Patents
Patents for C07D 239 - Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings (42,619)
10/2001
10/04/2001WO2001072696A1 Arthropodicidal carboxanilides
10/04/2001WO2001021577A3 Melanin concentrating hormone antagonist
10/04/2001WO1999061428A9 Quinazolines for treating brain tumor
10/04/2001US20010027198 Novel heterocyclic compounds and their use in medicine; process for their preparation and pharmaceutical compositions containing them
10/04/2001US20010027197 Antiproliverative, -carcinogenic and -tumor agents; mitogenesis-activated protein kinase inhibitors; noncytotoxic; binding with high affinity at the adenosine triphosphate binding site of the kinases
10/04/2001US20010027196 Adenosine receptor ligands and their use in the treatment of disease
10/04/2001EP1138675A2 Process for the preparation of 2-methyl-4-amino-5-aminomethylpyrimidine
10/04/2001EP1138328A1 Naphthalene derivatives as CNS drugs
10/04/2001EP1137649A2 Process for the preparation of pyrimidinone derivatives
10/04/2001EP1137642A1 Bis-sulfonamides
10/04/2001EP1137640A1 Cyclic hydrazine derivatives as tnf-alpha inhibitors
10/04/2001EP1137622A1 Method of preparing salts of dinitromethane
10/04/2001EP1137418A2 METHODS AND COMPOSITIONS FOR RESTORING CONFORMATIONAL STABILITY OF A PROTEIN OF THE p53 FAMILY
10/04/2001EP0973395A4 Diaryl ethers and processes for their preparation and herbicidal and desiccant compositions containing them
10/04/2001EP0698013B1 Fungicidal fused bicyclic pyrimidinones
10/04/2001EP0650482B1 Pesticidal pyrimidine compounds
10/04/2001EP0631575B1 Substituted pyrimidines and their use as pesticides
10/04/2001EP0613465B1 1,3-substituted cycloalkenes and cycloalkanes as central nervous system agents
10/04/2001EP0563384B1 Uracil derivative
10/04/2001CA2404712A1 Synergistic methods and compositions for treating cancer comprising antiproliferative cytotoxic and cytostatic agents
10/04/2001CA2402288A1 Naphtalene derivatives and their pharmaceutical use
10/04/2001CA2399864A1 4-amino-5-cyano-2-anilino-pyrimidine derivatives and their use as inhibitors of cell-cycle kinases
10/03/2001CN1315945A Nitrate salts of antihypertensive medicines
10/03/2001CN1315936A Compounds and compositions for delivering active agents
10/03/2001CN1072223C Halogen pyrimidines, its preparing process and pesticide containing same
10/03/2001CN1072221C 3-halo-3-heteroaryl carboxylic acid derivatives, method of preparing them and intermediates
10/02/2001US6297379 Thienopyrimidine compounds, their production and use
10/02/2001US6297374 Nitroimino-nitromethylene—azole or-azine heterocyclic compounds, insecticidal compositions containing them, and insecticidal methods of using them
10/02/2001US6297284 Aza-enediyne, aza-enyne allene, or an aza-diallene cationic compounds that bind to nucleic acids.
10/02/2001US6297277 Cysteine protease inhibitors containing heterocyclic leaving groups
10/02/2001US6297260 Nitrosated and nitrosylated nonsteroidal antiinflammatory compounds, compositions and methods of use
10/02/2001US6297253 Inactivating a nuclear localization signal of a protein comprising contacting the protein with an aryl carbonyl compound that forms stable reversible covalent interactions with neighboring basic amino acid residues
10/02/2001US6297223 Administering 5-substituted- or 5,6-dihydro-5-substituted-uracil derivative or a prodrug thereof; in conjunction with 5-fluorouracil or pro-drug thereof.
09/2001
09/27/2001WO2001070757A2 Thioketals and thioethers for inhibiting the expression of vcam-1
09/27/2001WO2001070737A2 Therapeutic heterocyclic compounds for the treatment of asthma and allergy and use thereof
09/27/2001WO2001070709A2 3-oxy-7-sulfamyl-3,4-dihydro-1,2,4-benzothiadazine-1,1-dioxide derivatives having diuretic and/or natriuretic activity
09/27/2001WO2001070707A2 Asymmetric synthesis of quinazolin-2-ones useful as hiv reverse transcriptase inhibitors
09/27/2001WO2001070675A2 Inhibitors of histone deacetylase
09/27/2001WO2001070671A2 Insecticidal anthranilamides
09/27/2001WO2001070670A1 Novel phenylalanine derivative
09/27/2001WO2001070255A2 Combined treatment with keratinocyte growth factor and epidermal growth factor inhibitor
09/27/2001WO2001070217A1 Dna-cleaving antitumor agents
09/27/2001US20010025044 A bicyclic nitrogen containing heteroaromatic compound useful for inhibiting protein kinase p38 which involved in cell proliferation, cell death and response to extracellular stimuli
09/27/2001US20010025033 Uracil substituted at 5-position by C2-4 alkynyl used as inactivator of uracil reductase enzyme
09/27/2001US20010025032 Administering mixture of nucleosides; anticancer agent
09/27/2001US20010024749 Surface modified carbonaceous materials
09/27/2001DE10014607A1 Production of asymmetric 4,6-bis(aryloxy)-pyrimidine derivatives comprises two stage reaction of 4,6-dichloro-pyrimidine with phenols using 1,4-diazabicyclo(2.2.2)octane in second reaction stage
