Patents
Patents for C07D 263 - Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings (20,978)
07/2003
07/22/2003CA2276203C N-(pyridinylamino)isoindolines and related compounds
07/17/2003WO2003057666A2 Inhibitors of dipeptidyl peptidase iv
07/17/2003WO2003057661A1 Prodrugs of excitatory amino acids
07/17/2003WO2003057144A2 Change inhibitors of dipeptidyl peptidase iv
07/17/2003US20030135051 Intermediates for making HIV-protease inhibitors and methods for making HIV-protease inhibitors
07/17/2003US20030134884 Benzyloxyiminohydrocarbylcarboxy compounds, such as E-4-(4-(5-methyl-2-phenyl-4-oxazolylmethoxy)benzyloxyimino)--4-phenylbutyric acid
07/17/2003US20030134859 Substituted 2-chloro-5-nitrobenzamides; treating retrograde osteoporosis and diabetes mellitus
07/17/2003US20030134237 Methine dyes, manufacturing methods thereof, and silver halide photoraphic materials contaning same dyes
07/17/2003CA2471204A1 Inhibitors of dipeptidyl peptidase iv
07/16/2003EP1326861A1 Alpha-aryl ethanolamines and their use as beta-3 adrenergic receptor agonists
07/16/2003EP1326850A1 A process for the preparation of bis-benzazolyl compounds
07/16/2003EP1326840A2 Substituted heterocyclic compounds for treating multidrug resistance
07/16/2003EP1326834A2 2-substituted heterocyclic compounds
07/16/2003EP1326833A2 Substituted heterocyclic compounds for treating multidrug resistance
07/16/2003CN1430618A Thiazine oxazolidinone
07/16/2003CN1430612A Hete rocyclic derivatives
07/16/2003CN1430607A Benzophenones as inhibitors of IL-1 beta and TNF-alpha
07/16/2003CN1430602A Ary-and heteroaryl sulfonates compounds
07/16/2003CN1430596A New gamma selective retinoids
07/16/2003CN1429822A Chiral dibenz [a,c] suberyl diallyl double oxazoline ligand compound and its preparation and application
07/15/2003US6593489 Catalytic stereoselective hydrogenation
07/15/2003US6593354 Substituted benzoxazole compounds
07/15/2003US6593347 Nitrosated and nitrosylated nonsteroidal antiinflammatory compounds, compositions and methods of use
07/10/2003WO2003055868A1 Benzothiazole- and benzoxazole-4,7-dione derivatives and their use as cdc25 phosphatase inhibitors
07/10/2003WO2003055861A1 Benzocyclodecane derivatives with antitumor activity
07/10/2003WO2003055850A1 β-AMYLOID PROTEIN PRODUCTION/SECRETION INHIBITORS
07/10/2003WO2003055847A1 Carboxylic acid derivative
07/10/2003WO2003055463A1 Composition comprising at least an oxazolin for inhibiting langerhans cell migration, and uses thereof
07/10/2003WO2003032908A3 Novel prodrugs of n-h bond-containing compounds and methods of making thereof
07/10/2003WO2003006440A8 Amide-containing compound having improved solubility and method of improving the solubility of an amide-containing compound
07/10/2003US20030130509 Process to produce 3-carbon amino alcohol salts
07/10/2003US20030130383 Ultraviolet radiation absorbents for thermoplastic polymers and methods of producing same
07/10/2003US20030130345 C2-substituted idan-1-ones and their derivatives, processes for their preparation and their use as pharmaceuticals
07/10/2003US20030130232 Amidine derivatives, the preparation and use thereof as medicaments with LTB4 antagonistic effect
07/10/2003CA2482392A1 Carboxylic acid derivative
07/10/2003CA2471910A1 Benzocyclodecane derivatives with antitumor activity
07/10/2003CA2471713A1 Benzothiazole- and benzoxazole-4,7-dione derivatives and their use as cdc25 phosphatase inhibitors
07/09/2003EP1325917A1 Radiolabelled alkylamino-benzothiazole and -benzoxazole derivatives and their use as D4 ligands
07/09/2003EP1324989A1 5-trityloxymethyl-oxazolidinones and process for the preparation thereof
07/09/2003EP1324988A1 Process for the preparation of 5-hydroxymethyl 2-oxazolidinone and novel intermediate
07/09/2003EP1156798B1 Felbamate derived compounds
07/09/2003EP0966465B1 Inhibitors of impdh enzyme
07/09/2003CN1429226A Piperazine and piperidine compounds
07/09/2003CN1429210A Substituted thioacetamides
07/09/2003CN1113875C Substituted aromatic thiocarboxylic acid amides and their use as herbicides
07/09/2003CN1113602C Tetra-substituted phenyl oxazolidone herbicides
07/08/2003US6589971 A method of treatment of a neoplastic disease in a patient in need of said treatment by administering a therapeutically effective amount of a compound of the formula: bind to specific sequences in the minor groove of duplex DNA, and to
07/08/2003US6589915 The invention relates to cyclohexenone derivatives of benzo-condensed, unsaturated 5-ring nitrogen heterocycles of general formula (I) wherein X represents N or a group C-R3, Y represents O, S, SO, SO2 or NR4 or X-Y represent S
07/08/2003US6589914 Dihalopropene compounds, insecticidal/acaridcidal agents containing same, and intermediates for their production
07/08/2003CA2285208C Improved method for producing thiazolidinediones, and new thiazolidinediones
07/08/2003CA2272640C Guanidinyl heterocycle compounds useful as alpha-2 adrenoceptor agonists
07/08/2003CA2264372C New benzocyclobutane compounds, their method of preparation, and pharmaceutical compositions containing them
