Patents
Patents for C07D 263 - Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings (20,978)
12/2002
12/19/2002WO2002100841A1 PROCESSES FOR PRODUCING OXAZOLIDINONE DERIVATIVE OF ß-HYDROXYETHYLAMINE COMPOUND AND FOR PRODUCING ß-HYDROXYETHYLAMINE COMPOUND
12/19/2002WO2002100835A1 Heterocyclic compounds having antitumor activity
12/19/2002WO2002100818A2 Aminediols as agents for the treatment of alzheimer's disease
12/19/2002WO2002100403A1 Modulators of peroxisome proliferator activated receptors (ppar)
12/19/2002WO2002070541A3 Peptide deformylase inhibitors
12/19/2002US20020193607 Enantioselective synthesis of azetidinone intermediate compounds
12/19/2002US20020193596 Inhibitors of protein isoprenyl transferases
12/19/2002US20020192693 Apparatus for polymer synthesis
12/19/2002DE10129940A1 Medicament used for treating central nervous system disorders e.g. psychosis, depression or neurological disorders, comprises new or known 4-phenylsulfonyl-oxazole-5-amine derivative which are serotonin 5-HT6 receptor ligands
12/19/2002CA2450269A1 Hiv protease inhibitors, compositions containing the same, their pharmaceutical uses and materials for their synthesis
12/19/2002CA2450265A1 Hiv protease inhibitors, compositions containing the same, their pharmaceutical uses and materials for their synthesis
12/19/2002CA2450205A1 Aminediols for the treatment of alzheimer's disease
12/19/2002CA2448552A1 Modulators of peroxisome proliferator activated receptors (ppar)
12/18/2002EP1265887A2 Carbocyclic side chain containing metalloprotease inhibitors
12/18/2002EP1265886A2 Carbocyclic side chain containing, n-substituted metalloprotease inhibitors
12/18/2002EP1265876A1 Preparation of mixtures of benzoxazolyl-stilbene compounds
12/18/2002EP1265853A1 Carboxylic acid derivatives as ip antagonists
12/18/2002EP1265606A1 Cell adhesion inhibitors
12/18/2002CN1386120A 萘酚衍生物 Naphthol derivative
12/18/2002CN1096446C N-(ortho-substd-benzyloxy)imine derivs, and their use as fungicides, acaricides or insecticides
12/18/2002CN1096265C Preparation of pharmaceutical composition containing novel thiazolidone and oxazolidone
12/17/2002US6495581 Drug for treating diabetes mellitus, hyperlipemia, impaired glucose tolerance, arterial sclerosis and improving insulin resistance, inflammatory disease
12/17/2002CA2216569C Use of oxazolidinone derivatives as anti-penetrating agents in a cosmetic and/or dermatological composition
12/12/2002WO2002098867A1 Production process for 5-alkyl-oxazolidin-2,4-dione
12/12/2002WO2002098850A2 Chemical compounds and pharmaceutical compositions as cathepsin s inhibitors
12/12/2002WO2002098406A1 Novel compounds and compositions as cathepsin inhibitors
12/12/2002US20020188133 Producing an isoxazolidinedione compound from beta - methyl L-aspartate via an important intermediate oxazolylethanol derivative
12/12/2002US20020188120 Such as 4-(4-methyoxy-benzenesulfonyl)-1-(3-phenyl-propyl)-piperidine-4-carboxylic acid hydroxyamide for treatment of arthritis, tumor metastasis, tissue ulceration, abnormal wound healing, periodontal disease, bone diseases, diabetes, and HIV
12/12/2002US20020188095 Method of manufacturing N-carboxyamino acid anhydride and polyamino acid
12/12/2002US20020187982 Glucagon antagonists/inverse agonists
12/12/2002US20020187979 3-heterocyclylpropanohydroxamic acid PCP inhibitors
12/12/2002CA2449021A1 Novel compounds and compositions as cathepsin inhibitors
12/12/2002CA2448418A1 Chemical compounds and pharmaceutical compositions as cathepsin s inhibitors
12/11/2002EP1264820A1 Novel amide compounds
12/11/2002EP1263744A1 Nematicidal trifluorobutenes
12/11/2002EP1263743A1 Heterocycle substituted diphenyl leukotriene antagonists
12/11/2002EP1263742A1 Oxazolidinone thioamides with piperazine amide substituents
12/11/2002EP1263718A1 Novel use of phenylheteroalkylamine derivatives
12/11/2002EP1263711A1 Novel use of phenylheteroalkylamine derivatives
12/11/2002EP0624155B2 Carbamates and plant-protecting agents containing them
12/11/2002CN1384824A Process for preparation of oxazole derivatives
12/11/2002CN1384823A Processes for preparation of oxo-oxazoline or alloamino acid derivatives
12/11/2002CN1095839C 4,5-diaryl oxazole derivatives
12/11/2002CN1095838C 4-cyclohexyl phenyl-oxazolines and their use for controlling animal pests
12/11/2002CN1095835C Tricyclo-substituted isohydroxyloxime acid derivative
12/10/2002US6492555 Reaction of a carbamate with either a (s)-secondary alcohol or (s)-epoxide or (s)-ester; bactericides
12/10/2002US6492396 Substituted thioacetamides
12/10/2002US6491871 System for determining receptor-ligand binding affinity
12/05/2002WO2002096872A1 Substituted imidates as pesticidal agents
12/05/2002WO2002096516A1 Use of compositions comprising cyclooxygenase-2 selective inhibitors in combination with radiation for inhibition or prevention of cardiovascular disease
12/05/2002WO2002051819A3 Heterocyclic compounds having antibacterial activity, process for their preparation and pharmaceutical compositions containing them
