Patents for C07D 237 - Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings (8,468) |
---|
09/10/2009 | US20090227592 Compounds effecting glucokinase |
09/10/2009 | US20090227591 Cyclopentene compounds |
09/09/2009 | EP2097382A1 Heteroaryl-substituted carboxamides and use thereof for the stimulation of the expression of no synthase |
09/09/2009 | CN101528714A Polymorphic form of 4-[3-(4-cyclopropanecarbonyl-piperazine-1-carbonyl)-4-fluoro-benzyl]-2h-phthalazin-1-one |
09/09/2009 | CN101528713A Pyridazine derivatives |
09/08/2009 | US7585976 chemical intermediate for Hemiasterlin, first isolated from the sponge Hemiasterella; anticarcinogenic agent for treatment of colon cancer, tumor; prevention of restenosis of blood vessels subject to traumas such as angioplasty and stenting |
09/08/2009 | US7585974 Derivatives of 5-(pyridin-3-yl)-1-azabicyclo[3.2.1]octane, their preparation and their therapeutic application |
09/08/2009 | CA2314339C N-benzyl-3-indenylacetamide derivatives for treating neoplasia |
09/03/2009 | US20090221546 Inhibitors of factor xa and other serine proteases involved in the coagulation cascade |
09/03/2009 | US20090221529 Heterocycles and derivatives thereof and methods of manufacture and therapeutic use |
09/02/2009 | EP2096108A1 Novel organic electroluminescent compounds and organic electroluminscent device using the same |
09/02/2009 | EP2094662A1 Polycyclic acid compounds useful as crth2 antagonists and antiallergic agents |
09/02/2009 | EP2094645A1 2-hydroxy-1,3-diaminopropane derivatives |
09/02/2009 | CN101522638A Pyridizinone derivatives |
09/01/2009 | US7582657 Vanilloid receptor ligands and their use in treatments |
08/27/2009 | WO2009103478A1 Pyridone and pyridazinone derivatives as mch antagonists |
08/27/2009 | US20090215834 Heterocyclic inhibitors of mek and methods of use thereof |
08/27/2009 | US20090215736 inhibitors of apoptosis and IL-1 beta secretion; mediate cell apoptosis and inflammation; good cell penetration and pharmacokinetic properties; [3S/R(2S)]3-[2-(Carbazol-9-yl-2-oxo-ethyl)-pentanoylamino]-5-fluoro-4-oxo-pentanoic acid |
08/26/2009 | CN101516838A Soluble epoxide hydrolase inhibitors |
08/25/2009 | US7579469 For therapy of disease characterized by inflammatory, allergic, or proliferative processes |
08/25/2009 | US7579465 For treatment of picornavirus infections in mammals |
08/25/2009 | US7579347 Vanilloid receptor ligands and their use in treatments |
08/20/2009 | US20090209542 mitogen activated protein kinase inhibitors; 4-(2-Fluoro-4-(methylthio)phenylamino)-N-(2-hydroxyethoxy)-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide; used in the treatment of hyperproliferative diseases, such as cancer and inflammation in mammals |
08/19/2009 | EP2089385A2 Inhibitors of hepatitis c virus |
08/19/2009 | CN101508677A Synthesis process of 6-methoxy pyridazine-3- carboxylic acid |
08/19/2009 | CN101508676A Synthesis process of 6-methoxy pyridazine-3- carboxylic acid |
08/18/2009 | US7576234 Synthesis of 2-alkyl amino acids |
08/18/2009 | US7576072 Heterocyclic inhibitors of MEK and methods of use thereof |
08/13/2009 | WO2005122682A3 Process for the preparation of esters of piperazic acid |
08/13/2009 | US20090203702 INHIBITORS OF p38 |
08/12/2009 | EP2086999A1 Inhibitors for disrupting the interaction of ubiquitination related enzymes and uses thereof |
08/12/2009 | EP2086967A2 Inhibitors of hepatitis c virus |
08/12/2009 | EP2086944A1 Process for preparing difluoromethylpyrazolyl carboxylates |
08/12/2009 | CN101506174A Caspase inhibitors based on pyridazinone scaffold |
08/12/2009 | CN101506155A Biphenyl derivatives and their use in treating hepatitis C |
