Patents
Patents for C07D 221 - Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups (10,931)
03/2001
03/07/2001EP1080080A1 Novel therapeutic agents that modulate neurokinin receptors
03/07/2001EP1080076A1 Improved method for preparing pharmaceutically valuable norbenzomorphane derivatives
03/07/2001CN1286685A Heterocyclic cytotoxic agents
03/06/2001US6197786 Anticholesterol agents
03/06/2001US6197785 Cardiovascular disorders
03/01/2001WO2001014380A1 Isomeric fused pyrrolocarbazoles and isoindolones
03/01/2001WO2001014375A1 Imidazo[1,2-a]pyridine and pyrazolo[2,3-a]pyridine derivatives
03/01/2001WO2001014328A2 Substituted ureas as cell adhesion inhibitors
03/01/2001DE19940708A1 Thermochrome Rylenfarbstoffe Thermochromic rylene dyes
03/01/2001CA2376293A1 Imidazo[1,2-a]pyridine and pyrazolo[2,3-a]pyridine derivatives
02/2001
02/28/2001EP1077946A1 Fused tricyclic compounds which inhibit parp activity
02/28/2001EP1077944A1 Carboxamide compounds, compositions, and methods for inhibiting parp activity
02/28/2001EP1077928A1 Novel substituted cyclic compounds, preparation method and pharmaceutical compositions containing them
02/28/2001EP1077927A1 Novel substituted cyclic compounds, preparation method and pharmaceutical compositions containing them
02/28/2001CN1285821A Aryl Fused azapolycyclic compounds
02/27/2001US6194439 Tricyclic polyhydroxylic tyrosine kinase inhibitors
02/27/2001US6194427 Brain disorders; psychological disorders; sleep disorders; anticonvulsants
02/27/2001US6194423 Fused isoquinolines as dopamine receptor ligands
02/27/2001US6193992 Administering apomorphine to increase intraclitoral blood flow and vaginal wall blood flow on stimulation but less than amount that induces nausea to treat sexual dysfunction
02/27/2001CA2111204C Piperidine derivatives having anxiolytic effect
02/22/2001WO1999063996A8 Multivalent agonists, partial agonists, inverse agonists and antagonists of the 5ht2 receptors
02/21/2001EP1076650A1 Aryl fused azapolycyclic compounds
02/21/2001EP1076646A1 Method for stereochemically controlled production of isomerically pure highly substituted azacyclic compounds
02/20/2001US6191160 Spiro-indolines as Y5 receptor antagonists
02/20/2001US6191138 Therapy for respiratory system disorders
02/20/2001CA2223624C Tricyclic 5,6-dihydro-9h-pyrazolo[3,4-c]-1,2,4-triazolo[4,3-.alpha.]pyridines
02/15/2001WO2001010840A1 Quaternized azafluorenones and their use in agents for dying fibers containing keratin
02/15/2001DE19937301A1 Quaternierte Azafluorenone und deren Verwendung in Mitteln zum Färben von keratinhaltigen Fasern Quaternized Azafluorenone and their use in compositions for dyeing keratin fibers
02/14/2001EP1075466A1 Cyclopentanone dihydropyridine compounds useful as potassium channel openers
02/14/2001EP0714897B1 Fused heteroaromatic cyclopentene derivative having endothelin-antagonist activity
02/13/2001US6187925 Intermediates and process for the synthesis of azasteroids
02/13/2001US6187783 Antitumor agents
02/08/2001WO2000066528A3 Quinones for treatment of diseases
02/07/2001CN1283186A Indole derivatives as XA factor inhibitors
02/07/2001CN1282738A Improved method for sgnthesizing 6,9-bis[(2-aminoethyl) amino] benz[g] isoquinoline-5, 10-diketone and its dimaleate
02/07/2001CN1061652C Endotheliomycine receptor antagonist
01/2001
01/31/2001EP1072263A1 Amide derivatives and nociceptin antagonists
01/31/2001EP1071666A1 Azacycloalkane derivatives, preparation and therapeutic application
01/31/2001CN1282321A Potassium channel openers
01/30/2001CA2191352C Quinoline derivatives as tachykinin nk3 receptor antagonists
01/30/2001CA1341173C Fungicides
01/25/2001WO2001005765A1 Cyclic amides and imides having selective antagonist activity at alpha-1d adrenergic receptor
01/24/2001EP1070065A1 Azabicyclic 5ht1 receptor ligands
01/24/2001EP1070062A1 Oxidation process using tempo
01/24/2001EP1070052A1 Fungicide compositions comprising a hydroximic or hydrazonic group
01/24/2001CN1281459A Piperidine derivatives
01/24/2001CN1281440A Perylene imide monocarboxylic acids as colorants
01/24/2001CN1281439A 4-Hydroxyquinoline-3-carboxamides and hydrazides as antiviral agents
01/24/2001CN1061044C Tricyclic 5,6-dihydro-9H-pyrazolo [3,4-C]-1,2,4-triaolo [4,3-alpha] pyridines
01/23/2001USRE37029 Antipsychotic and analgesic agents
01/23/2001US6177570 Reaction of dicarboxylic anhydride with an amine in the presence of a tertiary amine.
