Patents
Patents for C07D 237 - Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings (8,468)
04/2003
04/01/2003CA2288439C Biphenylsulfonamides and derivatives thereof that modulate the activity of endothelin
03/2003
03/27/2003WO2003024938A1 Phthalazinones and the use thereof in order to combat undesirable microorganisms
03/27/2003WO2003024441A1 Novel use of tricyclic compound
03/26/2003EP1294724A1 Pyrrolo[2,3-d]pyrimidine compounds as immunosuppressive agents
03/26/2003EP1294380A1 A method for treating septic shock
03/26/2003CN1406228A 4-oxo-1,4-dihydro-3-cinnolinecarboxamides as antiviral agents
03/25/2003US6538135 Amination of 4,5-dichloro-1-phenylpyridazin-6-one with aqueous ammonia in presence of phenolic catalyst
03/25/2003US6537991 A method of treating a peripheral neuropathic pain in a warm-blooded animal requiring such treatment which comprises administering to said animal a therapeutically effective amount of an EP1-type prostaglandin receptor antagonist
03/20/2003US20030055248 Il-8 receptor antagonists
03/20/2003US20030055093 For therapy of cardiovascular diseases, stable or unstable angina pectoris, coronary heart disease, stable or unstable angina pectoris, coronary heart disease, Prinzmetal angina, acute coronary syndrome, heart failure, myocardial infarction
03/20/2003US20030054298 Color photography; bleaching, fixing, development
03/18/2003US6534492 Uracil substituted phenyl sulfamoyl carboxamides
03/13/2003WO2002078625A3 Therapeutic combinations for cardiovascular and inflammatory indications
03/12/2003EP0672031B1 Catechol diethers as selective pde iv inhibitors
03/11/2003US6531473 Method of treatment using arylalkylpyridazinones
03/11/2003US6531241 Anions of equal number to cations to maintain charge neutrality, are disclosed. These spacer groups may be organic or inorganic in origin and may vary in length. The spacer groups may be saturated, containing single bonds, or may have
03/06/2003WO2003018563A1 Anti-inflammatory and protein kinase inhibitor composition and method of use
03/06/2003WO2003017765A1 Treatment for cystic fibrosis
03/05/2003EP1286968A2 Substituted iminoazines
03/04/2003US6528649 Imidazoloisoquinolines
03/04/2003US6528543 Glucokinase activating for treating type II diabetes; acylurea compound, phenylacetyl-substituted; 1-(2-(3-chloro-phenyl)-3cyclopentyl-propionyl)-3-methyl-urea
02/2003
02/27/2003WO2003016286A1 3-phenoxy-4-pyridazinol derivative and herbicide composition containing the same
02/27/2003WO2003015785A1 2h-phthalazin-1-ones and methods for use thereof
02/27/2003WO2003015774A1 Compounds effecting glucokinase
02/27/2003US20030040516 Pyrazinone inhibitors of fatty acid binding protein and method
02/27/2003CA2456985A1 2h-phthalazin-1-ones and methods for use thereof
02/26/2003EP0971901B1 Phthalazinones
02/26/2003CN1399573A Use of phthalazine derivatives
02/25/2003US6525072 Prevention and treatment of cellular disorders such as cancer
02/25/2003US6525053 2-Benzyl-5-(4-methylsulfonylphenyl)-6-(4-fluorophenyl)-3(2H) -pyridazinone; cyclooxygenase (COX) inhibitors pain, fever, inflammation, rheumatoid arthritis, osteoarthritis; minimizes GI and renal side-effects
02/20/2003WO2003014090A1 Amino-phthalazinone derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions containing them
02/20/2003WO2003013484A2 N-monoacylated derivatives of o-phenylenediamines, their six membered heterocyclic analogues and their use as pharmaceutical agents
02/20/2003WO2002096516A8 Use of compositions comprising cyclooxygenase-2 selective inhibitors in combination with radiation for inhibition or prevention of cardiovascular disease
02/20/2003WO2002068399B1 Aryl carbamate derivatives, preparation and use thereof
02/20/2003WO2002024635A3 Aminoalcohol derivatives
02/20/2003CA2455759A1 Amino-phthalazinone derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions containing them
02/19/2003CN1398258A 4-hydroxycinnoline-3-carboxyamides as antiviral agents
02/19/2003CN1398252A Dehydroamino acids compounds
02/13/2003US20030033089 Substituted quinazolines and analogs and the use thereof
02/11/2003US6518310 Non-peptidic; inhibits trypsin-like protease, thrombin and embolus formation; anticoagulant
02/06/2003WO2003010153A1 N-alkyl-n-phenylhydroxylamine compounds containing metal chelating groups, their preparation and their therapeutic uses
02/06/2003WO2003010150A1 Polymorph salt of a pyridazinone derivative for the treatment of arrythmia
02/06/2003CA2454774A1 Polymorph salt of a pyridazinone derivative for the treatment of arrythmia
02/05/2003EP1280780A2 Asymmetric synthesis of piperazic acid and derivatives thereof
02/05/2003CN1100748C Inhibition of matrix metalloproteases by 2-substituted-4-(4-substituted phenyl)-4-oxobutyric acids
02/04/2003US6515124 Dehydroamino acids
