Patents for C07D 249 - Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms (17,749) |
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07/30/2008 | CN101230044A Synthesis of 4-substituted methoxy acrylate-1,2,4-triazolinones derivatives and herbicidal activity |
07/29/2008 | US7405232 Long acting beta-2 agonists and their use as medicaments |
07/29/2008 | US7405231 Oxidized thioether derivatives |
07/29/2008 | CA2355711C Fungicide mixture |
07/29/2008 | CA2205811C Multifunctional cyanate ester and epoxy blends |
07/29/2008 | CA2175767C Adhesion receptor antagonists |
07/24/2008 | WO2008086857A1 Triazole derivative as an hsp 90 inhibitor |
07/24/2008 | US20080177081 Reacting 3,5-bis(2-cyanoisopropyl)toluene with a brominating reagent such as N-bromosuccinimide and 2,2'-azobis(2-methylpropionitrile) in solvent to produce 1-(bromomethyl)-3,5-bis(2-cyanoisopropyl)benzene; reacting with 1,2,4-triazole; purification, crystallization; avoids toxic solvents and reactants |
07/24/2008 | US20080176917 Schizophrenia; bioavailability, solubility, brain penetrancy; in vivo half life; synthesis; such as 3-[3-({4-methyl-5-[4-(pentafluoro-6-sulfanyl)phenyl]-4H-1,2,4-triazol-3-yl}thio)propyl]-1-[4-(trifluoromethyl)phenyl]-3-azabicyclo[3.1.0]hexane |
07/24/2008 | US20080176916 A-amino-n-hydroxy-acetamide derivatives |
07/24/2008 | US20080176850 able to inhibit various mutated RTs, including K103N, Y181C and Y188L |
07/24/2008 | DE102007002715A1 Triazolderivat Triazole derivative |
07/24/2008 | CA2675737A1 Triazole derivative |
07/23/2008 | EP1945705A1 Photolatent systems |
07/23/2008 | EP1945618A2 Process for the preparation of letrozole |
07/23/2008 | EP1945272A1 Method of scintigraphy |
07/23/2008 | EP1389223B1 Method for producing polyisocyanates |
07/23/2008 | CN101228137A Substituted triazole derivatives and their use as neurokinin 3 receptor antagonists |
07/23/2008 | CN101225074A Synthesis of compound containing aryl ether triazole |
07/23/2008 | CN100404536C Triazolopyrimidine derivatives as glycogen synthase kinase 3 inhibitors |
07/17/2008 | WO2008065123A3 Polymorphic forms of deferasirox ( icl670a) |
07/17/2008 | WO2008065123A2 Polymorphic forms of deferasirox ( icl670a) |
07/17/2008 | US20080171881 Method for Producing Organic Compound and Method for Decomposing Compound Having Dicarboximide Skeleton |
07/17/2008 | US20080171777 Biaryl substituted triazoles as sodium channel blockers |
07/17/2008 | US20080171692 Substituted amides |
07/17/2008 | US20080171662 Aminocarbonyl-Substituted Thiensulfonylamino(Thio)Carbonyl-Triazolin(Ethi)Ones, Processes For Their Preparation And Their Use |
07/16/2008 | EP1943234A1 Triazole compounds as lipoxygenase inhibitors |
07/16/2008 | EP1943224A2 Estrogen receptor modulators |
07/16/2008 | EP1943004A2 Ruthenium-catalyzed cycloaddition of alkynes and organic azides |
07/16/2008 | EP1942904A2 Cholesteryl ester transfer protein inhibitors |
07/16/2008 | CN100402507C Benzotriazole compound containing sulfur, and its preparing method |
07/16/2008 | CN100402499C 2-iminopyrrolidine derivatives |
07/15/2008 | US7399537 Organic electroluminescence device and phenylenediamine derivative |
07/10/2008 | WO2008083356A1 Substituted triazoles useful as axl inhibitors |
07/10/2008 | WO2008082198A1 Antifungal triazole derivatives, method for the preparation thereof and pharmaceutical composition containing same |
