Patents
Patents for C07D 221 - Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups (10,931)
12/2004
12/07/2004CA2316921C Aryl fused azapolycyclic compounds
12/02/2004US20040242572 New carboxamide compounds having melanin concentrating hormone antagonistic activity, pharmaceutical preparations comprising these compounds and process for their manufacture
12/02/2004CA2532059A1 Triaza-spiro compounds as nociceptin analogues and uses thereof
12/02/2004CA2526027A1 Process for making spirolactone compounds
12/01/2004EP1481970A1 Novel herbicides
12/01/2004EP1480647A1 Mono-ester and asymmetrically substituted di-ester pro-drugs of the dopamine d1 receptor agonists
12/01/2004EP1480628A1 Use of sodium/hydrogen exchange inhibitors for the treatment of thrombotic and inflammatory diseases
12/01/2004EP0886637B1 Inhibitors of microsomal triglyceride transfer protein and method
12/01/2004CN1177825C Substituted 1,2,3,4,5,6-hexahydro-2,6-methano-3-benzazocines and the use thereof as medicaments
11/2004
11/30/2004US6825351 Selective hydrogenation of amino-substituted fused bicyclic aromatic ring system, preparation of racemic amino substituted fused bicyclic ring system via nitrosation, enzymatic resolution of racemic mixture to produce (r)- and (s)-forms
11/30/2004US6825208 Selective inhibitors of serine protease enzymes, especially factor viia; modulation of the coagulation cascade.
11/30/2004US6824894 Retains high luminance or brightness for a long period and exhibiting a stability
11/30/2004CA2245142C New phenanthridines
11/25/2004WO2004101570A1 Sulfur-containing naphthoylimide derivatives
11/25/2004WO2004100891A2 Cytotoxic indeno and isoindoloisoquinolones
11/25/2004US20040235885 Novel composition and method for stabilizing the same
11/25/2004CA2525099A1 Cytotoxic indeno and isoindoloisoquinolones
11/24/2004EP1478626A2 Guanidino compounds
11/24/2004EP1200406B1 Cyclic amides and imides having selective antagonist activity at alpha-1d adrenergic receptor
11/24/2004EP1185536B1 Hemisynthetic method and intermediates thereof
11/24/2004EP0976732B1 1,4-substituted cyclic amine derivatives
11/24/2004CN1176909C Uses of thaliporphine or its derivatives in treatment of cardiac diseases and preparation of same
11/23/2004CA2171446C Pseudo- and non-peptide bradykinin receptor antagonists
11/18/2004US20040229895 Tetracyclic benzamide derivatives and methods of use thereof
11/18/2004US20040229847 Pyridinone and pyridinethione derivatives having hiv inhibiting properties
11/17/2004EP1477186A1 Antipruritics
11/17/2004EP1476429A1 Novel pyridine- and quinoline-derivatives
11/17/2004EP1476421A2 Novel amino acid derivatives, method for production thereof and pharmaceutical compositions comprising said derivative
11/17/2004EP1289999B1 Antitumoral analogs of et-743
11/17/2004EP1210333B1 p-Tolyl-heterocycles as herbicides
11/17/2004EP1206456B1 Thermochromic rylene dyes
11/17/2004EP1087953B1 Nitrate salts of antihypertensive medicines
11/11/2004WO2004096802A2 ANTIBIOTIC TETRAHYDRO-β-CARBOLINE DERIVATIVES
11/11/2004US20040224969 Salts of substituted 1,2,3,4-tetrahydroquinoline-2-carboxylic acid compounds
11/11/2004US20040224945 Novel substituted pyrazole derivatives
11/11/2004CA2524125A1 Antibiotic tetrahydro-.beta.-carboline derivatives
11/10/2004EP1475379A1 Use of scopine ester derivatives for the synthesis of drugs
11/10/2004EP1474398A1 N-allyloxyethyl-1,2,3,4,5,6-hexahydro-2,6-methano-3-benzazocines and the use of the same as pharmaceuticals
11/10/2004CN1545700A Optical data carrier that contains a cationic aminoheterocyclic dye as the light-absorbing compound in the information layer
11/10/2004CN1545503A Process of synthesis of a tricyclic ketone intermediate
11/10/2004CN1174981C Imidazole [1,2-A] pyridine and pyrazole [2,3-a] pyridine derivatives
11/10/2004CN1174745C Use of coating as taste masking agent for oral preparation
11/09/2004CA2144344C Cyclic benzylamino, benzylamido and benzylimido derivatives as antipsychotic agents
11/04/2004US20040220178 Substituted heterocycle fused gamma-carbolines
11/04/2004US20040219386 4,4'-bis-(spiro 9-fluorene-9'-acridin-10-yl)biphenyl for example, having visible light emissive, hole-transport, electron transport or bipolar-transport properties; use as emissive layer, charge transport layer, or as host material for such layers
11/03/2004CN1542011A Sulphur containing heterocyclic and naphthalimides compound and use thereof
11/03/2004CN1173953C Method for preparing 4-carboxyamino-2-substituted-1,2,3,4-tetrahydroquinoline
10/2004
10/28/2004WO2004091485A2 Aminoquinoline compounds
10/28/2004CA2521808A1 Computer-based model for identification and characterization of non-competitive inhibitors of nicotinic acetylcholine receptors and related ligand-gated ion channel receptors
10/28/2004CA2521619A1 Aminoquinoline compounds
