Patents
Patents for C07D 239 - Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings (42,619)
06/2003
06/11/2003EP1317414A2 Gamma-ketoacid dipeptides as inhibitors of caspase-3
06/11/2003EP1105372B1 Methoximinophenylacetic acid amides
06/11/2003EP1021413B1 The preparation and use of ortho-sulfonamido bicyclic heteroaryl hydroxamic acids as matrix metalloproteinase and tace inhibitors
06/11/2003EP0996614B1 Acrylonitrile compounds, process for their production and pesticides containing them
06/11/2003EP0892787B1 Novel alpha-hydroxylic acid derivatives, their production and use
06/11/2003EP0779894B1 Electrophilic polyethylene oxides for the modification of polysaccharides, polypeptides (proteins) and surfaces
06/11/2003CN1423632A Aromatic diamide derivatives or salts thereof, agricultural/norticultural chemicals and method of using the same
06/10/2003US6576643 Compounds containing dibenzo(A,D)cycloheptene or dibenz(B,F)oxepine derivatives are useful for treating osteoporosis, cardiovascular diosrders, cancer and inflammation
06/10/2003US6576637 Such as 3-(4-methyl-3-nitrophenyl)-3-(2-(4-(pyridin-2-yl-amino)butyryl amino)acetylamino)propionic acid; thrombosis, heart infarct, coronary heart diseases, arteriosclerosis, inflammations,
06/10/2003US6576635 Compositions comprising trimetrexate
06/10/2003US6576631 Broad disease control spectrum; residual effectiveness, rainfastness; nondamaging to crops
06/10/2003US6576159 Colorants, electroconductive materials; solubility, dissociation
06/10/2003CA2303577C Qt dispersion and heart rate variability improvement with crf antagonists to prevent sudden death
06/10/2003CA2192354C Corticotropin releasing factor against antagonist
06/10/2003CA2055670C Retroviral protease inhibiting compounds
06/05/2003WO2003045923A1 Preventives or remedies for alzheimer’s disease or amyloid protein fibrosis inhibitors containing nitrogen-containing heteroaryl compounds
06/05/2003WO2003045921A1 Heterocyclic amide compounds as apolipoprotein b inhibitors
06/05/2003WO2003045395A1 Quinazoline derivatives for the treatment of t cell mediated diseases
06/05/2003WO2002048137A3 Substituted heterocyclic phthalic acid diamide arthropodicides
06/05/2003US20030105142 Amide derivatives useful as inhibitors of the production of cytokines
06/05/2003US20030105119 For therapy of inflammation, immune disorders, asthma, chronic obstructive pulmonary disease (COPD), multiple sclerosis (MS), inflammatory bowel disease (IBD); side effect reduction
06/05/2003US20030105106 5-HT receptor ligands and uses thereof
06/05/2003US20030105102 Oxo-substituted compounds, process of making, and compositions and methods for inhibiting PARP activity
06/05/2003US20030105100 Substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamines useful for inhibiting cholesteryl ester transfer protein activity
06/05/2003US20030105092 Prevention of loss and restoration of bone mass by certain prostaglandin agonists
06/05/2003US20030105066 For use in producing antiviral, antifungal and antibacterial medicaments
06/05/2003CA2468716A1 Heterocyclic amide compounds as apolipoprotein b inhibitors
06/04/2003EP1315728A1 Process for the preparation of vitronectin receptor antagonists
06/04/2003EP1315727A2 7-oxo pyridopyrimidines
06/04/2003EP1315717A1 Quinazoline derivatives, medicaments containing these compounds, their use, and methods for the production thereof
06/04/2003EP1315715A1 Quinazoline derivatives as kinase inhibitors
06/04/2003EP1315705A1 Bicyclic heterocycles, medicaments containing these compounds, their use, and methods for the production thereof
06/04/2003EP1315704A1 2-guanidino-4-aryl-quinazoline
06/04/2003EP1315498A2 Use of ectoin or ectoin derivatives for stabilizing p53
06/04/2003EP1315473A2 Use of ectoine or ectoine derivatives for oral care
06/04/2003EP0980244B1 Use of quinazoline compounds for the treatment of polycystic kidney disease
06/04/2003EP0973844B1 Compounds and process for controlling cone tilt angle in mixtures of smectic liquid crystal compounds
06/04/2003EP0901487B1 2,3,6 trisubstituted-4(3h)-quinazolinones
06/04/2003EP0783507B1 Compounds useful as antiproliferative agents and garft inhibitors
06/04/2003EP0775120B1 Novel pyrimidine derivatives and processes for the preparation thereof
06/04/2003CN1422271A Pyrrolopyrimidinone derivatives, process of preparation and use
06/04/2003CN1422260A 2-guanidino-4-arylchinazolines as NHE-3 inhibitors
06/04/2003CN1422259A Crystalline pharmaceutical
06/04/2003CN1422254A Aryl substituted pyridines, pyrimidines, pyrazines and triazines and the use thereof
06/04/2003CN1422249A Novel alpha-sulfin-and alpha-sulfonamino acid amides
06/04/2003CN1421440A Synthesis of quinazoline-4 (3H) derivative
06/04/2003CN1110490C Sulfamide-substituted condensed seven-membered ring compound, used as medicine and medical preparation containing the same
06/04/2003CN1110483C Cyclic alkyleneureas containing monomers and polymers and latices therefrom
06/03/2003US6573278 Aryl sulfonamides and analogues thereof and their use in the treatment of neurodegenerative diseases
06/03/2003US6573270 Endothelin receptor antagonists
06/03/2003US6573269 Compounds for protecting surface of substrate from ultraviolet light