08/11/2009 | US7572793 Tau protein kinase 1 inhibitors; treatment for neurodegenerative disorders; Alzheimer's Disease, Parkinson's disease, Pick's Disease, vision defects; antiischemic, antidiabetic, anticarcinogenic, antitumor agents, antidepressants |
08/06/2009 | WO2009097306A1 Substituted pyridazine derivatives which have histamine h3 antagonist activity |
08/06/2009 | WO2009054952A3 Small molecule inhibitors of parp activity |
08/06/2009 | US20090197890 Pyridazine derivatives and their use as therapeutic agents |
08/06/2009 | CA2712885A1 Substituted pyridazine derivatives which have histamine h3 antagonist activity |
08/05/2009 | EP2085391A2 Inhibitors of factor XA and other serine proteases involved in the coagulation cascade |
08/05/2009 | EP1509506B1 Pyridazine derivatives |
08/05/2009 | EP1473289B1 Preventives or remedies for alzheimer's disease or amyloid protein fibrosis inhibitors containing nitrogen-containing heteroaryl compounds |
08/05/2009 | CN101501006A Pyridinone and pyridazinone derivatives as inhibitors of poly(ADP-ribose)polymerase (PARP) |
08/04/2009 | US7569518 3-chloro-5-(4-chlorophenyl)-6-methyl-4-(2,4,6-trifluorophenyl)pyridazine; 4,5-diphenyl-6-alkyl-,2H-pyridazin-3-one, 4-(2,6-difluoro-4-aminophenyl)-5-phenyl-6-alkylpyridazine, and 3,4-diphenyl-5-alkyl-5-hydroxy furanone intermediates; a fungicide controlling plant diseases for agriculture or gardening |
08/04/2009 | US7569517 4-biphenyl-substituted pyrazolidin-3 5-diones pesticide agent and/or microbicide and/or herbicide |
07/30/2009 | US20090192136 Benzoyl-piperazine derivatives |
07/29/2009 | EP2083014A2 Inhibitors of interleukin-1ß converting enzyme |
07/29/2009 | EP2082743A2 Inhibitors of GSK-3 and crystal structures of GSK-3beta protein and protein complexes |
07/29/2009 | EP1268443B1 2-hydroxy-mutilin carbamate derivatives for antibacterial use |
07/29/2009 | CN101495459A Monoazole ligand platinum analogs |
07/29/2009 | CN101492416A Compounds effecting glucokinase |
07/28/2009 | US7566781 melanin concentrating hormone receptor antagonist; preventing or treating vascular system diseases, nervous system disorders, metabolic disorders, urogenital diseases, respiratory diseases disorders; N-(2-ethyl-3-methylimidazo[1,2-a]pyridin-6-yl)-3-fluoro-4-(pyridin-2-ylmethoxy)benzamide |
07/23/2009 | US20090187018 Manufacture of Pure Hydralazine Salts |
07/23/2009 | US20090186155 Ink for ink-jet recording, ink cartridge, ink-jet recording apparatus, method of determining, and method of ink-jet recording |
07/22/2009 | EP2079710A1 Caspase inhibitors based on pyridazinone scaffold |
07/22/2009 | EP2079525A1 Calcium receptor modulating agents |
07/22/2009 | CN101486683A Pyridazinones and triazinones and medicinal use thereof |
07/21/2009 | US7563893 3-Phenyl-cinnoline analogue and antitumor agent using the same |
07/21/2009 | US7563790 Pyridazine derivatives |
07/16/2009 | US20090181973 Medicinal composition comprising 3-alkoxy-6-allylthiopyridazines for prevention or treatment of cancer of the pancreas |
07/15/2009 | EP2077998A1 Phthalazine, aza- and diaza-phthalazine compounds and methods of use |
07/15/2009 | EP2077997A1 Pyridazine derivatives |
07/15/2009 | EP1529037B1 Synthesis of 2-alkylcysteines, 2-(hydroxylated phenyl)-4-alkylthiazoline-4-carboxylic acids and derivatives thereof |
07/15/2009 | EP1426365B1 3-phenoxy-4-pyridazinol derivative and herbicide composition containing the same |
07/15/2009 | CN101484428A Alkyl-pyridazine derivatives as inhibitors of 11 beta hydroxysteroid dehydrogenase type 1(11b-HSD 1) |
07/14/2009 | US7560463 Diaryl ethers as opioid receptor antagonists |
