Patents
Patents for C07D 237 - Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings (8,468)
01/2005
01/20/2005DE10328888A1 Preparation of 1,2-disubstituted hexahydropyridazine-3-carboxylic acid derivatives, useful as intermediates for pharmaceuticals e.g. cilazapril, by reacting protected hydrazine with disubstituted valerate
01/19/2005EP1497269A1 Substituted 2-phenyl-3(2h)-pyridazinones
01/19/2005EP1496838A2 Substituted amides
01/19/2005CN1568187A 2H-2, 3-dinitrogen phenodiazine-1-ketone and using method thereof
01/19/2005CN1568185A Compounds effecting glucokinase
01/18/2005US6844032 Liquid crystal compounds having bis(trifluoromethyl) phenyl rings, liquid crystal compositions and liquid crystal display devices
01/13/2005WO2005003098A1 Heterocyclically substituted pentanol derivatives, method for the production thereof, and use thereof as anti-inflammatory agents
01/13/2005US20050009900 3-Substituted with a heterocyclic group, e.g., 2-Chloro-5-[1-(2,3-dihydroxy-propyl)-5-methyl-1H-pyrazol-3-yl]-N-(1-hydroxy-cycloheptylmethyl)-benzamide; treatment of IL-1 mediated disorders, including osteo- and rheumatoid arthritis, allergies, asthma, COPD, cancer, and reperfusion or ischemia in stroke
01/13/2005US20050009844 Inhibitors of p38
01/13/2005US20050009830 Fused ring cinnoline derivatives including naphthocinnolines, quinollinocinnolines and naphthopyridinopyridines, e.g., 2,3-Dimethoxydibenzo[ch]cinnoline and 2,3-Dimethoxy-8,9-methylenedioxy-dibenzo[c,h]cinnoline; treatment of anticancer agnets, fungicides and bactericides
01/13/2005CA2531060A1 Heterocyclically-substitued pentanol derivatives, process for their production and their use as anti-inflammatory agents
01/12/2005EP1495002A1 Benzamide derivatives useful as histone deacetylase inhibitors
01/12/2005CN1564687A Use of phosphodiesterase IV inhibitors
01/06/2005US20050004134 Adenosine antagonists; having 6-oxo-1,6-dihydro-3-pynidazinyl functionality; synthesis
01/06/2005US20050004127 Quinoline, isoquinoline and phthalazine derivatives as antagonists of the gonadotropin-releasing hormone
01/06/2005US20050004124 Synergistic mixture; antidiabetic agents; antiischemic agents
01/05/2005EP1493733A2 Fungicidal heterocyclic aromatic amides, their compositions and methods of use
01/05/2005EP1492757A1 (2-((2-alkoxy)-phenyl)-cyclopent-1-enyl) aromatic carbo- and heterocyclic carboxylic acid and derivatives
01/05/2005CN1561246A Compositions of cyclooxygenase-2 selective inhibitors and radiation for inhibition or prevention of cardiovascular disease
12/2004
12/30/2004US20040266774 Amide compounds
12/30/2004US20040266772 Polymorph salt of a pryridazinone derivative for the treatment of arrythmia
12/30/2004US20040261190 Hydrazono-malonitriles
12/29/2004EP1491201A1 Methods of reducing toxicity of 5-fluorouracil with acylated pyrimidine nucleosides
12/29/2004EP1490343A1 New aryl imidazoles and related compounds as c5a receptor modulators
12/29/2004EP1490340A1 Heteroaromatic urea derivatives as vr-1 receptor modulators for treating pain
12/29/2004EP1490062A1 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
12/29/2004EP1263723A4 Ningalin b analogs employable for reversing multidrug resistance
12/29/2004EP0994834A4 Ligated platinum group metal catalyst complex and improved process for catalytically converting alkanes to esters and derivatives thereof
12/29/2004EP0986545B1 Non-steroidal (hetero) cyclically substituted acylanilides with mixed gestagen and androgen activity
12/29/2004CN1558904A Substituted alkylaminopyridazinone derivatives, process for the preparation thereof and pharmaceutical composition containing the same
12/29/2004CN1558903A Water-soluble phenylpyridazine compounds and compositions containing the same
12/28/2004CA2268922C Methods of treating or preventing cardiac arrhythmia
12/28/2004CA2126072C Tri-substituted phenyl derivatives and processes for their preparation
12/23/2004US20040259863 Type 4 phosphodiesterase inhibitors and uses thereof
12/23/2004US20040259804 (Substituted)Acyl dipeptidyl inhibitors of the ICE/ced-3 family of cysteine proteases
12/23/2004CA2529729A1 New imidazopyridazinone and imidazopyridone derivatives, the preparation thereof and their use as pharmaceutical compositions
12/22/2004EP1487785A2 Novel florfenicol-type antibiotics
12/22/2004EP1133486B1 Nonsteroidal antiinflammatories
12/16/2004WO2004108690A1 Sulphonamide compounds that modulate chemokine receptor activity (ccr4)
12/15/2004EP1486489A2 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
12/15/2004EP1485365A1 Sulfonyl-derivatives as novel inhibitors of histone deacetylase
12/15/2004EP1430033A4 Anti-inflammatory and protein kinase inhibitor composition and method of use
12/15/2004CN1555366A Phthalazinones and the use thereof in order to combat undesirable microorganisms
12/09/2004WO2003104206A3 Herbicidally active heterocyclylalkynes
12/09/2004US20040248872 Safe for agricultural or gardening use; effective against insects and mammals