06/03/2003US6573268 Administering novel azolidinedione derivatives, tautomers, stereoisomers, polymorphs, pharmaceutically acceptable salts and solvates to treat diabetes
06/03/2003US6573218 Fused-benzene derivatives useful as herbicides
06/03/2003CA2088934C High contrast distorted helix effect electro-optic devices and tight ferroelectric pitch ferroelectric liquid crystal compositions useful therein
06/03/2003CA2053954C Process for the preparation of nitroguanidine derivatives
05/2003
05/30/2003WO2003043995A1 Process for the racemization of chiral quinazolinones
05/30/2003WO2003043994A1 Substituted acylaminophenyluracils
05/30/2003WO2003043993A1 5-phenylpyrimidines, agents comprising the same, method for production and use thereof
05/30/2003WO2003043988A1 Piperidin-2-one derivative compounds and drugs containing these compounds as the active ingredient
05/30/2003WO2003043979A2 Pharmaceutically active compounds and methods of use thereof
05/30/2003WO2003043961A2 Modulators of rho c activity
05/30/2003CA2467752A1 Piperidin-2-one derivative compounds and pharmaceutical composition comprising the same as active ingredient
05/29/2003US20030100769 Such s 2-(6-chloro-3-pyridyl)-2-imidazoline which has good affinity for and activate alpha-4-beta-2-nicotinic acetyl-choline receptors; for treatment and prevention of neuro-degenerative disorders (Alzheimer's/Parkinson's disease)
05/29/2003US20030100762 Membrane penetrative dyes sensitive to membrane potentials
05/29/2003US20030100755 For example (2S, 3S, 5S)-2-(2,6-dimethylphenoxyacetyl)amino-3-hydroxy-5-(2S-(1-tetrahydro-pyrimid-2-onyl)-3-methyl butanoyl)amino-1,6-diphenylhexane; HIV therapy
05/29/2003US20030100615 Antineoplastic polyamines capable of uptake by a target cell upon administration to a human or non-human animal, and upon uptake bind via an electrostatic interaction between positively charged nitrogen and biological counter- anions
05/29/2003US20030100608 1,4-disubstituted benzo-fused cycloalkyl urea compounds
05/29/2003US20030100575 Derivatives of barbituric and thiobarbituric acids; rapidly metabolized by blood and tissue enzymes to form polar metabolites with no hypnotic activity and which are rapidly eliminated
05/29/2003US20030100573 For treatment of debilitating bone disorders; anticancer agents
05/29/2003US20030100571 Such as 2-((6-(((4-(3,4-dimethoxyphenyl)methyl)amino)-7-ethyl-7H-purin-2-yl)amino) -4,5-methyl-N-phenyl-5-thiazole-carboxamide for treatment of lymphocyte mediated diseases such as transplant rejection and graft versus host disease
05/29/2003US20030100559 Such as 3-((3-(3-trifluoromethoxyphenoxy)phenyl)((3-(1,1,2,2-tetrafluoroethoxy) -phenyl)methyl)amino)-1,1,1-trifluoro-2-propanol for treatment of coronary artery disease
05/29/2003US20030100549 Inhibitors of c-Jun N-terminal kinases (JNK)
05/29/2003US20030100494 Containing growth hormone secretion promoting substance for prophylaxis and therapy of diseases involving degeneration or death of nerve cells
05/28/2003EP1314732A2 Substituted pyrimidine compounds and their use
05/28/2003EP1314731A2 Substituted pyrimidine compounds and their use
05/28/2003EP1313721A2 Non-imidazole aryloxyalkylamines as h3 receptor ligands
05/28/2003EP1313713A2 4-pyrimidinamine derivatives, pharmaceutical compositions and related methods
05/28/2003EP1313712A2 Process and intermediates for preparing retroviral protease inhibitors
05/28/2003EP1313704A2 Compounds useful as insecticides, compounds useful as acaricides, and processes to use and make same
05/28/2003EP1313701A1 Phenoxybenzylamine derivatives as selective serotonin re-uptake inhibitors
05/28/2003EP1313700A1 10-aryl-11h-benzo[b]fluorene derivatives and analogs as estrogenic compounds
05/28/2003EP1161428B1 Pyrimidine compounds
05/28/2003EP1027403B1 5-arylindane derivatives and ferroelectric liquid crystal mixture containing same
05/28/2003EP1015444B1 Pyrimidine derivatives and processes for the preparation thereof
05/28/2003EP0817784B1 Process for the synthesis of nucleoside analogues
05/28/2003CN1420887A 8-quinolinxanthine and 8-isoquinolinxanthine derivs. as PDE 5 inhibitors
05/28/2003CN1420873A Substd. phenyluracils
05/28/2003CN1420872A Caspase inhibitors and use thereof
05/28/2003CN1420114A 2,3-disubstd. -4(3H)-quinazolones
05/28/2003CN1109676C Substd. aminophenyluracils as herbicides and insecticides
05/28/2003CN1109675C Arylpyrimidine derivs.
05/28/2003CN1109499C Fungicide active substance combinations
05/27/2003US6570027 Method of preparing intermediates useful in synthesis of retroviral protease inhibitors
05/27/2003US6570015 Process for producing 2-substituted thiopyrimidine-4-carboxylate
05/27/2003US6569880 Bis(benzimidazole) derivatives serving as potassium blocking agents
05/27/2003US6569863 Bicyclic heteroamatic compounds useful as LH agonists
05/27/2003US6569504 Mesogenic materials with anomalous birefringence dispersion and high second order susceptibility (X(2))
05/22/2003WO2003042206A1 Pyridinone and pyrimidinone compounds
05/22/2003WO2003042186A1 Dithiocarbamate derivatives and their use as antibacterial agents
05/22/2003WO2003042168A1 NOVEL α-OXYGENATED OR α-THIOLATED CARBOXYLIC ACID PHENETHYLAMIDE DERIVATIVES