07/09/2009 | WO2009086041A1 Herbicidal pyridazinone derivatives |
07/09/2009 | US20090176789 Diazaspirodecane orexin receptor antagonists |
07/09/2009 | US20090176774 Compounds and methods of use |
07/09/2009 | US20090176765 Pyridinone and Pyridazinone Derivatives as Inhibitors of Poly (Adp-Ribose) Polymerase (Parp) |
07/09/2009 | CA2707520A1 Herbicidal pyridazinone derivatives |
07/08/2009 | CN101479238A Amine derivative having npyy5 receptor antagonist activity |
07/08/2009 | CN101475526A Carboxylic acid derivatives inhibiting the binding of integrins to receptors thereof |
07/08/2009 | CN100509759C Novel alpha-oxygenated or alpha-thiolated carboxylic acid penethylamide derivatives |
07/07/2009 | CA2539969C Process for the preparation of carboxylic acids of nitrogen-containing aromatic heterocyclic compounds |
07/07/2009 | CA2461510C Substituted alkylaminopyridazinone derivatives, process for the preparation thereof and pharmaceutical composition containing the same |
07/07/2009 | CA2438324C Acylated 6,7,8,9-tetrahydro-5h-benzocycloheptenyl amines and their use as pharmaceutical |
07/02/2009 | WO2009080314A1 Pyridazine derivatives useful as fungicides and for the treatment of cancer |
07/02/2009 | WO2009079797A1 Compounds and method for treatment of cancer |
07/02/2009 | CA2710039A1 Compounds and method for treatment of cancer |
07/02/2009 | CA2709169A1 Pyridazine derivatives useful as fungicides and for the treatment of cancer |
07/01/2009 | EP2074998A2 Use of cyclic bioisosteres of purine system derivatives for the treatment of diseases caused by disorders of nitrergic and dopaminergic systems |
07/01/2009 | EP2074097A2 Compounds for treating proliferative disorders |
07/01/2009 | EP1226127B1 Substituted phenyl sulfamoyl carboxamides |
07/01/2009 | CN101472899A 2-substituted 4-benzylphthalazinone derivatives as histamine H1 and H3 antagonists |
07/01/2009 | CN100506230C Vascular intimal hyperplasia inhibitor |
06/30/2009 | US7553976 Derivatives of 2-(iminomethyl)amino-phenyl, their preparation, their use as medicaments and the pharmaceutical compositions containing them |
06/30/2009 | US7553972 Benzamide inhibitors of the P2X7 receptor |
06/30/2009 | US7553966 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof |
06/30/2009 | US7553964 Useful in treating conditions or disorders prevented by or ameliorated by histamine-3 receptor ligands; for example, 5-{4-[3-({2R}-2-methyl-pyrrolidin-1-yl)-cis-cyclobutyl]-phenyl}-pyrimidine |
06/30/2009 | CA2307111C Novel pyridazine derivatives and drugs containing the same as the active ingredient |
06/25/2009 | WO2009007856A3 Novel polymorph of atorvastatin calcium and use thereof for the preparation of amorphous atorvastatin calcium |
06/25/2009 | US20090163501 Aurora kinase modulators and method of use |
06/24/2009 | EP1781614B1 Compounds which potentiate glutamate receptor and uses thereof in medicine |
06/23/2009 | USRE40793 treating conditions related to impairment of gastric emptying, gastromotility disorders; superior gastrokinetic properties; e.g. trans-4-amino-N-[(1-butyl-3-hydroxy-4-piperidinyl)methyl]-5-chloro-2,3-dihydro-7-benzofurancarboxamide |
06/23/2009 | US7550489 N-[3-(4-chlorophenyl)-2-(3-cyanophenyl)-1-methylpropyl]-2-(5-trifluoromethyl-2-pyridyloxy)-2-methylpropanamide and phentermine, metformin, or bupropion; obesity; antipsychotic agents; synergistic; cannabinoid receptor antagonists |
06/18/2009 | US20090155187 Drug for inhibiting vascular intimal hyperplasia |
06/17/2009 | EP2069312A2 Pyridizinone derivatives |
06/17/2009 | EP2069305A2 Nicotinic acid derivatives as modulators of metabotropic glutamate receptors |