02/04/2003US6514983 Inhibitors of the nucleic enzyme poly(adenosine 5'-diphospho-ribose)polymerase
02/04/2003US6514971 Cinnoline derivatives and use as medicine
01/2003
01/30/2003US20030023087 Nitrosated and nitrosylated phosphodiesterase inhibitors, compositions and methods of use
01/29/2003EP1278723A2 P-(sulfonyl)-aryl and -heteroaryl amines
01/28/2003US6512111 A method for preparing compounds of formula (I) ) wherein cyclization is carried out in a basic medium and in the presence of a phosphonic acid derivative and the use of said method as an intermediate step for preparing a compound
01/28/2003US6511987 Heterocyclic derivatives that bind to the benzodiazepine site of GABAA receptors for treatment of central nervous system disorders
01/23/2003WO2003006454A2 Heterocyclic carboxamides and their use as fungicides
01/23/2003WO2003006423A1 N-(3-amino-2-hydroxy-propyl) substituted alkylamide compounds
01/23/2003WO2003006023A1 Pyrazinone inhibitors of fatty acid binding protein and method
01/23/2003CA2453503A1 N-(3-amino-2-hydroxy-propyl) substituted alkylamide compounds
01/22/2003EP1277729A1 Ppar (gamma) modulators
01/22/2003CN1099417C New polycyclic 2,3-phthalazine derivatives and their use
01/16/2003WO2003004474A1 Pesticidally active aminoacetonitriles
01/16/2003WO2003004035A1 New use of a pyridazinone derivative
01/16/2003US20030013713 Compounds as PDE IV and TNF-inhibitors
01/16/2003CA2450821A1 New use of a pyridazinone derivative
01/15/2003EP1275301A1 Trisubstituted heterocyclic compounds and their use as fungicides
01/15/2003EP1274689A2 Sulfur containing dihydrophthalazine antagonists of excitatory amino acid receptors
01/15/2003EP1274428A2 Il-8 receptor antagonists
01/15/2003CN1390547A Therapy for tissue damage by local ischemia
01/09/2003WO2003002541A1 Pyridazinone
01/09/2003US20030009033 Substituted condensation products of N-benzyl-3-indenylacent amides with heterocyclic aldehydes for neoplasia
01/09/2003US20030008915 Acylated 6,7,8,9-tetrahydro-5H-benzocycloheptenyl amines and their use as pharmaceutical agents
01/09/2003US20030008871 Administering sulfonyl pyridazinone compounds for therapy and prophylaxis of tissue damage resulting from ischemia
01/09/2003CA2451755A1 Pyridazinone
01/08/2003EP1272476A1 2-phenyl-2h-pyridazine-3-ones
01/08/2003EP1272475A1 2-phenyl-2h-pyridazine-3-ones
01/08/2003EP1272474A1 Substituted 5-methyldihydropyridazinones and their use in the prophylaxis and/or treatment of anemias
01/08/2003EP1272456A1 Hydrazide and alkoxyamide angiogenesis inhibitors
01/08/2003CN1390217A Bicyclic and tricyclic heteroaromatic compounds
01/02/2003US20030004139 Antidiabetic agents
01/02/2003EP1268443A1 2-hydroxy-mutilin carbamate derivatives for antibacterial use
12/2002
12/31/2002US6500951 Process for preparing pyridazin-3-on derivatives
12/31/2002US6500847 Inhibition of matrix metalloproteases by substitued biaryl oxobutyric acids
12/27/2002WO2002044157A3 Parb inhibitors
12/26/2002US20020198208 Medicinal preparation and process for manufacturing thereof
12/26/2002US20020198207 Novel Hexanoic acid derivatives
12/24/2002US6498275 Use of compounds for the elevation of pyruvate dehydrogenase activity
12/24/2002US6498160 For therapy of emphysema, chronic bronchitis, asthma and allergic rhinitis
12/24/2002US6498159 Such as 4-((3-chloro-4-methoxybenzyl)amino)-1-((4-hydroxy-4 -hydroxymethyl)piperidino)-6-phthalazine carbonitrile
12/24/2002CA2150812C Catechol diethers as selective pde iv inhibitors
12/19/2002WO2002085906A3 Phthalazinones derivatives useful as pde4/7 inhibitors
12/19/2002WO2002055501A3 N-pyridyl carboxamide derivatives and pharmaceutical compositions containing them
12/19/2002US20020193596 Inhibitors of protein isoprenyl transferases
12/18/2002EP1266651A2 UV absorbing and photostabilizing agents and compositions and external preparation for skin
12/18/2002EP1265873A2 4-oxo-1,4-dihydro-3-cinnolinecarboxamides as antiviral agents
12/18/2002EP1265872A1 4-hydroxycinnoline-3-carboxyamides as antiviral agents
12/18/2002EP1265871A1 Pyridazinyl phenyl hydrazones useful against congestive heart failure
12/12/2002WO2002098849A2 Hydroxy alkyl amine derivatives as beta-secretase inhibitors and their use for the treatment of alzheimer’s disease and similar diseases
12/12/2002CA2448834A1 Hydroxy alkyl amine derivatives as beta-secretase inhibitors and their use for the treatment of alzheimer's disease and similar diseases
12/11/2002EP1264820A1 Novel amide compounds
12/11/2002EP1263723A1 Ningalin b analogs employable for reversing multidrug resistance
12/11/2002EP0752813B1 Inhibitors of metazoan parasite proteases
12/11/2002EP0624155B2 Carbamates and plant-protecting agents containing them
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