Patents for C07D 239 - Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings (42,619) |
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10/12/2010 | US7812160 G-protein-coupled chemoattractant receptor, expressed on T helper cells antagonists such as [4-(dimethylamino)-2-(4-{[4-(trifluoromethyl)benzoyl]amino}benzyl)-5-pyrimidinyl]acetic acid;, used for the treatment of allergic diseases, inflammatory diseases, eosinophil- and basophil-related diseases |
10/12/2010 | US7812038 such as vascular cell adhesion molecules and fibronectins, administered for the treatment of asthma, multiple sclerosis or inflammatory bowel diseases in mammals; (3S)-3-{[({1-[(2-chlorophenyl)methyl]-4-hydroxy-2-oxo-1,2-dihydro-3quinolinyl}amino)carbonyl]amino}-3-(4-methylphenyl)propanoic acid |
10/12/2010 | US7812031 Pyrimidine derivatives as orexin receptor antagonists |
10/12/2010 | US7812029 such as N4-[(2,2-Dimethyl-4H-benzo[1,4]oxazin-3-one)-6-yl]-5-fluoro-N2-[3-(methylaminocarbonylmethyleneoxy)phenyl]-2,4-pyrimidinediamine; Glomerulonephritis; rheumatoid arthritis; systemic lupus erythematosis; multiple sclerosis |
10/12/2010 | CA2467838C Pyrimidine derivatives as modulators of insuline-like growth factor-1 receptor (igf-i) |
10/12/2010 | CA2339761C Arylpiperazines and their use as metalloproteinase inhibiting agents (mmp) |
10/07/2010 | WO2010114493A1 Lanthanide metal complexes useful in treating cancer |
10/07/2010 | WO2010114292A2 Improved method for manufacturing dipeptidyl peptidase-iv inhibitor and intermediate |
10/07/2010 | WO2010113848A1 Isothiourea derivative or isourea derivative having bace1 inhibitory activity |
10/07/2010 | WO2010113834A1 Pyrimidine compound |
10/07/2010 | WO2010112411A1 Co-crystal of etravirine and nicotinamide |
10/07/2010 | WO2010112210A1 Methods for the identification of kinase interacting molecules and for the purification of kinase proteins |
10/07/2010 | US20100256168 Quinazolinones as inhibitors of human phosphatidylinositol 3-kinase delta |
10/07/2010 | US20100256167 Quinazolinones as inhibitors of human phosphatidylinositol 3-kinase delta |
10/07/2010 | US20100256166 Novel Hydantoin Derivatives as Metalloproteinase Inhibitors |
10/07/2010 | US20100256120 Amide derivatives |
10/07/2010 | DE102009016553A1 Sulfonamid- und Sulfoximin-substituierte Diaryldihydropyrimidinone und ihre Verwendung Sulfonamide and sulfoximine-substituted Diaryldihydropyrimidinone and their use |
10/07/2010 | CA2757671A1 Methods for the identification of kinase interacting molecules and for the purification of kinase proteins |
10/07/2010 | CA2757228A1 Co-crystal of etravirine and nicotinamide |
10/07/2010 | CA2757188A1 Pyrimidine compound |
10/07/2010 | CA2756915A1 Improved method for manufacturing dipeptidyl peptidase-iv inhibitor and intermediate |
10/06/2010 | EP2235009A1 Synthesis of paliperidone |
10/06/2010 | EP2234993A1 Bis- (sulf onylamino) derivatives for use in therapy |
10/06/2010 | EP2234986A2 Sulfamides as zap-70 inhibitors |
10/06/2010 | EP2234985A1 4-(4-cyano-2-thioaryl)dihydropyrimidinones and use thereof |
10/06/2010 | EP2234977A1 Viral polymerase inhibitors |
10/06/2010 | EP2234971A1 Process and intermediates for the synthesis of heterocyclic substituted piperazines with cxcr3 antagonist activity |
10/06/2010 | EP1776349B1 2-amino-quinazoline derivatives useful as inhibitors of beta-secretase (bace) |
10/06/2010 | EP1421105B1 Anti-cancer cyclopenta¬g quinazoline compounds |
10/06/2010 | EP1309569B1 N-aryl-{4-[7-(alkoxy)quinazolin-4-yl]piperazinyl}carboxamide derivatives as PDGFRs inhibitors |
10/06/2010 | EP1268446B1 Method for producing asymmetrical 4,6-bis(aryloxy)pyrimidine derivatives |
