| Patents for C07D 221 - Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups (10,931) |
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| 03/22/2000 | CN1248257A Compound for inhibition of gastric acid secretion |
| 03/22/2000 | CN1050605C Cycloalkano-indole and -azaindole derivatives, its prepn. and medical composition containing them |
| 03/21/2000 | US6040305 Enzyme inhibitor as antitumor agent treating pancreatic tumor, lung cancer, myeloid leukemia, thyroid follicular tumor, myelodysplastic tumor, epidermal carcinoma tumor, bladder tumor, colon tumor, breast tumor, prostate tumor |
| 03/17/2000 | CA2282112A1 Annulated 4-carboxyamino-2-methyl-1,2,3,4-tetrahydroquinolines |
| 03/15/2000 | EP0984969A1 Fused dihydropyrans |
| 03/15/2000 | EP0984942A1 Liquid benz-iso-quinoline derivatives |
| 03/15/2000 | EP0984777A1 Arylsubstituted piperazines useful in the treatement of benign prostatic hyperlasia |
| 03/08/2000 | EP0983507A1 Tricyclic tetrahydroquinoline derivatives and tricyclic tetrahydroquinoline combinatorial libraries |
| 03/08/2000 | EP0983247A1 Method for producing aromatic bisimides |
| 03/08/2000 | EP0983243A1 Novel quinoline- and naphthalenecarboxamides, pharmaceutical compositions and methods of inhibiting calpain |
| 03/07/2000 | US6034098 Inhibitors of microsomal triglyceride transfer protein and method |
| 03/02/2000 | WO2000011001A1 Muscarinic agonists and antagonists |
| 03/02/2000 | WO1999064043A9 Muscarinic receptor antagonists |
| 03/02/2000 | CA2340946A1 Muscarinic agonists and antagonists |
| 03/01/2000 | EP0982307A2 9 -Amino- and 9-nitro-camptothecin derivatives, process for their preparation and use as antitumor agents |
| 03/01/2000 | EP0981527A1 Salt of naphthyridine carboxylic acid derivative |
| 03/01/2000 | EP0641341B1 METHOD FOR PREPARING BENZO [b]NAPHTHYRIDINES |
| 03/01/2000 | CN1246033A Hexahydroindenopyridine compounds having antispermatogenic activity |
| 02/29/2000 | US6031101 Oxidation process using tempo |
| 02/29/2000 | US6031099 Piperidine derivates having anxiolytic effect |
| 02/29/2000 | US6030982 Analogs of a 4-(2-((3,10-dibromo-8-chloro-4-(2-((3,10-dibromo-8-chloro-6,11 -dihydro-5h-benzo(5,6)-cyclohepta(1,2-b)pyrid-11-yl)-1-piperidinyl)-2 -oxothyl-betaoxo-1-piperidine; antitumor agents |
| 02/29/2000 | US6030981 Phenanthridine derivatives, methods of producing them and medicaments containing phenanthridine derivatives |
| 02/29/2000 | US6030803 Dibenzodihydropyridinecarboxylic esters and their use in chemiluminescent assay methods |
| 02/24/2000 | WO2000009486A1 Substituted isoquinoline derivatives and their use as anticonvulsivants |
| 02/24/2000 | CA2340092A1 Substituted isoquinoline derivatives and their use as anticonvulsivants |
| 02/23/2000 | CN1245499A 8-azabicyclo [3,2,1] octane, 8-azabicyclo [3,2,1] oct-6-ene-,9-azabicyclo [3,2,1] nonane-, 9-aza-3-oxabicyclo [3,3,1] nonane- and 9-aza-3-thiabicyclo[3,3,1] nonane derivatives, their preparation and |
| 02/23/2000 | CN1245429A Leukotriene antagonists for oral squamous cell carcinoma |
| 02/22/2000 | US6028198 Pharmaceutical composition for prevention and treatment of motion sickness syndrome |
| 02/22/2000 | US6028195 Piperazine derivatives and process for the preparation thereof |
| 02/22/2000 | US6028079 Condensed-indan derivatives and pharmaceutically acceptable salts thereof |
