Patents
Patents for C07D 231 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings (25,550)
03/2006
03/02/2006WO2006021652A1 Method for preparing n-piperidino-1,5-diphenylpyrazole-3-carboxamide derivatives
03/02/2006WO2006021213A2 Vasopressin v1a antagonists
03/02/2006WO2005103010A3 Pyrazole derivatives useful for the treatment of cancer
03/02/2006WO2005079774A3 Management of ophthalmologic disorders, including macular degeneration
03/02/2006US20060047126 e.g. 3-[1-(2,4-dichlorobenzyl)-6-trifluoromethyl-1H-indazol-3-yl]-acrylic acid; anticarcinogenic agent; inhibitors of spermatogenesis, heat shock proteins and/or elongation factor 1 alpha; analogues of lonidamine
03/02/2006DE102004041531A1 Verfahren zum Herstellen von Biphenylaminen A method for producing biphenyl amines
03/02/2006CA2577837A1 Diarylsulfones as 5-ht2a antagonists
03/02/2006CA2577420A1 Lonidamine analogues and their use in male contraception and cancer treatment
03/02/2006CA2577089A1 Sigma receptor inhibitors
03/02/2006CA2564223A1 Method for preparing n-piperidino-1,5-diphenylpyrazole-3-carboxamide derivatives
03/01/2006EP1630164A1 Pyrazolopyrimidinones as phosphodiesterase inhibitors
03/01/2006EP1628963A1 Novel ureido - and amido-pyrazolone derivatives
03/01/2006EP1628962A1 Iodopyrazolyl carboxanilides
03/01/2006EP1628661A2 Modulators of vr1 receptor
03/01/2006EP1311507B1 Fused pyrazole derivatives being protein kinase inhibitors
03/01/2006EP1017382B1 Biarylalkanoic acids as cell adhesion inhibitors
03/01/2006CN1742013A Pyrazolopyrimidine compound and method for producing the same
03/01/2006CN1740179A N4-substituent pyrazolyl [4,5-e][1,2,4] thiadiazine derivative and its prepn process and medicine composition
03/01/2006CN1740162A Process for the preparation of pesticidal compounds
03/01/2006CN1243723C N-phenpropylcyclopentyl-substituted glutaramide derivatives as NEP inhibitors for FSAD
02/2006
02/28/2006US7005433 Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4
02/23/2006WO2005123688A3 3-aminoindazoles
02/23/2006WO2005048953A3 Amide derivatives as kinase modulators
02/23/2006US20060041095 Intermediate products, methods for their preparation and use thereof
02/23/2006US20060040973 Novel guanidine mimics as factor Xa inhibitors
02/23/2006DE102004039280A1 1,5-Diphenyl-pyrazole 1,5-diphenyl-pyrazoles
02/23/2006CA2576531A1 1,5-diphenylpyrazoles
02/23/2006CA2574078A1 Ophthalmic compositions for treating ocular hypertension
02/22/2006EP1627877A1 Processes for producing pyrazoloacridone derivative and intermediate therefor
02/22/2006EP1626967A1 Substituted pyrazoles
02/22/2006EP1626963A1 Substituted pyrazoline compounds, their preparation and use as medicaments
02/22/2006EP1626962A1 Benzamide inhibitors of the p2x7 receptor
02/22/2006EP1121431B1 Non-endogenous, constitutively activated human g protein-coupled receptors
02/22/2006CN1738804A 吡唑化合物 Pyrazole compounds
02/21/2006US7002023 Method for producing 1 substituted 5-chloro-4 methly pyrazoles
02/21/2006US7001917 2-(4-(4-(4-Fluorophenyl)-3,5-imethyl-1H-pyrazol-1-yl)phenyl) ethyl (4-methylphenyl)sulfonylcarbamate ammonium salt, e.g., as an antagonist for Prostoglandin E receptor; analgesics; antipyretics; antiinflammatory agents
02/16/2006WO2006017384A2 Indazoles useful in treating cardiovascular diseases
02/16/2006WO2006015860A2 Pyrazole derivatives for treating conditions mediated by activation of the adenosine a2b or a3 receptor
02/16/2006WO2005121097A3 Pyrazole derivatives, compositions containing such compounds and methods of use
02/16/2006WO2005080317A3 Therapeutic amide derivatives
02/16/2006US20060035934 Fused compounds that inhibit vanilloid subtype 1 (VR1) receptor
02/16/2006US20060035110 Electroluminescent materials and devices
02/16/2006CA2576407A1 Substituted phenylacetamides and their use as glucokinase activators
02/16/2006CA2576254A1 Compounds which potentiate glutamate receptor and uses thereof in medicine
02/16/2006CA2575180A1 Indazoles useful in treating cardiovascular diseases
02/16/2006CA2572752A1 Pyrazole derivatives for treating conditions mediated by activation of the adenosine a2b or a3 receptor
02/16/2006CA2572745A1 Pyrazole amide derivatives, compositions containing such compounds and methods of use
02/15/2006CN1735614A Pyrazolopyrimidines as cyclin-dependent kinase inhibitors
02/15/2006CN1241915C Prepn process and use of substituted pyrazole compound
02/14/2006US6998489 Methods of making indazoles
