Patents
Patents for C07D 263 - Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings (20,978)
10/1999
10/26/1999US5973111 Novel compounds that are capable of binding to the active site of interleukin-1b-converting enzyme (ice) and inhibiting activity of that enzyme; administering to treat inflammatory, autoimmune, and neurodegenerative diseases
10/26/1999US5972970 Oxazolidinedione derivatives, their production and use
10/26/1999US5972968 Interleukin inhibitor
10/26/1999US5972965 4,5-diaryl oxazole derivatives
10/26/1999US5972959 Oxime derivatives, their preparation and their therapeutic use
10/26/1999US5972241 Liquid crystal compounds having a chiral fluorinated terminal portion
10/21/1999WO1999052876A1 Azacycloalkane derivatives, preparation and therapeutic application
10/21/1999WO1999052874A1 Difluoroalkene derivatives, process for producing the same, and agricultural or horticultural pest control agent
10/21/1999WO1999052850A1 Oxidation process using periodic acid
10/21/1999WO1999052849A1 Oxidation process using tempo
10/21/1999DE19816880A1 New diaryl substituted heterocyclic compounds are AMPA receptor antagonists useful in treatment of neurodegenerative disorders and cerebral ischemia
10/21/1999CA2327929A1 Oxidation process using periodic acid
10/21/1999CA2327890A1 Oxidation process using tempo
10/20/1999EP0950056A2 N-(pyridinylamino)isoindolines and related compounds
10/20/1999EP0832078B1 N-hydroxyureas as antiinflammatory agents
10/20/1999EP0717738B1 Substituted oxazine and thiazine oxazolidinone antimicrobials
10/20/1999CN1232025A Pyrrolidine and piperidine derivatives
10/19/1999US5969147 Pesticides, parasiticides, miticides
10/19/1999US5968985 Benzoylguanidine derivatives as medicaments
10/19/1999US5968977 Ketonitrile derivatives and antibacterial agent and drugs containing the same
10/19/1999US5968970 Treatment of hiv
10/19/1999US5968962 Phenyloxazolidinones having a C-C bond to 4-8 membered heterocyclic rings
10/16/1999CA2269049A1 N-acyl and n-aroyl aralkyl amides
10/13/1999EP0949242A1 Aromatic amine derivatives having nos inhibitory effect
10/13/1999EP0949238A1 Substituted propionyl derivatives
10/13/1999EP0948490A1 Process for the preparation of 2-imino-5-phenyl-4-oxazolidinone and its intermediates
10/13/1999EP0948324A2 Methods and pharmaceutical compositions for inhibiting tumour cell growth
10/13/1999EP0783486B1 Novel prostaglandin synthase inhibitors
10/13/1999CN1045597C Alkylenediamine derivatives having heterocyclic group and medicinal composition thereof
10/12/1999US5965774 Substituted anilide derivative
10/12/1999US5965739 Oxazolidine protected taxol analogs of given formula, and methods of synthesis from an oxazolidine free acid and a baccatin compound in the presence of a dehydrating agent; useful intermediates to make various taxol analogues
10/12/1999US5965601 Novel compounds for inhibiting replication of a retrovirus; treating hiv
10/12/1999US5965584 Pharmaceutical composition
10/12/1999US5965558 2 or 2,3-di((2-carboxyethylenearyl)quinoxalines; purification of proteins and glycoproteins; units including protein tyrosine phosphatases and proteins with src-homology-2 domains; antidiabetics,-allergens,-coagulants
10/12/1999US5965539 Peptidomimetics; anti-cancer drugs
10/12/1999US5965054 Comprising salts consisting of alkyl substituted, nitrogen-containing heterocyclic delocalized aromatic cations, and their perfluoro derivatives; high energy, high voltage
10/12/1999CA1340785C Platelet activating factor antagonists
10/07/1999WO1999050267A1 Process for producing isooxazolidinedione compound
10/07/1999WO1999050205A2 Asymmetric grignard synthesis with cyclic 1,2 aminoalcohols
10/06/1999EP0946689A1 Antioxidants and antioxidant boosters capable of producing hydroperoxyl radicals
10/06/1999EP0946528A2 OXYGEN OR SULFUR CONTAINING 5-MEMBERED HETEROAROMATICS AS FACTOR Xa INHIBITORS
10/06/1999EP0946519A1 Benzamide derivatives having a vasopressin antagonistic activity
10/06/1999EP0946518A1 Modulators of proteins with phosphotyrosine recognition units
10/06/1999EP0946499A1 N-(aryl/heteroaryl/alkylacetyl) amino acid amides, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds
10/06/1999CN1230958A Oxazolone derivatives and their use as anti-helicobacter pylori agents
10/06/1999CN1230542A Sidechain-bearing taxanes
10/05/1999US5962725 Chemical intermediate; blocks reproduction of virus
10/05/1999US5962683 Oxazoline compounds as stabilizers
10/05/1999US5962640 Methods for preparing novel dipeptide compounds or pharmacuetically acceptable salts thereof
10/05/1999US5962495 Estrogen sensitive diseases; breast cancer; prostate tumors
10/05/1999US5962489 Fungicides
10/05/1999US5962470 Heterocyclic compounds having anti-diabetic activity and their use
10/05/1999US5962439 Cardiovascular disorder
09/1999
09/30/1999WO1999048897A2 Synthesis of compounds and libraries of compounds
09/30/1999CA2324016A1 Synthesis of compounds and libraries of compounds
09/29/1999EP0945448A1 5-alkoxy-2(3h)-oxazolone compounds and process for the preparation thereof
09/29/1999EP0945431A2 Process and intermediates for the preparation of phenylacetic derivatives
09/29/1999EP0944622A1 2-imidazolinylaminobenzoxazole compounds useful as alpha-2 adrenoceptor agonists
09/29/1999EP0944608A1 4-cyclohexylphenyl-oxazolines and their use for controlling animal pests
09/29/1999EP0944604A1 Guanidinyl heterocycle compounds useful as alpha-2 adrenoceptor agonists
09/29/1999EP0944590A2 Aminoguanidines and alkoxyguanidines as protease inhibitors
09/29/1999EP0811005B1 Herbicidal benzoyl derivatives
09/29/1999CN1230211A Antioxidants and antioxidant boosters capable of producing hydroperoxyl radicals
09/29/1999CN1230110A Cell adhesion inhibitors
09/29/1999CN1229795A Heterocyclic compounds
09/28/1999US5959114 Process to chloroketones using oxazolines
09/28/1999US5958839 Herbicidal compounds
09/28/1999US5958838 Controlling weeds in crops.