| 02/22/2000 | US6028052 Treating NIDDM with RXR agonists |
| 02/17/2000 | DE19830105C1 Acridinderivate Acridine |
| 02/16/2000 | CN1244528A Di- Or triaza-spiral [4,5] decane derivative |
| 02/15/2000 | US6025369 N-methyl-D-aspartate (NMDA) receptor blockers for the prevention of atherosclerosis |
| 02/15/2000 | US6025364 Method of treating asthma |
| 02/15/2000 | US6025355 Substituted indolinyl and derivatives thereof, neurological injury and neurodegenerative disorders. |
| 02/10/2000 | WO2000006577A1 OXAZOLO, THIAZOLO AND SELENAZOLO [4,5-c]-QUINOLIN-4-AMINES AND ANALOGS THEREOF |
| 02/10/2000 | WO2000006569A1 Substituted pyrazole derivatives condensed with six-membered heterocyclic rings |
| 02/10/2000 | WO2000006545A1 High affinity ligands for nociceptin receptor orl-1 |
| 02/10/2000 | WO2000006531A2 Nitric esters and nitrate salts of specific drugs |
| 02/10/2000 | WO2000006167A1 Tricyclic compounds |
| 02/10/2000 | WO1999063944A3 Novel therapeutic agents that modulate estrogen receptors |
| 02/10/2000 | CA2339071A1 Substituted pyrazole derivatives condensed with six-membered heterocyclic rings |
| 02/10/2000 | CA2338298A1 Tricyclic compounds |
| 02/09/2000 | EP0978282A2 Sublingual composition containing apomorphine for diagnosing functional impotence |
| 02/09/2000 | EP0977815A1 ALKYL, ALKENYL AND ALKYNYL CHRYSAMINE G DERIVATIVES FOR THE ANTEMORTEM DIAGNOSIS OF ALZHEIMER'S DISEASE AND $i(IN VIVO) IMAGING AND PREVENTION OF AMYLOID DEPOSITION |
| 02/09/2000 | EP0977739A1 Synthesis of intermediates useful in preparing tricyclic compounds |
| 02/09/2000 | CN1049219C Fused heteroaromatic cyclopentene derivative having endothelin-antagonist activity |
| 02/03/2000 | WO2000005215A1 A process for preparing benzocycloheptapyridin-11-ones |
| 02/03/2000 | WO1999063936A3 Novel therapeutic agents that modulate endothelin receptors |
| 02/03/2000 | WO1999063933A3 Multivalent agonists, partial agonists and antagonists of the gaba receptors |
| 02/03/2000 | WO1999061444A3 Bicyclic pyrimidines and bicyclic 3,4-dihydropyrimidines as inhibitors of cellular proliferation |
| 02/03/2000 | DE19834044A1 Neue substituierte Pyrazolderivate New substituted pyrazole derivatives |
| 02/02/2000 | EP0976732A1 1,4-substituted cyclic amine derivatives |
| 02/02/2000 | CN1243511A Preparation of -3,4-dicarboxylic anhydrides |
| 02/02/2000 | CN1243510A Tricyclicbenzo [3] isoindole and benzo (h) isoquinoline |
| 02/01/2000 | US6020362 Glycoprotein IIB IIIA antagonists |
| 01/27/2000 | WO2000004020A1 Compounds, compositions, and methods for stimulating neuronal growth and elongation |
| 01/27/2000 | WO2000004012A1 COMPOUNDS SPECIFIC FOR THE HUMAN α1d ADRENERGIC RECEPTOR AND USES THEREOF |
| 01/27/2000 | WO1999063930A3 Novel angiotensin receptor modulators and their uses |
| 01/27/2000 | CA2338037A1 Compounds specific for the human .alpha.1d adrenergic receptor and uses thereof |
| 01/27/2000 | CA2337377A1 Compounds, compositions, and methods for stimulating neuronal growth and elongation |
| 01/26/2000 | EP0973737A1 Efficient synthesis of a chiral mediator |
| 01/26/2000 | EP0758895B1 Sublingual dosage forms containing apomorphine for use in the treatment of erectile dysfunction |
| 01/26/2000 | EP0670839B1 Process for the preparation of 9-amino camptothecin |
