Patents
Patents for C07D 231 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings (25,550)
03/2006
03/30/2006US20060069269 e.g. N-(1-Benzyl-3-oxo-2,3-dihydro-1H-indazol-5-yl)-3-chloro-2-methyl-benzenesulfonamide; 11beta-hydroxysteroid dehydrogenases (11beta-HSD's) inhibitor; antidiabetic, hypoglycemic agent; non-insulin dependent diabetes, metabolic syndrome, obesity
03/30/2006US20060069255 Novel aryl ureido benzoic acid derivatives and their use
03/30/2006US20060069147 hydrolase enzyme antagonists such as N-{(6S,9R,11R)-2-[5-4-fluoroophenyl)-1-methyl-1H-pyrazol-3-yl]-5,6,7,8,9,10-hexahydro-6,9-methanobenzo[a][8]annulen-11-yl}-N'-(2,2,2-trifiuoroethyl)sulfamide that inhibit processing of amyloid precursor protein, useful in treating or preventing Alzheimer's disease
03/30/2006US20060069140 Pyrazolone compounds and thrombopoietin receptor activator
03/30/2006DE102004046308A1 Neues Verfahren zur Herstellung von 3,5-Dimethylpyrazol-blockierten Polysocyanaten New process for the preparation of 3,5-dimethylpyrazole-blocked Polysocyanaten
03/30/2006CA2580787A1 Heterocyclic derivatives for the treatment of diseases mediated by stearoyl-coa desaturase enzymes
03/30/2006CA2580265A1 Amino-containing compounds which inhibit memapsin 2 beta-secretase activity and methods of use thereof
03/29/2006EP1640003A2 Compositions comprising a Cyclooxygenase-2 Inhibitor and a Leukotriene B4 receptor antagonist
03/29/2006EP1638957A1 N-heterocyclyl phenyl-substituted cyclic ketoenols
03/29/2006EP1638946A2 2-aminoethyl substituted pyrimidin-2-ones, cyclopropanes, pyrazolines, pyrimidines and benzothiazepines and their use as urotensin ii urotensini ii and somatostatins 5 receptor ligands
03/29/2006EP1638945A1 Heterocyclically substituted pentanol derivatives, method for the production thereof, and use thereof as anti-inflammatory agents
03/29/2006EP1638941A1 Indazole, benzisoxazole, and benzisothiazole kinase inhibitors
03/29/2006EP1638928A1 N-alkynyl-2-(substituted aryloxy)alkylthioamide derivatives as fungicides
03/29/2006EP1638612A2 Cox-2-targeted imaging agents
03/29/2006EP1638540A2 Pyrazolidinedione derivatives and their use as platelet aggregation inhibitors
03/29/2006CN1247546C Pyrazolinone derivatives
03/28/2006US7019094 Intermediate products, methods for their preparation and use thereof
03/28/2006US7019019 Matriptase inhibitors and methods of use
03/28/2006US7019011 Aminoindazole derivatives as medicaments and pharmaceutical compositions including them
03/28/2006US7019006 Compounds useful as anti-inflammatory agents
03/28/2006US7019003 Bactericides
03/28/2006US7018999 Administering a stress-activated protein kinase inhibitor, particularly a fused pyrrolocarbazole compound.
