Patents
Patents for C07D 263 - Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings (20,978)
05/1999
05/19/1999CN1216978A New vitamin-D derivatives with carbo- or heterocyclic substitutents at C-25, process for the prodn. intermediate products and their use for producing medicaments
05/19/1999CN1216767A Novel 5-membered ring heterocycles, their prepn. their use and pharmaceutical preparations comprising them
05/19/1999CN1043422C Method for preparing polyhydroxycyclopentane derivatives
05/18/1999US5905151 Trimer catalyst for aliphatic and aromatic isocyanates
05/18/1999CA1340549C Method of preparing sphingosine derivatives
05/18/1999CA1340543C Pharmaceutically active compounds
05/14/1999WO1999023081A2 Trifluoromethylbiphenylyl-dihalophenylazolines as pesticides
05/14/1999WO1999022720A2 Selective cyclooxygenase-2 inhibitors against premature labor
05/14/1999WO1999007692A3 New epothilone derivatives, method for producing same and their pharmaceutical use
05/14/1999WO1999001124A9 Synthesis of epothilones, intermediates thereto, analogues and uses thereof
05/14/1999CA2308639A1 Method of using cyclooxygenase-2 inhibitors in maintaining the fetal ductus ateriosus during treatment and prevention of preterm labor
05/12/1999EP0914605A1 Molecular model for vla-4 inhibitors
05/12/1999CN1216545A Farnesyl transferase inhibitors
05/11/1999US5902818 N-halogenated, oxazolidinone monomers having an acrylic ester group at the 4-position release small amounts free halogens; disinfectants such as medical and dental coatings, fabrics; cost efficiency, performance
05/06/1999WO1999021843A1 4, 5-diaryloxazole compounds
05/06/1999WO1999021422A1 Treatment of schizophrenia with ampakines and neuroleptics
05/06/1999EP0912533A1 Alkylaminobenzothiazole and -benzoxazole derivatives
05/06/1999EP0912510A1 Nickel catalyzed addition of -nh- containing compounds to vinyl and aryl halides
05/06/1999EP0912504A1 Process to prepare taxol
05/06/1999EP0684242B1 Isoxazolidinedione derivative and use thereof
05/06/1999DE19749717A1 New epothilone derivatives
05/06/1999DE19747644A1 Sterically hindered phenols for stabilizing polymers, oils and lubricants
05/06/1999CA2307952A1 4, 5-diaryloxazole compounds
05/06/1999CA2306817A1 Treatment of schizophrenia with ampakines and neuroleptics
05/05/1999CN1216043A Substd. benzenesulfonamide derivs as prodrugs of COX-2 inhibitors
05/05/1999CN1216039A Process to prepare taxol
05/05/1999CN1215724A Novel compounds
04/1999
04/29/1999DE19748928A1 New epothilone derivatives
04/28/1999EP0911324A1 Process for the preparation of chiral succinic acid derivatives
04/28/1999EP0559738B1 Methods for detection and quantitation of cell subsets within subpopulations of a mixed cell population
04/28/1999CN1215400A Piperazine and piperidine compounds
04/28/1999CN1215393A Process to prepare oxazolidinones
04/22/1999WO1999019299A1 Heterocycles useful in the treatment of benign prostatic hyperplasia and intermediates thereof
04/22/1999WO1999019296A1 Aminobutanoic acid derivatives
04/22/1999WO1999018941A2 Ih-MODULATORS
04/22/1999WO1999006361A3 N-hydroxyformamide derivatives as inhibitors of matrix metalloproteinases
04/22/1999WO1999002146A8 Amino acid derivatives
04/22/1999CA2305353A1 Heterocycles useful in the treatment of benign prostatic hyperplasia and intermediates thereof
04/22/1999CA2305180A1 Ih-modulators
04/21/1999EP0695184B1 Hiv protease inhibitors
04/15/1999WO1999018091A1 Novel compounds useful as neuro-protective agents
04/15/1999WO1999018084A1 Method and reagents for n-alkylating ureides
04/15/1999DE19812409C1 Coupling agents for polymers, oligomers, organic compounds and inorganic substances
04/15/1999CA2305538A1 Novel compounds useful as neuro-protective agents
04/14/1999EP0908454A2 Oxazoles, thiazoles, oxazolines, oxadiazoles and benzoxazoles useful as neuro-protective agents
04/14/1999EP0908186A2 Method for treating pain
04/14/1999EP0908180A2 Use of phenyl oxazole or phenyl thiazole derivatives for treating pain
04/14/1999EP0907661A1 METHODS AND COMPOSITIONS USEFUL FOR INHIBITION OF alpha v beta 5 MEDIATED ANGIOGENESIS
04/14/1999EP0907653A1 Process for the preparation of penam and penem derivatives
04/14/1999EP0907634A1 Pesticides
04/14/1999EP0907633A1 New synthetic catechol derivatives, method for production and use thereof
04/14/1999CN1213663A Process for manufacture of chiral succinic acid derivatives of formula
04/13/1999CA1340492C Novel naphthyridine-and quinoline-carboxylic acids as bacterial agents