| 01/26/2000 | CN1242367A Spiro [Piperidine-4,1'-pyrrolo[3,4-c] pyrrole] |
| 01/26/2000 | CN1048719C Novel 7-(substituted)-8-(substituted)-9-(substituted amino)-6-demethyl-6-deoxytetracyclines, prepn. method, their compositions and use thereof |
| 01/26/2000 | CN1048718C Phenylethyl and phenylpropylamines compounds, prepn. method, pharmaceutical agent and use thereof |
| 01/25/2000 | US6017927 Quinuclidine derivatives and medicinal composition thereof |
| 01/20/2000 | WO2000002851A1 Sulfur substituted sulfonylaminocarboxylic acid n-arylamides, their preparation, their use and pharmaceutical preparations comprising them |
| 01/19/2000 | EP0972767A1 CYCLOALKA[b]PYRIDINE-3-CARBONYLGUANIDINE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, AND DRUGS CONTAINING THE SAME |
| 01/19/2000 | EP0971920A1 Compounds for inhibition of gastric acid secretion |
| 01/19/2000 | EP0971899A1 Hexahydroindenopyridine compounds having antispermatogenic activity |
| 01/18/2000 | US6015902 Intercalators having affinity for DNA and methods of use |
| 01/18/2000 | US6015458 Process for the preparation of highly chromatic perylene pigments |
| 01/13/2000 | WO2000001672A1 Naphthalimidobenzamide derivatives |
| 01/12/2000 | EP0970949A1 Acridine derivatives |
| 01/12/2000 | CN1240788A Acridine derivatives |
| 01/11/2000 | US6013803 Reducing aminopiperidine derivative with a reducing agent to reduce the dimers of the compound |
| 01/06/2000 | WO2000000472A1 5-ht7 receptor antagonists |
| 01/06/2000 | WO1999043661A3 Substituted cycloalkyl-4-oxonicotinic carboxamides; gaba brain receptor ligands |
| 01/05/2000 | EP0969003A2 Process for the preparation of benzo[f]quinolinone derivatives and intermediates |
| 01/05/2000 | EP0968250A1 Soluble chromophores having improved solubilising groups |
| 01/05/2000 | EP0968210A1 Method of making arylamino triazolopyridines |
| 01/05/2000 | CN1048015C Bicyclic tetrahydro pyrazolopyridines |
| 12/29/1999 | WO1999067231A1 Nitrate salts of antihypertensive medicines |
| 12/29/1999 | WO1999067220A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis |
| 12/29/1999 | WO1999066944A1 Methods for identifying novel multimeric agents that modulate receptors |
| 12/29/1999 | WO1999058500B1 Method for stereochemically controlled production of isomerically pure highly substituted azacyclic compounds |
| 12/29/1999 | EP0966457A1 Ring opening metathesis of alkenes |
| 12/29/1999 | EP0966443A1 Heteroaryl-hexanoic acid amide derivatives, their preparation and their use as selective inhibitors of mip-1-alpha binding to its ccr1 receptor |
| 12/29/1999 | CN1047774C Prepn. of azadiphenyl cycloheptyl ketenes compound |
| 12/29/1999 | CA2335356A1 Nitrate salts of antihypertensive medicines |
| 12/29/1999 | CA2325388A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis |
| 12/29/1999 | CA2319650A1 Methods for identifying novel multimeric agents that modulate receptors |
| 12/28/1999 | US6008230 Treating bone diseases caused by abnormal bone metabolism in human being or animals as the inhibitors of bone resorption or the inhibitors of bone metastasis |
| 12/23/1999 | WO1999066005A1 Novel chemiluminescent labeling compounds |
| 12/23/1999 | WO1999065878A1 Synthesis of benzo[f]quinolinones |
| 12/23/1999 | CA2334701A1 Synthesis of benzo¬f|quinolinones |
| 12/23/1999 | CA2301120A1 Novel chemiluminescent labeling compounds |