Patents for C07D 221 - Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups (10,931) |
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08/18/2005 | WO2005075459A1 Synthesis of cyanoimino-benzoimidazoles |
08/18/2005 | WO2005074872A1 Lightening direct dyestuffs for keratin fibers and dyes containing said compounds |
08/18/2005 | US20050182082 Modulators of the glucocorticoid receptor, AP-1, and/or NF-kB activity and use thereof |
08/18/2005 | CA2555219A1 Synthesis of cyanoimino-benzoimidazoles |
08/17/2005 | EP1562943A1 Fused heterocyclic compounds |
08/17/2005 | EP1562593A2 Topoisomerase-targeting agents |
08/17/2005 | EP1200446B1 OXATHIEPINO 6,5- i b /i ]DIHYDROPYRIDINES, AND RELATED COMPOSITIONS AND METHODS |
08/17/2005 | CN1656077A Process for preparing chiral diol sulfones and dihydroxy acid HMG CoA reductase inhibitors |
08/11/2005 | WO2005073204A1 Selective estrogen receptor modulators for the treatment of vasomotor symptoms |
08/11/2005 | WO2005072732A1 Modulators of the glucocorticoid receptor, ap-1, and/or nf-kb activity and use thereof |
08/11/2005 | WO2005051302A3 Bicyclic inhibitors of mek and methods of use thereof |
08/11/2005 | US20050176970 Field-effect transistor; mono- and diimide perylene and naphthalene compounds, core-substituted with one or more electron-withdrawing groups, generating the radical anions electrochemically |
08/11/2005 | US20050176780 2,5-disubstituted 3-mercaptopentanoic acid |
08/11/2005 | US20050176731 N-[5-({(2S)-3-[(4-{4-[(4-benzylpiperidin-1-yl)carbonyl]phenyl}cyclohexyl)amino]-2-hydroxypropyl}oxy)-2-hydroxyphenyl]methanesulfonamide; beta 3 receptors agonist; gastrointestinal diseases; antiobesity, antidiabetic, cicatrizing agents, tocolytics, dysmenorrhea, antiglaucomatous; amidation |
08/11/2005 | US20050176718 Aza- and polyaza-naphthalenyl carboxamides useful as HIV integrase inhibitors |
08/11/2005 | US20050176702 1,8-Annelated quinoline derivatives substituted with carbon-linked triazoles as farnesyl transferase inhibitors |
08/11/2005 | DE102004003735A1 Verfahren zur Herstellung von Terrylen-3,4:11,12-tetracarbonsäurediimiden Process for preparing terylene-3,4: 11,12-tetracarboxylic |
08/11/2005 | DE102004003734A1 Verfahren zur Herstellung von Terrylen-3,4:11,12-tetracarbonsäurediimiden durch Di-rektsynthese Process for preparing terylene-3,4: 11,12-tetracarboxylic by di-rektsynthese |
08/10/2005 | CN1653050A Opioid and opioid-like compounds and uses thereof |
08/10/2005 | CN1652786A Fluorinated 4-azasteroid derivatives as androgen receptor modulators |
08/09/2005 | US6927294 Nitrogen-containing heterocycles |
08/09/2005 | CA2327029C Method for making 4-carboxyamino-2-substituted-1,2,3,4-tetrahydroquinoline |
08/04/2005 | WO2005070895A1 Method for the production of terylene-3,4:11,12-tetracarboxydiimides by direct synthesis |
08/04/2005 | WO2005070894A1 Method for producing terrylen-3,4:11,12-tetracarbon acid di-imids |
08/04/2005 | WO2004091485A3 Aminoquinoline compounds |
08/04/2005 | US20050171355 important intermediate; without using an expensive catalyst and a special facilities; reacting a pyrimidinium derivative such as 1,3-dimethyl-2,3-dihydro-2-oxopyrimidinium chloride, an acetyl compound such as 4-acetylpyridine and an ammonia or an ammonium salt |
08/04/2005 | US20050171352 Process for the preparation of 4-(8-chloro-5 6-dihydro-11h-benzo-(5 6)-cyclohepta-(1 2b)-pyridin-11-ylidene-1-piperidiniecarboxylic acid ethyl ester (loratadine) |
08/04/2005 | US20050171252 provides protection from the damaging effects of light, and at least one organic material; Living and inanimate organic material such as human or animal skin, human or animal hair, paper, foods, perfumes, cosmetics, plastics, polymer dispersions, paints, photographic emulsions, photographic layers, etc |
