Patents for C07D 237 - Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings (8,468) |
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04/14/2010 | CN101693697A Pyrizdazine derivatives and their use as therapeutic agents |
04/13/2010 | US7696207 Therapeutic agents useful for treating pain |
04/13/2010 | US7695736 Powder of 30-90% a water-soluble cycloxygenase inhibitor, 5-60% of a buffer and 0-10% of other excipients |
04/08/2010 | US20100087479 Compositions Useful as Inhibitors of Voltage-Gated Sodium Channels |
04/07/2010 | EP2170065A1 Diphenyl substituted alkanes |
04/06/2010 | US7692006 Phthalazinone derivatives |
04/06/2010 | US7691865 4-(2-pyridin-2-yl-pyrazolo[1,5-a]pyridin-3-yl)-pyrimidin-2-ylamine; 4-[2-(6-methyl-pyridin-2-yl)-pyrazolo[1,5-a]pyrimidin-3-yl]-pyrimidin-2-ylamine; high affinity for Alk 5 and/or Alk 4 hence useful as antagonists thereof; fibrotic disorders |
04/01/2010 | WO2010036553A1 Fungicidal pyridazines |
03/31/2010 | EP2168576A2 New utilities of tricyclic compounds |
03/25/2010 | US20100077512 Pyridazin-4-ylmethyl-sulfonamides used as Fungicides and Against Arthropods |
03/25/2010 | US20100075972 Agent for treatment of multiple sclerosis |
03/24/2010 | CN101679304A Pyridazine-, pyridine- and pyrane-derivatives as GPBAR1 agonisis |
03/24/2010 | CN101679303A pyridazinone derivatives |
03/24/2010 | CN101679302A Fungicidal pyridazines, method for the production thereof, and use thereof for controlling fungi and agents containing the same |
03/24/2010 | CN101679274A phthalazine and isoquinoline derivatives with slp receptor modulating activities |
03/24/2010 | CN101678214A 芳基醚哒嗪酮衍生物 Aryl ether pyridazinones |
03/23/2010 | US7683062 of 7-chloro-N,N,5-trimethyl-4-oxo-3-phenyl-3,5-dihydro-4H-pyridazino[4,5-b]indole-1-acetamide; dysfunction of peripheral-type benzodiazepine receptors; anticarcinogenic, antiinflammatory agent, neurodegenerative diseases; stresses, arthritis; improved bioavailability, solubility, storage stability |
03/18/2010 | WO2010029379A1 Compounds for inhibiting semicarbazide-sensitive amine oxidase (ssao) / vascular adhesion protein-1 (vap-1) and uses thereof for treatment and prevention of diseases |
03/18/2010 | US20100069405 Derivatives of heteroaryl-alkylcarbamates, methods for their preparation and use thereof as fatty acid amido hydrolase enzyme inhibitors |
03/18/2010 | US20100069368 Organic Compounds and Their Uses |
03/18/2010 | US20100069351 Spiro compound and use thereof |
03/17/2010 | EP1651615B1 Pyridazinyl- piperazines and their use as histamine h3 receptor ligands |
03/17/2010 | CN101669952A Pyridazine derivatives and their use as therapeutic agents |
03/16/2010 | US7678812 Aminotetralin-derived urea modulators of vanilloid VR1 receptor |
03/16/2010 | US7678798 5-({4-[(3S)-4-(5-bromo-2,3-dihydro-1H-inden-1-yl)-3-methylpiperazin-1-yl]-4-methylpiperidin-1-yl}carbonyl)-4,6-dimethylpyrimidine; inflammatory diseases, immune diseases and viral infections; HIV |
03/16/2010 | US7678795 (1S,8R)-5-Cyclopropyl-1,11,11-trimethyl-3,4-diaza-tricyclo[6.2.1.02,7]undeca-2(7),3,5-triene; type II diabetes; 11beta-hydroxysteroid dehydrogenase type 1 (11beta-HSD1) |
03/16/2010 | US7678778 Salts of isophosphoramide mustard and analogs thereof as anti-tumor agents |
03/11/2010 | WO2010028051A2 Substituted heterocyclic mercaptosulfonamide metalloprotease inhibitors |
03/11/2010 | US20100063053 Heterocyclic inhibitors of mek and methods of use thereof |
03/10/2010 | EP1751113B1 Urea antagonists of p2y1 receptor useful in the treatment of thrombotic conditions |