12/09/2004US20040248740 for controlling undesirable plants
12/08/2004EP1482940A2 Prodrugs of substituted polycyclic compounds useful for selective inhibition of the coagulation cascade
12/08/2004CN1178906C N-hydroxyformamide derivatives as inhibitors of matrix metalloproteinases
12/02/2004US20040242886 Induction apoptosis in tumor cells; antitumor, anticancer agents
12/02/2004US20040242873 Substituted alkylaminopyridazinone derivatives, process for the preparation thereof and pharmaceutical composition containing the same
12/02/2004US20040242648 Compounds having simultaneous ability to block L-type calcium channels and to inhibit phosphodiesterase type 3 activity
12/01/2004EP1481970A1 Novel herbicides
12/01/2004EP1480957A1 Hppars activators
12/01/2004EP1480649A2 Stable pharmaceutical compositions
12/01/2004EP1181280B1 Substituted benzoyl ketones, methods for producing them and their use as herbicides
12/01/2004CN1177835C Substituted benzoylcyclohexandiones
11/2004
11/30/2004US6826033 Beta 3 adrenergic receptor agonists; treatment of pollakiuria, urinary incontinence, obesity or diabetes
11/30/2004US6825196 Stable pharmaceutical compositions
11/25/2004WO2004084842A3 Inhibitors of cathepsin s
11/25/2004WO2004050657A3 COMPOUNDS WITH MIXED PDE-INHIBITORY AND β-ADRENERGIC ANTAGONIST OR PARTIAL AGONIST ACTIVITY FOR TREATMENT OF HEART FAILURE
11/25/2004US20040235877 Novel use of tricyclic compound
11/25/2004US20040235853 Therapeutic agents useful for treating pain
11/25/2004US20040235848 Phenylalanine derivatives
11/25/2004US20040235845 Use of phosphodiesterase iv inhibitors
11/25/2004US20040235830 Substituted cyclohexane derivatives and the use thereof in medicaments for treating cardiovascular diseases
11/24/2004EP1478363A1 Fused azabicyclic compounds that inhibit vanilloid receptor subtype 1 (vr1) receptor
11/24/2004EP1478361A2 Arylsulfone derivatives
11/23/2004US6821974 Vasodilation; hypotensive agents; cardiovascular disorders
11/18/2004WO2004099158A1 Monocyclic diazodioxide based bcl-2 protein antagonists
11/18/2004WO2004099146A1 Benzamide inhibitors of the p2x7 receptor
11/18/2004US20040229819 Hemiasterlin derivatives and uses thereof
11/17/2004EP1477175A1 Fused pyridazine derivative compounds and drugs containing the compounds as the active ingredient
11/17/2004EP1476434A2 Pyridazine derivatives, use of the same as medicaments, pharmaceutical compositions and method for producing the same
11/17/2004EP1476423A2 Arylsulfonamidobenzylic compounds
11/17/2004EP1476419A2 N-biphenylmethyl aminocycloalkanecarboxamide derivatives
11/17/2004EP1248620B1 A new use of levosimendan
11/17/2004EP1210333B1 p-Tolyl-heterocycles as herbicides
11/17/2004EP1087953B1 Nitrate salts of antihypertensive medicines
11/11/2004US20040225013 Acylated 6,7,8,9-tetrahydro-5H-benzocycloheptenyl amines and their use as pharmaceutical agents
11/10/2004EP1474401A2 Novel aryl- and heteroarylpiperazines
11/10/2004EP1137641B1 Process for preparing pyridazin-3-on derivatives
11/10/2004CN1545505A Polymorph salt of a pyridazinone derivative for the treatment of arrythmia
11/04/2004WO2003077847A3 Substituted amides
11/04/2004US20040220172 Uracil substituted phenyl sulfamoyl carboxamides
11/03/2004EP1473289A1 Preventives or remedies for alzheimer's disease or amyloid protein fibrosis inhibitors containing nitrogen-containing heteroaryl compounds
11/03/2004EP1471910A2 Substituted quinazolin-4-ylamine analogues as modulators of capsaicin receptors
11/03/2004CN1543455A 3-phenoxy-4-pyridazinol derivative and herbicide composition containing the same
11/02/2004US6812229 Carbamate derivative and agricultural/horticultural fungicide
11/02/2004CA2129040C Styryl derivatives and processes for their preparation
10/2004
10/28/2004US20040214890 1,3-diamino-2-hydroxypropane derivatives are useful as inhibitors of the beta-secretase enzyme that are useful in the treatment of Alzheimer's disease and other diseases characterized by deposition of A beta peptide in a mammal
10/27/2004EP1471049A1 Novel thyroid hormone receptor ligand, medicinal compositions containing the same and use thereof
10/27/2004EP1470752A1 Insecticides containing hydrazone derivatives as the active ingredient and novel hydrazone derivatives
10/27/2004EP1470112A1 Substituted pyridazinones as inhibitors of p38
10/27/2004EP1469854A1 Condensed heterocyclic compounds
10/27/2004EP1272456B1 Hydrazide and alkoxyamide angiogenesis inhibitors
10/27/2004EP0960108B1 Matrix metalloproteinase inhibitors
10/27/2004CN1539828A Nitrogen-contg. heterocyclic carboxamide derivatives or salt thereof
10/26/2004US6809088 Derivatives of 2-(iminomethyl)amino-phenyl, their preparation, their use as medicaments and the pharmaceutical compositions containing them
10/21/2004WO2004089412A1 Specific nad(p)h oxidase inhibitor
10/21/2004US20040210053 Process for preparing hexahydropyridazine-3-carboxylic acid derivatives
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