Patents
Patents for C07D 239 - Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings (42,619)
03/2002
03/19/2002CA2151588C Antiproliferative substituted 5-thiapyrimidinone and 5-selenopyrimidinone
03/14/2002WO2002020500A2 Materials and methods to potentiate cancer treatment
03/14/2002WO2002020495A2 Inhibitors of glycogen synthase kinase 3
03/14/2002WO2002020494A1 Process for producing pyrimidine derivative and intermediate thereof
03/14/2002WO2002020488A2 Quinoline and quinazoline derivatives as ligands for the neuropeptide y receptor
03/14/2002WO2002020465A2 Gamma-ketoacid dipeptides as inhibitors of caspase-3
03/14/2002WO2002020017A2 Use of ectoin or ectoin derivatives for stabilizing p53
03/14/2002WO2002019978A2 Use of ectoine or ectoine derivatives for oral care
03/14/2002WO2001085760A8 Thrombin inhibitors
03/14/2002WO2001070757A3 Thioketals and thioethers for inhibiting the expression of vcam-1
03/14/2002WO2001070692A3 Heterocyclic acylsulfimides, a method for their production, agents containing the same and their use as pesticides
03/14/2002WO2001068612A3 Aryl substituted pyridines, pyrimidines, pyrazines and triazines and the use thereof
03/14/2002WO2001062743A3 Method for the simplified production of (3-chloro-4-fluoro-phenyl)-[7-(3-morpholino-4-yl-propoxy)-6-nitro-quinazoline-4-yl]-amine or (3-chloro-4-fluoro-phenyl)-[7-(3-morpholino-4-yl-propoxy)-6-amino-quinazoline-4-yl]-amine
03/14/2002WO2001058852A3 (r)-2-aryl-propionamides, useful in the inhibition of il-8-induced chemiotaxis of neutrophils
03/14/2002US20020032328 Heterocyclic acylsulfimides, processes for their preparation, compositions comprising them and their use as pesticides
03/14/2002US20020032223 Benzamidine derivatives and their use as anti-coagulants
03/14/2002US20020032208 Chemical compounds
03/14/2002US20020032206 Pharmaceutical compositions for prevention and treatment of central nervous system disorders
03/14/2002US20020032199 5-HT7 receptor antagonists
03/14/2002US20020032186 N-hydroxy-2-(alkyl, aryl, or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
03/14/2002US20020030179 Having negative and large dielectric anisotropy value and small optical anisotropy value at the same time
03/14/2002DE10043667A1 2-Guanidino-4-aryl-chinazoline 2-guanidino-4-aryl-quinazolines
03/14/2002DE10043456A1 Verwendung von Ectoin oder Ectoin-Derivaten zur Stabilisierung von p53 Use of ectoine or ectoine derivatives for the stabilization of p53
03/14/2002DE10042655A1 Verfahren zur Herstellung von Inhibitoren der Zell-Adhäsion Process for the preparation of inhibitors of cell adhesion
03/14/2002CA2421172A1 Gamma-ketoacid dipeptides as inhibitors of caspase-3
03/14/2002CA2420703A1 Quinoline and quinazoline derivatives as ligands for the neuropeptide y receptor
03/13/2002EP1186597A1 Process for the production of 2-pyridylpyridine derivatives
03/13/2002EP1185540A1 Ruthenium dimeric complexes suitable as antimetastatic and antineoplastic agents
03/13/2002EP1185522A1 Substituted phenyl compounds with immunosuppressing activity and pharmaceutical compositions containing them
03/13/2002EP1185517A1 Antibiotic prodrugs
03/13/2002EP1185505A1 Method of producing methoxyimino acetic amide
03/13/2002EP1185275A1 Aminopyrimidines as sorbitol dehydrogenase inhibitors
03/13/2002EP1185229A1 Method of treating hair loss
03/13/2002EP0975219B1 Fungicide active substance combinations
03/13/2002EP0912524B1 2-(o- pyrimidin-4-yl]methylene oxy)phenyl acetic acid derivatives and their use in combatting noxious fungi and animal pests