03/09/2010 | US7674828 Urea antagonists of P2Y1receptor useful in the treatment of thrombotic conditions |
03/09/2010 | US7674809 Anti-inflammatory and analgesic heterocyclic amidines that inhibit nitrogen oxide (NO) production |
03/04/2010 | WO2010004215A3 Substituted 1-benzyl-cinnolin-4(1h)-one derivatives, preparation thereof, and therapeutic use thereof |
03/03/2010 | EP1996557B1 Pyridazinone compound and use thereof as herbicides |
03/02/2010 | US7671050 (4-Methoxyphenyl)-[3-(4-methoxyphenyl)-[1,2,4]triazolo[3,4-a]phthalazin-6-yl]-amine; phosphodiesterase inhibitors |
02/25/2010 | US20100048590 N-(3-amino-2-hydroxy-propyl) substituted alkylamide compounds |
02/25/2010 | US20100048579 Pyridazine-, pyridine- and pyrane-derivatives as gpbar1 agonists |
02/25/2010 | US20100048578 Hydrazide compound and harmful arthropod-controlling agent containing the same |
02/24/2010 | EP2157084A1 5-phenyl-3-pyridazinone derivative |
02/24/2010 | CN101657430A organic compounds and their uses |
02/23/2010 | US7667037 Processes for preparation of ziprasidone |
02/23/2010 | US7667035 (R)-2-(-3-amino-piperidin-1-yl)-3-(but-2-ynyl)-5-(4-methyl-quinazolin-2-ylmethyl)-3,5-dihydro-imidazo[4,5-d]pyridazin-4-one; inhibitors of dipeptidylpeptidase IV (DPP IV) |
02/18/2010 | WO2010019417A2 Chymase inhibitors |
02/18/2010 | US20100041663 Organic Compounds as Smo Inhibitors |
02/18/2010 | US20100041661 Caspase inhibitors based on pyridazinone scaffold |
02/18/2010 | US20100041555 3-Phenoxy-4-pyridazinol derivatives and herbicidal composition containing the same |
02/18/2010 | CA2733128A1 Chymase inhibitors |
02/17/2010 | EP2152370A1 Aryl ether pyridazinone derivatives |
02/17/2010 | EP1511737B1 Aryloximes |
02/17/2010 | CN101648914A Method for preparing 6-methyl-3-(3,4-dichloroanilino)-4-(3-trifluoromethylphenyl)pyridazine and phytocidal activity thereof |
02/16/2010 | US7662959 Quaternary trifluoromethylcyclohexane derivatives for liquid crystals |
02/16/2010 | US7662821 Tetrahydronaphthalene derivatives, process for their production and their use as anti-inflammatory agents |
02/16/2010 | US7662818 e.g. 4-[5-(piperidine-1-carbonyl)-furan-2-ylmethyl]-2H-phthalazin-1-one; enzyme poly(ADP-ribose)polymerase (synthase)-1 or poly ADP-ribosyltransferase (PARP-1) inhibitor; anticarcinogenic agent with BRCA2 deficient phenotype; septic shock; ischemic injury; hemorrhagic shock; and multiple sclerosis |
02/16/2010 | CA2478183C Substituted amides |
02/16/2010 | CA2429109C Anti-inflammatory agents |
02/10/2010 | EP2150539A1 Pyridazinone derivatives |
02/10/2010 | EP1747196B1 Substituted aryl acylthioureas and related compounds; inhibitors of viral replication |
02/09/2010 | US7659307 Heterocyclic carboxamides and their use as fungicides |
02/09/2010 | US7659297 improved selectivity and pharmacokinetic properties; 6-Fluoro-1-[(1 H-indazol-4-yl)amino]-4,4-dimethyl-2-(trifluoromethyl)-1,2,3,4-tetrahydronaphthalene-2,5-diol; cyclization of imines |
02/09/2010 | US7659272 N-[phenyl or heteroaryl carbonoyl pyridyl] arylsulfonamides; antiinflammatory, antianaphylactic agents; transplant rejection, gastointestinal, respriatory system and skin disorders |
02/09/2010 | CA2413061C Serine protease inhibitors |
02/04/2010 | WO2009129267A3 Small molecule inhibitors of the pleckstrin homology domain and methods for using same |
02/04/2010 | US20100029689 Phosphodiesterase 4 inhibitors |
02/04/2010 | US20100029658 Heterocyclic derivatives, pharmaceutical compositions and methods of use thereof |
02/03/2010 | CN101641336A 3 - cinnolinecarboxamide derivatives and their use for treating cancer |