10/06/2010 | CN101851241A Anti-tumor compound and preparation method and application thereof |
10/06/2010 | CN101851212A Process for the preparation of aminopyrimidines |
10/06/2010 | CN101851211A Novel piperazinoamide compound |
10/06/2010 | CN101851173A Inhibitors of histone deacetylase |
10/06/2010 | CN101849953A Inflammatory cytokine release inhibitor |
10/06/2010 | CN101062928B Process for preparing 2-pyrrolidinyl-1h-pyrrolo[3,2-d]pyrimidine inhibitors of nucleoside metabolism |
10/05/2010 | US7807858 Process for production of fluoro derivative |
10/05/2010 | US7807842 Synthesis of tetracyclines and analogues thereof |
10/05/2010 | US7807832 oxidizing an alkyne compound containing pyrimidine and benzene rings with KMnO4 to form 1,2-diketone; reacting 2,4-dichloropyrimidine with (trimethylsilyl)acetylene to form( trimethylsilylethynyl-pyrimidine, reacting intermediate with an amine to form (trimethylsilyl)akyne, deportecting |
10/05/2010 | US7807701 Dibenzylamine compounds and pharmaceutical use thereof |
10/05/2010 | US7807689 such as 2-{6-[3(R)-Amino-piperidin-1-yl]-3-methyl-2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-ylmethyl}-benzonitrile, used for the treatment of breast cancer and non-insulin depepndent diabetes |
10/05/2010 | US7807654 Compositions and methods for treatment of mitochondrial diseases |
10/05/2010 | CA2400479C Platelet adp receptor inhibitors |
10/05/2010 | CA2369595C Conjugate having a cleavable linkage for use in a liposome |
09/30/2010 | WO2010111348A1 Process for preparing antiviral compound |
09/30/2010 | WO2010109443A1 Process for the preparation of erlotinib or its pharmaceutically acceptable salts thereof |
09/30/2010 | WO2010108856A1 Leukotriene b4 inhibitors |
09/30/2010 | WO2010108611A1 Pyrimindine-4-ylpropane dinitrile derivatives, method for the production thereof, and use thereof as herbicide and plant growth regulators |
09/30/2010 | WO2010079431A3 Compounds for the prevention and treatment of cardiovascular disease |
09/30/2010 | US20100249410 Process for preparing n-alkylated hydroxypyrimidinone compounds |
09/30/2010 | US20100249409 Process for stereoselective synthesis of lamivudine |
09/30/2010 | US20100249405 Organic Compounds |
09/30/2010 | US20100249181 HIV Protease Inhibiting Compounds |
09/30/2010 | US20100249161 2- ( 2 -hydroxyphenyl) -quinazolin-4-ones useful for treating obesity and diabetes |
09/30/2010 | US20100249158 Substituted amino-quinazolinones, medicaments comprising said compound, their use and their method of manufacture |
09/30/2010 | US20100249149 Inhibitors of Protein Kinases |
09/30/2010 | US20100249147 Sulfonyl-substituted 6-membered ring derivative |
09/30/2010 | US20100249124 2,3-diaryl- or heteroaryl-substituted 1,1,1-trifluoro-2-hydroxypropyl compounds |
09/30/2010 | US20100249123 Novel benzamide derivatives as modulators of the follicle stimulating hormone |
09/30/2010 | US20100249117 Factor xa inhibitors |
09/30/2010 | US20100249114 Selected CGRP-antagonists, process for preparing them and their use as pharmaceutical compositions |
09/30/2010 | US20100249100 Quinazolines useful as modulators of ion channels |
09/30/2010 | US20100249092 Heteroaryl compounds and uses thereof |
09/30/2010 | US20100249077 Pyridylmethyl-Sulfonamide Compounds |
09/30/2010 | US20100248264 Capture compounds, collections thereof and methods for analyzing the proteome and complex compositions |
09/30/2010 | US20100248241 Mutations in the bcr-abl tyrosine kinase associated with resistance to sti-571 |
09/30/2010 | US20100247534 Fused heterocyclic compounds as inhibitors of potassium channel function |