02/14/2006US6998415 Substituted sulfonylphenylheterocycles as cyclooxygenase-2 and 5-lipoxygenase inhibitors
02/14/2006US6998414 Substituted arylamides as IP antagonists
02/09/2006WO2006014290A2 Anti-inflammatory medicaments
02/09/2006WO2006014134A1 Novel piperidine derivative for the treatment of depression
02/09/2006WO2003090691A3 Method and compositions for identifying anti-hiv therapeutic compounds
02/09/2006US20060030618 Vanilloid receptor ligands and their use in treatments
02/09/2006US20060030612 2-Benzyl-3-(4-methoxyphenyl)-7-trifluoromethyl-2h-indazole; 3-[4-(2-benzyl-7-trifluoromethyl-2h-indazol-3-yl)-benzyl]-benzoic acid methyl ester, for example; useful in the treatment or inhibition of LXR (Liver X receptor) mediated diseases, e.g., cardiovascular diseases
02/09/2006CA2576073A1 Novel piperidine derivative for the treatment of depression
02/09/2006CA2573124A1 Anti-inflammatory medicaments
02/08/2006EP1623741A2 Cannabinoid receptor ligands for hair growth modulation
02/08/2006EP1622904A1 Cannabinoid receptor ligands and uses thereof
02/08/2006EP1622892A1 Indazoles having analgesic activity
02/08/2006EP1622890A2 Blockers of the quorum sensing system of gram-negative bacteria
02/08/2006EP1622876A1 Cannabinoid receptor ligands and uses thereof
02/08/2006EP1622870A2 Glutaminyl based dp iv-inhibitors
02/08/2006EP1622866A1 Aminopropanol derivatives as sphingosine-1-phosphate receptor modulators
02/08/2006EP1318978B1 N-acylsulfonamide apoptosis promoters
02/08/2006EP1309328A4 Cox-2 inhibitors and the prevention of the side effects of radiation therapy
02/08/2006EP1149082B1 Process for preparing pesticidal intermediates
02/08/2006CN1732161A 1,3-diamino-2-hydroxypropane pro-drug derivatives
02/08/2006CN1732158A Indazole derivatives as CRF antagonists
02/08/2006CN1732157A 1-alkyl-3-aminoindazoles
02/08/2006CN1732156A Biphenyl derivatives and their use as fungicides
02/08/2006CN1732155A 4-amino-5-methylpyrazole derivatives and process for production thereof
02/08/2006CN1731994A Prophylactic and therapeutic agent for neuropathy
02/08/2006CN1240679C 2- and 2,5-substituted phenylketoenols
02/07/2006US6995181 hyterocyclylaminomethyl- or aminocarbonyl-substituted 9,10-ethanoanthracenes or their aza derivatives; treating obesity, diabetes, inflammatory and immune disorders
02/07/2006US6995178 Insecticidal anthranilamides
02/02/2006WO2006011469A1 Novel cyclohexane derivative, prodrug thereof and salt thereof, and therapeutic agent containing the same for diabetes
02/02/2006WO2006011005A1 Derivatives of pyrazoline, procedure for obtaining them and use thereof as therapeutic agents
02/02/2006WO2005113511A9 Urea antagonists of p2y1 receptor useful in the treatment of thrombotic conditions
02/02/2006WO2005110994A3 Substituted pyrazolyl urea derivatives useful in the treatment of cancer
02/02/2006US20060025596 Method for deuteration or tritiation of heterocyclic ring
02/02/2006US20060025467 3-amino-1-arylpropyl indoles as monoamine reuptake inhibitors
02/02/2006US20060025466 E.g., N-[1-cyano-1-methyl-2-(5-nitroindazol-1-yl)-ethyl]-4-trifluoromethoxybenzamide; especially suitable for controlling parasites such as helminthes on warm-blooded animals.
02/02/2006US20060025454 Prenylation inhibitors and methods of their synthesis and use
02/02/2006US20060025448 Hair growth stimulators
02/02/2006US20060025416 Substituted aryl acylthioureas and related compounds; inhibitors of viral replication
02/02/2006US20060025415 Compositions useful as inhibitors of voltage-gated sodium channels
02/02/2006DE102004033021A1 Liquid pressure transmitting medium, useful in hydraulic component or machines, comprises ionic liquid as pressure transmitting medium
02/02/2006CA2578332A1 Derivatives of pyrazoline, procedure for obtaining them and use thereof as therapeutic agents
02/02/2006CA2574460A1 High stability diionic liquid salts
02/02/2006CA2574313A1 Inhibitors of hsp90
02/02/2006CA2573777A1 Novel cyclohexane derivative, prodrug thereof and salt thereof, and therapeutic agent containing the same for diabetes
02/01/2006EP1620445A2 Method and compositions for identifying anti-hiv therapeutic compounds
02/01/2006EP1620412A2 Heterocyclic compounds and hydro isomers thereof
02/01/2006EP1620405A2 Pyrazole-amides and sulfonamides as sodium channel modulators
02/01/2006EP1620108A2 Pyrazole-amine compounds useful as kinase inhibitors
02/01/2006EP1620091A2 Inhibitors of glutaminyl cyclase
02/01/2006EP1620090A1 Pyrazole compounds as hsp90 inhibitors for the treatment of cancer