03/13/2002EP0901473B1 Piperazinylalkylthiopyrimidine derivatives, pharmaceutical compositions containing the same and a process for the preparation of the novel compounds
03/13/2002EP0770067B1 Substituted cinnamic oxime and hydroxamide derivatives
03/13/2002CN1340052A Process for the production of tert-butyl (E)-(6[2-[4-(4-fluorophenyl)-6-isopropyl-2-[methyl(methylsulfonyl)amino] pyrimidin 5-yl] (4R,6S)-2,2-dimethyl [1,3] dioxan-4-yl) acetate
03/13/2002CN1340049A 4-heterocyclylsulfonamide)-5-methoxy-6-(2-methoxyphenoxy)-2-phenyl-or-pyridylpyrimidines as endothelin receptor antagonists
03/13/2002CN1340046A β-丙氨酸衍生物 β- alanine derivatives
03/12/2002US6355805 β3-adrenergic receptor agonists
03/12/2002US6355799 Substituted benzene compounds, process for their preparation, and herbicidal and defoliant compositions containing them
03/12/2002US6355796 Reacting beta-amino-beta-(perfluoroalkyl)acrylate compound with base and carbamoyl chloride compound to form urea compound, reacting urea compound with phosphorus pentahalide or oxalyl halide
03/12/2002US6355726 Multicomponent ugi reaction; antisense agents, antigens; diagnosis; controlling gene expression by polymeric peptide nucleic acids
03/12/2002US6355660 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
03/12/2002US6355655 Treating a cognitive disorder, a neuro-degenerative disorder; age-related dementia; age-induced memory impairment; a movement disorder, attention deficit disorder; attention deficit hyperactivity disorder; psychosis; cognitive deficits
03/12/2002US6355645 4-(3'-bromobenzoyl)-6,7-dimethoxyquinazoline; for lowering blood cholesterol, including reducing total cholesterol and ldl-cholesterol levels
03/12/2002US6355637 Local anesthetic compounds
03/12/2002CA2313783C Pharmaceutical compositions of (e)-7-[4-(4-fluorophenyl)-6-isopropyl-2-[methyl(methylsulfonyl)amino]pyrimidin-5-yl]-(3r,5s)-3,5-dihydroxyhept-6-enoic acid or a salt thereof
03/12/2002CA2187214C Aminostilbazole derivative and medicine
03/07/2002WO2002018384A1 Process for the preparation of vitronectin receptor antagonists
03/07/2002WO2002018379A2 7-oxo pyridopyrimidines
03/07/2002WO2002018373A1 Quinazoline derivatives, medicaments containing these compounds, their use, and methods for the production thereof
03/07/2002WO2002018350A1 Grk inhibitor
03/07/2002WO2002018349A2 Process and intermediates for preparing retroviral protease inhibitors
03/07/2002WO2002018339A2 Compounds useful as insecticides, compounds useful as acaricides, and processes to use and make same
03/07/2002WO2002018333A1 Phenoxybenzylamine derivatives as selective serotonin re-uptake inhibitors
03/07/2002WO2002017712A2 Disubstituted benzenes as insecticides
03/07/2002WO2001070707A3 Asymmetric synthesis of quinazolin-2-ones useful as hiv reverse transcriptase inhibitors
03/07/2002WO2001068645A3 N-cyanomethylcarboxamides and their use as protease inhibitors
03/07/2002US20020028946 Process for the preparation of heteroaryl-phenylalanines
03/07/2002US20020028933 Thioamide derivatives
03/07/2002US20020028842 Reducing the vomiting side effects of phosphodiesterase inhibitors, e.g. Rolipram, Ariflo, by benzylation by benzyl bromide or a derivative
03/07/2002US20020028836 Potassium channel openers
03/07/2002US20020028813 Isoquinoline inhibitors of the nucleic enzyme poly(adenosine 5'-diphospho-ribose) polymerase (PARP); treat tissue damage from necrosis or apoptosis, ischemia or reperfusion injury, stroke, senescence diseases