07/10/2008 | US20080167357 Azabicyclo (3.1.0) Hexane Derivatives Useful as Modulators of Dopamine D3 Receptors |
07/10/2008 | CA2710051A1 Substituted triazoles useful as axl inhibitors |
07/09/2008 | EP1940811A1 Heterocyclic compounds with carboxyl isostere groups and their use for the treatment of cardiovascular diseases |
07/09/2008 | EP1940807A1 Carbamoylbenzotriazole derivatives as inhibitors of lipases and phospholipases |
07/09/2008 | EP1940806A2 A process for the preparation of pure anastrozole |
07/09/2008 | CN100400520C Method for extracting methyl o-phenylendiamine from TDI organic residue and synthesizing TTA using same |
07/09/2008 | CN100400487C Glucocorticoid receptor modulators |
07/08/2008 | WO2008083353A1 Bicyclic aryl and bicyclic heteroaryl substituted triazoles useful as axl inhibitors |
07/08/2008 | CA2710043A1 Bicyclic aryl and bicyclic heteroaryl substituted triazoles useful as axl inhibitors |
07/03/2008 | WO2007137066A3 HETEROCYCLIC INHIBITORS OF 11-β HYDROXYL STEROID DEHYDROGENASE TYPE I AND METHODS OF USING THE SAME |
07/03/2008 | US20080161325 e.g. N1-[3-amino-4-(3,5-difluorophenyl)-2-hydroxybutyl]-3-(butylsulfonyl)-N1-(3-ethylbenzyl)-D-alaninamide dihydrochloride; inhibitors of amyloid beta-secretase enzyme; neurodegenerative diseases: Alzheimer's, Parkinson's diseases, Down's syndrome |
07/03/2008 | US20080156227 Benzotriazole compound other than 2-(2-hydroxy-3- alpha -cumyl-5-tert-octylphenyl)-2H-benzotriazole plus a hindered amine, a phosphite and a phenolic anti-oxidant compound; storage stability without using any volatile solvent |
07/03/2008 | CA2672727A1 Sphingosine-1-phosphate receptor agonist and antagonist compounds |
07/02/2008 | EP1939203A2 Inhibitors of human phosphatidyl-inositol 3-kinase delta isoform |
07/02/2008 | EP1939183A1 Novel nitrogenated heterocyclic compound |
07/02/2008 | EP1937638A1 Methods of treating amyloidosis using aryl-cyclopropyl derivative aspartyl protease inhibitors |
07/02/2008 | EP1501808B1 Tachykinin receptor antagonists |
07/02/2008 | EP1496838A4 Substituted amides |
07/02/2008 | CN101213657A Epoxy bleedout-preventing agent |
07/02/2008 | CN100398612C Azo compound, aqueous dye solutions containing the same, inks and use thereof |
07/02/2008 | CN100398536C Compounds, methods and formulations for the oral delivery of a glucagon like peptide (glp)-1 compound or an melanocortin 4 receptor (mc4) agonist peptide |
07/01/2008 | US7393873 Arylsulfonamide derivatives |
06/26/2008 | WO2008077138A1 3-benzofuranyl-4-indolyl maleimides as potent gsk3 inhibitors for neurogenerative disorders |
06/26/2008 | WO2008076225A2 Non-nucleoside reverse transcriptase inhibitors |
06/26/2008 | WO2008076223A1 Non-nucleoside reverse transcriptase inhibitors |
06/26/2008 | WO2008075955A2 Process for the preparation of 1,4,5-trisubstituted triazoles and 3,4,5-trisubstituted triazoles |
06/26/2008 | WO2008075152A1 1- [4- (sulfonyl) -phenyl] -5- (benzyl) -ih-i, 2, 4-triazol derivatives as inhibitors of carbonic anhydrase for treating glaucoma or ocular hypertension |
06/26/2008 | WO2008034644A3 Process for making anastrozole |
06/26/2008 | US20080153892 1-(Urea-, thiourea- and cyanoguanidine-methylene)benzyl)imidaoles, treatment of neuronal disorders, especially Alzheimer's disease, Down Syndrome, Parkinson's disease and Huntington's disease |
06/26/2008 | US20080153836 1H-Quinazoline-2,4-Diones |