08/04/2005 | US20050171102 Semicarbazide derivatives for combating thromboembolic diseases |
08/04/2005 | US20050171101 Neurodegenerative diseases; diseases ascribed by NMDA- and NO-induced neurotoxicity ; ischemia; antiinflammatory; anticancer; antidiabetic; 2-{3-[4-Phenyl-3,6-dihydro-1(2H)-pyridyl]propyl}-6(5H)-phenanthridinone |
08/03/2005 | EP1559711A1 Preparation of pyridine derivatives using pyrimidinium derivatives as intermediates |
08/03/2005 | EP1558576A2 Piperidinyl cyclopentyl aryl benzylamide modulators of chemokine receptor activity |
08/03/2005 | EP1558250A1 Gamma-aminoamide modulators of chemokine receptor activity |
08/03/2005 | CN1649967A Method for the production of perylen-3, 4:9, 10-tetracarboxylic acid diimides and perylen-3, 4:9, 10-tetracarboxylic acid dianhydride and naphtalene-1, 8-dicarboxylimides |
08/03/2005 | CN1649867A Novel 1, 2, 3-substituted indolizine derivatives, inhibitors of FGFs, method for making same and pharmaceutical compositions containing same |
08/03/2005 | CN1649845A Muscarinic antagonists |
08/02/2005 | US6923836 Preparation of dyed plastics or polymeric dye particles |
08/02/2005 | CA2132537C Basic derivatives of glutamic acid and aspartic acid as gastrin or cholecystokinin antagonists |
07/28/2005 | US20050165039 Fluorinated 4-azasteroid derivatives as androgen receptor modulators |
07/28/2005 | US20050164883 agronomically tolerable salts, isomers and enantiomers of those compounds, are suitable for use as herbicides |
07/28/2005 | DE10360745A1 Neue Amid-Verbindungen mit MCH-antagonistischer Wirkung und diese Verbindungen enthaltende Arzneimittel New amide compounds with MCH-antagonistic activity and pharmaceutical compositions containing them |
07/27/2005 | EP1557410A2 Bacterial gyrase inhibitors and uses thereof |
07/27/2005 | EP1556382A1 3-phenyl substituted pyridoindolone, preparation and therapeutic use thereof |
07/27/2005 | EP1556358A2 Enantioselective alkylation of tricyclic compounds |
07/27/2005 | EP1287004B1 Synthetic process for the manufacture of an ecteinascidin compound |
07/27/2005 | EP1274411B1 Phenylethylamines and condensed rings variants as prodrugs of catecholamines, and their use |
07/27/2005 | CN1212318C Fluorene-naphthalene imide derivative compound and its application |
07/26/2005 | US6921835 Carbocyclic carboxy amines such as 1-aminomethyl-3,4-dimethyl-cyclopentyl acetic acid or prodrugs used as antiepileptics, antidepressants, anxiolytics, analgesics, antiinflammatory agents and for prophylaxis of neurodegenerative disorders |
07/26/2005 | US6921759 For therapy, prophylaxis or delaying the onset of AIDS and infection by HIV |
07/26/2005 | CA2253948C Carboline derivatives |
07/26/2005 | CA2149007C Cyclohexane derivatives, process for their preparation, and the use of the compounds for the treatment of diseases |
07/21/2005 | WO2005065779A1 Calcitonin gene related peptide receptor antagonists |
07/21/2005 | WO2005043124A3 Chiral 1,8-diarylnaphthalenes, methods of making them, and their use as sensors |
07/21/2005 | WO2005018561A3 Nitrosated and nitrosylated cardiovascular compounds, compositions and methods of use |
07/21/2005 | US20050159487 Cyclic amino acids and derivatives thereof useful as pharmaceutical agents |
07/21/2005 | US20050159440 N-substituted groups such as 3-fluoropropyl; 2,2-dimethylethyl; 2-ethoxyethyl; 2-methoxyethyl; 2-propenyl; 2-propynyl; 2-cyanoethyl; 3-cyanopropyl; 3-iodoprop-(2E)-enyl; 3-iodoprop-(2Z)-enyl; therapy for drug abuse, in particular, cocaine abuse; side effect reduction |
07/21/2005 | CA2549330A1 Calcitonin gene related peptide receptor antagonists |
07/20/2005 | EP1554260A1 Aryloxyalkylamine derivatives as h3 receptor ligands |
07/20/2005 | EP1185493B1 Quinones for treatment of diseases |
07/20/2005 | EP1129077B9 Fluorinated 3,4-dihydroquinoline derivatives used as nos inhibitors |