04/08/1999WO1998054161A9 Oxazolidinone antibacterial agents having a thiocarbonyl functionality
04/07/1999EP0906755A2 Use of phenyl oxazole or phenyl thiazole derivatives for treating neuropathic pain
04/07/1999EP0906268A1 Alkyloxyamino substituted fluorenones and their use as protein kinase c inhibitors
04/07/1999EP0868182A4 Process for production of piperidine derivatives
04/07/1999EP0681474B1 Pharmaceutical composition containing 5-morpholinomethyl-3-(4-chlorobenzylideneamine)-2-oxazolidinone and its use for the treatment of cns disorders
04/07/1999EP0659181B1 Sulfonamide inhibitors of hiv-aspartyl protease
04/07/1999EP0609281B1 Benzoxazole, benzothiazole and benzimidazole derivatives as fungicides
04/06/1999US5892052 Process for making retroviral protease inhibiting compounds
04/06/1999US5891876 Alpha-amino-3-hydroxy-5-methyl-isoxazole-4-propionic acid (ampa); drugs that enhance these receptor currents will facilitate communication in brain networks responsible for perceptual-motor integration and higher order behaviors
04/03/1999CA2247580A1 Process for preparing chiral succinic acid derivatives
04/01/1999WO1999015894A2 Method of identification of leads or active compounds
04/01/1999WO1999014998A2 Method for preventing and treating hearing loss using sensorineurotrophic compounds
04/01/1999CA2304783A1 Method of identification of leads or active compounds
04/01/1999CA2304647A1 Method for preventing and treating hearing loss using sensorineurotophic compounds
03/1999
03/31/1999EP0905512A1 Method of identification of leads or active compounds
03/31/1999EP0905255A2 Process for the preparation of pharmaceutically active thiazolidine or oxazolidine compounds by a yeast reductase
03/31/1999EP0905139A2 5 ring heterocyles, process for preparation, use as inhibitors of leukocyte adhesion and pharmaceutical preparations comprising them
03/31/1999EP0904274A1 Farnesyl transferase inhibitors
03/31/1999EP0904262A1 Conformationally restricted aromatic inhibitors of microsomal triglyceride transfer protein and method
03/31/1999EP0904079A1 Antidiabetic agents
03/31/1999EP0904077A2 Methods for the preparation of biphenyl isoxazole sulfonamides
03/31/1999EP0877733A4 Process for production of piperidine derivatives
03/31/1999EP0773778B1 Hair styling composition and method
03/31/1999CN1212691A Tricyclic compound and its preparation and use
03/30/1999US5889165 Photolabile nucleoside protecting groups
03/30/1999US5889130 Monomeric and polymeric cyclic amine and N-halamine compounds
03/30/1999US5889059 Phenylacetic acid derivatives, preparation thereof and intermediates therefor, and compositions containing them
03/30/1999US5889037 Prevention, therapy tissue damage from lipid peroxidation
03/30/1999US5889014 Heterocyclic compounds for inhibiting phosphodiesterase IV
03/25/1999WO1999014205A1 New 2-(3h)-oxazolone derivatives
03/24/1999EP0902782A1 Urea derivatives as inhibitors of impdh enzyme
03/23/1999US5886043 Antiarthritic agents, antitumor agents, antiinflammatory agents
03/23/1999US5886036 Treating hiv infections
03/23/1999US5886024 Thiophene-containing butonic acid derivatives as matrix metalloprotease inhibitors
03/23/1999US5886022 Treatment of osteoarthritis, rheumatoid arthritis, septic arthritis, periodontal disease, corneal ulceration, proteinuria, aneurysmal aortic disease, dystrophobic epidermolysis bullosa
03/23/1999CA2247735A1 Novel 5-membered ring heterocycles, their preparation, their use and pharmaceutical preparations comprising them
03/18/1999WO1999012924A1 Piperidinylmethyloxazolidinone derivative
03/18/1999WO1999012914A1 Thiourea derivatives
03/18/1999WO1999012903A1 Benzimidazolinones, benzoxazolinones, benzopiperazinones, indanones, and derivatives thereof as inhibitors of factor xa
03/18/1999CA2303438A1 Benzimidazolinones, benzoxazolinones, benzopiperazinones, indanones, and derivatives thereof as inhibitors of factor xa
03/17/1999EP0902034A2 Very large scale immobilized peptide synthesis
03/17/1999EP0902017A1 Transesterification process
03/17/1999EP0902013A1 Novel amidine derivatives, their preparation and their use as medicaments with LTB-4 antagonistic effect
03/17/1999EP0901789A1 Method of treating tourette's syndrome
03/17/1999EP0901372A1 Potassium, sodium and tris oxaprozin salt pharmaceutical formulations
03/17/1999CN1211183A Methods for preparation of biphenyl isoxazole sulfonamides
03/17/1999CN1210858A Optically active bisoxazoline compounds production and use thereof