09/27/2001DE10014006A1 New heterocyclic acylsulfimide derivatives, useful as insecticides, acaricides and nematocides for plant protection or in veterinary medicine
09/27/2001CA2404002A1 Inhibitors of histone deacetylase
09/27/2001CA2403823A1 Thioketals and thioethers for inhibiting the expression of vcam-1
09/27/2001CA2403230A1 Asymmetric synthesis of quinazolin-2-ones useful as hiv reverse transcriptase inhibitors
09/27/2001CA2402572A1 3-oxy-7-sulfamyl-3,4-dihydro-1,2,4-benzothiadazine-1,1-dioxide derivatives having diuretic and/or natriuretic activity
09/26/2001EP1136472A1 Aryl- and heteroarylamides of carboalkoxysulfanilic acids
09/26/2001EP1135450A1 Chiral liquid crystal compounds having a fluorinated terminal portion
09/26/2001EP1135391A1 Novel triazolo(4,5-d)pyrimidine compounds
09/26/2001EP1135132A2 Inhibitors of multidrug transporters
09/26/2001EP1135131A1 Aryl and heterocyclyl substituted pyrimidine derivatives as anti-coagulants
09/26/2001EP1031570A4 Immuno-modulator exhibiting anti-microbial and anti-mycobacterial activities, method for producing the same and pharmaceutical preparation for treating mycobacterioses as well as lung chronic and non specific conditions, sexually transmitted diseases and the resulting immuno-deficiency
09/26/2001EP0934252B1 Amide derivatives and their use as pesticides
09/26/2001EP0900214B1 Process for preparation of pyrimidine derivatives
09/26/2001EP0775141B1 Phenyl xanthine derivatives
09/26/2001EP0773943B1 Compounds useful as antiproliferative agents and garft inhibitors
09/26/2001CN1314894A Substituted phenyl uracils compound
09/26/2001CN1071748C Method for preparing sulphonyl ureas with herbicidal properties and N-(pyrimidinyl or triazinyl)-carbamates as intermediates
09/25/2001US6294542 Pyrimidinone compounds, pharmaceutical compositions containing the compounds and the process for preparing the same
09/25/2001US6294538 Antidiabetic agents and diabetic neuropathy, treatment with oxidoreductase enzymes
09/25/2001US6294535 Uracil derivatives and antitumor effect potentiator and antitumor agent containing the same
09/25/2001US6294533 Calcium channel blockers
09/25/2001US6294517 Compositions and kits comprising alpha-adrenergic receptor antagonists and nitric oxide donors and methods of use
09/25/2001CA2091005C Microbiological process for hydroxylation of nitrogen-heterocyclic-carboxylic acids
09/20/2001WO2001068645A2 N-cyanomethylcarboxamides and their use as protease inhibitors
09/20/2001WO2001068615A1 Quinazoline synthesis
09/20/2001WO2001068614A2 5-substituted arylpyrimidines
09/20/2001WO2001068613A1 Pyrimidinone derivatives and herbicides
09/20/2001WO2001068612A2 Aryl substituted pyridines, pyrimidines, pyrazines and triazines and the use thereof
09/20/2001WO2001068609A1 1,2,3,4-tetrahydroisoquinoline derivatives
09/20/2001WO2001068600A2 Benzylated pde4 inhibitors
09/20/2001WO2001068585A1 Novel amide compounds
09/20/2001WO2000071506A9 Naphthalene ureas as glucose uptake enhancers
09/20/2001WO2000047553A8 ALKENYL AND ALKYNYL COMPOUNDS AS INHIBITORS OF FACTOR Xa
09/20/2001CA2402384A1 Benzylated pde4 inhibitors
09/20/2001CA2373411A1 5-substituted arylpyrimidines
09/19/2001EP1133488A1 Propanoic acid derivatives as integrin inhibitors
09/19/2001EP1133478A1 Novel acylguanidine derivatives, method for preparing same, application as medicines and pharmaceutical compositions containing them
09/19/2001EP0853616B1 Bicyclic 4-aralkylaminopyrimidine derivatives as tyrosine kinase inhibitors
09/19/2001CN1313854A Antiviral pyrimidinedione derivatives and process for the preparation thereof
09/19/2001CN1313846A C-terminal modified oxamyl dipeptides as inhibitors of the ICE/ced-3 family of cystenine proteases
09/19/2001CN1313769A Pharmaceutical combination comprising A COX-2 inhibitor and a iNOS inhibitor
09/19/2001CN1313768A Nitrogenous heterocyclic carboxamide derivatives or salts thereof and antivirual agents containing both
09/19/2001CN1313766A DNA-cleaving antitumor agents
09/19/2001CN1071325C Thiol derivatives with metallopeptidase inhibitory activity
09/19/2001CN1071320C Preparation of arylamides of heteroaromatic carboxylic acids
09/18/2001US6291500 Administering an antifungal agent
09/18/2001US6291468 Pyrimidine 3-oxide compounds for inducing/stimulating hair growth and/or retarding hair loss
09/18/2001US6291455 Producing an antiangiogenic and/or vascular permeability reducing effect
09/18/2001US6291400 Herbicidal compounds
09/18/2001US6291034 Naphthyl organic compounds
09/18/2001CA2236814C Quinoline and quinazoline compounds useful in therapy
09/13/2001WO2001066534A2 Cyclic and bicyclic diamino histamine-3 receptor antagonists
09/13/2001WO2001066527A1 Substituted benzoylcyclohexenones