07/20/2005 | CN1642580A Radiolabelled quinoline and quinolinone derivatives and their use as metabotropic glutamate receptor ligands |
07/20/2005 | CN1640869A Method for preparing 8-chloro-10, 11-dihydro-4-aza-5H-dibenzo[a, d]-5-cycloheptanone |
07/20/2005 | CN1211386C Antitumoral analogue of Et-743 |
07/19/2005 | US6919445 Detecting with a multicolor fluorescent dyes, for automated 4-DNA sequencing systems, identifying the classes of the polynucleotides |
07/14/2005 | WO2005063680A1 Process for the preparation of arylamines |
07/14/2005 | WO2005063239A1 3-(4-piperidine-1ylmethyl-phenyl)-propion acid-phenylamide-derivatives and related compounds used in the form of mch antagonists (melanine concentrating hormone) for treating eating disorders |
07/14/2005 | WO2005062894A2 Co-administration of dopamine-receptor binding compounds |
07/14/2005 | US20050153997 Fredericamycin derivatives |
07/14/2005 | US20050153942 Heterocyclic inhibitors of MEK and methods of use thereof |
07/14/2005 | CA2550650A1 Co-administration of dopamine-receptor binding compounds |
07/14/2005 | CA2550649A1 3-(4-piperidine-1ylmethyl-phenyl)-propion acid-phenylamide-derivatives and related compounds used in the form of mch antagonists (melanine concentrating hormone) for treating eating disorders |
07/13/2005 | CN1638762A Azabicyclic, azatricyclic and azaspirocyclic derivatives of aminocyclohexane NMDA, 5HT3, and neuronal nicotinic receptor antagonists |
07/13/2005 | CN1636982A Synthesis of intermediates useful in preparing tricyclic compounds |
07/12/2005 | US6916830 Substituted tetrahydroisoquinolines as C5a receptor modulators |
07/12/2005 | US6916823 Method of treatment of dopamine-related dysfunction |
07/07/2005 | WO2005047258A3 Methods and compositions for selectin inhibition |
07/07/2005 | WO2004048340A8 Sinomenine and sinomenine compounds, synthesis and use |
07/07/2005 | US20050148591 Tartrate salts of 5,8,14-triazatetracyclo [10.3.1.02,11.04,9]-hexadeca-2(11),3,5,7,9-pentaen and pharmaceutical compositions thereof |
07/07/2005 | CA2548494A1 Novel tricyclic spiroderivatives as modulators of chemokine receptor activity |
07/07/2005 | CA2547814A1 Spiropiperidine derivatives for controlling pests |
07/06/2005 | EP1280809B1 Antitumoral ecteinascidin derivatives |
07/06/2005 | CN1635998A Tricyclic analgesics |
07/06/2005 | CN1634894A Spiro[benzocyclo-4'-piperidine-2'-one] template compound and method for preparing same |
07/06/2005 | CN1634893A 4, 5-disubstituted-1, 8-naphthoyl imide compounds and use thereof |
06/30/2005 | WO2005058836A1 Insecticidal spiroindane derivatives |
06/30/2005 | WO2005058298A2 Fk228 analogs and their use as hdac-inhibitors |
06/30/2005 | WO2004089926A3 Genipin derivatives and uses thereof |
06/30/2005 | US20050143408 Aporphine esters and their use in therapy |
06/30/2005 | CA2557004A1 Pyrazolo [3,4-b] pyridine compounds, and their use as phosphodiesterase inhibitors |
06/29/2005 | EP1545502A2 Keto cannabinoids with therapeutic indications |
06/29/2005 | EP1373272B1 Tert. alkylphenoxy substituted polycyclic compounds |
06/29/2005 | CN1633472A Thermochromic rylene dyes |
06/29/2005 | CN1633412A Novel amino acid derivatives, method for production thereof and pharmaceutical compositions comprising said derivative |
06/23/2005 | WO2004089307A8 Acylated spiropiperidine derivatives as melanocortin-4 receptor agonists |
06/22/2005 | EP1542990A1 Novel imidazole compounds as transforming growth factor (tgf) inhibitors |
06/22/2005 | EP1542983A1 Heterodiamondoids |
06/22/2005 | EP1542975A2 9-cyano-substituted perylene-3,4-dicarboxylic acid monoimides |
06/22/2005 | CN1630641A Farnesyl protein transferase inhibitors as antitumor agents |
06/22/2005 | CN1630639A Novel pyridine- and quinoline-derivatives |
06/22/2005 | CN1207285C Method of extracting Huperzine A from Chinese herbal medicine multi-layer tower |