06/26/2008 | US20080153812 Novel compounds |
06/26/2008 | CA2673368A1 3-benzofuranyl-4-indolyl maleimides as potent gsk3 inhibitors for neurogenerative disorders |
06/26/2008 | CA2673093A1 Non-nucleoside reverse transcriptase inhibitors |
06/25/2008 | EP1935869A1 Retinoids for the treatment of emphysema |
06/25/2008 | EP1934188A2 Alpha, alpha`-dihydroxy ketone derivatives and use thereof as uv filter |
06/25/2008 | CN101208312A Method of synthesis of anastrozole and purification of one of its intermediate |
06/25/2008 | CN101208088A Phenylalkyl substituted heteroaryl devivatives |
06/25/2008 | CN101208082A Niacin receptor agonists, compositions containing such compounds and methods of treatment |
06/25/2008 | CN101205216A Benzotriazole ammonium salts, preparation and uses thereof |
06/25/2008 | CN100396679C Piperazinyl-, piperidinyl- and morpholinyl-derivatives as novel inhibitors of histone deacetylase |
06/24/2008 | US7390835 Aralkyl amines as cannabinoid receptor modulators |
06/19/2008 | WO2008073461A2 Ion channel modulators |
06/19/2008 | US20080146632 Fc Receptor Modulating Compounds and Compositions |
06/19/2008 | US20080146620 Dibenzylamine Compounds and Pharmaceutical Use Thereof |
06/19/2008 | US20080145946 Impurity of anastrozole intermediate, and uses thereof |
06/18/2008 | EP1932833A1 Nitrogenated heterocyclic compound and pharmaceutical composition comprising the same |
06/18/2008 | EP1931647A2 Selected cgrp antagonists, methods for the production thereof and their use as medicaments |
06/18/2008 | EP1931646A2 Selected cgrp antagonists, a method for the production thereof and use in the form of drugs |
06/17/2008 | US7387668 Azo compound, aqueous dye solutions containing the same, inks and use thereof |
06/17/2008 | CA2286772C Fungicide active substance combinations |
06/12/2008 | US20080139599 e.g. 4-[6-(5-methyl-2-phenyloxazol-4-ylmethoxy)-1-oxoindan-5-yl]benzoic acid; antidiabetic and antilipemic agent, obesity; atherosclerosis; coupling benzene derivatives folowed by hydration and alkylation |
06/12/2008 | US20080139560 Ion Channel Modulators |
06/11/2008 | EP1928846A2 Triazole compounds that modulate hsp90 activity |
06/11/2008 | EP1928822A1 Violet laser excitable dyes and their method of use |
06/11/2008 | EP1449836B1 Low dusting crystal transformations of 2, 2'-methylenbis 4-(1,1,3,3-tetramethylbutyl)-6-benzotriazolylphenol and mixture thereof, method for preparing them, and ultraviolet absorbent using the same |
06/11/2008 | EP1180107B1 Novel ruthenium metal alkylidene complexes coordinated with triazolylidene ligands that exhibit high olefin metathesis activity |
06/10/2008 | US7385054 For use as contrast media; x-ray diagnosis and magnetic resonance imaging |
06/10/2008 | CA2296665C Triazolo[4,5-d]pyrimidine derivatives as anti-thromobotic agents |
06/05/2008 | WO2008014811A8 PROCESS FOR THE PREPARATION OF ε-ALKOXYCARBONYLLYSINES AND THEIR ANALOGUES |
06/05/2008 | WO2007018431A3 Triazole-containing releasable linkers and conjugates comprising the same |
06/05/2008 | US20080132556 3-hydroxymethyl-4hydroxy-phenyl- derivatives for the treatment of respiratory diseases |
06/05/2008 | US20080132524 Ortho-heterocyclic substituted aryl amides for controlling invertebrate pests |
06/05/2008 | US20080132507 Hydrazide Derivatives |
06/05/2008 | US20080132506 Anti-inflammatory medicaments |
06/05/2008 | US20080132459 Inhibitors of Histone Deacetylase |