03/28/2006CA2343459C Pyrazole derivatives as anti-inflammatory/analgesic agents
03/28/2006CA2125104C Substituted benzoylguanidines, process for their preparation, their use as a medicament or diagnostic, and medicament containing them
03/28/2006CA2120374C 9-[(substituted glycyl) amido]-6-(substituted)-5-hydroxy-6-deoxytetracyclines
03/23/2006WO2006030211A2 Acyclic sulphonamides
03/23/2006WO2006030124A1 Condensed pyrazole derivatives, preparation method thereof and therapeutic use of same
03/23/2006WO2005095348A3 Pyrazole-amine compounds for the treatment of neurodegenerative disorders
03/23/2006US20060063938 Compounds to treat hiv infection and aids
03/23/2006US20060063820 2,6-dihalo-4-(3,3-dichloro-allyloxy)-benzylalcohole derivatives having insecticidal and acaricidal properties
03/23/2006US20060063798 Heterocyclic aromatic compounds useful as growth hormone secretagogues
03/23/2006US20060063765 5-[({[({(2S)-4-[(3,4-dichlorophenyl)methyl]-2-morpholinyl}methyl)amino]carbonyl}amino)methyl]-N-methyl-3-furancarboxamide; free of N-{[4-(3,4-dichlorobenzyl)morpholin-2-yl]methyl}-N'-(2-furylmethyl)urea; CCR3/chemokine recetptor/ antagonists
03/23/2006US20060063759 e.g. 5-(10,11-Dihydro-dibenzo[a,d]cyclohepten-5-ylidenemethyl)-3H-benzooxazol-2-one; antiinflammatory, antidiabetic agent; electrolytes and water retention modulator; hypotensive, hypoglycemic agent; arrhythmias, myocardial fibrosis, osteoporosis, polyuria, polydipsia, Crohn's disease
03/23/2006DE102004044827A1 Jod-phenylsubstituierte cyclische Ketoenole Iodine-substituted cyclic ketoenols
03/23/2006CA2579799A1 Benzoyl-substituted serine amides
03/22/2006EP1637539A1 Pyrazole derivative, drug composition containing the same and production intermediate therefor
03/22/2006EP1637522A1 Substituted pyrazoline compounds for reducing triglycerides in blood
03/22/2006EP1636192A1 3-alkylidenehydrazino substituted heteroaryl compounds as thrombopoietin receptor activators
03/22/2006EP1635821A2 4-bromo-5-(2-chloro-benzoylamino)-1h-pyrazole-3-carboxylic acid (phenyl)amide derivatives and related compounds as bradykinin b1 receptor antagonists for the treatment of inflammatory diseases
03/22/2006CN1751037A Sulfonamide derivatives as PPAR modulators
03/22/2006CN1751029A 2-aminoethyl substituted pyrimidin-2-ones, cyclopropanes, pyrazolines, pyrimidines and benzothiazepines and their use as urotensin ii and somatostatin 5 receptor ligands
03/22/2006CN1751028A Non-nucleoside reverse transcriptase inhibitors
03/22/2006CN1246304C Intermediate product for preparing benzamidoxime derivative
03/21/2006US7015233 Fused compounds that inhibit vanilloid subtype 1 (VR1) receptor
03/21/2006US7015218 Amide compounds and medicinal use thereof
03/21/2006US7014663 Compounds derived from diaminopyrazoles substituted by an aminoalkyl or aminoalkenyl radical and their use in oxidation dyeing of keratinous fibres
03/21/2006CA2072416C Cyclopropenone derivatives
03/16/2006WO2006028035A1 Oxidation reaction catalyst and process for producing compound using the same
03/16/2006WO2005034850A3 Cycloalkyl heterocycles for treating hepatitis c virus
03/16/2006US20060058366 Jnk inhibitor
03/16/2006US20060058363 Nitric oxide releasing selective cyclooxygenase-2 inhibitors
03/16/2006US20060058315 2-Oxo-ethanesulfonamide derivates
03/15/2006EP1634873A1 Sigma receptor inhibitors
03/15/2006EP1634872A1 Pyrazole derivatives as sigma receptor inhibitors
03/15/2006EP1633354A2 N-(((((1,3-thiazol-2-yl)amino)carbonyl)phenyl)sulfonyl)phenylalanine derivatives and related compounds for the treatment of diabetes
03/15/2006EP1633351A1 5-substituted 2h-pyrazole-3-carboxylic acid derivatives as agonists for the nicotinic acid receptor rup25 for the treatment of dyslipidemia and related diseases
03/15/2006EP1633350A2 Acylated amino acid amidyl pyrazoles and related compounds
03/15/2006EP1633349A1 4-bromo-5- (2-chloro-benzoylamino)-1h-pyrazole-3-carboxylic acid (1-(aminocarbonyl) eth-1-yl) amide derivatives and related compounds as bradykinin b1 receptor antagonists for the treatment of inflammatory diseases