12/05/2002WO2001093840A2 Ligands of integrin receptors
12/05/2002US20020183551 Process for the preparation of N-carboxyanhydrides
12/05/2002US20020183397 Substituted n-phenyl-n-fused-benzyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
12/05/2002US20020183371 Oxazolidinone combinatorial libraries, compositions and methods of preparation
12/05/2002US20020183334 For therapy of sleepiness, promotion of wakefulness, treatment of Parkinson's disease, cerebral ischemia, stroke, sleep apneas, eating disorders, stimulation of appetite and weight gain, treatment of attention deficit hyperactivity disorder
12/05/2002US20020183315 Amino-substituted compounds useful as inhibitors of impdh enzyme
12/05/2002DE10125963A1 Substituierte Imidate Substituted Imidates
12/05/2002CA2447657A1 Use of compositions comprising cyclooxygenase-2 selective inhibitors in combination with radiation for inhibition or prevention of cardiovascular disease
12/05/2002CA2411549A1 Ligands of integrin receptors
12/04/2002EP1262480A1 Process for the preparation of N-carboxyanhydrides of amino acids
12/04/2002EP1261600A1 Heteroaromatic carboxamide derivatives and their use as inhibitors of the enzyme ikk-2
12/04/2002EP1111993A4 Fused-benzene derivatives useful as herbicides
12/04/2002EP1001930B1 N-hydroxyformamide derivatives as inhibitors of matrix metalloproteinases
12/03/2002US6489365 Ltb4-antagonistic compounds for treatment of inflammation, allergy or gastropathy induced by non-steroidal antiinflammatory agents in a warm-blooded animals
12/03/2002US6489268 Highly selective herbicidal phenoxypropionic acid alkoxycarbonyl anilid compounds and method of preparing the same
12/03/2002CA2263500C Malonate derivatives useful as intermediates for producing isoxazolidinadione hypoglycemic agents
12/03/2002CA2074933C Thiazole derivatives as active superoxide radical inhibitors
11/2002
11/28/2002WO2002094809A1 3-quinoline-2-(1h)-ylideneindolin-2-one derivatives
11/28/2002WO2002094770A2 Aminoalcohol derivatives
11/28/2002WO2002094765A2 Substituted aromatic amide derivative, intermediate thereof, agrohorticultural insecticide containing thereof and method for the use thereof
11/28/2002WO2002079753A3 2-aminobenzoxazole derivatives and combinatorial libraries thereof
11/28/2002WO2002048106A3 Isoindolin-1-one glucokinase activators
11/28/2002WO2002009759A3 Aldosterone antagonist and cyclooxygenase-2 inhibitor combination therapy to prevent or treat inflammation-related cardiovascular disorders
11/28/2002US20020177707 Aminoaryl oxazolidinone n-oxides
11/28/2002US20020177595 Novel compounds useful as neuro-protective agents
11/28/2002US20020177594 Inhibitors of histone deacetylase
11/28/2002CA2448076A1 3-quinoline-2-(1h)-ylideneindolin-2-one derivatives
11/27/2002EP1259495A2 Indane derivatives and their use as cell adhesion inhibitors
11/27/2002EP1259491A1 4-imidazole derivatives of benzyl and restricted benzyl sulfonamides, sulfamides, ureas, carbamates and amides and their use as alpha-1a agonists
11/27/2002EP0862557B1 SYMMETRICAL bis-HETEROARYLMETHOXYPHENYLALKYL CARBOXYLATES AS INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS
11/27/2002CN1381454A Method for preparing oxazolidone amine
11/27/2002CN1381447A Method for preparing N-[1-(S)-carbethoxy-3-hydrocinnamyl] -L-alanine-N-carboxy acid anhydride
11/27/2002CN1094943C Urethanes and ureas that induce cytokine production
11/26/2002US6486098 Herbicidal phenoxypropionic acid N-alkyl-N-2-fluorophenyl amide compounds
11/26/2002CA2148103C Process for preparing taxane derivatives
11/25/2002WO2001090087A1 Heterocyclic compounds
11/25/2002CA2410382A1 Heterocyclic compounds
11/21/2002WO2002092734A1 Antioxidants and antioxidant boosters capable of producing hydroperoxyl radicals
11/21/2002WO2002092595A1 Broadspectrum 2-amino-benzoxazole sulfonamide hiv protease inhibitors
11/21/2002WO2002092084A1 Carboxylic acid substituted oxazole derivatives for use as ppar-alpha and -gamma activators in the treatment of diabetes
11/21/2002WO2002028841B1 Reagents for labeling biomolecules having aldehyde or ketone moieties
11/21/2002US20020173664 An 3-acyl-4-substituted-oxazolidin-2,5-dione that readily reacts with nucleophilic reagents such as free amino acids; use in peptide synthesis for example
11/21/2002US20020173526 Heterocyclic compounds their production and use
11/20/2002EP1258491A1 Amino acid hydroxyethylamino sulfonamide retroviral protease inhibitors
11/20/2002EP1258473A1 Benzoic acid derivatives, process for producing the same and drugs containing the same as the active ingredient
11/20/2002EP1165472A4 Methods for the preparation of biphenyl isoxazole sulfonamides
11/20/2002EP1147101B1 Reverse hydroxamate inhibitors of matrix metalloproteinases
11/20/2002EP1077966B1 Biphenyl sulfonyl aryl carboxylic acids useful in the treatment of insulin resistance and hyperglycemia
11/20/2002CN1380881A Methods for crystallization of N-(1-(s)-ethoxycarbonyl-3-phenylpropyl)-L-alanine N-carboxyanhydride