09/30/2010 | US20100247468 Compounds that modulate PPAR gamma-type receptors and cosmetic/pharmaceutical compositions comprising said compounds |
09/30/2010 | US20100242792 Synthesis of colorants in mixing apparatus |
09/30/2010 | DE19840447B4 Fluorierte Derivate des Indans und ihre Verwendung in flüssigkristallinen Mischungen Fluorinated derivatives of indane and their use in liquid crystal mixtures |
09/30/2010 | CA2756007A1 Pyrimindine-4-ylpropane dinitrile derivatives, method for the production thereof, and use thereof as herbicide and plant growth regulators |
09/30/2010 | CA2755348A1 Antiviral compounds and uses thereof |
09/30/2010 | CA2753825A1 Process for preparing antiviral compound |
09/30/2010 | CA2747327A1 Leukotriene b4 inhibitors |
09/29/2010 | EP2233483A1 Indole or Benzimidazole derivatives as IkB-kinase modulators and intermediates in their preparation. |
09/29/2010 | EP2233472A1 Heterocyclic compounds and uses thereof in the treatment of sexual disorders |
09/29/2010 | EP2231622A1 Preparations containing amino acids and orotic acid |
09/29/2010 | EP2231621A1 Process for preparing n-substituted hydroxypyrimidinone carboxamides |
09/29/2010 | EP2231620A1 Diaminopyridines for the treatment of diseases which are characterised by excessive or anomal cell proliferation |
09/29/2010 | EP2231619A1 Inhibitors of stearoyl-coa desaturase |
09/29/2010 | EP2004641B1 Hiv inhibiting 5-(hydroxymethylene and aminomethylene) substituted pyrimidines |
09/29/2010 | EP1789398B1 2-amino-quinazoline derivatives useful as inhibitors of b-secretase (bace) |
09/29/2010 | EP1638928B1 N-alkynyl-2-(substituted aryloxy)alkylthioamide derivatives as fungicides |
09/29/2010 | CN1794987B Nitrooxyderivatives of fluvastatin, pravastatin, cerivastatin, atorvastatin and rosuvastatin as cholesterol-reducing agents with improved anti-inflammatory, antithrombotic and antiplatelet activity |
09/29/2010 | CN101848641A Use of sulfonanilide compounds as herbicide |
09/29/2010 | CN101845021A Quinazoline ketones alkaloid and preparation method and application thereof |
09/29/2010 | CN101279949B Method for synthesizing 2-hydroxyl-4,6-dimethylpyrimidine |
09/28/2010 | US7803941 Process for preparing ring-fluorinated aromatics |
09/28/2010 | US7803939 N2,N4-bis(4-ethoxyphenyl)-5-fluoro-2,4-pyrimidinediamine; inhibit the IgE and/or IgG receptor signaling cascades that lead to the release of chemical mediators; Syk kinase inhibitors |
09/28/2010 | US7803938 3-{[4-(4-acetyl-3-hydroxy-2-propylphenoxymethyl)-phenyl]-(S)-hydroxymethyl}-benzoic acid; anxiolytic, neuroleptic agent and antidepressant as glutamate receptor agonist; antiinflammatory agent as leukotriene receptor agonist; |
09/28/2010 | US7803806 protein kinase inhibitors such as 1-{3-[4-(5-Bromo-thiophen-2-yl)-pyrimidin-2-ylamino]-phenyl}-ethanol, used for the treatment of breast cancer or rheumatoid arthritis |
09/28/2010 | US7803399 Delivery system for nucleic acids |
09/28/2010 | CA2387016C Acrylamide derivatives as fab i inhibitors |
09/28/2010 | CA2383524C Thiazolyl alkynyl compounds and methods of use thereof |
09/28/2010 | CA2382631C Poly(ether-thioether), poly(ether-sulfoxide) and poly(ether-sulfone) nucleic acids |
09/28/2010 | CA2308201C Use of anti-fungal agents for the treatment of fungus-induced mucositis |
09/24/2010 | CA2719523A1 Polymorphic forms of 4-phenylamino quinazoline derivatives, the preparation methods and uses thereof |
09/23/2010 | WO2010108059A1 Substituted pyrimidine derivatives as antagonists of the histamine h4 receptor |
09/23/2010 | WO2010107768A1 Bicyclic compounds as inhibitors of diacylglycerol acyltransferase |