03/15/2006EP1633348A1 4- BROMO - 5 - (2- CHLORO - BENZOYLAMINO) - 1H - PYRAZOLE - 3 - CARBOXYLIC ACID AMIDE DERIVATIVES AND RELATED COMPOUNDS AS BRADYKININ B sb 1 /sb RECEPTOR ANTAGONISTS FOR THE TREATMENT OF INFLAMMATORY DISEASES
03/15/2006EP1567151B1 3-(2-hydroxy-phenyl)-1h-pyrazole-4-carboxylic acid amide derivatives as hsp90 inhibitors for the treatment of cancer
03/15/2006EP1465864B1 Inhibitors of factor xa and other serine proteases involved in the coagulation cascade
03/15/2006EP1309593B1 Substituted pyrazoles
03/15/2006EP1296679B1 Dermal therapeutic system containing non-steroidal antiphlogistics with selective cox-2 inhibition
03/15/2006EP1129078B1 Indazole derivatives with 5-ht2 receptor activity
03/15/2006CN1747950A 2-(1h-indazole-6-ylamino)-benzamide compounds as protein kinases inhibitors useful for the treatment of ophthalmic diseases
03/15/2006CN1747730A Pyrazole derivatives modulators of hepatocyte growth factor (scatter factor) activity
03/15/2006CN1245388C Process for synthesis of lonidamine
03/15/2006CN1245384C Carboxamides as fungicides in agriculture
03/14/2006US7012119 Cleaving and replacing thio control agent moieties from polymers made by living-type free radical polymerization
03/14/2006US7012075 Cathepsin cysteine protease inhibitors
03/14/2006CA2267879C Heteroaryl succinamides and their use as metalloproteinase inhibitors
03/14/2006CA2103838C Novel 7-(substituted)-8-(substituted-9-[(substituted glycyl)amido]-6-demethyl-6-deoxytetracyclines
03/09/2006WO2006025069A2 Tricyclic pyrazole derivatives as cannabinoid receptor modulators
03/09/2006WO2006024930A1 Novel co-crystals between polyethylene glycols and 5-phenylpyrazolyl-1-benzenesulfonamides
03/09/2006WO2006024858A1 4-arylazo-3,5-diamino-pyrazole compounds and use thereof
03/09/2006WO2006024388A1 Method for the production of biphenylamines
03/09/2006WO2005105770A3 Arylphenylamino-, arylphenylamide-, and arylphenylether-sulfide derivatives
03/09/2006US20060052614 Such as 5-amino-3-cyano-1-(2,6-dichloro-4-trifluoromethylphenyl)pyrazole by reacting hydrazine and dicyanoacetylene in chloroform, stirring, heating, the crystallizing in hexane/toluene solvent; for preparation of pesicidal intermediates
03/09/2006US20060052613 1-alkyl-3-aminoindazoles
03/09/2006US20060052597 Aryloxyalkylamine derivatives as h3 receptor ligands
03/09/2006US20060052445 Diarylsulfones as 5-HT2A antagonists
03/09/2006US20060052358 Modulators of ATP-binding cassette transporters
03/09/2006DE10231627B4 Heterozyklisch substituierte Benzoylharnstoffe und ihre Verwendung als Arzneimittel Heterocyclic unsubstituted benzoyl ureas and their use as a medicament
03/08/2006EP1632483A1 Heterocyclic substituted carbonyl derivatives and their use as dopamine d3 receptor ligands
03/08/2006EP1632477A1 Benzamide derivative or salt thereof
03/08/2006EP1631568A1 Pyrazole derivatives as phosphodiesterase 4 inhibitors
03/08/2006EP1631560A2 C-fms kinase inhibitors
03/08/2006EP1631143A1 Hydrazone derivatives for combatting harmful insects and arachnids
03/08/2006EP1482924A4 Cathepsin cysteine protease inhibitors
03/08/2006EP1325009B1 Amino-substituted tetracyclic compounds useful as anti-inflammatory agents and pharmaceutical compositions comprising same
03/08/2006CN1745068A Pyrazolyl-n-carboxylanilide compound for preventing and controlling harm microbes
03/08/2006CN1745067A Biphenylcarboxamide compound
03/08/2006CN1744894A 3-(2-hydroxy-phenyl)-1H-pyrazole-4-carboxylic acid amide derivatives as HSP90 inhibitor for the treatment of cancer
03/08/2006CN1244564C Process for prepn. of pesticidal compounds
03/08/2006CN1244542C Aromatic amine derivatives having NOS inhibitory effect
03/07/2006US7009056 Glaucoma; multiple sclerosis
03/02/2006WO2006023783A1 Novel anthranilamides useful for controlling invertebrate pests
03/02/2006WO2006023704A2 Lonidamine analogues and their use in male contraception and cancer treatment
03/02/2006WO2006021806A1 Arylsulphonylstilbene derivatives for treatment of insomnia and related conditions
03/02/2006WO2006021805A1 Diarylsulfones as 5-ht2a antagonists