02/03/2010 | CN101638390A Method for industrial preparation of 6-methyl-3-amino pyridazine |
02/02/2010 | US7655749 contacting pyridines or pyrimidines monomer with a particlulate catalyst containing metal or alloy (e.g. magnesium or alloy substrate) having a second reduced metal or alloy ( Ni, Cu, Co etc.) coated on the substrate to form dimer ( bi-pyridine) or polymer |
02/02/2010 | US7655666 Substituted 1H-quinazoline-2,4-diones useful as AMPA receptor ligands |
02/02/2010 | US7655649 Inhibitors of Akt activity |
01/28/2010 | US20100022547 Compounds and Methods for Treating Mammalian Gastrointestinal Parasitic Infections |
01/28/2010 | US20100022526 Pyridazine derivatives, processes for their preparation and their use as fungicides |
01/28/2010 | US20100019657 Novel organic electroluminescent compounds and organic electroluminescent device using the same |
01/27/2010 | CN100584831C Pyridazinyl- piperazines and their use as histamine h3 receptor |
01/26/2010 | US7652144 Compounds as PDE IV and TNF inhibitors |
01/26/2010 | US7652006 Substituted 1(2H)-phthalazinones and pharmaceutical compositions thereof |
01/26/2010 | CA2469380C Heteroaryl-substituted aminocyclohexane derivatives |
01/21/2010 | WO2010006940A1 Tetrahydrocinnolines as 11 beta hsd1 inhibitors for diabetes |
01/21/2010 | US20100016545 Process for the covalent coupling of two molecules by means of a diels-alder reaction with inverse electron requirement |
01/21/2010 | US20100016339 Fungicidal compounds and compositions |
01/21/2010 | US20100016325 Tetrahydrocinnoline derivatives |
01/21/2010 | CA2730059A1 Tetrahydrocinnolines as 11 beta hsd1 inhibitors for diabetes |
01/20/2010 | CN100581543C Tetrahydronaphthalene derivatives, process for their production and their use as anti-inflammatory agents |
01/14/2010 | WO2010004215A2 Substituted 1-benzyl-cinnolin-4(1h)-one derivatives, preparation thereof, and therapeutic use thereof |
01/14/2010 | WO2010003624A2 Heterocyclic compounds, processes for their preparation, medicaments comprising these compounds, and the use thereof |
01/14/2010 | US20100010220 Process for Preparing Amidrazones |
01/14/2010 | US20100010015 Heterocyclic spiro-compounds as aldosterone synthase inhibitors |
01/14/2010 | US20100009991 Polycyclic acid compounds useful as crth2 antagonists and antiallergic agents |
01/14/2010 | US20100009850 Iodine-phenyl-substituted cyclic cetoenols |
01/14/2010 | CA2729896A1 Substituted 1-benzyl-cinnolin-4(1h)-one derivatives, preparation thereof, and therapeutic use thereof |
01/13/2010 | EP2143715A1 Method for obtaining pure enantiomers of a pyridazinone derivative |
01/13/2010 | EP2086944B1 Process for preparing difluoromethylpyrazolyl carboxylates |
01/13/2010 | EP1910298B1 Phenylglycinamide and pyridylglycinamide derivatives useful as anticoagulants |
01/13/2010 | EP1144388B1 Acyl derivatives which treat vla-4 related disorders |
01/12/2010 | US7645757 Derivatives of heteroaryl-alkylcarbamates, methods for their preparation and use thereof as fatty acid amido hydrolase enzyme inhibitors |
01/12/2010 | CA2442906C Reconstitutable parenteral composition containing a cox-2 inhibitor |
01/07/2010 | WO2010000456A1 Substituted 6- (1-piperazinyl) -pyridazines as 5-ht6 receptor antagonists |
01/07/2010 | CA2729313A1 Substituted 6-(1-piperazinyl)-pyridazines as 5-ht6 receptor antagonists |
01/06/2010 | CN100577163C Compounds effecting glucokinase |
01/05/2010 | CA2185397C Arylalkyl-diazinones |
12/31/2009 | US20090326222 Benzothiazole cyclobutyl amine derivatives |