09/28/1999US5958683 Screening method using the RZR receptor family
09/28/1999CA2157032C Isoxazolidinedione derivative and use thereof
09/23/1999WO1999047525A1 Herbicidally active 3-hydroxy-4-aryl-5-oxopyrazoline derivatives
09/23/1999DE19813821A1 New epothilone derivatives
09/23/1999DE19812408A1 Oxazoline- or oxazine-carboxylic acids which undergo polyaddition reactions to give linear polyester-amide or copolymers, useful as blend components
09/22/1999CN1229080A Processes for preparing intermediate product used in method of diastereoselective syntheses of nucleosides
09/22/1999CN1229079A Processes for preparing intermediate product used in method of diastereoselective syntheses of nucleosides
09/22/1999CN1229078A Processes for preparing intermediate product used in method of diastereoselective syntheses of nucleosides
09/22/1999CN1045206C Method for preparing cyclic amide derivative
09/16/1999WO1999046252A1 Process for producing oxazolidin-2-one derivatives
09/16/1999WO1999046246A1 Hetaryl-substituted benzyl phenyl ethers, method for the production thereof, and their use for combating harmful fungi and animal pests
09/16/1999WO1999046243A1 Process for the enantioselective synthesis of hydroxypyrrolidines from amino acids and products thereof
09/16/1999WO1999046232A1 Carboxylic acid derivatives and drugs containing the same as the active ingredient
09/16/1999DE19807502A1 Verfahren zur Nachvernetzung von Hydrogelen mit 2-Oxazolidinonen Method for post-crosslinking of hydrogels with 2-oxazolidinones
09/15/1999EP0941215A1 Glyoxylic acid amides and their use as pesticides
09/15/1999EP0749421B1 Sulphonamide derivatives as aspartyl protease inhibitors
09/15/1999EP0741697B1 Amino acid derivatives and their use as phospholipase a2 inhibitors
09/15/1999CN1228414A New benzocyclobutane compounds, process for their preparation and pharmaceutical compositions containing them
09/15/1999CN1045084C Novel compound with platelet aggregation inhibitor activity and its use, and drug composition containing the same
09/14/1999US5952507 Process for manufacture of chiral succinic acid derivatives
09/14/1999US5952362 2-imidazoline, 2-oxazoline, 2-thiazoline, and 4-imidazole derivatives of methylphenyl, methoxyphenyl, and aminophenyl alkylsulfonamides and ureas and their use
09/14/1999US5952360 Admisnistering to a mammal certain phenyl oxazoles or phenyl thiazoles
09/14/1999US5952359 Thiazoles and their agricultural compositions
09/14/1999US5952356 Treating diabetes in a mammal with an active material and a glucosidase inhibitor
09/14/1999US5952316 2-amino-1,3-propanediol compound and immunosuppressant
09/14/1999CA2144125C Use of sulfonic acids as antiageing agents in a cosmetic or dermatologic composition
09/08/1999EP0940386A1 Benzocyclobutan compounds, their process for preparation and pharmaceutical compositions containing them
09/08/1999EP0940139A2 Substituted guanidines and derivatives thereof as modulators of neurotransmitter release and novel methodology for identifying neurotransmitter release blockers
09/08/1999EP0939755A1 Oxazoline arthropodicides
09/08/1999EP0749415B1 Benzamide analogs, useful as parp (adp-ribosyltransferase, adprt) dna repair enzyme inhibitors
09/02/1999WO1999043730A1 Epoxy resin hardener and one-pack type epoxy resin composition
09/02/1999WO1999043720A1 Method for cross-linking hydrogels with bis- and poly-2-oxazolidinones