10/27/2004EP1470110A2 Method for the production of substituted 1,2,3,4-tetrahydroquinoline-2-carboxylic acids
10/27/2004EP0929527B1 Pictet-spengler reaction for the synthesis of tetrahydroisoquinolines and related heterocyclic compounds
10/27/2004CN1172917C Steroid receptor modulator compounds and methods
10/26/2004US6809203 Oxazolo, thiazolo and selenazolo [4,5-C]-quinolin-4-amines and analogs thereof
10/26/2004US6809199 (Halo-benzo carbonyl)heterocyclo fused phenyl p38 kinase inhibiting agents
10/26/2004CA2261827C Use of amines to produce drugs for preventing tumour cell proliferation
10/21/2004WO2004089926A2 Genipin derivatives and uses thereof
10/21/2004WO2004089909A1 2-azabicyclo[3.3.1]nonane derivatives as opioid receptor antagonists
10/21/2004WO2004089908A2 3-azabicyclo[3.2.1]octane derivatives
10/21/2004WO2004089307A2 Acylated spiropiperidine derivatives as melanocortin-4 receptor agonists
10/21/2004WO2004072046A3 Quinoline derivatives and their use for modulation of lxr activity
10/21/2004WO2004024728A3 Pyrazolo[3,4-b]pyridine compounds, and their use as phosphodiesterase inhibitors
10/21/2004US20040209902 Aminoquinoline compounds
10/21/2004US20040209876 Bicyclic and tricyclic amines as modulators of chemokine receptor activity
10/21/2004US20040209864 Substituted heterocycle fused gamma-carbolines
10/21/2004US20040209846 Heterocyclic analgesic compounds and methods of use thereof
10/21/2004CA2520114A1 Acylated spiropiperidine derivatives as melanocortin-4 receptor agonists
10/20/2004EP1206473B1 Isomeric fused pyrrolocarbazoles and isoindolones
10/14/2004WO2004086861A2 Fungicidal properties of sampangine and its analogs to agriculturally important fungal plant pathogens
10/14/2004WO2004037853A3 Quinolones with anti-hiv activity
10/14/2004US20040204446 Nitrogen compounds such as N-(2-Fluoro-benzyl)-N-indan-2-yl-2-(3-methyl-2-o-tolyl-piperidin-1-yl) -acetamide, administered for prophylaxis arthritis, psoriasis, cardiovascular disorders, reperfusion injury or respiratory system disorders
10/14/2004US20040204445 2-Azabicyclo[3.3.1]nonane derivatives
10/13/2004EP1465893A1 Derivatives of 5-(pyridin-3-yl)-1-azabicyclo (3.2.1) octane, the preparation thereof and the application of same in therapeutics
10/13/2004EP1465629A1 5-ht3 receptor antagonists and methods of use
10/07/2004WO2003068748A9 Novel pyridine- and quinoline-derivatives
10/07/2004US20040198759 Aporphine and oxoaporphine compounds and pharmaceutical use thereof
10/07/2004US20040198716 Cysteine protease inhimbitors
10/07/2004US20040194665 Perylene derivatives and their application as dispersants
10/06/2004EP1037892B1 Piperidine derivatives
10/05/2004US6800650 For therapy and prophylaxis of diabetes, particularly non-insulin dependent diabetes mellitus and impaired glucose tolerance.
10/05/2004US6800634 Anticancer agents
10/05/2004CA2282834C Novel hexanoic acid derivatives
09/2004
09/30/2004WO2004082698A1 Quaternary chelidonine and alkaloid derivatives, process for their preparation and their use in manufacture of medicaments
09/30/2004WO2004082682A1 Amino cyclobutylamide modulators of chemokine receptor activity
09/30/2004WO2003022785A3 Synthesis of enantiomerically pure amino-substituted fused bicyclic rings
09/30/2004US20040192920 Condensing a suitable alcohol with a piperidone in the presence of polyphosphoric acid.
09/30/2004US20040192721 Fungicidal properties of sampangine and its analogs to agriculturally important fungal plant pathogens
09/30/2004US20040192681 N-acylsulfonamide apoptosis promoters
09/30/2004CA2519220A1 Amino cyclobutylamide modulators of chemokine receptor activity
09/29/2004EP1189905B1 Substituted heterocycle fused gamma-carbolines
09/29/2004CN1532198A Quaternary chelidonine derivatives
09/23/2004US20040186145 Sulfur substituted sulfonylaminocarboxylic acid N-arylamides, their preparation, their use and pharmaceutical preparations comprising them
09/23/2004US20040186132 Steroid receptor modulator compounds and methods
09/23/2004US20040185352 Photothermographic element comprising improved base precursors and methods for their use
09/22/2004EP1460072A1 Bicyclic heteroaromatic compounds as protein tyrosine kinase inhibitors
09/22/2004EP1459753A1 Quaternary chelidonine and alkaloid derivatives, process for their preparation and their use in the manufacture of medicaments
09/22/2004EP1458724A1 Total synthesis of galanthamine, analogues and derivatives thereof
09/22/2004EP1458720A1 1,8-annelated quinoline derivatives substituted with carbon-linked triazoles as farnesyl transferase inhibitors
09/22/2004EP1458677A1 3-phenyl-2-arylalkylthiopropionic acid derivatives as selective agonists of ppar-alpha
09/22/2004EP1458676A2 Compounds for the treatment of inflammatory disorders
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