07/03/2003WO2003053927A1 Piperazine derivative
07/03/2003WO2003053885A1 Method for forming a carbon-carbon or carbon-heteroatom linkage
07/03/2003WO2003053435A1 Broadspectrum heterocyclic substituted phenyl containing sulfonamide hiv protease inhibitors
07/03/2003US20030125567 Converting alpha- isocyanoalkanoate esters in the presence of assistants at temperatures above 80 degrees C. into the 5-alkoxy-substituted oxazoles, and removing the reaction product from the reaction mixture
07/03/2003US20030125367 Administering a patient with bacterial infections a oxazolidinones having a bicylcic/3.1.0/ hexane containing group as antibiotic
07/03/2003US20030125365 Inhibitors of the beta-secretase enzyme that are useful in the treatment of Alzheimer's disease
07/03/2003US20030125362 Synthesis of epothilones, intermediates thereto, analogues and uses thereof
07/03/2003US20030125329 Treating atherosclerosis and other coronary artery diseases
07/03/2003US20030125328 Treating atherosclerosis and other coronary artery diseases
07/03/2003CA2470964A1 Broadspectrum heterocyclic substituted phenyl containing sulfonamide hiv protease inhibitors
07/03/2003CA2470808A1 Piperazine derivative
07/03/2003CA2470141A1 Method for forming a carbon-carbon or carbon-heteroatom linkage
07/02/2003EP1322625A2 Reagents for labeling biomolecules having aldehyde or ketone moieties
07/02/2003CN1427834A Process for preparation of citalopram
07/01/2003US6586471 Halogenated 2-amino-3, 4 heptenoic acid derivatives useful as nitric oxide synthase inhibitors
07/01/2003US6586433 Anticholesterol agents; antilipemic agents; cardiovascular disorders
06/2003
06/26/2003WO2003051852A1 Intermediate and process for producing optically active compound from the intermediate
06/26/2003WO2003051842A2 Compositions decreasing activity of hormone-sensitive lipase
06/26/2003WO2003051841A2 Compounds and uses thereof for decreasing activity of hormone-sensitive lipase
06/26/2003US20030120082 Cyclization and acidification of 4-methyl-5-n-butoxyoxazole within tubular reactor
06/26/2003US20030119902 Novel aminobenzoephenones
06/26/2003US20030119886 Nonsteroidal antiinflammatory agents, e.g., N-hydroxy-1-(4-sulfonyl or aminosulfonyl)phenyl)-(ring- substituted hetero-cyclyl)alkanamide or -urea; dual enzyme inhibitors with minimal side effects; asthma; antiallergens; antipyretics
06/26/2003US20030119868 Gyrase inhibitors and uses thereof
06/26/2003US20030119849 Piperazine and piperidine compounds
06/26/2003US20030119833 Treating cardiovascular diseases
06/26/2003US20030119814 Novel prodrugs of N-H bond-containing compounds and methods of making thereof
06/26/2003US20030119807 Inhibit Procollagen C-proteinase; antiscarring treatment for wounds.
06/26/2003US20030119031 Fluroescence analysis; controlling transcription factors; bactericides, viricides, anticancer agents, fungicides, antiprotozoa agents
06/26/2003US20030119008 Nucleotides and analogs having photoremovable protecting groups
06/26/2003CA2468413A1 Compounds and uses thereof for decreasing activity of hormone-sensitive lipase
06/25/2003EP1320518A2 Preparation of enantiomerically-enriched cyclopropylalanine derivatives
06/25/2003EP1320365A1 Substituted azole derivatives as inhibitors of corticotropin releasing factor
06/25/2003EP1224178B1 Crystals of an oxyiminoalkanoic acid derivative and their use as antidiabetics
06/25/2003CN1426303A Thiazole, imidazole and oxazole compounds and treatments of disorder associated with protein aging
06/24/2003US6583292 Method for the esterification of alcohols and compounds useful therefor as potential anticancer agents
06/24/2003US6583183 Substituted n-phenyl-n-fused-benzyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
06/24/2003US6583090 Hetaryl-substituted benzyl phenyl ethers, method for the production thereof, and their use for combating harmful fungi and animal pests
06/24/2003CA2126337C 2-amino-1,3-propanediol compound and immunosuppressant
06/19/2003WO2003050095A1 Substituted benzoxazoles and analogues as estrogenic agents
06/19/2003WO2003050073A1 Substituted hydroxyethylamines
06/19/2003WO2003050063A2 PROCESS FOR THE SYNTHESIS OF CHIRALLY PURE β-AMINO-ALCOHOLS
06/19/2003WO2003049702A2 Vanilloid receptor ligands and their use in treatments
06/19/2003WO2003028650A3 Benzimidazolidinone derivatives as muscarinic agents
06/19/2003US20030114681 C2-substituted indan-1-ols and their derivatives, processes for their preparation and their use as pharmaceuticals
06/19/2003US20030114502 Substituted thiazoles and oxazoles as corticotropin releasing hormone ligands
06/19/2003US20030114454 Substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamines useful for inhibiting cholesteryl ester transfer protein activity
06/19/2003US20030114447 Controlling apoptosis; central nervous system disorders
06/19/2003US20030114435 Benzoic acid derivatives, processes for producing the same and drugs containing the same as the active ingredient