgesic, antipyretic; respiratory system disorders: asthma and rhinitis; coupling amino/thio-phenyl derivatives with ester followed by hydrolysis to acid |
05/14/2008 | EP1919464A1 Oxadiazole compounds as urokinase inhibitors |
05/14/2008 | EP1446375B1 Dihalogenpropene compounds, method for the production thereof, agents containing said compounds and the use thereof as pest control agents |
05/08/2008 | WO2008039431A3 Crystalline forms of 3-[5-(2-fhjorophenyl)-[1,2,4]oxadiazol-3-yl]-benzoic acid |
05/08/2008 | US20080108811 Aromatic Amine Derivative and Organic Electroluminescent Device Using Same |
05/07/2008 | EP1917323A1 Novel materials for organic electroluminescent devices |
05/07/2008 | CN101175736A Compound, composition, phase difference plate, elliptically polarizing plate and liquid crystal display device |
05/07/2008 | CN101172983A Substituted phenylacetic acids |
05/06/2008 | US7368479 Alpha-sulfonylamino-acetonitriles |
05/02/2008 | WO2008050200A1 Oxadiazole compounds as calcium channel antagonists |
04/29/2008 | US7365196 Sulphonamido-substituted bridged bicycloalkyl derivatives |
04/29/2008 | US7365074 Pyridazine, pyrimidine and pyrazine ethyne compounds |
04/29/2008 | US7365068 Hepatitis C virus infections; -(3-cyclopropyl-4-(pentyloxy)phenyl)-3-nicotinoylthiourea;methyl 2-oxo-2-(5-((3-(4-(pentyloxy)-3-(trifluoromethyl)phenyl)thioureido)carbonyl)pyridin-2-ylamino)acetate |
04/29/2008 | US7364670 Liquid crystalline compound, liquid crystalline composition and retardation film |
04/24/2008 | US20080096874 Oxadiazole Derivative as Dgat Inhibitors |
04/23/2008 | EP1914225A1 Salt molten at room temperature and display device |
04/23/2008 | EP1912971A2 Di-substituted oxadiazoles as cxc-chemokine receptor ligands |
04/23/2008 | EP1912958A1 Substituted malononitrile compounds for combating animal pests |
04/17/2008 | US20080090854 Cxcr2 inhibitors |
04/17/2008 | US20080090840 Heterocyclic GPR40 Modulators |
04/16/2008 | CN101163690A 苯并噻吩异羟肟酸衍生物 Benzothiophene hydroxamic acid derivatives |
04/15/2008 | US7358265 Oxa-and thiadiazoles and their use as metalloproteinase inhibitors |
04/15/2008 | CA2410303C Beta-amino acid nitrile derivatives |
04/10/2008 | US20080086009 Reacting a alkyl nitrile selected from acetonitrile, propionitrile, or butyronitrile with acetone or acetophenone in presence of ferric nitrate to produce 3-acetyl-5-methyl or ethyl or other alkyl-1,2,4-oxadiazole derivative or a 3-benzoyl-5- ethyl or methyl or other alkyl-l 1,2,4-oxadiazole derivatives |
04/10/2008 | US20080085894 Alpha-(n-sulfonamido)acetamide derivatives as beta-amyloid inhibitors |
04/09/2008 | EP1907383A1 Gpcr agonists |
04/09/2008 | EP1907382A1 Nitrocatechol derivatives as comt inhibitors |
04/09/2008 | CN101157661A Method for producing molsidomine |
04/09/2008 | CN100379415C Hetero biaryl derivatives as matrix metalloproteinase inhibitors |
04/03/2008 | WO2008039431A2 Crystalline forms of 3-[5-(2-fhjorophenyl)-[1,2,4]oxadiazol-3-yl]-benzoic acid |
04/03/2008 | WO2008039023A1 Heteroaryl-pyrazole derivatives as cannabinoid cb1 receptor antagonists |
04/03/2008 | WO2008037476A1 Oxadiazole derivatives with anti-inflammatory and immunosuppressive properties |
04/03/2008 | US20080081812 and inverse agonist; 2-(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazol-3-yl)-5-(pyridin-4-yl)-1,3,4-oxadiazole; obesity and obesity-related metabolic disorders |
04/03/2008 | CA2664268A1 Diaryl oxadiazol derivatives |
04/03/2008 | CA2663574A1 Crystalline forms of 3-[5-(2-fluorophenyl)-[1,2,4]oxadiazol-3-yl]-benzoic acid |
04/02/2008 | CN100378086C Novel piperazine derivatives and their use as synthesis intermediates |
04/02/2008 | CN100378085C Preparation process of 5-alkyl-1,3,4-oxidazole ketone |
04/02/2008 | CN100378084C 2,5-diaryl substituting group-1,3,4-oxidazole derivative, its synthesis and use |
04/01/2008 | US7351825 4-[5-((1S,2R)-1-Carboxy-2-phenyl-cyclopropylsulfamoyl)-thiophen-2-yl]-3,6-dihydro-2H-pyridine-1-carboxylic acid tert-butyl ester; aggrecanase and matrix metalloproteinase (with zinc in the catalytic active center) (MMP) inhibitor; antiarthritic agent: osteoarthritis, rheumatoid arthritis |