03/07/2002US20020028812 Phenylalanine derivatives
03/07/2002US20020028811 Use as pesticides such as 2-fluoromethoxyimino-N-methyl-2-((6-aryl-s-triazin-2-yloxy)-phenyl) -acetamide; use on crops as fungicide; microbiocide on wood; chemical synthesis
03/07/2002US20020028774 C-terminal modified oxamyl dipeptides as inhibitors of the ICE/ced-3 family of cysteine proteases
03/07/2002DE10042064A1 Chinazoline, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung Quinazolines, medicaments containing these compounds, their use and process for their preparation
03/07/2002DE10042060A1 Bicyclische Heterocyclen, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung Bicyclic heterocycles, pharmaceutical compositions containing them, their use and process for their preparation
03/07/2002DE10042058A1 Bicyclische Heterocyclen, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung Bicyclic heterocycles, pharmaceutical compositions containing them, their use and process for their preparation
03/07/2002CA2731273A1 Processes and intermediates for preparing retroviral protease inhibitors
03/07/2002CA2420969A1 Phenoxybenzylamine derivatives as selective serotonin re-uptake inhibitors
03/07/2002CA2420122A1 7-oxo pyridopyrimidines
03/06/2002EP1184376A1 Novel heterocyclic carboxamide derivatives
03/06/2002EP1183091A1 Optimization of ligand affinity for rna targets using mass spectrometry
03/06/2002EP1017683A4 Protecting and linking groups for organic synthesis
03/06/2002EP0695296B1 3-aryloxy carboxylic acid derivatives and method of preparing them
03/06/2002EP0695295B1 3-(hetero)aryl carboxylic acid derivatives, methods of preparing them and intermediates used in their preparation
03/06/2002CN1339029A Method of producing thiobarbituric acid derivatives
03/06/2002CN1339028A Pyrimidine-2,4,6-triones as inhibitors of matrix metalloproteinases
03/06/2002CN1080264C Oxathiolanes, method for their preparation and pharmaceutical compoistions containing same
03/06/2002CN1080257C Guanidine derivatives
03/05/2002US6352993 Pyrimidine derivatives and processes for the preparation thereof
03/05/2002US6352991 2-hydroxymethylcyclopropylidenemethylpurines and -pyrimidines as antiviral agents
03/05/2002US6352989 Nitrogenous heterocyclic derivatives and medicine thereof
03/05/2002US6352958 Pre- and post-emergence herbicides
03/05/2002CA2049850C 4-substituted dihydropyrido[4,3-d]pyrimidines as analgesics and topical antiinflammatory agents for the treatment of skin disorders
02/2002
02/28/2002WO2002016362A2 Nitrogenous heterocyclic compounds
02/28/2002WO2002016361A2 Nitrogenous heterocyclic compounds
02/28/2002WO2002016360A2 Nitrogenous heterocyclic compounds
02/28/2002WO2002016351A1 Quinazoline derivatives as kinase inhibitors
02/28/2002WO2002016319A1 Novel thiourea compounds and the pharmaceutical compositions containing the same
02/28/2002WO2002016318A1 Novel thiourea derivatives and the pharmaceutical compositions containing the same
02/28/2002WO2002016316A1 10-ARYL-11-HBENZO [b]FLUORENE DERIVATIVES AND ANALOGS FOR MEDICINAL USE
02/28/2002WO2001085699A3 Prodrugs of hiv replication inhibiting pyrimidines
02/28/2002WO2001070255A3 Combined treatment with keratinocyte growth factor and epidermal growth factor inhibitor
02/28/2002WO2001068600A3 Benzylated pde4 inhibitors
02/28/2002WO2001046200A8 Novel piperidine and piperazine derivatives
02/28/2002WO2001042216A3 Caspase inhibitors and uses thereof