01/23/2001US6177464 Bactericides
01/23/2001US6177442 Bicyclic amine derivatives
01/23/2001US6177423 N-(hydroxy or protected hydroxy)-benzo(de)isoquinoline-1,3-dione derivatives; bacterial dna gyrase and dna topoisomerase inhibitors useful for antibacterial agents having reduced drug resistance and reduced side effects
01/18/2001WO2001004124A1 OXATHIEPINO[6,5-b]DIHYDROPYRIDINES, AND RELATED COMPOSITIONS AND METHODS
01/18/2001WO2001004094A1 Processes for the preparation of ipidacrine or ipidacrine hydrochloride hydrate
01/18/2001WO2000034245A3 Crystalline form of benzoquinoline-3-one derivatve as inhibitor of 5-alpha reductase
01/18/2001CA2379199A1 Oxathiepino[6,5-b]dihydropyridines, and related compositions and methods
01/18/2001CA2379030A1 Processes for the preparation of ipidacrine or ipidacrine hydrochloride hydrate
01/17/2001EP1068193A1 Benzylpiperazinyl- and benzylpiperidinyl ethanone derivatives, their preparation and their use as dopamine d 4? receptor antagonists
01/17/2001CN1280560A Adamantane derivatives
01/16/2001US6174896 Quinuclidine derivatives and medicinal composition thereof
01/16/2001CA2223404C Novel crystal form of anhydrous 7-(¬1.alpha., 5.alpha., 6.alpha.|-6-amino-3-azabicyclo¬3.1.0|hex-3-yl)-6-fluoro-1-(2,4-difluorophenyl)-1,4-dihydro-4-oxo-1,8-naphthyridine-3-carboxylic acid, methanesulfonic acid salt
01/10/2001EP0777655B1 Process for preparing chiral tetracyclic dopaminergic compounds
01/09/2001US6172113 Bicyclic amino derivatives and PGD2 antagonist containing the same
01/09/2001US6171866 N-substituted iminodiacetic acid derivatives
01/04/2001WO2000030589A3 Synthesis of intermediates useful in preparing tricyclic compounds
01/03/2001EP1064284A1 Hypnotic beta-carboline derivatives, process for their preparation and their use as medicinal products
01/03/2001CN1278797A Oxo-substituted compouns, process of making, and compositions and methods for inhibiting parp activity
01/02/2001US6168776 Alkyl, alkenyl and alkynyl Chrysamine G derivatives for the antemortem diagnosis of Alzheimer's disease and in vivo imaging and prevention of amyloid deposition
01/02/2001CA1341162C Sbustituted aminomethyltetralins and their heterocyclic analogues
12/2000
12/28/2000WO2000078768A1 Potassium channel openers
12/28/2000WO2000078722A1 Process for the preparation of intermediate compounds of drugs
12/28/2000CA2375289A1 Process for the preparation of intermediate compounds of pharmaceuticals
12/28/2000CA2375282A1 Potassium channel openers
12/27/2000EP1061919A1 Novel opiate compounds, methods of making and methods of use
12/27/2000CN1277961A Novel 2,3-methylene amino acid compound, prepn. method therefor, pharmaceutical compositions contg. same
12/26/2000US6166210 Perylene imide monocarboxylic acids
12/26/2000US6166209 Piperidine derivatives
12/21/2000WO2000077010A2 Substituted heterocycle fused gamma-carbolines
12/21/2000WO2000077005A1 Naphthopyrans annelated in c5-c6 with a lactam-type c6 ring and compositions and (co)polymer containing them
12/21/2000WO2000077002A1 Substituted heterocycle fused gamma-carbolines
12/21/2000WO2000077001A1 Substituted heterocycle fused gamma-carbolines
12/21/2000WO2000077000A1 New bispidine compounds useful in the treatment of cardiac arrhythmias
12/21/2000CA2381322A1 Substituted heterocycle fused gamma-carbolines
12/21/2000CA2375857A1 Naphthopyrans annelated in c5-c6 with a lactam-type c6 ring and compositions and (co)polymer containing them
12/21/2000CA2375841A1 New bispidine compounds useful in the treatment of cardiac arrhythmias
12/21/2000CA2374239A1 Substituted heterocycle fused gamma-carbolines
12/21/2000CA2373920A1 Substituted heterocycle fused gamma-carbolines
12/20/2000EP1061076A1 N-acyl cyclic amine derivatives
12/19/2000US6162822 Bisimide compounds
12/14/2000WO2000075236A1 Extended rhodamine compounds useful as fluorescent labels
12/14/2000WO2000075141A1 Bicyclic polyaminoacid metal complexes, method for preparing same and use in medical imaging
12/14/2000WO2000075116A2 Tricyclic analgesics
12/14/2000WO2000074678A1 Analgesics
12/14/2000CA2390948A1 Cell adhesion-inhibiting antiinflammatory compounds
12/14/2000CA2376076A1 Tricyclic analgesics
12/14/2000CA2365075A1 Extended rhodamine compounds useful as fluorescent labels
12/13/2000EP1058698A1 Preparation for prevention and healing of inflammation affections
12/13/2000EP1058549A1 THROMBIN OR FACTOR Xa INHIBITORS
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