03/27/2008 | WO2008035239A1 Phenyl derivatives and their use as immunomodulators |
03/27/2008 | CA2662673A1 Phenyl derivatives and their use as immunomodulators |
03/26/2008 | EP1901731A1 Niacin receptor agonists, compositions containing such compounds and methods of treatment |
03/26/2008 | EP0971878B1 Amine compounds, their production and use as amyloid-beta production inhibitors |
03/25/2008 | US7348440 Mitotic kinesin inhibitors |
03/25/2008 | US7348345 Nonnucleoside reverse transcriptase inhibitors |
03/20/2008 | WO2008016692A3 Chemical compounds |
03/20/2008 | US20080070957 p-(2-alkoxy-2-acylethyl)biphenyl compounds; 1-[4'-(2-ethoxy-3-morpholin-4-yl-3-oxopropyl)biphenyl-3-yl]-3-heptyl-1-methylurea; human or veterinary medicine: dermatology, cardiovascular diseases, immune diseases,; lipid metabolism diseases; Peroxisome Proliferator-Activated Receptor modulator |
03/19/2008 | EP1149091B1 4-(heterocyclylsulfonamido)-5-methoxy-6-(2-methoxyphenoxy)-2-phenyl- or pyridylpyrimidines as endothelin receptor antagonists |
03/18/2008 | US7345095 Alpha, beta -peptide inhibitors; Alzheimer's disease; 2-(4-Chloro-benzenesulfonylamino)-3-phenyl-propionic acid methyl ester |
03/13/2008 | WO2008030570A1 Processes for the preparation of 1,2,4-oxadiazole benzoic acids |
03/13/2008 | US20080064879 Compound ,Composition And Thin Film |
03/13/2008 | US20080064728 Heterocyclic Compounds Useful as Dpp-Iv Inhibitors |
03/13/2008 | CA2842625A1 Processes for the preparation of 1,2,4-oxadiazole benzoic acids |
03/13/2008 | CA2662749A1 Processes for the preparation of 1,2,4-oxadiazole benzoic acids |
03/06/2008 | US20080058335 Pain, inflammatory or immune disorders, neurological disorders, cancers of the immune system, respiratory disorders, cardiovascular disorders, neuroprotection; e.g. 5-chloro-N-[(2Z)-5-(1-hydroxy-1-methylethyl)-3-[((cis)-3-methoxycyclobutyl)methyl]-4-methyl-1,3-thiazol-2(3H)-ylidene]-2-methoxybenzamide |
03/06/2008 | US20080058314 Novel dicarboxylic acid derivatives with pharmaceutical properties |
03/05/2008 | EP1893592A1 Oxadiazole derivatives as dgat inhibitors |
03/05/2008 | EP1893591A1 POLYCYCLIC OXADIAZOLES OR I SOXAZOLES AND THEIR USE AS SlP RECEPTOR LIGANDS |
03/05/2008 | EP1718967A4 METHODS OF DETECTING Lp-PLA2 ACTIVITY |
02/28/2008 | WO2008023783A1 Amine compound |
02/28/2008 | WO2008023157A1 Nitrogen containing heterocyclic compounds useful as m3-receptor modulators |
02/28/2008 | WO2007016136A3 Organic nitric oxide enhancing salts of cyclooxygenase-2 selective inhibitors, compositons and methods of use |
02/28/2008 | WO2007016095A3 Cyclooxygenase-2 selective inhibitor compounds comprising nitric oxide enhancing groups, compositions and methods of use |
02/28/2008 | US20080051441 Aryl Sulphonamide Modulators |
02/28/2008 | CA2660524A1 Compounds for treating proliferative disorders |
02/27/2008 | EP1891000A1 Sphingolipids |
02/27/2008 | EP1399423B9 Anthranilic acid amides with a heteroarylsulfonyl side chain, method for the production thereof, use thereof as a medicament or diagnostic agent and pharmaceutical preparations containing said compounds |
02/26/2008 | CA2322195C Novel diphenyl-substituted 5-ring-heterocycles, method for producing them and their use as medicaments |
02/21/2008 | WO2006134317A8 Oxadiazole derivatives as dgat inhibitors |
02/21/2008 | US20080045571 Additional heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists |
02/20/2008 | EP1888512A2 Chemical compounds |
02/20/2008 | CN101128413A Substituted oxyarenes |
02/19/2008 | US7332514 Dibenzylamine compound and medicinal use thereof |
02/14/2008 | US20080039510 (1,5-diphenyl-1h-pyrazol-3-yl)oxadiazole derivatives, preparation method thereof and use of same in therapeutics |
02/13/2008 | EP1513796B1 Phenyloxyalkanoic acid derivatives as hppar activators |
02/13/2008 | CN101124201A Parp抑制剂 Parp inhibitors |
02/12/2008 | US7329756 Process for the manufacture of Isradipine |
02/07/2008 | WO2008016692A2 Chemical compounds |
02/07/2008 | WO2008016139A1 Fluorescent oleamide derivative and use thereof |
02/07/2008 | US20080033022 Inhibitors of c-Jun N-terminal kinases (JNK) |
02/07/2008 | CA2659473A1 Chemical compounds |